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Titolo Data di pubblicazione Autore(i) File
Synthesis of New Classes of MMPs Sugars-Based Inhibitors 1-gen-2014 Gragnani, Tiziana; D'Andrea, Felicia; Cuffaro, D.; Giorgelli, Francesco; Nuti, Elisa; Rosalia, Lea; Orlandini, Elisabetta; Rossello, Armando
New arylsulfonamido-based MMP inhibitors with improved water solubility 1-gen-2016 Cuffaro, Doretta; D'Andrea, Felicia; Cargioli, Laura; Nuti, Elisa; Rossello, Armando
Sugar-Based Arylsulfonamide Carboxylates as Selective and Water-Soluble Matrix Metalloproteinase-12 Inhibitors 1-gen-2016 Nuti, Elisa; Cuffaro, Doretta; D'Andrea, Felicia; Rosalia, Lea; Tepshi, Livia; Fabbi, Marina; Carbotti, Grazia; Ferrini, Silvano; Santamaria, Salvatore; Camodeca, Caterina; Ciccone, Lidia; Orlandini, Elisabetta; Nencetti, Susanna; Stura, Enrico A.; Dive, Vincent; Rossello, Armando
Crystal structure of the catalytic domain of MMP-12 in complex with a selective sugar-conjugated arylsulfonamide carboxylate water-soluble inhibitor (DC27) 1-gen-2016 Stura, E. A.; Rosalia, L.; Cuffaro, D.; Tepshi, L.; Ciccone, L.; Rossello, A.
Crystal structure of the catalytic domain of MMP-9 in complex with a selective sugar-conjugated arylsulfonamide carboxylate water-soluble inhibitor (DC27) 1-gen-2016 Stura, E. A.; Rosalia, L.; Cuffaro, D.; Tepshi, L.; Ciccone, L.; Rossello, A.
Crystal structure of the catalytic domain of MMP-12 in complex with a selective sugar-conjugated thiourea-linked carboxylate zinc-chelator water-soluble inhibitor (DC31) 1-gen-2016 Stura, E. A.; Rosalia, L.; Cuffaro, D.; Tepshi, L.; Ciccone, L.; Rossello, A.
Crystal structure of the catalytic domain of MMP-12 in complex with a selective sugar-conjugated triazole-linked carboxylate chelating water-soluble inhibitor (DC24) 1-gen-2016 Stura, E. A.; Rosalia, L.; Cuffaro, D.; Tepshi, L.; Ciccone, L.; Rossello, A.
Crystal structure of the catalytic domain of MMP-12 in complex with a selective sugar-conjugated triazole-linked carboxylate chelator water-soluble inhibitor (DC32) 1-gen-2016 Stura, E. A.; Rosalia, L.; Cuffaro, D.; Tepshi, L.; Ciccone, L.; Rossello, A.
Crystal structure of the catalytic domain of MMP-12 in complex with a selective sugar-conjugated triazole-linked carboxylate zinc-chelator water-soluble inhibitor (DC28) 1-gen-2016 Stura, E. A.; Rosalia, L.; Cuffaro, D.; Tepshi, L.; Ciccone, L.; Rossello, A.
SUGAR-BASED ARYLSULFONAMIDE CARBOXYLATES AS SELECTIVE AND WATER SOLUBLE MMP-12 INHIBITORS 1-gen-2016 Cuffaro, Doretta; Nuti, Elisa; D'Andrea, Felicia; Enrico A., Stura; Grazia, Carbotti; Marina, Fabbi; Silvano, Ferrini; Rossello, Armando
Bifunctional Inhibitors as a New Tool To Reduce Cancer Cell Invasion by Impairing MMP-9 Homodimerization 1-gen-2017 Nuti, Elisa; Rosalia, Lea; Cuffaro, Doretta; Camodeca, Caterina; Giacomelli, Chiara; DA POZZO, Eleonora; Tuccinardi, Tiziano; Costa, Barbara; Antoni, Claudia; Vera, Laura; Ciccone, Lidia; Orlandini, Elisabetta; Nencetti, Susanna; Dive, Vincent; Martini, Claudia; Stura, Enrico A.; Rossello, Armando
Matrix metalloproteinase-12 inhibitors: synthesis, structure-activity relationships and intestinal absorption of novel sugar-based biphenylsulfonamide carboxylates 1-gen-2018 Cuffaro, Doretta; Camodeca, Caterina; D'Andrea, Felicia; Piragine, Eugenia; Testai, Lara; Calderone, Vincenzo; Orlandini, Elisabetta; Nuti, Elisa; Rossello, Armando
Development of Thioaryl-Based Matrix Metalloproteinase-12 Inhibitors with Alternative Zinc-Binding Groups: Synthesis, Potentiometric, NMR, and Crystallographic Studies 1-gen-2018 Nuti, Elisa; Cuffaro, Doretta; Bernardini, Elisa; Camodeca, Caterina; Panelli, Laura; Chaves, Sílvia; Ciccone, Lidia; Tepshi, Livia; Vera, Laura; Orlandini, Elisabetta; Nencetti, Susanna; Stura, Enrico A.; Santos, M. Amélia; Dive, Vincent; Rossello, Armando
Selectively Charged and Zwitterionic Analogues of the Smallest Immunogenic Structure of Streptococcus Pneumoniae Type 14 1-gen-2019 Gragnani, Tiziana; Cuffaro, Doretta; Fallarini, Silvia; Lombardi, Grazia; D'Andrea, Felicia; Guazzelli, Lorenzo
Preparation of 1,6-di-deoxy-D-galacto and 1,6-di-deoxy-L-altro nojirimycin derivatives by aminocyclization of a 1,5-dicarbonyl derivative 1-gen-2019 Cuffaro, D.; Landi, M.; D'Andrea, F.; Guazzelli, L.
Age-related macular degeneration: Current knowledge of zinc metalloproteinases involvement 1-gen-2019 Liva, Francesca; Cuffaro, D.; Nuti, E.; Nencetti, S.; Orlandini, E.; Vozzi, G.; Rossello, A.
Design and Synthesis of Ionic Liquid-Based Matrix Metalloproteinase Inhibitors (MMPIs): A Simple Approach to Increase Hydrophilicity and to Develop MMPI-Coated Gold Nanoparticles 1-gen-2019 D'Andrea, Felicia; Nuti, Elisa; Becherini, Stefano; Cuffaro, Doretta; Husanu, Elena; Camodeca, Caterina; De Vita, Elena; Zocchi, Maria Raffaella; Poggi, Alessandro; D'Arrigo, Cristina; Cappello, Valentina; Gemmi, Mauro; Nencetti, Susanna; Chiappe, Cinzia; Rossello, Armando
Design, synthesis and biological evaluation of bifunctional inhibitors of membrane type 1 matrix metalloproteinase (MT1-MMP) 1-gen-2019 Cuffaro, Doretta; Nuti, Elisa; Gifford, Valentina; Ito, Noriko; Camodeca, Caterina; Tuccinardi, Tiziano; Nencetti, Susanna; Orlandini, Elisabetta; Itoh, Yoshifumi; Rossello, Armando
ADAM metalloproteinases as potential drug targets 1-gen-2019 Camodeca, Caterina; Cuffaro, Doretta; Nuti, Elisa; Rossello, Armando
Identification of histone deacetylase inhibitors with (arylidene)aminoxy scaffold active in uveal melanoma cell lines 1-gen-2020 Nencetti, S.; Cuffaro, D.; Nuti, E.; Ciccone, L.; Rossello, A.; Fabbi, M.; Ballante, F.; Ortore, G.; Carbotti, G.; Campelli, F.; Banti, I.; Gangemi, R.; Marshall, G. R.; Orlandini, E.
Mostra risultati da 1 a 20 di 45
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