Sfoglia per Autore
Synthesis of New Classes of MMPs Sugars-Based Inhibitors
2014-01-01 Gragnani, Tiziana; D'Andrea, Felicia; Cuffaro, D.; Giorgelli, Francesco; Nuti, Elisa; Rosalia, Lea; Orlandini, Elisabetta; Rossello, Armando
New arylsulfonamido-based MMP inhibitors with improved water solubility
2016-01-01 Cuffaro, Doretta; D'Andrea, Felicia; Cargioli, Laura; Nuti, Elisa; Rossello, Armando
Sugar-Based Arylsulfonamide Carboxylates as Selective and Water-Soluble Matrix Metalloproteinase-12 Inhibitors
2016-01-01 Nuti, Elisa; Cuffaro, Doretta; D'Andrea, Felicia; Rosalia, Lea; Tepshi, Livia; Fabbi, Marina; Carbotti, Grazia; Ferrini, Silvano; Santamaria, Salvatore; Camodeca, Caterina; Ciccone, Lidia; Orlandini, Elisabetta; Nencetti, Susanna; Stura, Enrico A.; Dive, Vincent; Rossello, Armando
Crystal structure of the catalytic domain of MMP-12 in complex with a selective sugar-conjugated arylsulfonamide carboxylate water-soluble inhibitor (DC27)
2016-01-01 Stura, E. A.; Rosalia, L.; Cuffaro, D.; Tepshi, L.; Ciccone, L.; Rossello, A.
Crystal structure of the catalytic domain of MMP-9 in complex with a selective sugar-conjugated arylsulfonamide carboxylate water-soluble inhibitor (DC27)
2016-01-01 Stura, E. A.; Rosalia, L.; Cuffaro, D.; Tepshi, L.; Ciccone, L.; Rossello, A.
Crystal structure of the catalytic domain of MMP-12 in complex with a selective sugar-conjugated thiourea-linked carboxylate zinc-chelator water-soluble inhibitor (DC31)
2016-01-01 Stura, E. A.; Rosalia, L.; Cuffaro, D.; Tepshi, L.; Ciccone, L.; Rossello, A.
Crystal structure of the catalytic domain of MMP-12 in complex with a selective sugar-conjugated triazole-linked carboxylate chelating water-soluble inhibitor (DC24)
2016-01-01 Stura, E. A.; Rosalia, L.; Cuffaro, D.; Tepshi, L.; Ciccone, L.; Rossello, A.
Crystal structure of the catalytic domain of MMP-12 in complex with a selective sugar-conjugated triazole-linked carboxylate chelator water-soluble inhibitor (DC32)
2016-01-01 Stura, E. A.; Rosalia, L.; Cuffaro, D.; Tepshi, L.; Ciccone, L.; Rossello, A.
Crystal structure of the catalytic domain of MMP-12 in complex with a selective sugar-conjugated triazole-linked carboxylate zinc-chelator water-soluble inhibitor (DC28)
2016-01-01 Stura, E. A.; Rosalia, L.; Cuffaro, D.; Tepshi, L.; Ciccone, L.; Rossello, A.
SUGAR-BASED ARYLSULFONAMIDE CARBOXYLATES AS SELECTIVE AND WATER SOLUBLE MMP-12 INHIBITORS
2016-01-01 Cuffaro, Doretta; Nuti, Elisa; D'Andrea, Felicia; Enrico A., Stura; Grazia, Carbotti; Marina, Fabbi; Silvano, Ferrini; Rossello, Armando
Bifunctional Inhibitors as a New Tool To Reduce Cancer Cell Invasion by Impairing MMP-9 Homodimerization
2017-01-01 Nuti, Elisa; Rosalia, Lea; Cuffaro, Doretta; Camodeca, Caterina; Giacomelli, Chiara; DA POZZO, Eleonora; Tuccinardi, Tiziano; Costa, Barbara; Antoni, Claudia; Vera, Laura; Ciccone, Lidia; Orlandini, Elisabetta; Nencetti, Susanna; Dive, Vincent; Martini, Claudia; Stura, Enrico A.; Rossello, Armando
Matrix metalloproteinase-12 inhibitors: synthesis, structure-activity relationships and intestinal absorption of novel sugar-based biphenylsulfonamide carboxylates
2018-01-01 Cuffaro, Doretta; Camodeca, Caterina; D'Andrea, Felicia; Piragine, Eugenia; Testai, Lara; Calderone, Vincenzo; Orlandini, Elisabetta; Nuti, Elisa; Rossello, Armando
Development of Thioaryl-Based Matrix Metalloproteinase-12 Inhibitors with Alternative Zinc-Binding Groups: Synthesis, Potentiometric, NMR, and Crystallographic Studies
2018-01-01 Nuti, Elisa; Cuffaro, Doretta; Bernardini, Elisa; Camodeca, Caterina; Panelli, Laura; Chaves, Sílvia; Ciccone, Lidia; Tepshi, Livia; Vera, Laura; Orlandini, Elisabetta; Nencetti, Susanna; Stura, Enrico A.; Santos, M. Amélia; Dive, Vincent; Rossello, Armando
Selectively Charged and Zwitterionic Analogues of the Smallest Immunogenic Structure of Streptococcus Pneumoniae Type 14
2019-01-01 Gragnani, Tiziana; Cuffaro, Doretta; Fallarini, Silvia; Lombardi, Grazia; D'Andrea, Felicia; Guazzelli, Lorenzo
Preparation of 1,6-di-deoxy-D-galacto and 1,6-di-deoxy-L-altro nojirimycin derivatives by aminocyclization of a 1,5-dicarbonyl derivative
2019-01-01 Cuffaro, D.; Landi, M.; D'Andrea, F.; Guazzelli, L.
Age-related macular degeneration: Current knowledge of zinc metalloproteinases involvement
2019-01-01 Liva, Francesca; Cuffaro, D.; Nuti, E.; Nencetti, S.; Orlandini, E.; Vozzi, G.; Rossello, A.
Design and Synthesis of Ionic Liquid-Based Matrix Metalloproteinase Inhibitors (MMPIs): A Simple Approach to Increase Hydrophilicity and to Develop MMPI-Coated Gold Nanoparticles
2019-01-01 D'Andrea, Felicia; Nuti, Elisa; Becherini, Stefano; Cuffaro, Doretta; Husanu, Elena; Camodeca, Caterina; De Vita, Elena; Zocchi, Maria Raffaella; Poggi, Alessandro; D'Arrigo, Cristina; Cappello, Valentina; Gemmi, Mauro; Nencetti, Susanna; Chiappe, Cinzia; Rossello, Armando
Design, synthesis and biological evaluation of bifunctional inhibitors of membrane type 1 matrix metalloproteinase (MT1-MMP)
2019-01-01 Cuffaro, Doretta; Nuti, Elisa; Gifford, Valentina; Ito, Noriko; Camodeca, Caterina; Tuccinardi, Tiziano; Nencetti, Susanna; Orlandini, Elisabetta; Itoh, Yoshifumi; Rossello, Armando
ADAM metalloproteinases as potential drug targets
2019-01-01 Camodeca, Caterina; Cuffaro, Doretta; Nuti, Elisa; Rossello, Armando
Identification of histone deacetylase inhibitors with (arylidene)aminoxy scaffold active in uveal melanoma cell lines
2020-01-01 Nencetti, S.; Cuffaro, D.; Nuti, E.; Ciccone, L.; Rossello, A.; Fabbi, M.; Ballante, F.; Ortore, G.; Carbotti, G.; Campelli, F.; Banti, I.; Gangemi, R.; Marshall, G. R.; Orlandini, E.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Synthesis of New Classes of MMPs Sugars-Based Inhibitors | 1-gen-2014 | Gragnani, Tiziana; D'Andrea, Felicia; Cuffaro, D.; Giorgelli, Francesco; Nuti, Elisa; Rosalia, Lea; Orlandini, Elisabetta; Rossello, Armando | |
New arylsulfonamido-based MMP inhibitors with improved water solubility | 1-gen-2016 | Cuffaro, Doretta; D'Andrea, Felicia; Cargioli, Laura; Nuti, Elisa; Rossello, Armando | |
Sugar-Based Arylsulfonamide Carboxylates as Selective and Water-Soluble Matrix Metalloproteinase-12 Inhibitors | 1-gen-2016 | Nuti, Elisa; Cuffaro, Doretta; D'Andrea, Felicia; Rosalia, Lea; Tepshi, Livia; Fabbi, Marina; Carbotti, Grazia; Ferrini, Silvano; Santamaria, Salvatore; Camodeca, Caterina; Ciccone, Lidia; Orlandini, Elisabetta; Nencetti, Susanna; Stura, Enrico A.; Dive, Vincent; Rossello, Armando | |
Crystal structure of the catalytic domain of MMP-12 in complex with a selective sugar-conjugated arylsulfonamide carboxylate water-soluble inhibitor (DC27) | 1-gen-2016 | Stura, E. A.; Rosalia, L.; Cuffaro, D.; Tepshi, L.; Ciccone, L.; Rossello, A. | |
Crystal structure of the catalytic domain of MMP-9 in complex with a selective sugar-conjugated arylsulfonamide carboxylate water-soluble inhibitor (DC27) | 1-gen-2016 | Stura, E. A.; Rosalia, L.; Cuffaro, D.; Tepshi, L.; Ciccone, L.; Rossello, A. | |
Crystal structure of the catalytic domain of MMP-12 in complex with a selective sugar-conjugated thiourea-linked carboxylate zinc-chelator water-soluble inhibitor (DC31) | 1-gen-2016 | Stura, E. A.; Rosalia, L.; Cuffaro, D.; Tepshi, L.; Ciccone, L.; Rossello, A. | |
Crystal structure of the catalytic domain of MMP-12 in complex with a selective sugar-conjugated triazole-linked carboxylate chelating water-soluble inhibitor (DC24) | 1-gen-2016 | Stura, E. A.; Rosalia, L.; Cuffaro, D.; Tepshi, L.; Ciccone, L.; Rossello, A. | |
Crystal structure of the catalytic domain of MMP-12 in complex with a selective sugar-conjugated triazole-linked carboxylate chelator water-soluble inhibitor (DC32) | 1-gen-2016 | Stura, E. A.; Rosalia, L.; Cuffaro, D.; Tepshi, L.; Ciccone, L.; Rossello, A. | |
Crystal structure of the catalytic domain of MMP-12 in complex with a selective sugar-conjugated triazole-linked carboxylate zinc-chelator water-soluble inhibitor (DC28) | 1-gen-2016 | Stura, E. A.; Rosalia, L.; Cuffaro, D.; Tepshi, L.; Ciccone, L.; Rossello, A. | |
SUGAR-BASED ARYLSULFONAMIDE CARBOXYLATES AS SELECTIVE AND WATER SOLUBLE MMP-12 INHIBITORS | 1-gen-2016 | Cuffaro, Doretta; Nuti, Elisa; D'Andrea, Felicia; Enrico A., Stura; Grazia, Carbotti; Marina, Fabbi; Silvano, Ferrini; Rossello, Armando | |
Bifunctional Inhibitors as a New Tool To Reduce Cancer Cell Invasion by Impairing MMP-9 Homodimerization | 1-gen-2017 | Nuti, Elisa; Rosalia, Lea; Cuffaro, Doretta; Camodeca, Caterina; Giacomelli, Chiara; DA POZZO, Eleonora; Tuccinardi, Tiziano; Costa, Barbara; Antoni, Claudia; Vera, Laura; Ciccone, Lidia; Orlandini, Elisabetta; Nencetti, Susanna; Dive, Vincent; Martini, Claudia; Stura, Enrico A.; Rossello, Armando | |
Matrix metalloproteinase-12 inhibitors: synthesis, structure-activity relationships and intestinal absorption of novel sugar-based biphenylsulfonamide carboxylates | 1-gen-2018 | Cuffaro, Doretta; Camodeca, Caterina; D'Andrea, Felicia; Piragine, Eugenia; Testai, Lara; Calderone, Vincenzo; Orlandini, Elisabetta; Nuti, Elisa; Rossello, Armando | |
Development of Thioaryl-Based Matrix Metalloproteinase-12 Inhibitors with Alternative Zinc-Binding Groups: Synthesis, Potentiometric, NMR, and Crystallographic Studies | 1-gen-2018 | Nuti, Elisa; Cuffaro, Doretta; Bernardini, Elisa; Camodeca, Caterina; Panelli, Laura; Chaves, Sílvia; Ciccone, Lidia; Tepshi, Livia; Vera, Laura; Orlandini, Elisabetta; Nencetti, Susanna; Stura, Enrico A.; Santos, M. Amélia; Dive, Vincent; Rossello, Armando | |
Selectively Charged and Zwitterionic Analogues of the Smallest Immunogenic Structure of Streptococcus Pneumoniae Type 14 | 1-gen-2019 | Gragnani, Tiziana; Cuffaro, Doretta; Fallarini, Silvia; Lombardi, Grazia; D'Andrea, Felicia; Guazzelli, Lorenzo | |
Preparation of 1,6-di-deoxy-D-galacto and 1,6-di-deoxy-L-altro nojirimycin derivatives by aminocyclization of a 1,5-dicarbonyl derivative | 1-gen-2019 | Cuffaro, D.; Landi, M.; D'Andrea, F.; Guazzelli, L. | |
Age-related macular degeneration: Current knowledge of zinc metalloproteinases involvement | 1-gen-2019 | Liva, Francesca; Cuffaro, D.; Nuti, E.; Nencetti, S.; Orlandini, E.; Vozzi, G.; Rossello, A. | |
Design and Synthesis of Ionic Liquid-Based Matrix Metalloproteinase Inhibitors (MMPIs): A Simple Approach to Increase Hydrophilicity and to Develop MMPI-Coated Gold Nanoparticles | 1-gen-2019 | D'Andrea, Felicia; Nuti, Elisa; Becherini, Stefano; Cuffaro, Doretta; Husanu, Elena; Camodeca, Caterina; De Vita, Elena; Zocchi, Maria Raffaella; Poggi, Alessandro; D'Arrigo, Cristina; Cappello, Valentina; Gemmi, Mauro; Nencetti, Susanna; Chiappe, Cinzia; Rossello, Armando | |
Design, synthesis and biological evaluation of bifunctional inhibitors of membrane type 1 matrix metalloproteinase (MT1-MMP) | 1-gen-2019 | Cuffaro, Doretta; Nuti, Elisa; Gifford, Valentina; Ito, Noriko; Camodeca, Caterina; Tuccinardi, Tiziano; Nencetti, Susanna; Orlandini, Elisabetta; Itoh, Yoshifumi; Rossello, Armando | |
ADAM metalloproteinases as potential drug targets | 1-gen-2019 | Camodeca, Caterina; Cuffaro, Doretta; Nuti, Elisa; Rossello, Armando | |
Identification of histone deacetylase inhibitors with (arylidene)aminoxy scaffold active in uveal melanoma cell lines | 1-gen-2020 | Nencetti, S.; Cuffaro, D.; Nuti, E.; Ciccone, L.; Rossello, A.; Fabbi, M.; Ballante, F.; Ortore, G.; Carbotti, G.; Campelli, F.; Banti, I.; Gangemi, R.; Marshall, G. R.; Orlandini, E. |
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