Sfoglia per Autore
Mimicking the intramolecular hydrogen bond: Synthesis, biological evaluation, andmolecular modeling of benzoxazines and quinazolines as potential antimalarial agents
2012-01-01 Gemma, S.; Camodeca, C.; Brindisi, M.; Brogi, S.; Kukreja, G.; Kunjir, S.; Gabellieri, E.; Lucantoni, L.; Habluetzel, A.; Taramelli, D.; Basilico, N.; Gualdani, R.; Tadini-Buoninsegni, F.; Bartolommei, G.; Moncelli, M. R.; Martin, R. E.; Summers, R. L.; Lamponi, S.; Savini, L.; Fiorini, I.; Valoti, M.; Novellino, E.; Campiani, G.; Butini, S.
Optimization of 4-aminoquinoline/clotrimazole-based hybrid antimalarials: Further structure-activity relationships, in vivo studies, and preliminary toxicity profiling
2012-01-01 Gemma, S.; Camodeca, C.; Sanna Coccone, S.; Joshi, B. P.; Bernetti, M.; Moretti, V.; Brogi, S.; De Marcos, M. C. B.; Savini, L.; Taramelli, D.; Basilico, N.; Parapini, S.; Rottmann, M.; Brun, R.; Lamponi, S.; Caccia, S.; Guiso, G.; Summers, R. L.; Martin, R. E.; Saponara, S.; Gorelli, B.; Novellino, E.; Campiani, G.; Butini, S.
N-O-Isopropyl Sulfonamido-Based Hydroxamates as Matrix Metalloproteinase Inhibitors: Hit Selection and in Vivo Antiangiogenic Activity
2015-01-01 Nuti, Elisa; Cantelmo, Anna Rita; Gallo, Cristina; Bruno, Antonino; Bassani, Barbara; Camodeca, Caterina; Tuccinardi, Tiziano; Vera, Laura; Orlandini, Elisabetta; Nencetti, Susanna; Stura, Enrico A; Martinelli, Adriano; Dive, Vincent; Albini, Adriana; Rossello, Armando
MMP-8 Is Critical for Dexamethasone Therapy in Alkali-Burned Corneas Under Dry Eye Conditions
2016-01-01 Bian, Fang; Wang, Changjun; Tukler Henriksson, Johanna; Pflugfelder, Stephen C.; Camodeca, Caterina; Nuti, Elisa; Rossello, Armando; Li, De Quan; de Paiva, Cintia S.
Synthesis, experimental evaluation and molecular modelling of hydroxamate derivatives as zinc metalloproteinase inhibitors
2016-01-01 Sjøli, Stian; Nuti, Elisa; Camodeca, Caterina; Bilto, Irina; Rossello, Armando; Winberg, Jan Olof; Sylte, Ingebrigt; Adekoya, Olayiwola A.
Sugar-Based Arylsulfonamide Carboxylates as Selective and Water-Soluble Matrix Metalloproteinase-12 Inhibitors
2016-01-01 Nuti, Elisa; Cuffaro, Doretta; D'Andrea, Felicia; Rosalia, Lea; Tepshi, Livia; Fabbi, Marina; Carbotti, Grazia; Ferrini, Silvano; Santamaria, Salvatore; Camodeca, Caterina; Ciccone, Lidia; Orlandini, Elisabetta; Nencetti, Susanna; Stura, Enrico A.; Dive, Vincent; Rossello, Armando
ADAM10 new selective inhibitors reduce NKG2D ligand release sensitizing Hodgkin lymphoma cells to NKG2D-mediated killing
2016-01-01 Zocchi, Maria Raffaella; Camodeca, Caterina; Nuti, Elisa; Rossello, Armando; Venè, Roberta; Tosetti, Francesca; Dapino, Irene; Costa, Delfina; Musso, Alessandra; Poggi, Alessandro
Discovery of a new selective inhibitor of A Disintegrin And Metalloprotease 10 (ADAM-10) able to reduce the shedding of NKG2D ligands in Hodgkin's lymphoma cell models
2016-01-01 Camodeca, Caterina; Nuti, Elisa; Tepshi, Livia; Boero, Silvia; Tuccinardi, Tiziano; Stura, Enrico A; Poggi, Alessandro; Zocchi, Maria Raffaella; Rossello, Armando
Bifunctional Inhibitors as a New Tool To Reduce Cancer Cell Invasion by Impairing MMP-9 Homodimerization
2017-01-01 Nuti, Elisa; Rosalia, Lea; Cuffaro, Doretta; Camodeca, Caterina; Giacomelli, Chiara; DA POZZO, Eleonora; Tuccinardi, Tiziano; Costa, Barbara; Antoni, Claudia; Vera, Laura; Ciccone, Lidia; Orlandini, Elisabetta; Nencetti, Susanna; Dive, Vincent; Martini, Claudia; Stura, Enrico A.; Rossello, Armando
Synthesis and antiangiogenic activity study of new hop chalcone Xanthohumol analogues
2017-01-01 Nuti, Elisa; Bassani, Barbara; Camodeca, Caterina; Rosalia, Lea; Cantelmo, Annarita; Gallo, Cristina; Baci, Denisa; Bruno, Antonino; Orlandini, Elisabetta; Nencetti, Susanna; Noonan, Douglas M.; Albini, Adriana; Rossello, Armando
Development of Thioaryl-Based Matrix Metalloproteinase-12 Inhibitors with Alternative Zinc-Binding Groups: Synthesis, Potentiometric, NMR, and Crystallographic Studies
2018-01-01 Nuti, Elisa; Cuffaro, Doretta; Bernardini, Elisa; Camodeca, Caterina; Panelli, Laura; Chaves, Sílvia; Ciccone, Lidia; Tepshi, Livia; Vera, Laura; Orlandini, Elisabetta; Nencetti, Susanna; Stura, Enrico A.; Santos, M. Amélia; Dive, Vincent; Rossello, Armando
Specific ADAM10 inhibitors localize in exosome-like vesicles released by Hodgkin lymphoma and stromal cells and prevent sheddase activity carried to bystander cells
2018-01-01 Tosetti, Francesca; Venè, Roberta; Camodeca, Caterina; Nuti, Elisa; Rossello, Armando; D'Arrigo, Cristina; Galante, Denise; Ferrari, Nicoletta; Poggi, Alessandro; Zocchi, Maria Raffaella
Matrix metalloproteinase-12 inhibitors: synthesis, structure-activity relationships and intestinal absorption of novel sugar-based biphenylsulfonamide carboxylates
2018-01-01 Cuffaro, Doretta; Camodeca, Caterina; D'Andrea, Felicia; Piragine, Eugenia; Testai, Lara; Calderone, Vincenzo; Orlandini, Elisabetta; Nuti, Elisa; Rossello, Armando
Synthesis and in vitro Evaluation of ADAM10 and ADAM17 Highly Selective Bioimaging Probes
2018-01-01 Camodeca, Caterina; Nuti, Elisa; Tosetti, Francesca; Poggi, Alessandro; D'Arrigo, Cristina; Zocchi, Maria Raffaella; Rossello, Armando
Design, synthesis and biological evaluation of bifunctional inhibitors of membrane type 1 matrix metalloproteinase (MT1-MMP)
2019-01-01 Cuffaro, Doretta; Nuti, Elisa; Gifford, Valentina; Ito, Noriko; Camodeca, Caterina; Tuccinardi, Tiziano; Nencetti, Susanna; Orlandini, Elisabetta; Itoh, Yoshifumi; Rossello, Armando
ADAM metalloproteinases as potential drug targets
2019-01-01 Camodeca, Caterina; Cuffaro, Doretta; Nuti, Elisa; Rossello, Armando
Matrix metalloproteinase inhibitors prevent the release and proteolytic activity of monocyte/macrophage-derived microparticles
2019-01-01 Fogli, Stefano; Neri, Tommaso; Nuti, Elisa; Mattii, Letizia; Camodeca, Caterina; Rossello, Armando
Design and Synthesis of Ionic Liquid-Based Matrix Metalloproteinase Inhibitors (MMPIs): A Simple Approach to Increase Hydrophilicity and to Develop MMPI-Coated Gold Nanoparticles
2019-01-01 D'Andrea, Felicia; Nuti, Elisa; Becherini, Stefano; Cuffaro, Doretta; Husanu, Elena; Camodeca, Caterina; De Vita, Elena; Zocchi, Maria Raffaella; Poggi, Alessandro; D'Arrigo, Cristina; Cappello, Valentina; Gemmi, Mauro; Nencetti, Susanna; Chiappe, Cinzia; Rossello, Armando
Bivalent Inhibitor with Selectivity for Trimeric MMP-9 Amplifies Neutrophil Chemotaxis and Enables Functional Studies on MMP-9 Proteoforms
2020-01-01 Nuti, E.; Rossello, A.; Cuffaro, D.; Camodeca, C.; Van Bael, J.; van der Maat, D.; Martens, E.; Fiten, P.; Pereira, R. V. S.; Ugarte-Berzal, E.; Gouwy, M.; Opdenakker, G.; Vandooren, J.
Focus on Human Monoamine Transporter Selectivity. New Human DAT and NET Models, Experimental Validation, and SERT Affinity Exploration
2020-01-01 Ortore, G.; Orlandini, E.; Betti, L.; Giannaccini, G.; Mazzoni, M. R.; Camodeca, C.; Nencetti, S.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Mimicking the intramolecular hydrogen bond: Synthesis, biological evaluation, andmolecular modeling of benzoxazines and quinazolines as potential antimalarial agents | 1-gen-2012 | Gemma, S.; Camodeca, C.; Brindisi, M.; Brogi, S.; Kukreja, G.; Kunjir, S.; Gabellieri, E.; Lucantoni, L.; Habluetzel, A.; Taramelli, D.; Basilico, N.; Gualdani, R.; Tadini-Buoninsegni, F.; Bartolommei, G.; Moncelli, M. R.; Martin, R. E.; Summers, R. L.; Lamponi, S.; Savini, L.; Fiorini, I.; Valoti, M.; Novellino, E.; Campiani, G.; Butini, S. | |
Optimization of 4-aminoquinoline/clotrimazole-based hybrid antimalarials: Further structure-activity relationships, in vivo studies, and preliminary toxicity profiling | 1-gen-2012 | Gemma, S.; Camodeca, C.; Sanna Coccone, S.; Joshi, B. P.; Bernetti, M.; Moretti, V.; Brogi, S.; De Marcos, M. C. B.; Savini, L.; Taramelli, D.; Basilico, N.; Parapini, S.; Rottmann, M.; Brun, R.; Lamponi, S.; Caccia, S.; Guiso, G.; Summers, R. L.; Martin, R. E.; Saponara, S.; Gorelli, B.; Novellino, E.; Campiani, G.; Butini, S. | |
N-O-Isopropyl Sulfonamido-Based Hydroxamates as Matrix Metalloproteinase Inhibitors: Hit Selection and in Vivo Antiangiogenic Activity | 1-gen-2015 | Nuti, Elisa; Cantelmo, Anna Rita; Gallo, Cristina; Bruno, Antonino; Bassani, Barbara; Camodeca, Caterina; Tuccinardi, Tiziano; Vera, Laura; Orlandini, Elisabetta; Nencetti, Susanna; Stura, Enrico A; Martinelli, Adriano; Dive, Vincent; Albini, Adriana; Rossello, Armando | |
MMP-8 Is Critical for Dexamethasone Therapy in Alkali-Burned Corneas Under Dry Eye Conditions | 1-gen-2016 | Bian, Fang; Wang, Changjun; Tukler Henriksson, Johanna; Pflugfelder, Stephen C.; Camodeca, Caterina; Nuti, Elisa; Rossello, Armando; Li, De Quan; de Paiva, Cintia S. | |
Synthesis, experimental evaluation and molecular modelling of hydroxamate derivatives as zinc metalloproteinase inhibitors | 1-gen-2016 | Sjøli, Stian; Nuti, Elisa; Camodeca, Caterina; Bilto, Irina; Rossello, Armando; Winberg, Jan Olof; Sylte, Ingebrigt; Adekoya, Olayiwola A. | |
Sugar-Based Arylsulfonamide Carboxylates as Selective and Water-Soluble Matrix Metalloproteinase-12 Inhibitors | 1-gen-2016 | Nuti, Elisa; Cuffaro, Doretta; D'Andrea, Felicia; Rosalia, Lea; Tepshi, Livia; Fabbi, Marina; Carbotti, Grazia; Ferrini, Silvano; Santamaria, Salvatore; Camodeca, Caterina; Ciccone, Lidia; Orlandini, Elisabetta; Nencetti, Susanna; Stura, Enrico A.; Dive, Vincent; Rossello, Armando | |
ADAM10 new selective inhibitors reduce NKG2D ligand release sensitizing Hodgkin lymphoma cells to NKG2D-mediated killing | 1-gen-2016 | Zocchi, Maria Raffaella; Camodeca, Caterina; Nuti, Elisa; Rossello, Armando; Venè, Roberta; Tosetti, Francesca; Dapino, Irene; Costa, Delfina; Musso, Alessandra; Poggi, Alessandro | |
Discovery of a new selective inhibitor of A Disintegrin And Metalloprotease 10 (ADAM-10) able to reduce the shedding of NKG2D ligands in Hodgkin's lymphoma cell models | 1-gen-2016 | Camodeca, Caterina; Nuti, Elisa; Tepshi, Livia; Boero, Silvia; Tuccinardi, Tiziano; Stura, Enrico A; Poggi, Alessandro; Zocchi, Maria Raffaella; Rossello, Armando | |
Bifunctional Inhibitors as a New Tool To Reduce Cancer Cell Invasion by Impairing MMP-9 Homodimerization | 1-gen-2017 | Nuti, Elisa; Rosalia, Lea; Cuffaro, Doretta; Camodeca, Caterina; Giacomelli, Chiara; DA POZZO, Eleonora; Tuccinardi, Tiziano; Costa, Barbara; Antoni, Claudia; Vera, Laura; Ciccone, Lidia; Orlandini, Elisabetta; Nencetti, Susanna; Dive, Vincent; Martini, Claudia; Stura, Enrico A.; Rossello, Armando | |
Synthesis and antiangiogenic activity study of new hop chalcone Xanthohumol analogues | 1-gen-2017 | Nuti, Elisa; Bassani, Barbara; Camodeca, Caterina; Rosalia, Lea; Cantelmo, Annarita; Gallo, Cristina; Baci, Denisa; Bruno, Antonino; Orlandini, Elisabetta; Nencetti, Susanna; Noonan, Douglas M.; Albini, Adriana; Rossello, Armando | |
Development of Thioaryl-Based Matrix Metalloproteinase-12 Inhibitors with Alternative Zinc-Binding Groups: Synthesis, Potentiometric, NMR, and Crystallographic Studies | 1-gen-2018 | Nuti, Elisa; Cuffaro, Doretta; Bernardini, Elisa; Camodeca, Caterina; Panelli, Laura; Chaves, Sílvia; Ciccone, Lidia; Tepshi, Livia; Vera, Laura; Orlandini, Elisabetta; Nencetti, Susanna; Stura, Enrico A.; Santos, M. Amélia; Dive, Vincent; Rossello, Armando | |
Specific ADAM10 inhibitors localize in exosome-like vesicles released by Hodgkin lymphoma and stromal cells and prevent sheddase activity carried to bystander cells | 1-gen-2018 | Tosetti, Francesca; Venè, Roberta; Camodeca, Caterina; Nuti, Elisa; Rossello, Armando; D'Arrigo, Cristina; Galante, Denise; Ferrari, Nicoletta; Poggi, Alessandro; Zocchi, Maria Raffaella | |
Matrix metalloproteinase-12 inhibitors: synthesis, structure-activity relationships and intestinal absorption of novel sugar-based biphenylsulfonamide carboxylates | 1-gen-2018 | Cuffaro, Doretta; Camodeca, Caterina; D'Andrea, Felicia; Piragine, Eugenia; Testai, Lara; Calderone, Vincenzo; Orlandini, Elisabetta; Nuti, Elisa; Rossello, Armando | |
Synthesis and in vitro Evaluation of ADAM10 and ADAM17 Highly Selective Bioimaging Probes | 1-gen-2018 | Camodeca, Caterina; Nuti, Elisa; Tosetti, Francesca; Poggi, Alessandro; D'Arrigo, Cristina; Zocchi, Maria Raffaella; Rossello, Armando | |
Design, synthesis and biological evaluation of bifunctional inhibitors of membrane type 1 matrix metalloproteinase (MT1-MMP) | 1-gen-2019 | Cuffaro, Doretta; Nuti, Elisa; Gifford, Valentina; Ito, Noriko; Camodeca, Caterina; Tuccinardi, Tiziano; Nencetti, Susanna; Orlandini, Elisabetta; Itoh, Yoshifumi; Rossello, Armando | |
ADAM metalloproteinases as potential drug targets | 1-gen-2019 | Camodeca, Caterina; Cuffaro, Doretta; Nuti, Elisa; Rossello, Armando | |
Matrix metalloproteinase inhibitors prevent the release and proteolytic activity of monocyte/macrophage-derived microparticles | 1-gen-2019 | Fogli, Stefano; Neri, Tommaso; Nuti, Elisa; Mattii, Letizia; Camodeca, Caterina; Rossello, Armando | |
Design and Synthesis of Ionic Liquid-Based Matrix Metalloproteinase Inhibitors (MMPIs): A Simple Approach to Increase Hydrophilicity and to Develop MMPI-Coated Gold Nanoparticles | 1-gen-2019 | D'Andrea, Felicia; Nuti, Elisa; Becherini, Stefano; Cuffaro, Doretta; Husanu, Elena; Camodeca, Caterina; De Vita, Elena; Zocchi, Maria Raffaella; Poggi, Alessandro; D'Arrigo, Cristina; Cappello, Valentina; Gemmi, Mauro; Nencetti, Susanna; Chiappe, Cinzia; Rossello, Armando | |
Bivalent Inhibitor with Selectivity for Trimeric MMP-9 Amplifies Neutrophil Chemotaxis and Enables Functional Studies on MMP-9 Proteoforms | 1-gen-2020 | Nuti, E.; Rossello, A.; Cuffaro, D.; Camodeca, C.; Van Bael, J.; van der Maat, D.; Martens, E.; Fiten, P.; Pereira, R. V. S.; Ugarte-Berzal, E.; Gouwy, M.; Opdenakker, G.; Vandooren, J. | |
Focus on Human Monoamine Transporter Selectivity. New Human DAT and NET Models, Experimental Validation, and SERT Affinity Exploration | 1-gen-2020 | Ortore, G.; Orlandini, E.; Betti, L.; Giannaccini, G.; Mazzoni, M. R.; Camodeca, C.; Nencetti, S. |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile