POLI, GIULIO Statistiche
POLI, GIULIO
DIPARTIMENTO DI FARMACIA
An update on antibacterial AlkylGuanidino Ureas: Design of new derivatives, synergism with colistin and data analysis of the whole library
2024-01-01 Ardino, Claudia; Sannio, Filomena; Poli, Giulio; Galati, Salvatore; Dreassi, Elena; Botta, Lorenzo; Docquier, Jean-Denis; D'Agostino, Ilaria
Design, synthesis, ADME and biological evaluation of benzylpiperidine and benzylpiperazine derivatives as novel reversible monoacylglycerol lipase (MAGL) inhibitors
2024-01-01 Di Stefano, Miriana; Masoni, Samuele; Bononi, Giulia; Poli, Giulio; Galati, Salvatore; Gado, Francesca; Manzi, Simone; Vagaggini, Chiara; Brai, Annalaura; Caligiuri, Isabella; Asif, Kanwal; Rizzolio, Flavio; Macchia, Marco; Chicca, Andrea; Sodi, Andrea; Di Bussolo, Valeria; Minutolo, Filippo; Meier, Philip; Gertsch, Jürg; Granchi, Carlotta; Dreassi, Elena; Tuccinardi, Tiziano
Nuovi agenti antivirali a struttura N-idrossiindrol-carbossamidica
2024-01-01 Minutolo, Filippo; Pistello, Mauro; DI BUSSOLO, Valeria; Freer, Giulia; Quaranta, Paola; Granchi, Carlotta; Tuccinardi, Tiziano; Poli, Giulio; Bononi, Giulia; Masoni, Samuele
A Multitarget Approach against Neuroinflammation: Alkyl Substituted Coumarins as Inhibitors of Enzymes Involved in Neurodegeneration
2023-01-01 Berrino, Emanuela; Carradori, Simone; Carta, Fabrizio; Melfi, Francesco; Gallorini, Marialucia; Poli, Giulio; Tuccinardi, Tiziano; Fernández-Bolaños, José G; López, Óscar; Petzer, Jacobus P; Petzer, Anél; Guglielmi, Paolo; Secci, Daniela; Supuran, Claudiu T
An in silico toolbox for the prediction of the potential pathogenic effects of missense mutations in the dimeric region of hRPE65
2023-01-01 Poli, Giulio; Demontis, Gian Carlo; Sodi, Andrea; Saba, Alessandro; Rizzo, Stanislao; Macchia, Marco; Tuccinardi, Tiziano
Identification of New GSK3β Inhibitors through a Consensus Machine Learning-Based Virtual Screening
2023-01-01 Galati, Salvatore; Di Stefano, Miriana; Bertini, Simone; Granchi, Carlotta; Giordano, Antonio; Gado, Francesca; Macchia, Marco; Tuccinardi, Tiziano; Poli, Giulio
miRNA-203b-3p Induces Acute and Chronic Pruritus through 5-HTR2B and TRPV4
2023-01-01 De Logu, Francesco; Maglie, Roberto; Titiz, Mustafa; Poli, Giulio; Landini, Lorenzo; Marini, Matilde; Souza Monteiro de Araujo, Daniel; De Siena, Gaetano; Montini, Marco; Cabrini, Daniela Almeida; Otuki, Michel Fleith; Pawloski, Priscila Lúcia; Antiga, Emiliano; Tuccinardi, Tiziano; Calixto, João Batista; Geppetti, Pierangelo; Nassini, Romina; André, Eunice
MolBook UNIPI─Create, Manage, Analyze, and Share Your Chemical Data for Free
2023-01-01 Galati, Salvatore; Di Stefano, Miriana; Macchia, Marco; Poli, Giulio; Tuccinardi, Tiziano
New Insights into Bitopic Orthosteric/Allosteric Ligands of Cannabinoid Receptor Type 2
2023-01-01 Ferrisi, Rebecca; Polini, Beatrice; Ricardi, Caterina; Gado, Francesca; Mohamed, Kawthar A; Baron, Giovanna; Faiella, Salvatore; Poli, Giulio; Rapposelli, Simona; Saccomanni, Giuseppe; Aldini, Giancarlo; Chiellini, Grazia; Laprairie, Robert B; Manera, Clementina; Ortore, Gabriella
Sirtuin 1-activating derivatives belonging to the anilinopyridine class displaying in vivo cardioprotective activities
2023-01-01 Bononi, G.; Citi, V.; Martelli, A.; Poli, G.; Tuccinardi, T.; Granchi, C.; Testai, L.; Calderone, V.; Minutolo, F.
Antibacterial alkylguanidino ureas: Molecular simplification approach, searching for membrane-based MoA
2022-01-01 D'Agostino, Ilaria; Ardino, Claudia; Poli, Giulio; Sannio, Filomena; Lucidi, Massimiliano; Poggialini, Federica; Visaggio, Daniela; Rango, Enrico; Filippi, Silvia; Petricci, Elena; Visca, Paolo; Botta, Lorenzo; Docquier, Jean-Denis; Dreassi, Elena
Co-Inhibition of P-gp and Hsp90 by an Isatin-Derived Compound Contributes to the Increase of the Chemosensitivity of MCF7/ADR-Resistant Cells to Doxorubicin
2022-01-01 Abdalla, Ashraf N; Di Stefano, Miriana; Poli, Giulio; Tuccinardi, Tiziano; Bader, Ammar; Vassallo, Antonio; Abdallah, Mohamed E; El-Readi, Mahmoud Zaki; Refaat, Bassem; Algarni, Alanood S; Ahmad, Rizwan; Alkahtani, Hamad M; Abdel-Aziz, Alaa A-M; El-Azab, Adel S; Alqathama, Aljawharah
Dissecting the Activity of Catechins as Incomplete Aldose Reductase Differential Inhibitors through Kinetic and Computational Approaches
2022-01-01 Balestri, Francesco; Poli, Giulio; Piazza, Lucia; Cappiello, Mario; Moschini, Roberta; Signore, Giovanni; Tuccinardi, Tiziano; Mura, Umberto; Del Corso, Antonella
From Anti-infective Agents to Cancer Therapy: a Drug Repositioning Study Revealed a New Use for Nitrofuran Derivatives
2022-01-01 Ortore, Gabriella; Poli, Giulio; Martinelli, Adriano; Tuccinardi, Tiziano; Rizzolio, Flavio; Caligiuri, Isabella
Identification of Human Dihydroorotate Dehydrogenase Inhibitor by a Pharmacophore-Based Virtual Screening Study
2022-01-01 Galati, Salvatore; Sainas, Stefano; Giorgis, Marta; Boschi, Donatella; Lolli, Marco L; Ortore, Gabriella; Poli, Giulio; Tuccinardi, Tiziano
Machine Learning-Based Virtual Screening for the Identification of Cdk5 Inhibitors
2022-01-01 Di Stefano, Miriana; Galati, Salvatore; Ortore, Gabriella; Caligiuri, Isabella; Rizzolio, Flavio; Ceni, Costanza; Bertini, Simone; Bononi, Giulia; Granchi, Carlotta; Macchia, Marco; Poli, Giulio; Tuccinardi, Tiziano
New PIN1 inhibitors identified through a pharmacophore-driven, hierarchical consensus docking strategy
2022-01-01 Poli, Giulio; Di Stefano, Miriana; Estevez, Joan Arias; Minutolo, Filippo; Granchi, Carlotta; Giordano, Antonio; Parisi, Salvatore; Mauceri, Matteo; Canzonieri, Vincenzo; Macchia, Marco; Caligiuri, Isabella; Tuccinardi, Tiziano; Rizzolio, Flavio
New Synthetic Analogues of Natural Polyphenols as Sirtuin 1-Activating Compounds
2022-01-01 Bononi, G.; Flori, L.; Citi, V.; Acciai, C.; Nocilla, V.; Martelli, A.; Poli, G.; Tuccinardi, T.; Granchi, C.; Testai, L.; Calderone, V.; Minutolo, F.
Novel Potent and Selective Agonists of the GPR55 Receptor Based on the 3-Benzylquinolin-2(1H)-One Scaffold
2022-01-01 Ceni, Costanza; Benko, Michael J; Mohamed, Kawthar A; Poli, Giulio; Di Stefano, Miriana; Tuccinardi, Tiziano; Digiacomo, Maria; Valoti, Massimo; Laprairie, Robert B; Macchia, Marco; Bertini, Simone
Predicting potentially pathogenic effects of hRPE65 missense mutations: a computational strategy based on molecular dynamics simulations
2022-01-01 Poli, Giulio; Barravecchia, Ivana; Demontis, Gian Carlo; Sodi, Andrea; Saba, Alessandro; Rizzo, Stanislao; Macchia, Marco; Tuccinardi, Tiziano
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
An update on antibacterial AlkylGuanidino Ureas: Design of new derivatives, synergism with colistin and data analysis of the whole library | 1-gen-2024 | Ardino, Claudia; Sannio, Filomena; Poli, Giulio; Galati, Salvatore; Dreassi, Elena; Botta, Lorenzo; Docquier, Jean-Denis; D'Agostino, Ilaria | |
Design, synthesis, ADME and biological evaluation of benzylpiperidine and benzylpiperazine derivatives as novel reversible monoacylglycerol lipase (MAGL) inhibitors | 1-gen-2024 | Di Stefano, Miriana; Masoni, Samuele; Bononi, Giulia; Poli, Giulio; Galati, Salvatore; Gado, Francesca; Manzi, Simone; Vagaggini, Chiara; Brai, Annalaura; Caligiuri, Isabella; Asif, Kanwal; Rizzolio, Flavio; Macchia, Marco; Chicca, Andrea; Sodi, Andrea; Di Bussolo, Valeria; Minutolo, Filippo; Meier, Philip; Gertsch, Jürg; Granchi, Carlotta; Dreassi, Elena; Tuccinardi, Tiziano | |
Nuovi agenti antivirali a struttura N-idrossiindrol-carbossamidica | 1-gen-2024 | Minutolo, Filippo; Pistello, Mauro; DI BUSSOLO, Valeria; Freer, Giulia; Quaranta, Paola; Granchi, Carlotta; Tuccinardi, Tiziano; Poli, Giulio; Bononi, Giulia; Masoni, Samuele | |
A Multitarget Approach against Neuroinflammation: Alkyl Substituted Coumarins as Inhibitors of Enzymes Involved in Neurodegeneration | 1-gen-2023 | Berrino, Emanuela; Carradori, Simone; Carta, Fabrizio; Melfi, Francesco; Gallorini, Marialucia; Poli, Giulio; Tuccinardi, Tiziano; Fernández-Bolaños, José G; López, Óscar; Petzer, Jacobus P; Petzer, Anél; Guglielmi, Paolo; Secci, Daniela; Supuran, Claudiu T | |
An in silico toolbox for the prediction of the potential pathogenic effects of missense mutations in the dimeric region of hRPE65 | 1-gen-2023 | Poli, Giulio; Demontis, Gian Carlo; Sodi, Andrea; Saba, Alessandro; Rizzo, Stanislao; Macchia, Marco; Tuccinardi, Tiziano | |
Identification of New GSK3β Inhibitors through a Consensus Machine Learning-Based Virtual Screening | 1-gen-2023 | Galati, Salvatore; Di Stefano, Miriana; Bertini, Simone; Granchi, Carlotta; Giordano, Antonio; Gado, Francesca; Macchia, Marco; Tuccinardi, Tiziano; Poli, Giulio | |
miRNA-203b-3p Induces Acute and Chronic Pruritus through 5-HTR2B and TRPV4 | 1-gen-2023 | De Logu, Francesco; Maglie, Roberto; Titiz, Mustafa; Poli, Giulio; Landini, Lorenzo; Marini, Matilde; Souza Monteiro de Araujo, Daniel; De Siena, Gaetano; Montini, Marco; Cabrini, Daniela Almeida; Otuki, Michel Fleith; Pawloski, Priscila Lúcia; Antiga, Emiliano; Tuccinardi, Tiziano; Calixto, João Batista; Geppetti, Pierangelo; Nassini, Romina; André, Eunice | |
MolBook UNIPI─Create, Manage, Analyze, and Share Your Chemical Data for Free | 1-gen-2023 | Galati, Salvatore; Di Stefano, Miriana; Macchia, Marco; Poli, Giulio; Tuccinardi, Tiziano | |
New Insights into Bitopic Orthosteric/Allosteric Ligands of Cannabinoid Receptor Type 2 | 1-gen-2023 | Ferrisi, Rebecca; Polini, Beatrice; Ricardi, Caterina; Gado, Francesca; Mohamed, Kawthar A; Baron, Giovanna; Faiella, Salvatore; Poli, Giulio; Rapposelli, Simona; Saccomanni, Giuseppe; Aldini, Giancarlo; Chiellini, Grazia; Laprairie, Robert B; Manera, Clementina; Ortore, Gabriella | |
Sirtuin 1-activating derivatives belonging to the anilinopyridine class displaying in vivo cardioprotective activities | 1-gen-2023 | Bononi, G.; Citi, V.; Martelli, A.; Poli, G.; Tuccinardi, T.; Granchi, C.; Testai, L.; Calderone, V.; Minutolo, F. | |
Antibacterial alkylguanidino ureas: Molecular simplification approach, searching for membrane-based MoA | 1-gen-2022 | D'Agostino, Ilaria; Ardino, Claudia; Poli, Giulio; Sannio, Filomena; Lucidi, Massimiliano; Poggialini, Federica; Visaggio, Daniela; Rango, Enrico; Filippi, Silvia; Petricci, Elena; Visca, Paolo; Botta, Lorenzo; Docquier, Jean-Denis; Dreassi, Elena | |
Co-Inhibition of P-gp and Hsp90 by an Isatin-Derived Compound Contributes to the Increase of the Chemosensitivity of MCF7/ADR-Resistant Cells to Doxorubicin | 1-gen-2022 | Abdalla, Ashraf N; Di Stefano, Miriana; Poli, Giulio; Tuccinardi, Tiziano; Bader, Ammar; Vassallo, Antonio; Abdallah, Mohamed E; El-Readi, Mahmoud Zaki; Refaat, Bassem; Algarni, Alanood S; Ahmad, Rizwan; Alkahtani, Hamad M; Abdel-Aziz, Alaa A-M; El-Azab, Adel S; Alqathama, Aljawharah | |
Dissecting the Activity of Catechins as Incomplete Aldose Reductase Differential Inhibitors through Kinetic and Computational Approaches | 1-gen-2022 | Balestri, Francesco; Poli, Giulio; Piazza, Lucia; Cappiello, Mario; Moschini, Roberta; Signore, Giovanni; Tuccinardi, Tiziano; Mura, Umberto; Del Corso, Antonella | |
From Anti-infective Agents to Cancer Therapy: a Drug Repositioning Study Revealed a New Use for Nitrofuran Derivatives | 1-gen-2022 | Ortore, Gabriella; Poli, Giulio; Martinelli, Adriano; Tuccinardi, Tiziano; Rizzolio, Flavio; Caligiuri, Isabella | |
Identification of Human Dihydroorotate Dehydrogenase Inhibitor by a Pharmacophore-Based Virtual Screening Study | 1-gen-2022 | Galati, Salvatore; Sainas, Stefano; Giorgis, Marta; Boschi, Donatella; Lolli, Marco L; Ortore, Gabriella; Poli, Giulio; Tuccinardi, Tiziano | |
Machine Learning-Based Virtual Screening for the Identification of Cdk5 Inhibitors | 1-gen-2022 | Di Stefano, Miriana; Galati, Salvatore; Ortore, Gabriella; Caligiuri, Isabella; Rizzolio, Flavio; Ceni, Costanza; Bertini, Simone; Bononi, Giulia; Granchi, Carlotta; Macchia, Marco; Poli, Giulio; Tuccinardi, Tiziano | |
New PIN1 inhibitors identified through a pharmacophore-driven, hierarchical consensus docking strategy | 1-gen-2022 | Poli, Giulio; Di Stefano, Miriana; Estevez, Joan Arias; Minutolo, Filippo; Granchi, Carlotta; Giordano, Antonio; Parisi, Salvatore; Mauceri, Matteo; Canzonieri, Vincenzo; Macchia, Marco; Caligiuri, Isabella; Tuccinardi, Tiziano; Rizzolio, Flavio | |
New Synthetic Analogues of Natural Polyphenols as Sirtuin 1-Activating Compounds | 1-gen-2022 | Bononi, G.; Flori, L.; Citi, V.; Acciai, C.; Nocilla, V.; Martelli, A.; Poli, G.; Tuccinardi, T.; Granchi, C.; Testai, L.; Calderone, V.; Minutolo, F. | |
Novel Potent and Selective Agonists of the GPR55 Receptor Based on the 3-Benzylquinolin-2(1H)-One Scaffold | 1-gen-2022 | Ceni, Costanza; Benko, Michael J; Mohamed, Kawthar A; Poli, Giulio; Di Stefano, Miriana; Tuccinardi, Tiziano; Digiacomo, Maria; Valoti, Massimo; Laprairie, Robert B; Macchia, Marco; Bertini, Simone | |
Predicting potentially pathogenic effects of hRPE65 missense mutations: a computational strategy based on molecular dynamics simulations | 1-gen-2022 | Poli, Giulio; Barravecchia, Ivana; Demontis, Gian Carlo; Sodi, Andrea; Saba, Alessandro; Rizzo, Stanislao; Macchia, Marco; Tuccinardi, Tiziano |