POLI, GIULIO Statistiche
POLI, GIULIO
DIPARTIMENTO DI FARMACIA
1,3-Dipolar Cycloaddition, HPLC Enantioseparation, and Docking Studies of Saccharin/Isoxazole and Saccharin/Isoxazoline Derivatives as Selective Carbonic Anhydrase IX and XII Inhibitors
2020-01-01 D'Ascenzio, M.; Secci, D.; Carradori, S.; Zara, S.; Guglielmi, P.; Cirilli, R.; Pierini, M.; Poli, G.; Tuccinardi, T.; Angeli, A.; Supuran, C. T.
3D Pharmacophore Modeling Techniques in Computer-Aided Molecular Design Using LigandScout
2017-01-01 Seidel, Thomas; Bryant, Sharon D.; Ibis, Gökhan; Poli, Giulio; Langer, Thierry
A Virtual Screening Study for Lactate Dehydrogenase 5 Inhibitors by using a Pharmacophore-Based Approach
2016-01-01 Tuccinardi, Tiziano; Poli, Giulio; Corchia, Isacco; Granchi, Carlotta; Lapillo, Margherita; Macchia, Marco; Minutolo, Filippo; Ortore, GABRIELLA MARIA PIA; Martinelli, Adriano
Aldose reductase differential inhibitors in green tea
2020-01-01 Balestri, F.; Poli, G.; Pineschi, C.; Moschini, R.; Cappiello, M.; Mura, U.; Tuccinardi, T.; Corso, A. D.
An updated patent review of monoacylglycerol lipase (MAGL) inhibitors (2018-present)
2021-01-01 Bononi, G.; Poli, G.; Rizzolio, F.; Tuccinardi, T.; Macchia, M.; Minutolo, F.; Granchi, C.
Antibacterial alkylguanidino ureas: Molecular simplification approach, searching for membrane-based MoA
2022-01-01 D'Agostino, Ilaria; Ardino, Claudia; Poli, Giulio; Sannio, Filomena; Lucidi, Massimiliano; Poggialini, Federica; Visaggio, Daniela; Rango, Enrico; Filippi, Silvia; Petricci, Elena; Visca, Paolo; Botta, Lorenzo; Docquier, Jean-Denis; Dreassi, Elena
Antibacterial and ATP Synthesis Modulating Compounds from Salvia tingitana
2020-01-01 Bisio, A.; Schito, A. M.; Pedrelli, F.; Danton, O.; Reinhardt, J. K.; Poli, G.; Tuccinardi, T.; Burgi, T.; De Riccardis, F.; Giacomini, M.; Calzia, D.; Panfoli, I.; Schito, G. C.; Hamburger, M.; De Tommasi, N.
Anticancer activity of euplotin C, isolated from the marine ciliate euplotes crassus, against human melanoma cells
2018-01-01 Carpi, Sara; Polini, Beatrice; Poli, Giulio; ALCANTARA BARATA, Gabriela; Fogli, Stefano; Romanini, Antonella; Tuccinardi, Tiziano; Guella, Graziano; Frontini, FRANCESCO PAOLO; Nieri, Paola; Di Giuseppe, Graziano
Application of a FLAP-Consensus Docking Mixed Strategy for the Identification of New FAAH Inhibitors
2015-01-01 Poli, Giulio; Giuntini, N; Martinelli, Adriano; Tuccinardi, Tiziano
Application of MM-PBSA methods in virtual screening
2020-01-01 Poli, G.; Granchi, C.; Rizzolio, F.; Tuccinardi, T.
Binding investigation and preliminary optimisation of the 3-amino-1,2,4-triazin-5(2H)-one core for the development of new Fyn inhibitors
2018-01-01 Poli, Giulio; Lapillo, Margherita; Granchi, Carlotta; Caciolla, Jessica; Mouawad, Nayla; Caligiuri, Isabella; Rizzolio, Flavio; Langer, Thierry; Minutolo, Filippo; Tuccinardi, Tiziano
Carbonic Anhydrase Inhibitors: Identifying Therapeutic Cancer Agents Through Virtual Screening
2021-01-01 Poli, G.; Supuran, C. T.; Tuccinardi, T.
Co-Inhibition of P-gp and Hsp90 by an Isatin-Derived Compound Contributes to the Increase of the Chemosensitivity of MCF7/ADR-Resistant Cells to Doxorubicin
2022-01-01 Abdalla, Ashraf N; Di Stefano, Miriana; Poli, Giulio; Tuccinardi, Tiziano; Bader, Ammar; Vassallo, Antonio; Abdallah, Mohamed E; El-Readi, Mahmoud Zaki; Refaat, Bassem; Algarni, Alanood S; Ahmad, Rizwan; Alkahtani, Hamad M; Abdel-Aziz, Alaa A-M; El-Azab, Adel S; Alqathama, Aljawharah
Computational Approaches for the Identification and Optimization of Src Family Kinases Inhibitors.
2014-01-01 Poli, Giulio; Martinelli, Adriano; Tuccinardi, Tiziano
Computationally driven discovery of phenyl(piperazin-1-yl)methanone derivatives as reversible monoacylglycerol lipase (MAGL) inhibitors
2019-01-01 Poli, Giulio; Lapillo, Margherita; Jha, Vibhu; Mouawad, Nayla; Caligiuri, Isabella; Macchia, Marco; Minutolo, Filippo; Rizzolio, Flavio; Tuccinardi, Tiziano; Granchi, Carlotta
Conformational sampling of small molecules with iCon: Performance assessment in comparison with OMEGA
2018-01-01 Poli, Giulio; Seidel, Thomas; Langer, Thierry
Consensus Docking in Drug Discovery
2020-01-01 Poli, Giulio; Tuccinardi, Tiziano
Continued exploration of 1,2,4-oxadiazole periphery for carbonic anhydrase-targeting primary arene sulfonamides: Discovery of subnanomolar inhibitors of membrane-bound hCA IX isoform that selectively kill cancer cells in hypoxic environment
2019-01-01 Krasavin, Mikhail; Shetnev, Anton; Sharonova, Tatyana; Baykov, Sergey; Kalinin, Stanislav; Nocentini, Alessio; Sharoyko, Vladimir; Poli, Giulio; Tuccinardi, Tiziano; Presnukhina, Sofia; Tennikova, Tatiana B.; Supuran, Claudiu T.
Design, synthesis and biological evaluation of second-generation benzoylpiperidine derivatives as reversible monoacylglycerol lipase (MAGL) inhibitors
2021-01-01 Granchi, C.; Bononi, G.; Ferrisi, R.; Gori, E.; Mantini, G.; Glasmacher, S.; Poli, G.; Palazzolo, S.; Caligiuri, I.; Rizzolio, F.; Canzonieri, V.; Perin, T.; Gertsch, J.; Sodi, A.; Giovannetti, E.; Macchia, M.; Minutolo, F.; Tuccinardi, T.; Chicca, A.
Design, synthesis, docking studies and monoamine oxidase inhibition of a small library of 1-acetyl- and 1-thiocarbamoyl-3,5-diphenyl-4,5-dihydro-(1h)-pyrazoles
2019-01-01 Guglielmi, P.; Carradori, S.; Poli, G.; Secci, D.; Cirilli, R.; Rotondi, G.; Chimenti, P.; Petzer, A.; Petzer, J. P.
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 1,3-Dipolar Cycloaddition, HPLC Enantioseparation, and Docking Studies of Saccharin/Isoxazole and Saccharin/Isoxazoline Derivatives as Selective Carbonic Anhydrase IX and XII Inhibitors | 1-gen-2020 | D'Ascenzio, M.; Secci, D.; Carradori, S.; Zara, S.; Guglielmi, P.; Cirilli, R.; Pierini, M.; Poli, G.; Tuccinardi, T.; Angeli, A.; Supuran, C. T. | |
| 3D Pharmacophore Modeling Techniques in Computer-Aided Molecular Design Using LigandScout | 1-gen-2017 | Seidel, Thomas; Bryant, Sharon D.; Ibis, Gökhan; Poli, Giulio; Langer, Thierry | |
| A Virtual Screening Study for Lactate Dehydrogenase 5 Inhibitors by using a Pharmacophore-Based Approach | 1-gen-2016 | Tuccinardi, Tiziano; Poli, Giulio; Corchia, Isacco; Granchi, Carlotta; Lapillo, Margherita; Macchia, Marco; Minutolo, Filippo; Ortore, GABRIELLA MARIA PIA; Martinelli, Adriano | |
| Aldose reductase differential inhibitors in green tea | 1-gen-2020 | Balestri, F.; Poli, G.; Pineschi, C.; Moschini, R.; Cappiello, M.; Mura, U.; Tuccinardi, T.; Corso, A. D. | |
| An updated patent review of monoacylglycerol lipase (MAGL) inhibitors (2018-present) | 1-gen-2021 | Bononi, G.; Poli, G.; Rizzolio, F.; Tuccinardi, T.; Macchia, M.; Minutolo, F.; Granchi, C. | |
| Antibacterial alkylguanidino ureas: Molecular simplification approach, searching for membrane-based MoA | 1-gen-2022 | D'Agostino, Ilaria; Ardino, Claudia; Poli, Giulio; Sannio, Filomena; Lucidi, Massimiliano; Poggialini, Federica; Visaggio, Daniela; Rango, Enrico; Filippi, Silvia; Petricci, Elena; Visca, Paolo; Botta, Lorenzo; Docquier, Jean-Denis; Dreassi, Elena | |
| Antibacterial and ATP Synthesis Modulating Compounds from Salvia tingitana | 1-gen-2020 | Bisio, A.; Schito, A. M.; Pedrelli, F.; Danton, O.; Reinhardt, J. K.; Poli, G.; Tuccinardi, T.; Burgi, T.; De Riccardis, F.; Giacomini, M.; Calzia, D.; Panfoli, I.; Schito, G. C.; Hamburger, M.; De Tommasi, N. | |
| Anticancer activity of euplotin C, isolated from the marine ciliate euplotes crassus, against human melanoma cells | 1-gen-2018 | Carpi, Sara; Polini, Beatrice; Poli, Giulio; ALCANTARA BARATA, Gabriela; Fogli, Stefano; Romanini, Antonella; Tuccinardi, Tiziano; Guella, Graziano; Frontini, FRANCESCO PAOLO; Nieri, Paola; Di Giuseppe, Graziano | |
| Application of a FLAP-Consensus Docking Mixed Strategy for the Identification of New FAAH Inhibitors | 1-gen-2015 | Poli, Giulio; Giuntini, N; Martinelli, Adriano; Tuccinardi, Tiziano | |
| Application of MM-PBSA methods in virtual screening | 1-gen-2020 | Poli, G.; Granchi, C.; Rizzolio, F.; Tuccinardi, T. | |
| Binding investigation and preliminary optimisation of the 3-amino-1,2,4-triazin-5(2H)-one core for the development of new Fyn inhibitors | 1-gen-2018 | Poli, Giulio; Lapillo, Margherita; Granchi, Carlotta; Caciolla, Jessica; Mouawad, Nayla; Caligiuri, Isabella; Rizzolio, Flavio; Langer, Thierry; Minutolo, Filippo; Tuccinardi, Tiziano | |
| Carbonic Anhydrase Inhibitors: Identifying Therapeutic Cancer Agents Through Virtual Screening | 1-gen-2021 | Poli, G.; Supuran, C. T.; Tuccinardi, T. | |
| Co-Inhibition of P-gp and Hsp90 by an Isatin-Derived Compound Contributes to the Increase of the Chemosensitivity of MCF7/ADR-Resistant Cells to Doxorubicin | 1-gen-2022 | Abdalla, Ashraf N; Di Stefano, Miriana; Poli, Giulio; Tuccinardi, Tiziano; Bader, Ammar; Vassallo, Antonio; Abdallah, Mohamed E; El-Readi, Mahmoud Zaki; Refaat, Bassem; Algarni, Alanood S; Ahmad, Rizwan; Alkahtani, Hamad M; Abdel-Aziz, Alaa A-M; El-Azab, Adel S; Alqathama, Aljawharah | |
| Computational Approaches for the Identification and Optimization of Src Family Kinases Inhibitors. | 1-gen-2014 | Poli, Giulio; Martinelli, Adriano; Tuccinardi, Tiziano | |
| Computationally driven discovery of phenyl(piperazin-1-yl)methanone derivatives as reversible monoacylglycerol lipase (MAGL) inhibitors | 1-gen-2019 | Poli, Giulio; Lapillo, Margherita; Jha, Vibhu; Mouawad, Nayla; Caligiuri, Isabella; Macchia, Marco; Minutolo, Filippo; Rizzolio, Flavio; Tuccinardi, Tiziano; Granchi, Carlotta | |
| Conformational sampling of small molecules with iCon: Performance assessment in comparison with OMEGA | 1-gen-2018 | Poli, Giulio; Seidel, Thomas; Langer, Thierry | |
| Consensus Docking in Drug Discovery | 1-gen-2020 | Poli, Giulio; Tuccinardi, Tiziano | |
| Continued exploration of 1,2,4-oxadiazole periphery for carbonic anhydrase-targeting primary arene sulfonamides: Discovery of subnanomolar inhibitors of membrane-bound hCA IX isoform that selectively kill cancer cells in hypoxic environment | 1-gen-2019 | Krasavin, Mikhail; Shetnev, Anton; Sharonova, Tatyana; Baykov, Sergey; Kalinin, Stanislav; Nocentini, Alessio; Sharoyko, Vladimir; Poli, Giulio; Tuccinardi, Tiziano; Presnukhina, Sofia; Tennikova, Tatiana B.; Supuran, Claudiu T. | |
| Design, synthesis and biological evaluation of second-generation benzoylpiperidine derivatives as reversible monoacylglycerol lipase (MAGL) inhibitors | 1-gen-2021 | Granchi, C.; Bononi, G.; Ferrisi, R.; Gori, E.; Mantini, G.; Glasmacher, S.; Poli, G.; Palazzolo, S.; Caligiuri, I.; Rizzolio, F.; Canzonieri, V.; Perin, T.; Gertsch, J.; Sodi, A.; Giovannetti, E.; Macchia, M.; Minutolo, F.; Tuccinardi, T.; Chicca, A. | |
| Design, synthesis, docking studies and monoamine oxidase inhibition of a small library of 1-acetyl- and 1-thiocarbamoyl-3,5-diphenyl-4,5-dihydro-(1h)-pyrazoles | 1-gen-2019 | Guglielmi, P.; Carradori, S.; Poli, G.; Secci, D.; Cirilli, R.; Rotondi, G.; Chimenti, P.; Petzer, A.; Petzer, J. P. |