GRANCHI, CARLOTTA Statistiche
GRANCHI, CARLOTTA
DIPARTIMENTO DI FARMACIA
4-Aryliden-2-methyloxazol-5(4H)-one as a new scaffold for selective reversible MAGL inhibitors
2016-01-01 Granchi, Carlotta; Rizzolio, F; Bordoni, Vittorio; Caligiuri, I; Manera, Clementina; Macchia, Marco; Minutolo, Filippo; Martinelli, Adriano; Giordano, A; Tuccinardi, Tiziano
A carrier free delivery system of a monoacylglycerol lipase hydrophobic inhibitor
2022-01-01 Adeel, Muhammad; Saorin, Gloria; Boccalon, Giacomo; Sfriso, Andrea Augusto; Parisi, Salvatore; Moro, Isabella; Palazzolo, Stefano; Caligiuri, Isabella; Granchi, Carlotta; Corona, Giuseppe; Cemazar, Maja; Canzonieri, Vincenzo; Tuccinardi, Tiziano; Rizzolio, Flavio
A guide to PIN1 function and mutations across cancers
2019-01-01 El Boustani, Maguie; De Stefano, Lucia; Caligiuri, Isabella; Mouawad, Nayla; Granchi, Carlotta; Canzonieri, Vincenzo; Tuccinardi, Tiziano; Giordano, Antonio; Rizzolio, Flavio
A patent review of Monoacylglycerol Lipase (MAGL) inhibitors (2013-2017)
2017-01-01 Granchi, Carlotta; Caligiuri, Isabella; Minutolo, Filippo; Rizzolio, Flavio; Tuccinardi, Tiziano
A Virtual Screening Study for Lactate Dehydrogenase 5 Inhibitors by using a Pharmacophore-Based Approach
2016-01-01 Tuccinardi, Tiziano; Poli, Giulio; Corchia, Isacco; Granchi, Carlotta; Lapillo, Margherita; Macchia, Marco; Minutolo, Filippo; Ortore, GABRIELLA MARIA PIA; Martinelli, Adriano
Abstract 3082: Targeting hypoxic pancreatic cancer cells with glucose conjugated lactate dehydrogenase inhibitor NHI-Glc-2
2019-01-01 Hassouni, Btissame El; Sciarrillo, Rocco; Gómez, Valentina Edith; Maftouh, Mina; Mantini, Giulia; Vonk, Christian M.; Granchi, Carlotta; Funel, Niccola; Minutolo, Filippo; Peters, Godefridus J.; Giovannetti, Elisa
Activators of Sirtuin-1 and their Involvement in Cardioprotection
2018-01-01 Granchi, Carlotta; Minutolo, Filippo
AGENTI TERAPEUTICI IN GRADO DI RIDURRE LA PRODUZIONE CELLULARE DI ACIDO LATTICO E COMPOSIZIONI FARMACEUTICHE CHE COMPRENDONO TALI COMPOSTI
2011-01-01 Minutolo, Filippo; Macchia, Marco; Granchi, Carlotta; DI BUSSOLO, Valeria; Giannaccini, Gino; Lucacchini, Antonio; Paul J., Hergenrother; Emilia C., Calvaresi
alpha-Naphthylaminopropan-2-ol Derivatives as BACE1 Inhibitors
2008-01-01 V., Asso; E., Ghilardi; Bertini, Simone; Digiacomo, Maria; Granchi, Carlotta; Minutolo, Filippo; Rapposelli, Simona; A., Bortolato; S., Moro; Macchia, Marco
alpha-Naphtylaminopropan-2-ol derivatives as BACE1 inhibitors
2008-01-01 V., Asso; E., Ghilardi; Bertini, Simone; Digiacomo, Maria; Granchi, Carlotta; Minutolo, Filippo; Rapposelli, Simona; A., Bortolato; S., Moro; Macchia, Marco
Aminobenzothiazoles as inhibitors of tau-fibril formation in Alzheimer's and other neurodegenerative diseases
2008-01-01 Minutolo, Filippo; G., Bellini; Bertini, Simone; Granchi, Carlotta; Macchia, Marco; C., Ballatore; A., Crowe; E., Hyde; K., Brunden; J. Q., Trojanowski; V. M. Y., Lee
An Update on Patents Covering Agents That Interfere with the Cancer Glycolytic Cascade
2018-01-01 Fortunato, Serena; Bononi, Giulia; Granchi, Carlotta; Minutolo, Filippo
An update on therapeutic opportunities offered by cancer glycolytic metabolism
2014-01-01 Granchi, Carlotta; Fancelli, D.; Minutolo, Filippo
An updated patent review of monoacylglycerol lipase (MAGL) inhibitors (2018-present)
2021-01-01 Bononi, G.; Poli, G.; Rizzolio, F.; Tuccinardi, T.; Macchia, M.; Minutolo, F.; Granchi, C.
Anticancer agents interacting with membrane glucose transporters
2016-01-01 Granchi, Carlotta; Fortunato, Serena; Minutolo, Filippo
Anticancer Agents That Counteract Tumor Glycolysis
2012-01-01 Granchi, Carlotta; Minutolo, Filippo
Antiproliferative oxime derivatives that inhibit glucose transporter 1 (GLUT1) in cancer cells
2013-01-01 Tuccinardi, Tiziano; Granchi, Carlotta; Jessica, Iegre; Paterni, Ilaria; Bertini, Simone; Macchia, Marco; Martinelli, Adriano; Yanrong, Qian; Xiaozhuo, Chen; Minutolo, Filippo
Application of MM-PBSA methods in virtual screening
2020-01-01 Poli, G.; Granchi, C.; Rizzolio, F.; Tuccinardi, T.
Assessing the differential action on cancer cells of LDH-A inhibitors based on the N-hydroxyindole-2-carboxylate (NHI) and malonic (Mal) scaffolds
2013-01-01 Granchi, Carlotta; Emilia C., Calvaresi; Tuccinardi, Tiziano; Paterni, Ilaria; Macchia, Marco; Martinelli, Adriano; Paul J., Hergenrother; Minutolo, Filippo
ATP citrate lyase (ACLY) inhibitors: An anti-cancer strategy at the crossroads of glucose and lipid metabolism
2018-01-01 Granchi, Carlotta
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
4-Aryliden-2-methyloxazol-5(4H)-one as a new scaffold for selective reversible MAGL inhibitors | 1-gen-2016 | Granchi, Carlotta; Rizzolio, F; Bordoni, Vittorio; Caligiuri, I; Manera, Clementina; Macchia, Marco; Minutolo, Filippo; Martinelli, Adriano; Giordano, A; Tuccinardi, Tiziano | |
A carrier free delivery system of a monoacylglycerol lipase hydrophobic inhibitor | 1-gen-2022 | Adeel, Muhammad; Saorin, Gloria; Boccalon, Giacomo; Sfriso, Andrea Augusto; Parisi, Salvatore; Moro, Isabella; Palazzolo, Stefano; Caligiuri, Isabella; Granchi, Carlotta; Corona, Giuseppe; Cemazar, Maja; Canzonieri, Vincenzo; Tuccinardi, Tiziano; Rizzolio, Flavio | |
A guide to PIN1 function and mutations across cancers | 1-gen-2019 | El Boustani, Maguie; De Stefano, Lucia; Caligiuri, Isabella; Mouawad, Nayla; Granchi, Carlotta; Canzonieri, Vincenzo; Tuccinardi, Tiziano; Giordano, Antonio; Rizzolio, Flavio | |
A patent review of Monoacylglycerol Lipase (MAGL) inhibitors (2013-2017) | 1-gen-2017 | Granchi, Carlotta; Caligiuri, Isabella; Minutolo, Filippo; Rizzolio, Flavio; Tuccinardi, Tiziano | |
A Virtual Screening Study for Lactate Dehydrogenase 5 Inhibitors by using a Pharmacophore-Based Approach | 1-gen-2016 | Tuccinardi, Tiziano; Poli, Giulio; Corchia, Isacco; Granchi, Carlotta; Lapillo, Margherita; Macchia, Marco; Minutolo, Filippo; Ortore, GABRIELLA MARIA PIA; Martinelli, Adriano | |
Abstract 3082: Targeting hypoxic pancreatic cancer cells with glucose conjugated lactate dehydrogenase inhibitor NHI-Glc-2 | 1-gen-2019 | Hassouni, Btissame El; Sciarrillo, Rocco; Gómez, Valentina Edith; Maftouh, Mina; Mantini, Giulia; Vonk, Christian M.; Granchi, Carlotta; Funel, Niccola; Minutolo, Filippo; Peters, Godefridus J.; Giovannetti, Elisa | |
Activators of Sirtuin-1 and their Involvement in Cardioprotection | 1-gen-2018 | Granchi, Carlotta; Minutolo, Filippo | |
AGENTI TERAPEUTICI IN GRADO DI RIDURRE LA PRODUZIONE CELLULARE DI ACIDO LATTICO E COMPOSIZIONI FARMACEUTICHE CHE COMPRENDONO TALI COMPOSTI | 1-gen-2011 | Minutolo, Filippo; Macchia, Marco; Granchi, Carlotta; DI BUSSOLO, Valeria; Giannaccini, Gino; Lucacchini, Antonio; Paul J., Hergenrother; Emilia C., Calvaresi | |
alpha-Naphthylaminopropan-2-ol Derivatives as BACE1 Inhibitors | 1-gen-2008 | V., Asso; E., Ghilardi; Bertini, Simone; Digiacomo, Maria; Granchi, Carlotta; Minutolo, Filippo; Rapposelli, Simona; A., Bortolato; S., Moro; Macchia, Marco | |
alpha-Naphtylaminopropan-2-ol derivatives as BACE1 inhibitors | 1-gen-2008 | V., Asso; E., Ghilardi; Bertini, Simone; Digiacomo, Maria; Granchi, Carlotta; Minutolo, Filippo; Rapposelli, Simona; A., Bortolato; S., Moro; Macchia, Marco | |
Aminobenzothiazoles as inhibitors of tau-fibril formation in Alzheimer's and other neurodegenerative diseases | 1-gen-2008 | Minutolo, Filippo; G., Bellini; Bertini, Simone; Granchi, Carlotta; Macchia, Marco; C., Ballatore; A., Crowe; E., Hyde; K., Brunden; J. Q., Trojanowski; V. M. Y., Lee | |
An Update on Patents Covering Agents That Interfere with the Cancer Glycolytic Cascade | 1-gen-2018 | Fortunato, Serena; Bononi, Giulia; Granchi, Carlotta; Minutolo, Filippo | |
An update on therapeutic opportunities offered by cancer glycolytic metabolism | 1-gen-2014 | Granchi, Carlotta; Fancelli, D.; Minutolo, Filippo | |
An updated patent review of monoacylglycerol lipase (MAGL) inhibitors (2018-present) | 1-gen-2021 | Bononi, G.; Poli, G.; Rizzolio, F.; Tuccinardi, T.; Macchia, M.; Minutolo, F.; Granchi, C. | |
Anticancer agents interacting with membrane glucose transporters | 1-gen-2016 | Granchi, Carlotta; Fortunato, Serena; Minutolo, Filippo | |
Anticancer Agents That Counteract Tumor Glycolysis | 1-gen-2012 | Granchi, Carlotta; Minutolo, Filippo | |
Antiproliferative oxime derivatives that inhibit glucose transporter 1 (GLUT1) in cancer cells | 1-gen-2013 | Tuccinardi, Tiziano; Granchi, Carlotta; Jessica, Iegre; Paterni, Ilaria; Bertini, Simone; Macchia, Marco; Martinelli, Adriano; Yanrong, Qian; Xiaozhuo, Chen; Minutolo, Filippo | |
Application of MM-PBSA methods in virtual screening | 1-gen-2020 | Poli, G.; Granchi, C.; Rizzolio, F.; Tuccinardi, T. | |
Assessing the differential action on cancer cells of LDH-A inhibitors based on the N-hydroxyindole-2-carboxylate (NHI) and malonic (Mal) scaffolds | 1-gen-2013 | Granchi, Carlotta; Emilia C., Calvaresi; Tuccinardi, Tiziano; Paterni, Ilaria; Macchia, Marco; Martinelli, Adriano; Paul J., Hergenrother; Minutolo, Filippo | |
ATP citrate lyase (ACLY) inhibitors: An anti-cancer strategy at the crossroads of glucose and lipid metabolism | 1-gen-2018 | Granchi, Carlotta |