GRANCHI, CARLOTTA Statistiche
GRANCHI, CARLOTTA
DIPARTIMENTO DI FARMACIA
A carrier free delivery system of a MAGL inhibitor is effective on ovarian cancer
2024-01-01 Palazzolo, Stefano; Saorin, Gloria; Corona, Giuseppe; Granchi, Carlotta; Tuccinardi, Tiziano; Kamensek, Urska; Brezar, Simona Kranjc; Cemazar, Maja; Canzonieri, Vincenzo; Rizzolio, Flavio
A patent review of lactate dehydrogenase inhibitors (2014-present)
2024-01-01 Bononi, Giulia; Di Bussolo, Valeria; Tuccinardi, Tiziano; Minutolo, Filippo; Granchi, Carlotta
Design, synthesis, ADME and biological evaluation of benzylpiperidine and benzylpiperazine derivatives as novel reversible monoacylglycerol lipase (MAGL) inhibitors
2024-01-01 Di Stefano, Miriana; Masoni, Samuele; Bononi, Giulia; Poli, Giulio; Galati, Salvatore; Gado, Francesca; Manzi, Simone; Vagaggini, Chiara; Brai, Annalaura; Caligiuri, Isabella; Asif, Kanwal; Rizzolio, Flavio; Macchia, Marco; Chicca, Andrea; Sodi, Andrea; Di Bussolo, Valeria; Minutolo, Filippo; Meier, Philip; Gertsch, Jürg; Granchi, Carlotta; Dreassi, Elena; Tuccinardi, Tiziano
Glycoconjugate coumarins exploiting metabolism-enhanced fluorescence and preferential uptake: New optical tools for tumor cell staining
2024-01-01 Iacopini, Dalila; Santi, Melissa; Santangelo, Maria Chiara; Sardelli, Gemma; Piazza, Lucia; Mosca, Rossella; Comparini, Lucrezia Margherita; Granchi, Carlotta; Pineschi, Mauro; Di Pietro, Sebastiano; Signore, Giovanni; Di Bussolo, Valeria
Nuovi agenti antivirali a struttura N-idrossiindrol-carbossamidica
2024-01-01 Minutolo, Filippo; Pistello, Mauro; DI BUSSOLO, Valeria; Freer, Giulia; Quaranta, Paola; Granchi, Carlotta; Tuccinardi, Tiziano; Poli, Giulio; Bononi, Giulia; Masoni, Samuele
Sirtuin 1-activating derivatives belonging to the anilinopyridine class displaying in vivo cardioprotective activities
2024-01-01 Bononi, G.; Citi, V.; Martelli, A.; Poli, G.; Tuccinardi, T.; Granchi, C.; Testai, L.; Calderone, V.; Minutolo, F.
SMS121, a new inhibitor of CD36, impairs fatty acid uptake and viability of acute myeloid leukemia
2024-01-01 Åbacka, Hannah; Masoni, Samuele; Poli, Giulio; Huang, Peng; Gusso, Francesco; Granchi, Carlotta; Minutolo, Filippo; Tuccinardi, Tiziano; Hagström-Andersson, Anna K; Lindkvist-Petersson, Karin
The Benzoylpiperidine Fragment as a Privileged Structure in Medicinal Chemistry: A Comprehensive Review
2024-01-01 Bononi, Giulia; Lonzi, Chiara; Tuccinardi, Tiziano; Minutolo, Filippo; Granchi, Carlotta
VenomPred 2.0: A Novel In Silico Platform for an Extended and Human Interpretable Toxicological Profiling of Small Molecules
2024-01-01 Di Stefano, Miriana; Galati, Salvatore; Piazza, Lisa; Granchi, Carlotta; Mancini, Simone; Fratini, Filippo; Macchia, Marco; Poli, Giulio; Tuccinardi, Tiziano
WaSPred: A reliable AI-based water solubility predictor for small molecules
2024-01-01 Di Stefano, Miriana; Galati, Salvatore; Lonzi, Chiara; Granchi, Carlotta; Poli, Giulio; Tuccinardi, Tiziano; Macchia, Marco
Watermelon: setup and validation of an in silico fragment-based approach
2024-01-01 Di Stefano, Miriana; Galati, Salvatore; Piazza, Lisa; Gado, Francesca; Granchi, Carlotta; Macchia, Marco; Giordano, Antonio; Tuccinardi, Tiziano; Poli, Giulio
Combined inhibition of pyruvate dehydrogenase kinase 1 and lactate dehydrogenase a induces metabolic and signaling reprogramming and enhances lung adenocarcinoma cell killing
2023-01-01 Zhou, Yan; Guo, Yizhen; Ran, Maoxin; Shan, Wenying; Granchi, Carlotta; Giovannetti, Elisa; Minutolo, Filippo; Peters, Godefridus J.; Tam, Kin Yip
Enhanced activity of a pluronic F127 formulated Pin1 inhibitor for ovarian cancer therapy
2023-01-01 Saorin, G.; Mauceri, M.; Cavarzerani, E.; Caligiuri, I.; Bononi, G.; Granchi, C.; Bartoletti, M.; Perin, T.; Tuccinardi, T.; Canzonieri, V.; Adeel, M.; Rizzolio, F.
First-in-Class Dual Targeting Compounds for the Management of Seizures in Glucose Transporter Type 1 Deficiency Syndrome
2023-01-01 Angeli, Andrea; Ferraroni, Marta; Granchi, Carlotta; Minutolo, Filippo; Chen, Xiaozhuo; Shriwas, Pratik; Russo, Emilio; Leo, Antonio; Selleri, Silvia; Carta, Fabrizio; Supuran, Claudiu T
Identification of New GSK3β Inhibitors through a Consensus Machine Learning-Based Virtual Screening
2023-01-01 Galati, Salvatore; Di Stefano, Miriana; Bertini, Simone; Granchi, Carlotta; Giordano, Antonio; Gado, Francesca; Macchia, Marco; Tuccinardi, Tiziano; Poli, Giulio
Metabolic Effects of New Glucose Transporter (GLUT-1) and Lactate Dehydrogenase-A (LDH-A) Inhibitors against Chemoresistant Malignant Mesothelioma
2023-01-01 Franczak, Marika A.; Krol, Oliwia; Harasim, Gabriela; Jedrzejewska, Agata; Zaffaroni, Nadia; Granchi, Carlotta; Minutolo, Filippo; Avan, Amir; Giovannetti, Elisa; Smolenski, Ryszard T.; Peters, Godefridus J.
A carrier free delivery system of a monoacylglycerol lipase hydrophobic inhibitor
2022-01-01 Adeel, Muhammad; Saorin, Gloria; Boccalon, Giacomo; Sfriso, Andrea Augusto; Parisi, Salvatore; Moro, Isabella; Palazzolo, Stefano; Caligiuri, Isabella; Granchi, Carlotta; Corona, Giuseppe; Cemazar, Maja; Canzonieri, Vincenzo; Tuccinardi, Tiziano; Rizzolio, Flavio
ATP-citrate lyase (ACLY) inhibitors as therapeutic agents: a patenting perspective
2022-01-01 Granchi, Carlotta
Biological Activity of Natural and Synthetic Compounds
2022-01-01 Granchi, Carlotta
Functionalized aliphatic polyketones with germicide activity
2022-01-01 Araya-Hermosilla, E.; Parlanti, P.; Gemmi, M.; Mattoli, V.; Di Pietro, S.; Iacopini, D.; Granchi, C.; Turchi, B.; Fratini, F.; Di Bussolo, V.; Minutolo, F.; Picchioni, F.; Pucci, A.
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| A carrier free delivery system of a MAGL inhibitor is effective on ovarian cancer | 1-gen-2024 | Palazzolo, Stefano; Saorin, Gloria; Corona, Giuseppe; Granchi, Carlotta; Tuccinardi, Tiziano; Kamensek, Urska; Brezar, Simona Kranjc; Cemazar, Maja; Canzonieri, Vincenzo; Rizzolio, Flavio | |
| A patent review of lactate dehydrogenase inhibitors (2014-present) | 1-gen-2024 | Bononi, Giulia; Di Bussolo, Valeria; Tuccinardi, Tiziano; Minutolo, Filippo; Granchi, Carlotta | |
| Design, synthesis, ADME and biological evaluation of benzylpiperidine and benzylpiperazine derivatives as novel reversible monoacylglycerol lipase (MAGL) inhibitors | 1-gen-2024 | Di Stefano, Miriana; Masoni, Samuele; Bononi, Giulia; Poli, Giulio; Galati, Salvatore; Gado, Francesca; Manzi, Simone; Vagaggini, Chiara; Brai, Annalaura; Caligiuri, Isabella; Asif, Kanwal; Rizzolio, Flavio; Macchia, Marco; Chicca, Andrea; Sodi, Andrea; Di Bussolo, Valeria; Minutolo, Filippo; Meier, Philip; Gertsch, Jürg; Granchi, Carlotta; Dreassi, Elena; Tuccinardi, Tiziano | |
| Glycoconjugate coumarins exploiting metabolism-enhanced fluorescence and preferential uptake: New optical tools for tumor cell staining | 1-gen-2024 | Iacopini, Dalila; Santi, Melissa; Santangelo, Maria Chiara; Sardelli, Gemma; Piazza, Lucia; Mosca, Rossella; Comparini, Lucrezia Margherita; Granchi, Carlotta; Pineschi, Mauro; Di Pietro, Sebastiano; Signore, Giovanni; Di Bussolo, Valeria | |
| Nuovi agenti antivirali a struttura N-idrossiindrol-carbossamidica | 1-gen-2024 | Minutolo, Filippo; Pistello, Mauro; DI BUSSOLO, Valeria; Freer, Giulia; Quaranta, Paola; Granchi, Carlotta; Tuccinardi, Tiziano; Poli, Giulio; Bononi, Giulia; Masoni, Samuele | |
| Sirtuin 1-activating derivatives belonging to the anilinopyridine class displaying in vivo cardioprotective activities | 1-gen-2024 | Bononi, G.; Citi, V.; Martelli, A.; Poli, G.; Tuccinardi, T.; Granchi, C.; Testai, L.; Calderone, V.; Minutolo, F. | |
| SMS121, a new inhibitor of CD36, impairs fatty acid uptake and viability of acute myeloid leukemia | 1-gen-2024 | Åbacka, Hannah; Masoni, Samuele; Poli, Giulio; Huang, Peng; Gusso, Francesco; Granchi, Carlotta; Minutolo, Filippo; Tuccinardi, Tiziano; Hagström-Andersson, Anna K; Lindkvist-Petersson, Karin | |
| The Benzoylpiperidine Fragment as a Privileged Structure in Medicinal Chemistry: A Comprehensive Review | 1-gen-2024 | Bononi, Giulia; Lonzi, Chiara; Tuccinardi, Tiziano; Minutolo, Filippo; Granchi, Carlotta | |
| VenomPred 2.0: A Novel In Silico Platform for an Extended and Human Interpretable Toxicological Profiling of Small Molecules | 1-gen-2024 | Di Stefano, Miriana; Galati, Salvatore; Piazza, Lisa; Granchi, Carlotta; Mancini, Simone; Fratini, Filippo; Macchia, Marco; Poli, Giulio; Tuccinardi, Tiziano | |
| WaSPred: A reliable AI-based water solubility predictor for small molecules | 1-gen-2024 | Di Stefano, Miriana; Galati, Salvatore; Lonzi, Chiara; Granchi, Carlotta; Poli, Giulio; Tuccinardi, Tiziano; Macchia, Marco | |
| Watermelon: setup and validation of an in silico fragment-based approach | 1-gen-2024 | Di Stefano, Miriana; Galati, Salvatore; Piazza, Lisa; Gado, Francesca; Granchi, Carlotta; Macchia, Marco; Giordano, Antonio; Tuccinardi, Tiziano; Poli, Giulio | |
| Combined inhibition of pyruvate dehydrogenase kinase 1 and lactate dehydrogenase a induces metabolic and signaling reprogramming and enhances lung adenocarcinoma cell killing | 1-gen-2023 | Zhou, Yan; Guo, Yizhen; Ran, Maoxin; Shan, Wenying; Granchi, Carlotta; Giovannetti, Elisa; Minutolo, Filippo; Peters, Godefridus J.; Tam, Kin Yip | |
| Enhanced activity of a pluronic F127 formulated Pin1 inhibitor for ovarian cancer therapy | 1-gen-2023 | Saorin, G.; Mauceri, M.; Cavarzerani, E.; Caligiuri, I.; Bononi, G.; Granchi, C.; Bartoletti, M.; Perin, T.; Tuccinardi, T.; Canzonieri, V.; Adeel, M.; Rizzolio, F. | |
| First-in-Class Dual Targeting Compounds for the Management of Seizures in Glucose Transporter Type 1 Deficiency Syndrome | 1-gen-2023 | Angeli, Andrea; Ferraroni, Marta; Granchi, Carlotta; Minutolo, Filippo; Chen, Xiaozhuo; Shriwas, Pratik; Russo, Emilio; Leo, Antonio; Selleri, Silvia; Carta, Fabrizio; Supuran, Claudiu T | |
| Identification of New GSK3β Inhibitors through a Consensus Machine Learning-Based Virtual Screening | 1-gen-2023 | Galati, Salvatore; Di Stefano, Miriana; Bertini, Simone; Granchi, Carlotta; Giordano, Antonio; Gado, Francesca; Macchia, Marco; Tuccinardi, Tiziano; Poli, Giulio | |
| Metabolic Effects of New Glucose Transporter (GLUT-1) and Lactate Dehydrogenase-A (LDH-A) Inhibitors against Chemoresistant Malignant Mesothelioma | 1-gen-2023 | Franczak, Marika A.; Krol, Oliwia; Harasim, Gabriela; Jedrzejewska, Agata; Zaffaroni, Nadia; Granchi, Carlotta; Minutolo, Filippo; Avan, Amir; Giovannetti, Elisa; Smolenski, Ryszard T.; Peters, Godefridus J. | |
| A carrier free delivery system of a monoacylglycerol lipase hydrophobic inhibitor | 1-gen-2022 | Adeel, Muhammad; Saorin, Gloria; Boccalon, Giacomo; Sfriso, Andrea Augusto; Parisi, Salvatore; Moro, Isabella; Palazzolo, Stefano; Caligiuri, Isabella; Granchi, Carlotta; Corona, Giuseppe; Cemazar, Maja; Canzonieri, Vincenzo; Tuccinardi, Tiziano; Rizzolio, Flavio | |
| ATP-citrate lyase (ACLY) inhibitors as therapeutic agents: a patenting perspective | 1-gen-2022 | Granchi, Carlotta | |
| Biological Activity of Natural and Synthetic Compounds | 1-gen-2022 | Granchi, Carlotta | |
| Functionalized aliphatic polyketones with germicide activity | 1-gen-2022 | Araya-Hermosilla, E.; Parlanti, P.; Gemmi, M.; Mattoli, V.; Di Pietro, S.; Iacopini, D.; Granchi, C.; Turchi, B.; Fratini, F.; Di Bussolo, V.; Minutolo, F.; Picchioni, F.; Pucci, A. |