RAPPOSELLI, SIMONA Statistiche
RAPPOSELLI, SIMONA
DIPARTIMENTO DI FARMACIA
New Insights into Bitopic Orthosteric/Allosteric Ligands of Cannabinoid Receptor Type 2
2023-01-01 Ferrisi, Rebecca; Polini, Beatrice; Ricardi, Caterina; Gado, Francesca; Mohamed, Kawthar A; Baron, Giovanna; Faiella, Salvatore; Poli, Giulio; Rapposelli, Simona; Saccomanni, Giuseppe; Aldini, Giancarlo; Chiellini, Grazia; Laprairie, Robert B; Manera, Clementina; Ortore, Gabriella
New Insights into Bitopic Orthosteric/Allosteric Ligands of Cannabinoid Receptor Type 2
2023-01-01 Ferrisi, Rebecca; Polini, Beatrice; Ricardi, Caterina; Gado, Francesca; Mohamed, Kawthar A; Baron, Giovanna; Faiella, Salvatore; Poli, Giulio; Rapposelli, Simona; Saccomanni, Giuseppe; Aldini, Giancarlo; Chiellini, Grazia; Laprairie, Robert B; Manera, Clementina; Ortore, Gabriella
Potential use of TG68 - A novel thyromimetic - for the treatment of non-alcoholic fatty liver (NAFLD)-associated hepatocarcinogenesis
2023-01-01 Caddeo, Andrea; Serra, Marina; Sedda, Francesca; Bacci, Andrea; Manera, Clementina; Rapposelli, Simona; Columbano, Amedeo; Perra, Andrea; Kowalik, Marta Anna
Abstract 2569: Development of potent dual PDK1/AurA kinase inhibitors for Ewing sarcoma therapy
2022-01-01 Riveiro, Maria Eugenia; Huguet, Samuel; Vazquez, Ramiro; Frapolli, Roberta; Puricelli, Guido; Sestito, Simona; Madar, Olivier; Rezai, Keyvan; Garau, Gianpiero; Rapposelli, Simona
Design, synthesis and biological evaluation of novel orthosteric-allosteric ligands of the cannabinoid receptor type 2 (CB2R)
2022-01-01 Ferrisi, Rebecca; Gado, Francesca; Polini, Beatrice; Ricardi, Caterina; Mohamed, Kawthar A.; Stevenson, Lesley A.; Ortore, GABRIELLA MARIA PIA; Rapposelli, Simona; Saccomanni, Giuseppe; Pertwee, Roger G.; Laprairie, Robert B.; Manera, Clementina; Chiellini, Grazia
Design, Synthesis, and Biological Activity of New CB2 Receptor Ligands: from Orthosteric and Allosteric Modulators to Dualsteric/Bitopic Ligands
2022-01-01 Gado, Francesca; Ferrisi, Rebecca; Polini, Beatrice; Mohamed, Kawthar A.; Ricardi, Caterina; Lucarini, Elena; Carpi, Sara; Domenichini, Federica; Stevenson, Lesley A.; Rapposelli, Simona; Saccomanni, Giuseppe; Nieri, Paola; Ortore, GABRIELLA MARIA PIA; Pertwee, Roger G.; Ghelardini, Carla; Di Cesare Mannelli, Lorenzo; Chiellini, Grazia; Laprairie, Robert B.; Manera, Clementina
Design, Synthesis, and In Vitro Evaluation of Novel 8-Amino-Quinoline Combined with Natural Antioxidant Acids
2022-01-01 Bacci, Andrea; Corsi, Francesca; Runfola, Massimiliano; Sestito, Simona; Piano, Ilaria; Manera, Clementina; Saccomanni, Giuseppe; Gargini, Claudia; Rapposelli, Simona
Editorial: New insights into the mechanisms of resistance to anti-cancer drugs
2022-01-01 Bertoni, Francesco; Rapposelli, Simona
Multi-Target Mechanisms of Phytochemicals in Alzheimer's Disease: Effects on Oxidative Stress, Neuroinflammation and Protein Aggregation
2022-01-01 Sharifi-Rad, Javad; Rapposelli, Simona; Sestito, Simona; Herrera-Bravo, Jesús; Arancibia-Diaz, Alejandra; Salazar, Luis A; Yeskaliyeva, Balakyz; Beyatli, Ahmet; Leyva-Gómez, Gerardo; González-Contreras, Carlos; Gürer, Eda Sönmez; Martorell, Miquel; Calina, Daniela
Synthesis and In Vitro Characterization of Selective Cannabinoid CB2 Receptor Agonists: Biological Evaluation against Neuroblastoma Cancer Cells
2022-01-01 Gado, Francesca; Ferrisi, Rebecca; Di Somma, Sarah; Napolitano, Fabiana; Mohamed, Kawthar A; Stevenson, Lesley A; Rapposelli, Simona; Saccomanni, Giuseppe; Portella, Giuseppe; Pertwee, Roger G; Laprairie, Robert B; Malfitano, Anna Maria; Manera, Clementina
14-3-3 PROTEIN MODULATORS AS ANTITUMOR AGENTS
2021-01-01 Rapposelli, Simona; Gaudio, Eugenio; Dal Piaz, Fabrizio
Abstract 1294: Dual targeting of PDK1 and Aurora A using first-in class OXID-pyridonyl compounds in preclinical models of Ewing sarcoma
2021-01-01 Riveiro, Maria Eugenia; Rapposelli, Simona; Huguet, Samuel; Vazquez, Ramiro; Bekradda, Mohamed; Puricelli, Guido; Sestito, Simona; Madar, Olivier; Rezai, Keyvan
Beyond antioxidant effects: Nature-based templates unveil new strategies for neurodegenerative diseases
2021-01-01 Bacci, A.; Runfola, M.; Sestito, S.; Rapposelli, S.
Chitosan nanoparticles as a promising tool in nanomedicine with particular emphasis on oncological treatment
2021-01-01 Sharifi-Rad, J.; Quispe, C.; Butnariu, M.; Rotariu, L. S.; Sytar, O.; Sestito, S.; Rapposelli, S.; Akram, M.; Iqbal, M.; Krishna, A.; Kumar, N. V. A.; Braga, S. S.; Cardoso, S. M.; Jafernik, K.; Ekiert, H.; Cruz-Martins, N.; Szopa, A.; Villagran, M.; Mardones, L.; Martorell, M.; Docea, A. O.; Calina, D.
Development of potent dual PDK1/AurA kinase inhibitors for cancer therapy: Lead-optimization, structural insights, and ADME-Tox profile
2021-01-01 Sestito, S.; Bacci, A.; Chiarugi, S.; Runfola, M.; Gado, F.; Margheritis, E.; Gul, S.; Riveiro, M. E.; Vazquez, R.; Huguet, S.; Manera, C.; Rezai, K.; Garau, G.; Rapposelli, S.
Diphenyl-methane based thyromimetic inhibitors for transthyretin amyloidosis
2021-01-01 Kim, B.; Ko, Y. H.; Runfola, M.; Rapposelli, S.; Ortore, G.; Chiellini, G.; Kim, J. H.
Editorial: Protein-Protein Interactions: Drug Discovery for the Future
2021-01-01 Rapposelli, Simona; Gaudio, Eugenio; Bertozzi, Fabio; Gul, Sheraz
Identification of a Thyroid Hormone Derivative as a Pleiotropic Agent for the Treatment of Alzheimer's Disease
2021-01-01 Runfola, Massimiliano; Perni, Michele; Yang, Xiaoting; Marchese, Maria; Bacci, Andrea; Mero, Serena; Santorelli, Filippo M; Polini, Beatrice; Chiellini, Grazia; Giuliani, Daniela; Vilella, Antonietta; Bodria, Martina; Daini, Eleonora; Vandini, Eleonora; Rudge, Simon; Gul, Sheraz; Wakelam, Michale O J; Vendruscolo, Michele; Rapposelli, Simona
Late breaker posters
2021-01-01 Perra, Andrea; Anna Kowalik, Marta; Serra, Marina; Runfola, Massimiliano; Rapposelli, Simona; Columbano., Amedeo
Paving Luteolin Therapeutic Potentialities and Agro-Food-Pharma Applications: Emphasis on in Vivo Pharmacological Effects and Bioavailability Traits
2021-01-01 Taheri, Y.; Sharifi-Rad, J.; Antika, G.; Yilmaz, Y. B.; Tumer, T. B.; Abuhamdah, S.; Chandra, S.; Saklani, S.; Kilic, C. S.; Sestito, S.; Dastan, S. D.; Kumar, M.; Alshehri, M. M.; Rapposelli, S.; Cruz-Martins, N.; Cho, W. C.
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| New Insights into Bitopic Orthosteric/Allosteric Ligands of Cannabinoid Receptor Type 2 | 1-gen-2023 | Ferrisi, Rebecca; Polini, Beatrice; Ricardi, Caterina; Gado, Francesca; Mohamed, Kawthar A; Baron, Giovanna; Faiella, Salvatore; Poli, Giulio; Rapposelli, Simona; Saccomanni, Giuseppe; Aldini, Giancarlo; Chiellini, Grazia; Laprairie, Robert B; Manera, Clementina; Ortore, Gabriella | |
| New Insights into Bitopic Orthosteric/Allosteric Ligands of Cannabinoid Receptor Type 2 | 1-gen-2023 | Ferrisi, Rebecca; Polini, Beatrice; Ricardi, Caterina; Gado, Francesca; Mohamed, Kawthar A; Baron, Giovanna; Faiella, Salvatore; Poli, Giulio; Rapposelli, Simona; Saccomanni, Giuseppe; Aldini, Giancarlo; Chiellini, Grazia; Laprairie, Robert B; Manera, Clementina; Ortore, Gabriella | |
| Potential use of TG68 - A novel thyromimetic - for the treatment of non-alcoholic fatty liver (NAFLD)-associated hepatocarcinogenesis | 1-gen-2023 | Caddeo, Andrea; Serra, Marina; Sedda, Francesca; Bacci, Andrea; Manera, Clementina; Rapposelli, Simona; Columbano, Amedeo; Perra, Andrea; Kowalik, Marta Anna | |
| Abstract 2569: Development of potent dual PDK1/AurA kinase inhibitors for Ewing sarcoma therapy | 1-gen-2022 | Riveiro, Maria Eugenia; Huguet, Samuel; Vazquez, Ramiro; Frapolli, Roberta; Puricelli, Guido; Sestito, Simona; Madar, Olivier; Rezai, Keyvan; Garau, Gianpiero; Rapposelli, Simona | |
| Design, synthesis and biological evaluation of novel orthosteric-allosteric ligands of the cannabinoid receptor type 2 (CB2R) | 1-gen-2022 | Ferrisi, Rebecca; Gado, Francesca; Polini, Beatrice; Ricardi, Caterina; Mohamed, Kawthar A.; Stevenson, Lesley A.; Ortore, GABRIELLA MARIA PIA; Rapposelli, Simona; Saccomanni, Giuseppe; Pertwee, Roger G.; Laprairie, Robert B.; Manera, Clementina; Chiellini, Grazia | |
| Design, Synthesis, and Biological Activity of New CB2 Receptor Ligands: from Orthosteric and Allosteric Modulators to Dualsteric/Bitopic Ligands | 1-gen-2022 | Gado, Francesca; Ferrisi, Rebecca; Polini, Beatrice; Mohamed, Kawthar A.; Ricardi, Caterina; Lucarini, Elena; Carpi, Sara; Domenichini, Federica; Stevenson, Lesley A.; Rapposelli, Simona; Saccomanni, Giuseppe; Nieri, Paola; Ortore, GABRIELLA MARIA PIA; Pertwee, Roger G.; Ghelardini, Carla; Di Cesare Mannelli, Lorenzo; Chiellini, Grazia; Laprairie, Robert B.; Manera, Clementina | |
| Design, Synthesis, and In Vitro Evaluation of Novel 8-Amino-Quinoline Combined with Natural Antioxidant Acids | 1-gen-2022 | Bacci, Andrea; Corsi, Francesca; Runfola, Massimiliano; Sestito, Simona; Piano, Ilaria; Manera, Clementina; Saccomanni, Giuseppe; Gargini, Claudia; Rapposelli, Simona | |
| Editorial: New insights into the mechanisms of resistance to anti-cancer drugs | 1-gen-2022 | Bertoni, Francesco; Rapposelli, Simona | |
| Multi-Target Mechanisms of Phytochemicals in Alzheimer's Disease: Effects on Oxidative Stress, Neuroinflammation and Protein Aggregation | 1-gen-2022 | Sharifi-Rad, Javad; Rapposelli, Simona; Sestito, Simona; Herrera-Bravo, Jesús; Arancibia-Diaz, Alejandra; Salazar, Luis A; Yeskaliyeva, Balakyz; Beyatli, Ahmet; Leyva-Gómez, Gerardo; González-Contreras, Carlos; Gürer, Eda Sönmez; Martorell, Miquel; Calina, Daniela | |
| Synthesis and In Vitro Characterization of Selective Cannabinoid CB2 Receptor Agonists: Biological Evaluation against Neuroblastoma Cancer Cells | 1-gen-2022 | Gado, Francesca; Ferrisi, Rebecca; Di Somma, Sarah; Napolitano, Fabiana; Mohamed, Kawthar A; Stevenson, Lesley A; Rapposelli, Simona; Saccomanni, Giuseppe; Portella, Giuseppe; Pertwee, Roger G; Laprairie, Robert B; Malfitano, Anna Maria; Manera, Clementina | |
| 14-3-3 PROTEIN MODULATORS AS ANTITUMOR AGENTS | 1-gen-2021 | Rapposelli, Simona; Gaudio, Eugenio; Dal Piaz, Fabrizio | |
| Abstract 1294: Dual targeting of PDK1 and Aurora A using first-in class OXID-pyridonyl compounds in preclinical models of Ewing sarcoma | 1-gen-2021 | Riveiro, Maria Eugenia; Rapposelli, Simona; Huguet, Samuel; Vazquez, Ramiro; Bekradda, Mohamed; Puricelli, Guido; Sestito, Simona; Madar, Olivier; Rezai, Keyvan | |
| Beyond antioxidant effects: Nature-based templates unveil new strategies for neurodegenerative diseases | 1-gen-2021 | Bacci, A.; Runfola, M.; Sestito, S.; Rapposelli, S. | |
| Chitosan nanoparticles as a promising tool in nanomedicine with particular emphasis on oncological treatment | 1-gen-2021 | Sharifi-Rad, J.; Quispe, C.; Butnariu, M.; Rotariu, L. S.; Sytar, O.; Sestito, S.; Rapposelli, S.; Akram, M.; Iqbal, M.; Krishna, A.; Kumar, N. V. A.; Braga, S. S.; Cardoso, S. M.; Jafernik, K.; Ekiert, H.; Cruz-Martins, N.; Szopa, A.; Villagran, M.; Mardones, L.; Martorell, M.; Docea, A. O.; Calina, D. | |
| Development of potent dual PDK1/AurA kinase inhibitors for cancer therapy: Lead-optimization, structural insights, and ADME-Tox profile | 1-gen-2021 | Sestito, S.; Bacci, A.; Chiarugi, S.; Runfola, M.; Gado, F.; Margheritis, E.; Gul, S.; Riveiro, M. E.; Vazquez, R.; Huguet, S.; Manera, C.; Rezai, K.; Garau, G.; Rapposelli, S. | |
| Diphenyl-methane based thyromimetic inhibitors for transthyretin amyloidosis | 1-gen-2021 | Kim, B.; Ko, Y. H.; Runfola, M.; Rapposelli, S.; Ortore, G.; Chiellini, G.; Kim, J. H. | |
| Editorial: Protein-Protein Interactions: Drug Discovery for the Future | 1-gen-2021 | Rapposelli, Simona; Gaudio, Eugenio; Bertozzi, Fabio; Gul, Sheraz | |
| Identification of a Thyroid Hormone Derivative as a Pleiotropic Agent for the Treatment of Alzheimer's Disease | 1-gen-2021 | Runfola, Massimiliano; Perni, Michele; Yang, Xiaoting; Marchese, Maria; Bacci, Andrea; Mero, Serena; Santorelli, Filippo M; Polini, Beatrice; Chiellini, Grazia; Giuliani, Daniela; Vilella, Antonietta; Bodria, Martina; Daini, Eleonora; Vandini, Eleonora; Rudge, Simon; Gul, Sheraz; Wakelam, Michale O J; Vendruscolo, Michele; Rapposelli, Simona | |
| Late breaker posters | 1-gen-2021 | Perra, Andrea; Anna Kowalik, Marta; Serra, Marina; Runfola, Massimiliano; Rapposelli, Simona; Columbano., Amedeo | |
| Paving Luteolin Therapeutic Potentialities and Agro-Food-Pharma Applications: Emphasis on in Vivo Pharmacological Effects and Bioavailability Traits | 1-gen-2021 | Taheri, Y.; Sharifi-Rad, J.; Antika, G.; Yilmaz, Y. B.; Tumer, T. B.; Abuhamdah, S.; Chandra, S.; Saklani, S.; Kilic, C. S.; Sestito, S.; Dastan, S. D.; Kumar, M.; Alshehri, M. M.; Rapposelli, S.; Cruz-Martins, N.; Cho, W. C. |