TUCCINARDI, TIZIANO Statistiche
TUCCINARDI, TIZIANO
DIPARTIMENTO DI FARMACIA
1,3-Dipolar Cycloaddition, HPLC Enantioseparation, and Docking Studies of Saccharin/Isoxazole and Saccharin/Isoxazoline Derivatives as Selective Carbonic Anhydrase IX and XII Inhibitors
2020-01-01 D'Ascenzio, M.; Secci, D.; Carradori, S.; Zara, S.; Guglielmi, P.; Cirilli, R.; Pierini, M.; Poli, G.; Tuccinardi, T.; Angeli, A.; Supuran, C. T.
1,8-Naphthyridin-4-one derivatives as new ligands of A2A adenosine receptors.
2005-01-01 Manera, Clementina; Betti, Laura; Cavallini, T.; Giannaccini, Gino; Martinelli, Adriano; Ortore, G.; Saccomanni, Giuseppe; Trincavelli, MARIA LETIZIA; Tuccinardi, Tiziano; Ferrarini, P. L.
3D-QSAR and virtual screening studies for the translocator protein(TSPO)
2008-01-01 Tuccinardi, Tiziano; Taliani, Sabrina; Bellandi, M; DA POZZO, Eleonora; Greco, G; Novellino, E; Martinelli, Adriano; DA SETTIMO PASSETTI, Federico; Martini, Claudia
4-Aryliden-2-methyloxazol-5(4H)-one as a new scaffold for selective reversible MAGL inhibitors
2016-01-01 Granchi, Carlotta; Rizzolio, F; Bordoni, Vittorio; Caligiuri, I; Manera, Clementina; Macchia, Marco; Minutolo, Filippo; Martinelli, Adriano; Giordano, A; Tuccinardi, Tiziano
5-Amino-2-phenyl[1,2,3]triazolo[1,2-a][1,2,4]benzotriazin-1-one: a Versatile Scaffold to Obtain Potent and Selective A3 Adenosine Receptor Antagonists
2007-01-01 DA SETTIMO PASSETTI, Federico; Primofiore, G.; Taliani, Sabrina; Marini, ANNA MARIA; LA MOTTA, Concettina; Simorini, Francesca; Salerno, Silvia; Sergianni, V.; Tuccinardi, Tiziano; Martinelli, Adriano; Cosimelli, B.; Greco, G.; Novellino, E.; Ciampi, O.; Trincavelli, MARIA LETIZIA; Martini, Claudia
A carrier free delivery system of a monoacylglycerol lipase hydrophobic inhibitor
2022-01-01 Adeel, Muhammad; Saorin, Gloria; Boccalon, Giacomo; Sfriso, Andrea Augusto; Parisi, Salvatore; Moro, Isabella; Palazzolo, Stefano; Caligiuri, Isabella; Granchi, Carlotta; Corona, Giuseppe; Cemazar, Maja; Canzonieri, Vincenzo; Tuccinardi, Tiziano; Rizzolio, Flavio
A guide to PIN1 function and mutations across cancers
2019-01-01 El Boustani, Maguie; De Stefano, Lucia; Caligiuri, Isabella; Mouawad, Nayla; Granchi, Carlotta; Canzonieri, Vincenzo; Tuccinardi, Tiziano; Giordano, Antonio; Rizzolio, Flavio
A new development of matrix metalloproteinase inhibitors: twin hydroxamic acids as potent inhibitors of MMPs
2005-01-01 Rossello, Armando; Nuti, Elisa; CATALANI M., P; Carelli, P; Orlandini, Elisabetta; Rapposelli, Simona; Tuccinardi, Tiziano; ATKINSON S., J; Murphy, G; Balsamo, A.
A patent review of Monoacylglycerol Lipase (MAGL) inhibitors (2013-2017)
2017-01-01 Granchi, Carlotta; Caligiuri, Isabella; Minutolo, Filippo; Rizzolio, Flavio; Tuccinardi, Tiziano
A theoretical study to investigate D2DAR/D4DAR selectivity: Receptor modeling and molecular docking of dopaminergic ligands
2006-01-01 Ortore, GABRIELLA MARIA PIA; Tuccinardi, Tiziano; Bertini, Simone; Martinelli, Adriano
A Virtual Screening Study for Lactate Dehydrogenase 5 Inhibitors by using a Pharmacophore-Based Approach
2016-01-01 Tuccinardi, Tiziano; Poli, Giulio; Corchia, Isacco; Granchi, Carlotta; Lapillo, Margherita; Macchia, Marco; Minutolo, Filippo; Ortore, GABRIELLA MARIA PIA; Martinelli, Adriano
A Virtual Screening Study of the 18 kDa Translocator Protein using Pharmacophore Models Combined with 3D-QSAR Studies
2009-01-01 Tuccinardi, Tiziano; Taliani, Sabrina; Bellandi, Marusca; DA SETTIMO PASSETTI, Federico; DA POZZO, Eleonora; Martini, Claudia; Martinelli, Adriano
Adenosine Receptor Ligands in Clinical Trials
2010-01-01 Rizzolio, F; La Montagna, R; Tuccinardi, Tiziano; Russo, G; Caputi, M; Giordano, A.
Adenosine Receptor Ligands: Where Are We, and Where Are We Going?
2010-01-01 Tuccinardi, Tiziano; Martinelli, Adriano
Adenosine receptor modelling. A1/A2a selectivity
2006-01-01 Tuccinardi, Tiziano; Ortore, GABRIELLA MARIA PIA; Manera, Clementina; Saccomanni, Giuseppe; Martinelli, Adriano
Aldose reductase differential inhibitors in green tea
2020-01-01 Balestri, F.; Poli, G.; Pineschi, C.; Moschini, R.; Cappiello, M.; Mura, U.; Tuccinardi, T.; Corso, A. D.
Amber force field implementation, molecular modelling study, synthesis and MMP-1/MMP-2 inhibition profile of (R)- and (S)-N-hydroxy-2-(N-isopropoxybiphenyl-4-ylsulfonamido)-3-methylbutanamides
2006-01-01 Tuccinardi, Tiziano; Martinelli, Adriano; Nuti, Elisa; Carelli, P; Balzano, Federica; UCCELLO BARRETTA, Gloria; Murphy, G; Rossello, Armando
An overview of recent developments in GPCR modelling: methods and validation
2006-01-01 Martinelli, Adriano; Tuccinardi, Tiziano
An updated patent review of monoacylglycerol lipase (MAGL) inhibitors (2018-present)
2021-01-01 Bononi, G.; Poli, G.; Rizzolio, F.; Tuccinardi, T.; Macchia, M.; Minutolo, F.; Granchi, C.
Analysis of Human Carbonic Anhydrase II: Docking Reliability and Receptor-Based 3D-QSAR Study
2007-01-01 Tuccinardi, Tiziano; Nuti, Elisa; Ortore, GABRIELLA MARIA PIA; Supuran, Ct; Rossello, Armando; Martinelli, Adriano
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
1,3-Dipolar Cycloaddition, HPLC Enantioseparation, and Docking Studies of Saccharin/Isoxazole and Saccharin/Isoxazoline Derivatives as Selective Carbonic Anhydrase IX and XII Inhibitors | 1-gen-2020 | D'Ascenzio, M.; Secci, D.; Carradori, S.; Zara, S.; Guglielmi, P.; Cirilli, R.; Pierini, M.; Poli, G.; Tuccinardi, T.; Angeli, A.; Supuran, C. T. | |
1,8-Naphthyridin-4-one derivatives as new ligands of A2A adenosine receptors. | 1-gen-2005 | Manera, Clementina; Betti, Laura; Cavallini, T.; Giannaccini, Gino; Martinelli, Adriano; Ortore, G.; Saccomanni, Giuseppe; Trincavelli, MARIA LETIZIA; Tuccinardi, Tiziano; Ferrarini, P. L. | |
3D-QSAR and virtual screening studies for the translocator protein(TSPO) | 1-gen-2008 | Tuccinardi, Tiziano; Taliani, Sabrina; Bellandi, M; DA POZZO, Eleonora; Greco, G; Novellino, E; Martinelli, Adriano; DA SETTIMO PASSETTI, Federico; Martini, Claudia | |
4-Aryliden-2-methyloxazol-5(4H)-one as a new scaffold for selective reversible MAGL inhibitors | 1-gen-2016 | Granchi, Carlotta; Rizzolio, F; Bordoni, Vittorio; Caligiuri, I; Manera, Clementina; Macchia, Marco; Minutolo, Filippo; Martinelli, Adriano; Giordano, A; Tuccinardi, Tiziano | |
5-Amino-2-phenyl[1,2,3]triazolo[1,2-a][1,2,4]benzotriazin-1-one: a Versatile Scaffold to Obtain Potent and Selective A3 Adenosine Receptor Antagonists | 1-gen-2007 | DA SETTIMO PASSETTI, Federico; Primofiore, G.; Taliani, Sabrina; Marini, ANNA MARIA; LA MOTTA, Concettina; Simorini, Francesca; Salerno, Silvia; Sergianni, V.; Tuccinardi, Tiziano; Martinelli, Adriano; Cosimelli, B.; Greco, G.; Novellino, E.; Ciampi, O.; Trincavelli, MARIA LETIZIA; Martini, Claudia | |
A carrier free delivery system of a monoacylglycerol lipase hydrophobic inhibitor | 1-gen-2022 | Adeel, Muhammad; Saorin, Gloria; Boccalon, Giacomo; Sfriso, Andrea Augusto; Parisi, Salvatore; Moro, Isabella; Palazzolo, Stefano; Caligiuri, Isabella; Granchi, Carlotta; Corona, Giuseppe; Cemazar, Maja; Canzonieri, Vincenzo; Tuccinardi, Tiziano; Rizzolio, Flavio | |
A guide to PIN1 function and mutations across cancers | 1-gen-2019 | El Boustani, Maguie; De Stefano, Lucia; Caligiuri, Isabella; Mouawad, Nayla; Granchi, Carlotta; Canzonieri, Vincenzo; Tuccinardi, Tiziano; Giordano, Antonio; Rizzolio, Flavio | |
A new development of matrix metalloproteinase inhibitors: twin hydroxamic acids as potent inhibitors of MMPs | 1-gen-2005 | Rossello, Armando; Nuti, Elisa; CATALANI M., P; Carelli, P; Orlandini, Elisabetta; Rapposelli, Simona; Tuccinardi, Tiziano; ATKINSON S., J; Murphy, G; Balsamo, A. | |
A patent review of Monoacylglycerol Lipase (MAGL) inhibitors (2013-2017) | 1-gen-2017 | Granchi, Carlotta; Caligiuri, Isabella; Minutolo, Filippo; Rizzolio, Flavio; Tuccinardi, Tiziano | |
A theoretical study to investigate D2DAR/D4DAR selectivity: Receptor modeling and molecular docking of dopaminergic ligands | 1-gen-2006 | Ortore, GABRIELLA MARIA PIA; Tuccinardi, Tiziano; Bertini, Simone; Martinelli, Adriano | |
A Virtual Screening Study for Lactate Dehydrogenase 5 Inhibitors by using a Pharmacophore-Based Approach | 1-gen-2016 | Tuccinardi, Tiziano; Poli, Giulio; Corchia, Isacco; Granchi, Carlotta; Lapillo, Margherita; Macchia, Marco; Minutolo, Filippo; Ortore, GABRIELLA MARIA PIA; Martinelli, Adriano | |
A Virtual Screening Study of the 18 kDa Translocator Protein using Pharmacophore Models Combined with 3D-QSAR Studies | 1-gen-2009 | Tuccinardi, Tiziano; Taliani, Sabrina; Bellandi, Marusca; DA SETTIMO PASSETTI, Federico; DA POZZO, Eleonora; Martini, Claudia; Martinelli, Adriano | |
Adenosine Receptor Ligands in Clinical Trials | 1-gen-2010 | Rizzolio, F; La Montagna, R; Tuccinardi, Tiziano; Russo, G; Caputi, M; Giordano, A. | |
Adenosine Receptor Ligands: Where Are We, and Where Are We Going? | 1-gen-2010 | Tuccinardi, Tiziano; Martinelli, Adriano | |
Adenosine receptor modelling. A1/A2a selectivity | 1-gen-2006 | Tuccinardi, Tiziano; Ortore, GABRIELLA MARIA PIA; Manera, Clementina; Saccomanni, Giuseppe; Martinelli, Adriano | |
Aldose reductase differential inhibitors in green tea | 1-gen-2020 | Balestri, F.; Poli, G.; Pineschi, C.; Moschini, R.; Cappiello, M.; Mura, U.; Tuccinardi, T.; Corso, A. D. | |
Amber force field implementation, molecular modelling study, synthesis and MMP-1/MMP-2 inhibition profile of (R)- and (S)-N-hydroxy-2-(N-isopropoxybiphenyl-4-ylsulfonamido)-3-methylbutanamides | 1-gen-2006 | Tuccinardi, Tiziano; Martinelli, Adriano; Nuti, Elisa; Carelli, P; Balzano, Federica; UCCELLO BARRETTA, Gloria; Murphy, G; Rossello, Armando | |
An overview of recent developments in GPCR modelling: methods and validation | 1-gen-2006 | Martinelli, Adriano; Tuccinardi, Tiziano | |
An updated patent review of monoacylglycerol lipase (MAGL) inhibitors (2018-present) | 1-gen-2021 | Bononi, G.; Poli, G.; Rizzolio, F.; Tuccinardi, T.; Macchia, M.; Minutolo, F.; Granchi, C. | |
Analysis of Human Carbonic Anhydrase II: Docking Reliability and Receptor-Based 3D-QSAR Study | 1-gen-2007 | Tuccinardi, Tiziano; Nuti, Elisa; Ortore, GABRIELLA MARIA PIA; Supuran, Ct; Rossello, Armando; Martinelli, Adriano |