ORTORE, GABRIELLA MARIA PIA Statistiche

ORTORE, GABRIELLA MARIA PIA  

DIPARTIMENTO DI FARMACIA  

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Risultati 1 - 20 di 77 (tempo di esecuzione: 0.026 secondi).
Titolo Data di pubblicazione Autore(i) File
New Insights into Bitopic Orthosteric/Allosteric Ligands of Cannabinoid Receptor Type 2 1-gen-2023 Ferrisi, Rebecca; Polini, Beatrice; Ricardi, Caterina; Gado, Francesca; Mohamed, Kawthar A; Baron, Giovanna; Faiella, Salvatore; Poli, Giulio; Rapposelli, Simona; Saccomanni, Giuseppe; Aldini, Giancarlo; Chiellini, Grazia; Laprairie, Robert B; Manera, Clementina; Ortore, Gabriella
New Insights into Bitopic Orthosteric/Allosteric Ligands of Cannabinoid Receptor Type 2 1-gen-2023 Ferrisi, Rebecca; Polini, Beatrice; Ricardi, Caterina; Gado, Francesca; Mohamed, Kawthar A; Baron, Giovanna; Faiella, Salvatore; Poli, Giulio; Rapposelli, Simona; Saccomanni, Giuseppe; Aldini, Giancarlo; Chiellini, Grazia; Laprairie, Robert B; Manera, Clementina; Ortore, Gabriella
Thyroxine metabolite-derived 3-iodothyronamine (T1AM) and synthetic analogs as efficient suppressors of transthyretin amyloidosis 1-gen-2023 Kim, Bokyung; Ho Ko, Young; Si, Jinbeom; Na, Jongbum; Ortore, Gabriella; Chiellini, Grazia; Hae Kim, Jin
CB1 receptor binding sites for NAM and PAM: A first approach for studying, new n‑butyl‑diphenylcarboxamides as allosteric modulators 1-gen-2022 Gado, F.; Ceni, C.; Ferrisi, R.; Sbrana, G.; Stevenson, L. A.; Macchia, M.; Pertwee, R. G.; Bertini, S.; Manera, C.; Ortore, G.
Design, synthesis and biological evaluation of novel orthosteric-allosteric ligands of the cannabinoid receptor type 2 (CB2R) 1-gen-2022 Ferrisi, Rebecca; Gado, Francesca; Polini, Beatrice; Ricardi, Caterina; Mohamed, Kawthar A.; Stevenson, Lesley A.; Ortore, GABRIELLA MARIA PIA; Rapposelli, Simona; Saccomanni, Giuseppe; Pertwee, Roger G.; Laprairie, Robert B.; Manera, Clementina; Chiellini, Grazia
Design, Synthesis, and Biological Activity of New CB2 Receptor Ligands: from Orthosteric and Allosteric Modulators to Dualsteric/Bitopic Ligands 1-gen-2022 Gado, Francesca; Ferrisi, Rebecca; Polini, Beatrice; Mohamed, Kawthar A.; Ricardi, Caterina; Lucarini, Elena; Carpi, Sara; Domenichini, Federica; Stevenson, Lesley A.; Rapposelli, Simona; Saccomanni, Giuseppe; Nieri, Paola; Ortore, GABRIELLA MARIA PIA; Pertwee, Roger G.; Ghelardini, Carla; Di Cesare Mannelli, Lorenzo; Chiellini, Grazia; Laprairie, Robert B.; Manera, Clementina
From Anti-infective Agents to Cancer Therapy: a Drug Repositioning Study Revealed a New Use for Nitrofuran Derivatives 1-gen-2022 Ortore, Gabriella; Poli, Giulio; Martinelli, Adriano; Tuccinardi, Tiziano; Rizzolio, Flavio; Caligiuri, Isabella
Identification of Human Dihydroorotate Dehydrogenase Inhibitor by a Pharmacophore-Based Virtual Screening Study 1-gen-2022 Galati, Salvatore; Sainas, Stefano; Giorgis, Marta; Boschi, Donatella; Lolli, Marco L; Ortore, Gabriella; Poli, Giulio; Tuccinardi, Tiziano
Machine Learning-Based Virtual Screening for the Identification of Cdk5 Inhibitors 1-gen-2022 Di Stefano, Miriana; Galati, Salvatore; Ortore, Gabriella; Caligiuri, Isabella; Rizzolio, Flavio; Ceni, Costanza; Bertini, Simone; Bononi, Giulia; Granchi, Carlotta; Macchia, Marco; Poli, Giulio; Tuccinardi, Tiziano
Reversible Monoacylglycerol Lipase Inhibitors: Discovery of a New Class of Benzylpiperidine Derivatives 1-gen-2022 Bononi, Giulia; Di Stefano, Miriana; Poli, Giulio; Ortore, Gabriella; Meier, Philip; Masetto, Francesca; Caligiuri, Isabella; Rizzolio, Flavio; Macchia, Marco; Chicca, Andrea; Avan, Amir; Giovannetti, Elisa; Vagaggini, Chiara; Brai, Annalaura; Dreassi, Elena; Valoti, Massimo; Minutolo, Filippo; Granchi, Carlotta; Gertsch, Jürg; Tuccinardi, Tiziano
Synthesis and Evaluation of Monoaryl Derivatives as Transthyretin Fibril Formation Inhibitors 1-gen-2022 Ciccone, Lidia; Nencetti, Susanna; Camodeca, Caterina; Ortore, Gabriella; Cuffaro, Doretta; Socci, Simone; Orlandini, Elisabetta
Virtual screening and crystallographic studies reveal an unexpected γ-lactone derivative active against MptpB as a potential antitubercular agent 1-gen-2022 Cazzaniga, G.; Mori, M.; Meneghetti, F.; Chiarelli, L. R.; Stelitano, G.; Caligiuri, I.; Rizzolio, F.; Ciceri, S.; Poli, G.; Staver, D.; Ortore, G.; Tuccinardi, T.; Villa, S.
Diphenyl-methane based thyromimetic inhibitors for transthyretin amyloidosis 1-gen-2021 Kim, B.; Ko, Y. H.; Runfola, M.; Rapposelli, S.; Ortore, G.; Chiellini, G.; Kim, J. H.
Focus on Human Monoamine Transporter Selectivity. New Human DAT and NET Models, Experimental Validation, and SERT Affinity Exploration 1-gen-2020 Ortore, G.; Orlandini, E.; Betti, L.; Giannaccini, G.; Mazzoni, M. R.; Camodeca, C.; Nencetti, S.
Identification of histone deacetylase inhibitors with (arylidene)aminoxy scaffold active in uveal melanoma cell lines 1-gen-2020 Nencetti, S.; Cuffaro, D.; Nuti, E.; Ciccone, L.; Rossello, A.; Fabbi, M.; Ballante, F.; Ortore, G.; Carbotti, G.; Campelli, F.; Banti, I.; Gangemi, R.; Marshall, G. R.; Orlandini, E.
Discovery of Novel Adenosine Receptor Antagonists through a Combined Structure- and Ligand-Based Approach Followed by Molecular Dynamics Investigation of Ligand Binding Mode 1-gen-2018 Lagarias, Panagiotis; Vrontaki, Eleni; Lambrinidis, George; Stamatis, Dimitrios; Convertino, Marino; Ortore, Gabriella; Mavromoustakos, Thomas; Klotz, Karl-Norbert; Kolocouris, Antonios
Identification of Transthyretin Fibril Formation Inhibitors Using Structure-Based Virtual Screening 1-gen-2017 Ortore, GABRIELLA MARIA PIA; Martinelli, Adriano
A STRUCTURE-BASED VIRTUAL SCREENING TO IDENTIFY NEW SCAFFOLDS FOR TRANSTHYRETIN FIBRIL FORMATION INHIBITORS 1-gen-2016 Ortore, G.; Martinelli, A.
A Virtual Screening Study for Lactate Dehydrogenase 5 Inhibitors by using a Pharmacophore-Based Approach 1-gen-2016 Tuccinardi, Tiziano; Poli, Giulio; Corchia, Isacco; Granchi, Carlotta; Lapillo, Margherita; Macchia, Marco; Minutolo, Filippo; Ortore, GABRIELLA MARIA PIA; Martinelli, Adriano
Exploring the binding of quercetin-3-O-metabolites with transthyretin 1-gen-2016 Ortore, GABRIELLA MARIA PIA; Ciccone, Lidia; Orlandini, Elisabetta; Stura, E.; Braca, Alessandra; Rossello, Armando; Nencetti, Susanna