Sfoglia per Autore
4-Aryliden-2-methyloxazol-5(4H)-one as a new scaffold for selective reversible MAGL inhibitors
2016-01-01 Granchi, Carlotta; Rizzolio, F; Bordoni, Vittorio; Caligiuri, I; Manera, Clementina; Macchia, Marco; Minutolo, Filippo; Martinelli, Adriano; Giordano, A; Tuccinardi, Tiziano
Anticancer agents interacting with membrane glucose transporters
2016-01-01 Granchi, Carlotta; Fortunato, Serena; Minutolo, Filippo
A Virtual Screening Study for Lactate Dehydrogenase 5 Inhibitors by using a Pharmacophore-Based Approach
2016-01-01 Tuccinardi, Tiziano; Poli, Giulio; Corchia, Isacco; Granchi, Carlotta; Lapillo, Margherita; Macchia, Marco; Minutolo, Filippo; Ortore, GABRIELLA MARIA PIA; Martinelli, Adriano
Natural compounds as inhibitors of lactate dehydrogenase
2017-01-01 Braca, Alessandra; DE LEO, Marinella; Granchi, Carlotta; Tuccinardi, Tiziano; Minutolo, Filippo; De Tommasi, Nunziatina
Reactive Oxygen Species Synergize to Potently and Selectively Induce Cancer Cell Death
2017-01-01 Lee, Hyang Yeon; Parkinson, Elizabeth I; Granchi, Carlotta; Paterni, Ilaria; Panigrahy, Dipak; Seth, Pankaj; Minutolo, Filippo; Hergenrother, Paul J.
Phospho-Akt overexpression is prognostic and can be used to tailor the synergistic interaction of Akt inhibitors with gemcitabine in pancreatic cancer
2017-01-01 Massihnia, Daniela; Avan, Amir; Funel, Niccola; Maftouh, Mina; Van Krieken, Anne; Granchi, Carlotta; Raktoe, Rajiv; Boggi, Ugo; Aicher, Babette; Minutolo, Filippo; Russo, Antonio; Leon, Leticia G.; Peters, Godefridus J.; Giovannetti, Elisa
Inhibitors of lactate dehydrogenase (hLDH5) from Polygala flavescens subsp. flavescens
2017-01-01 Braca, Alessandra; DE LEO, Marinella; Peruzzi, Lorenzo; Granchi, Carlotta; Tuccinardi, Tiziano; Minutolo, Filippo; De Tommasi, N.
Constituents of Polygala flavescens ssp. flavescens and their activity as inhibitors of human lactate dehydrogenase
2017-01-01 DE LEO, Marinella; Peruzzi, Lorenzo; Granchi, Carlotta; Tuccinardi, Tiziano; Minutolo, Filippo; De Tommasi, N.; Braca, Alessandra
Glucose transporters: production, crystallization and inhibition
2017-01-01 Raminta, Venskutonytė; Jesper S., Hansen; Peter Aasted, Paulsen; Fortunato, Serena; Granchi, Carlotta; Minutolo, Filippo; Bjørn Panyella, Pedersen; Karin Lindkvist, Petersson
A patent review of Monoacylglycerol Lipase (MAGL) inhibitors (2013-2017)
2017-01-01 Granchi, Carlotta; Caligiuri, Isabella; Minutolo, Filippo; Rizzolio, Flavio; Tuccinardi, Tiziano
Three-dimensional analysis of the interactions between hLDH5 and its inhibitors
2017-01-01 Poli, Giulio; Granchi, Carlotta; Aissaoui, Mohamed; Minutolo, Filippo; Tuccinardi, Tiziano
Development of terphenyl-2-methyloxazol-5(4H)-one derivatives as selective reversible MAGL inhibitors
2017-01-01 Granchi, Carlotta; Caligiuri, Isabella; Bertelli, Eleonora; Poli, Giulio; Rizzolio, Flavio; Macchia, Marco; Martinelli, Adriano; Minutolo, Filippo; Tuccinardi, Tiziano
Characterization of the Saffron Derivative Crocetin as an Inhibitor of Human Lactate Dehydrogenase 5 in the Antiglycolytic Approach against Cancer
2017-01-01 Granchi, Carlotta; Fortunato, Serena; Meini, Serena; Rizzolio, Flavio; Caligiuri, Isabella; Tuccinardi, Tiziano; Lee, Hyang Yeon; Hergenrother, Paul J; Minutolo, Filippo
Risks and Benefits Related to Alimentary Exposure to Xenoestrogens
2017-01-01 Paterni, Ilaria; Granchi, Carlotta; Minutolo, Filippo
Clerodanes from Salvia pseudorosmarinus and their activity as inhibitors of monoacylglycerol lipase (MAGL)
2018-01-01 Guillen Huallpa, C.; Iannuzzi, A. M.; De Leo, M.; De Tommasi, N.; Granchi, C.; Braca, A.
GLUT1 and LOX inhibitors as perspective anticancer agents tackling glucose avidity and ECM remodeling in tumors
2018-01-01 Granchi, C.; Bononi, G.; Fortunato, S.; Tuccinardi, T.; Funel, N.; Firuzi, O.; Peters, G. J.; Giovannetti, E.; Minutolo, F.
Phenylethanoid glycosides from Cistanche phelypaea acting as monoacylglycerol lipase inhibitors
2018-01-01 De Leo, M.; Beladjila, K. A.; Berrehal, D.; De Tommasi, N.; Granchi, C.; Bononi, G.; Braca, A.
Discovery and optimization of benzoylpiperidine derivatives as new reversible, potent and selective MAGL inhibitors
2018-01-01 Granchi, Carlotta; Bononi, Giulia; Rizzolio, Flavio; Chicca, Andrea; Tuccinardi, Tiziano; Minutolo, Filippo
Salicylketoximes as inhibitors of Glucose Transporters
2018-01-01 Fortunato, Serena; Granchi, Carlotta; Venskutonyté, Raminta; Hansen, Jesper S.; Lindkvist-Petersson, Karin; Minutolo, Filippo
Nuovi attivatori dell’enzima SIRT1 per il trattamento delle patologie cardiovascolari e cardiometaboliche
2018-01-01 Calderone, Vincenzo; Minutolo, Filippo; Tuccinardi, Tiziano; Testai, Lara; Granchi, Carlotta; Martelli, Alma; Citi, Valentina; DE LORENZO GARDINAL, Virginia; Lenzi, Giulia; Leo, Francesca; Malloggi, Giulia.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
4-Aryliden-2-methyloxazol-5(4H)-one as a new scaffold for selective reversible MAGL inhibitors | 1-gen-2016 | Granchi, Carlotta; Rizzolio, F; Bordoni, Vittorio; Caligiuri, I; Manera, Clementina; Macchia, Marco; Minutolo, Filippo; Martinelli, Adriano; Giordano, A; Tuccinardi, Tiziano | |
Anticancer agents interacting with membrane glucose transporters | 1-gen-2016 | Granchi, Carlotta; Fortunato, Serena; Minutolo, Filippo | |
A Virtual Screening Study for Lactate Dehydrogenase 5 Inhibitors by using a Pharmacophore-Based Approach | 1-gen-2016 | Tuccinardi, Tiziano; Poli, Giulio; Corchia, Isacco; Granchi, Carlotta; Lapillo, Margherita; Macchia, Marco; Minutolo, Filippo; Ortore, GABRIELLA MARIA PIA; Martinelli, Adriano | |
Natural compounds as inhibitors of lactate dehydrogenase | 1-gen-2017 | Braca, Alessandra; DE LEO, Marinella; Granchi, Carlotta; Tuccinardi, Tiziano; Minutolo, Filippo; De Tommasi, Nunziatina | |
Reactive Oxygen Species Synergize to Potently and Selectively Induce Cancer Cell Death | 1-gen-2017 | Lee, Hyang Yeon; Parkinson, Elizabeth I; Granchi, Carlotta; Paterni, Ilaria; Panigrahy, Dipak; Seth, Pankaj; Minutolo, Filippo; Hergenrother, Paul J. | |
Phospho-Akt overexpression is prognostic and can be used to tailor the synergistic interaction of Akt inhibitors with gemcitabine in pancreatic cancer | 1-gen-2017 | Massihnia, Daniela; Avan, Amir; Funel, Niccola; Maftouh, Mina; Van Krieken, Anne; Granchi, Carlotta; Raktoe, Rajiv; Boggi, Ugo; Aicher, Babette; Minutolo, Filippo; Russo, Antonio; Leon, Leticia G.; Peters, Godefridus J.; Giovannetti, Elisa | |
Inhibitors of lactate dehydrogenase (hLDH5) from Polygala flavescens subsp. flavescens | 1-gen-2017 | Braca, Alessandra; DE LEO, Marinella; Peruzzi, Lorenzo; Granchi, Carlotta; Tuccinardi, Tiziano; Minutolo, Filippo; De Tommasi, N. | |
Constituents of Polygala flavescens ssp. flavescens and their activity as inhibitors of human lactate dehydrogenase | 1-gen-2017 | DE LEO, Marinella; Peruzzi, Lorenzo; Granchi, Carlotta; Tuccinardi, Tiziano; Minutolo, Filippo; De Tommasi, N.; Braca, Alessandra | |
Glucose transporters: production, crystallization and inhibition | 1-gen-2017 | Raminta, Venskutonytė; Jesper S., Hansen; Peter Aasted, Paulsen; Fortunato, Serena; Granchi, Carlotta; Minutolo, Filippo; Bjørn Panyella, Pedersen; Karin Lindkvist, Petersson | |
A patent review of Monoacylglycerol Lipase (MAGL) inhibitors (2013-2017) | 1-gen-2017 | Granchi, Carlotta; Caligiuri, Isabella; Minutolo, Filippo; Rizzolio, Flavio; Tuccinardi, Tiziano | |
Three-dimensional analysis of the interactions between hLDH5 and its inhibitors | 1-gen-2017 | Poli, Giulio; Granchi, Carlotta; Aissaoui, Mohamed; Minutolo, Filippo; Tuccinardi, Tiziano | |
Development of terphenyl-2-methyloxazol-5(4H)-one derivatives as selective reversible MAGL inhibitors | 1-gen-2017 | Granchi, Carlotta; Caligiuri, Isabella; Bertelli, Eleonora; Poli, Giulio; Rizzolio, Flavio; Macchia, Marco; Martinelli, Adriano; Minutolo, Filippo; Tuccinardi, Tiziano | |
Characterization of the Saffron Derivative Crocetin as an Inhibitor of Human Lactate Dehydrogenase 5 in the Antiglycolytic Approach against Cancer | 1-gen-2017 | Granchi, Carlotta; Fortunato, Serena; Meini, Serena; Rizzolio, Flavio; Caligiuri, Isabella; Tuccinardi, Tiziano; Lee, Hyang Yeon; Hergenrother, Paul J; Minutolo, Filippo | |
Risks and Benefits Related to Alimentary Exposure to Xenoestrogens | 1-gen-2017 | Paterni, Ilaria; Granchi, Carlotta; Minutolo, Filippo | |
Clerodanes from Salvia pseudorosmarinus and their activity as inhibitors of monoacylglycerol lipase (MAGL) | 1-gen-2018 | Guillen Huallpa, C.; Iannuzzi, A. M.; De Leo, M.; De Tommasi, N.; Granchi, C.; Braca, A. | |
GLUT1 and LOX inhibitors as perspective anticancer agents tackling glucose avidity and ECM remodeling in tumors | 1-gen-2018 | Granchi, C.; Bononi, G.; Fortunato, S.; Tuccinardi, T.; Funel, N.; Firuzi, O.; Peters, G. J.; Giovannetti, E.; Minutolo, F. | |
Phenylethanoid glycosides from Cistanche phelypaea acting as monoacylglycerol lipase inhibitors | 1-gen-2018 | De Leo, M.; Beladjila, K. A.; Berrehal, D.; De Tommasi, N.; Granchi, C.; Bononi, G.; Braca, A. | |
Discovery and optimization of benzoylpiperidine derivatives as new reversible, potent and selective MAGL inhibitors | 1-gen-2018 | Granchi, Carlotta; Bononi, Giulia; Rizzolio, Flavio; Chicca, Andrea; Tuccinardi, Tiziano; Minutolo, Filippo | |
Salicylketoximes as inhibitors of Glucose Transporters | 1-gen-2018 | Fortunato, Serena; Granchi, Carlotta; Venskutonyté, Raminta; Hansen, Jesper S.; Lindkvist-Petersson, Karin; Minutolo, Filippo | |
Nuovi attivatori dell’enzima SIRT1 per il trattamento delle patologie cardiovascolari e cardiometaboliche | 1-gen-2018 | Calderone, Vincenzo; Minutolo, Filippo; Tuccinardi, Tiziano; Testai, Lara; Granchi, Carlotta; Martelli, Alma; Citi, Valentina; DE LORENZO GARDINAL, Virginia; Lenzi, Giulia; Leo, Francesca; Malloggi, Giulia. |
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