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Titolo Data di pubblicazione Autore(i) File
Design of Selective Collagenase 3 (MMP-13) Inhibitors as Potential Therapeutic Agents in Rheumatoid Arthritis 1-gen-2008 Nuti, Elisa; Casalini, F; Avramova, S. I.; Orlandini, Elisabetta; Nencetti, Susanna; Tuccinardi, Tiziano; Nagase, H; Visse, R; Murphy, G; Rossello, Armando
D3 dopamine receptor subtype: which binding modes for such different ligands? 1-gen-2008 Martinelli, Adriano; Orlandini, Elisabetta; Tuccinardi, Tiziano; Ortore, GABRIELLA MARIA PIA
Design, synthesis, and biological evaluation of 1,8-naphthyridin-2(1H)-on-3-carboxamide, quinolin-2(1H)-on-3-carboxamide and 2-oxo-1,2-dihydropyridine-3-carboxamide derivatives as CB2 selective ligands 1-gen-2008 Manera, Clementina; M., Allarà; V., Benetti; M., Conti; A., Fazzini; A., Ligresti; V., Lucchesi; Saccomanni, Giuseppe; F., Taddei; Tuccinardi, Tiziano; V., DI MARZO; Martinelli, Adriano; P. L., Ferrarini
Design, synthesis, binding, and molecular modeling studies of new potent ligands of cannabinoid receptors 1-gen-2008 A., Brizzi; F., Corelli; M. G., Cascio; Martinelli, Adriano; Tuccinardi, Tiziano; T., Bisogno; V., DI MARZO
Synthesis and antitumor evaluation of 1,8-naphthyridine-2-(1H)-on-3carboxamide derivatives as CB2 selective agonists 1-gen-2008 M., Conti; Adinolfi, Barbara; M., Allarà; V., Benetti; V., DI MARZO; Manera, Clementina; Saccomanni, Giuseppe; Tuccinardi, Tiziano; P. L., Ferrarini
D3 dopamine receptor subtype: which binding modes for such different ligands?, 1-gen-2008 Martinelli, Adriano; Orlandini, Elisabetta; Tuccinardi, Tiziano; Ortore, GABRIELLA MARIA PIA
Arylsulfonamide derivatives as metalloproteases inhibitors and their preparation, pharmaceutical compositions and use in the treatment of degenerative disorders 1-gen-2008 Rossello, Armando; Nuti, Elisa; Orlandini, Elisabetta; Balsamo, Aldo; Tuccinardi, Tiziano
Synthesis and biological evaluation of folic acid derivatives as histone deacetylase inhibitors 1-gen-2008 M. A., Santos; E. A., Enyedy; M., Carrasco; N. I., Krupenko; S. A., Krupenko; Nuti, Elisa; Tuccinardi, Tiziano; Rossello, Armando; Martinelli, Adriano
Synthesis, Modeling, and RET Protein Kinase Inhibitory Activity of 3-and 4-Substituted beta-Carbolin-1-ones 1-gen-2008 Cincinelli, Raffaella; Cassinelli, Giuliana; Dallavalle, Sabrina; Lanzi, Cinzia; Merlini, Lucio; Botta, Maurizio; Tuccinardi, Tiziano; Martinelli, Adriano; Penco, Sergio; Zunino, Franco
Synthesis and AT1 affinity evaluation of benzamidophenyl analogs of known AT1 receptor ligands with similar aromatic skeleton 1-gen-2008 Rapposelli, Simona; Cuboni, S; Digiacomo, Maria; Lapucci, Annalina; Trincavelli, MARIA LETIZIA; Tuccinardi, Tiziano; Balsamo, A.
Derivatives of 4-Amino-6-hydroxy-2-mercaptopyrimidine as Novel, Potent, and Selective A3 Adenosine Receptor Antagonists 1-gen-2008 B., Cosimelli; G., Greco; M., Ehlardo; E., Novellino; DA SETTIMO PASSETTI, Federico; Taliani, Sabrina; LA MOTTA, Concettina; M., Bellandi; Tuccinardi, Tiziano; Martinelli, Adriano; O., Ciampi; Trincavelli, MARIA LETIZIA; Martini, Claudia
Development of a receptor-based 3D-QSAR study for the analysis of MMP2, MMP3, and MMP9 inhibitors 1-gen-2008 Tuccinardi, Tiziano; Nuti, Elisa; Ortore, GABRIELLA MARIA PIA; Rossello, Armando; Avramova, Si; Martinelli, Adriano
Novel aminopteroil-sulfonamide derivatives as inhibitors of dihydrofolate reductase and carbonic anhydrase, with potential anti tumor activity 1-gen-2008 S. M., Marques; E. A., Enyedy; Tuccinardi, Tiziano; Martinelli, Adriano; C. T., Supuran; N. I., Krupenko; S. A., Krupenko; M. A., Santos
Dual Inhibitors of Matrix Metalloproteinases and Carbonic Anhydrases: Iminodiacetyl-Based Hydroxamate-Benzenesulfonamide Conjugates 1-gen-2008 Marques, Sergio; Nuti, Elisa; Rossello, Armando; SUPURAN CLAUDIU, T; Tuccinardi, Tiziano; Martinelli, Adriano; SANTOS M., Amelia
Molecular Modeling of adenosine receptors: New results and trends 1-gen-2008 Martinelli, Adriano; Tuccinardi, Tiziano
Indoles and Related Compounds as Cannabinoid Ligands, 1-gen-2008 Manera, Clementina; Tuccinardi, Tiziano; Martinelli, Adriano; MINI REVIEWS IN MEDICINAL, Chemistry
QSAR of Carbonic Anhydrase Inhibitors and Their Impact on Drug Design 1-gen-2009 Martinelli, Adriano; Tuccinardi, Tiziano
Computational Studies of Epidermal Growth Factor Receptor for Docking Reliability, Three-Dimensional Quantitative Structure-Activity Relationship Analysis, and Virtual Screening Studies 1-gen-2009 LA MOTTA, Concettina; Sartini, Stefania; Tuccinardi, Tiziano; Nerini, Erika; DA SETTIMO PASSETTI, Federico; Martinelli, Adriano
New Resorcinol-Anandamide "Hybrids" as Potent Cannabinoid Receptor Ligands Endowed with Antinociceptive Activity in Vivo 1-gen-2009 Brizzi, Antonella; Brizzi, Vittorio; CASCIO MARIA, Grazia; Corelli, Federico; Guida, Francesca; Ligresti, Alessia; Maione, Sabatino; Martinelli, Adriano; Pasquini, Serena; Tuccinardi, Tiziano; DI MARZO, Vincenzo
Structural Evolutions of Salicylaldoximes as Selective Agonists for Estrogen Receptor Beta 1-gen-2009 Minutolo, Filippo; Bertini, Simone; Granchi, Carlotta; Marchitiello, T; Prota, G; Rapposelli, Simona; Tuccinardi, Tiziano; Martinelli, Adriano; GUNTHER J., R; CARLSON K., E; KATZENELLENBOGEN J., A; Macchia, Marco
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