Sfoglia per Autore
Design, Synthesis and biological evaluation of new 1,8-naphthyridin-4(1h)-on-3-carboxamide and quinolin-4(1h)-on-3-carboxamide derivatives as CB2 selective agonists
2006-01-01 M. P., Castelli; Manera, Clementina; V., Benetti; Martinelli, Adriano; A. P., Piras; Saccomanni, Giuseppe; Tuccinardi, Tiziano; A., Vannacci
MMPs: “Receptor Based” 3D QSAR
2006-01-01 S. L., Baroncini; Tuccinardi, Tiziano; Martinelli, Adriano
Design, Synthesis, and Biological Evaluation of New 1,8-Naphthyridin-4(1H)-one-3-carboxamide and Quinolin-4(1H)-one-3-carboxamide Derivatives as CB2 Selective Agonists
2006-01-01 Manera, Clementina; Benetti, V; Castelli, Mp; Cavallini, C; Lazzarotti, S; Pibiri, F; Saccomanni, Giuseppe; Tuccinardi, Tiziano; Vannacci, A; Martinelli, Adriano; Ferrarini, Pl
Adenosine receptor modelling. A1/A2a selectivity
2006-01-01 Tuccinardi, Tiziano; Ortore, GABRIELLA MARIA PIA; Manera, Clementina; Saccomanni, Giuseppe; Martinelli, Adriano
Iminodiacetyl-monohydroxamate derivatives as potent and selective MMP inhibitors
2006-01-01 Marques, Sm; Chaves, S; Rossello, Armando; Tuccinardi, Tiziano; Santos, Ma
Salicylaldoximes and anthranylaldoximes as alternatives to phenol-based estrogen receptor ligands
2006-01-01 Minutolo, Filippo; Bertini, Simone; Martinelli, Adriano; Ortore, GABRIELLA MARIA PIA; Placanica, Giorgio; G., Prota; Rapposelli, Simona; Tuccinardi, Tiziano; S., Sheng; K. E., Carlson; B. S., Katzenellenbogen; J. A., Katzenellenbogen; Macchia, Marco
Design, synthesis and molecular modeling study of iminodiacetyl monohydroxamic acid derivatives as MMP inhibitors
2006-01-01 Santos, M. A.; Marques, S. M.; Tuccinardi, Tiziano; Carelli, P; Panelli, L; Rossello, Armando
An overview of recent developments in GPCR modelling: methods and validation
2006-01-01 Martinelli, Adriano; Tuccinardi, Tiziano
Pharmacophore based receptor modeling: the case of adenosine A3 receptor antagonists. An approach to the optimization of protein models
2006-01-01 Tafi, A; Bernardini, C; Botta, M; Corelli, F; Andreini, M; Martinelli, Adriano; Ortore, GABRIELLA MARIA PIA; Baraldi, Pg; Fruttarolo, F; Borea, Pa; Tuccinardi, Tiziano
Synthesis of stable analogues of geranylgeranyl diphosphate possessing a (Z,E,E)-geranylgeranyl side chain, docking analysis, and biological assays for prenyl protein transferase inhibition
2006-01-01 Minutolo, Filippo; Bertini, Simone; Betti, Laura; Danesi, Romano; Gervasi, G; Giannaccini, Gino; Martinelli, Adriano; Papini, Am; Peroni, E; Placanica, Giorgio; Rapposelli, Simona; Tuccinardi, Tiziano; Macchia, Marco
Cannabinoid CB2/CB1 Selectivity. Receptor Modeling and Automated Docking Analysis
2006-01-01 Tuccinardi, Tiziano; Ferrarini, PIER LUIGI; Manera, Clementina; Ortore, GABRIELLA MARIA PIA; Saccomanni, Giuseppe; Martinelli, Adriano
A theoretical study to investigate D2DAR/D4DAR selectivity: Receptor modeling and molecular docking of dopaminergic ligands
2006-01-01 Ortore, GABRIELLA MARIA PIA; Tuccinardi, Tiziano; Bertini, Simone; Martinelli, Adriano
Proposal of a new binding orientation for non-peptide AT1 antagonists: Homology modeling, docking and three-dimensional quantitative structure-activity relationship analysis
2006-01-01 Tuccinardi, Tiziano; Calderone, Vincenzo; Rapposelli, Simona; Martinelli, Adriano
Salicylaldoximes and anthranylaldoximes as alternatives to phenol-based estrogen receptor ligands
2006-01-01 Minutolo, Filippo; Bertini, Simone; Martinelli, Adriano; Ortore, GABRIELLA MARIA PIA; Placanica, Giorgio; Prota, G; Rapposelli, Simona; Tuccinardi, Tiziano; Sheng, S; Carlson, K. E.; Katzenellenbogen, B. S.; Katzenellenbogen, J. A.; Macchia, Marco
Amber force field implementation, molecular modelling study, synthesis and MMP-1/MMP-2 inhibition profile of (R)- and (S)-N-hydroxy-2-(N-isopropoxybiphenyl-4-ylsulfonamido)-3-methylbutanamides
2006-01-01 Tuccinardi, Tiziano; Martinelli, Adriano; Nuti, Elisa; Carelli, P; Balzano, Federica; UCCELLO BARRETTA, Gloria; Murphy, G; Rossello, Armando
5-Amino-2-phenyl[1,2,3]triazolo[1,2-a][1,2,4]benzotriazin-1-one: a Versatile Scaffold to Obtain Potent and Selective A3 Adenosine Receptor Antagonists
2007-01-01 DA SETTIMO PASSETTI, Federico; Primofiore, G.; Taliani, Sabrina; Marini, ANNA MARIA; LA MOTTA, Concettina; Simorini, Francesca; Salerno, Silvia; Sergianni, V.; Tuccinardi, Tiziano; Martinelli, Adriano; Cosimelli, B.; Greco, G.; Novellino, E.; Ciampi, O.; Trincavelli, MARIA LETIZIA; Martini, Claudia
Synthesis and biological evaluation of 1,8-naphthyridine and quinoline derivatives as CB2 selective agonists
2007-01-01 Manera, Clementina; V., Benetti; Martinelli, Adriano; Saccomanni, Giuseppe; Tuccinardi, Tiziano; M. G., Cascio; V., DI MARZO; P. L., Ferrarini
Design of transthyretin amyloidosis inhibitors: A docking and virtual screening approach
2007-01-01 Ortore, GABRIELLA MARIA PIA; Orlandini, Elisabetta; Tuccinardi, Tiziano; E., Romagnoli; Martinelli, Adriano
Transthyretin amyloidosis: a computational approach toward the design of new inhibitors
2007-01-01 Ortore, GABRIELLA MARIA PIA; Tuccinardi, Tiziano; E., Romagnoli; Orlandini, Elisabetta; Martinelli, Adriano
MMPs selectivity: Docking and 3D-QSAR evaluation
2007-01-01 Tuccinardi, Tiziano; Ortore, GABRIELLA MARIA PIA; S. L., Baroncini; Martinelli, Adriano
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Design, Synthesis and biological evaluation of new 1,8-naphthyridin-4(1h)-on-3-carboxamide and quinolin-4(1h)-on-3-carboxamide derivatives as CB2 selective agonists | 1-gen-2006 | M. P., Castelli; Manera, Clementina; V., Benetti; Martinelli, Adriano; A. P., Piras; Saccomanni, Giuseppe; Tuccinardi, Tiziano; A., Vannacci | |
MMPs: “Receptor Based” 3D QSAR | 1-gen-2006 | S. L., Baroncini; Tuccinardi, Tiziano; Martinelli, Adriano | |
Design, Synthesis, and Biological Evaluation of New 1,8-Naphthyridin-4(1H)-one-3-carboxamide and Quinolin-4(1H)-one-3-carboxamide Derivatives as CB2 Selective Agonists | 1-gen-2006 | Manera, Clementina; Benetti, V; Castelli, Mp; Cavallini, C; Lazzarotti, S; Pibiri, F; Saccomanni, Giuseppe; Tuccinardi, Tiziano; Vannacci, A; Martinelli, Adriano; Ferrarini, Pl | |
Adenosine receptor modelling. A1/A2a selectivity | 1-gen-2006 | Tuccinardi, Tiziano; Ortore, GABRIELLA MARIA PIA; Manera, Clementina; Saccomanni, Giuseppe; Martinelli, Adriano | |
Iminodiacetyl-monohydroxamate derivatives as potent and selective MMP inhibitors | 1-gen-2006 | Marques, Sm; Chaves, S; Rossello, Armando; Tuccinardi, Tiziano; Santos, Ma | |
Salicylaldoximes and anthranylaldoximes as alternatives to phenol-based estrogen receptor ligands | 1-gen-2006 | Minutolo, Filippo; Bertini, Simone; Martinelli, Adriano; Ortore, GABRIELLA MARIA PIA; Placanica, Giorgio; G., Prota; Rapposelli, Simona; Tuccinardi, Tiziano; S., Sheng; K. E., Carlson; B. S., Katzenellenbogen; J. A., Katzenellenbogen; Macchia, Marco | |
Design, synthesis and molecular modeling study of iminodiacetyl monohydroxamic acid derivatives as MMP inhibitors | 1-gen-2006 | Santos, M. A.; Marques, S. M.; Tuccinardi, Tiziano; Carelli, P; Panelli, L; Rossello, Armando | |
An overview of recent developments in GPCR modelling: methods and validation | 1-gen-2006 | Martinelli, Adriano; Tuccinardi, Tiziano | |
Pharmacophore based receptor modeling: the case of adenosine A3 receptor antagonists. An approach to the optimization of protein models | 1-gen-2006 | Tafi, A; Bernardini, C; Botta, M; Corelli, F; Andreini, M; Martinelli, Adriano; Ortore, GABRIELLA MARIA PIA; Baraldi, Pg; Fruttarolo, F; Borea, Pa; Tuccinardi, Tiziano | |
Synthesis of stable analogues of geranylgeranyl diphosphate possessing a (Z,E,E)-geranylgeranyl side chain, docking analysis, and biological assays for prenyl protein transferase inhibition | 1-gen-2006 | Minutolo, Filippo; Bertini, Simone; Betti, Laura; Danesi, Romano; Gervasi, G; Giannaccini, Gino; Martinelli, Adriano; Papini, Am; Peroni, E; Placanica, Giorgio; Rapposelli, Simona; Tuccinardi, Tiziano; Macchia, Marco | |
Cannabinoid CB2/CB1 Selectivity. Receptor Modeling and Automated Docking Analysis | 1-gen-2006 | Tuccinardi, Tiziano; Ferrarini, PIER LUIGI; Manera, Clementina; Ortore, GABRIELLA MARIA PIA; Saccomanni, Giuseppe; Martinelli, Adriano | |
A theoretical study to investigate D2DAR/D4DAR selectivity: Receptor modeling and molecular docking of dopaminergic ligands | 1-gen-2006 | Ortore, GABRIELLA MARIA PIA; Tuccinardi, Tiziano; Bertini, Simone; Martinelli, Adriano | |
Proposal of a new binding orientation for non-peptide AT1 antagonists: Homology modeling, docking and three-dimensional quantitative structure-activity relationship analysis | 1-gen-2006 | Tuccinardi, Tiziano; Calderone, Vincenzo; Rapposelli, Simona; Martinelli, Adriano | |
Salicylaldoximes and anthranylaldoximes as alternatives to phenol-based estrogen receptor ligands | 1-gen-2006 | Minutolo, Filippo; Bertini, Simone; Martinelli, Adriano; Ortore, GABRIELLA MARIA PIA; Placanica, Giorgio; Prota, G; Rapposelli, Simona; Tuccinardi, Tiziano; Sheng, S; Carlson, K. E.; Katzenellenbogen, B. S.; Katzenellenbogen, J. A.; Macchia, Marco | |
Amber force field implementation, molecular modelling study, synthesis and MMP-1/MMP-2 inhibition profile of (R)- and (S)-N-hydroxy-2-(N-isopropoxybiphenyl-4-ylsulfonamido)-3-methylbutanamides | 1-gen-2006 | Tuccinardi, Tiziano; Martinelli, Adriano; Nuti, Elisa; Carelli, P; Balzano, Federica; UCCELLO BARRETTA, Gloria; Murphy, G; Rossello, Armando | |
5-Amino-2-phenyl[1,2,3]triazolo[1,2-a][1,2,4]benzotriazin-1-one: a Versatile Scaffold to Obtain Potent and Selective A3 Adenosine Receptor Antagonists | 1-gen-2007 | DA SETTIMO PASSETTI, Federico; Primofiore, G.; Taliani, Sabrina; Marini, ANNA MARIA; LA MOTTA, Concettina; Simorini, Francesca; Salerno, Silvia; Sergianni, V.; Tuccinardi, Tiziano; Martinelli, Adriano; Cosimelli, B.; Greco, G.; Novellino, E.; Ciampi, O.; Trincavelli, MARIA LETIZIA; Martini, Claudia | |
Synthesis and biological evaluation of 1,8-naphthyridine and quinoline derivatives as CB2 selective agonists | 1-gen-2007 | Manera, Clementina; V., Benetti; Martinelli, Adriano; Saccomanni, Giuseppe; Tuccinardi, Tiziano; M. G., Cascio; V., DI MARZO; P. L., Ferrarini | |
Design of transthyretin amyloidosis inhibitors: A docking and virtual screening approach | 1-gen-2007 | Ortore, GABRIELLA MARIA PIA; Orlandini, Elisabetta; Tuccinardi, Tiziano; E., Romagnoli; Martinelli, Adriano | |
Transthyretin amyloidosis: a computational approach toward the design of new inhibitors | 1-gen-2007 | Ortore, GABRIELLA MARIA PIA; Tuccinardi, Tiziano; E., Romagnoli; Orlandini, Elisabetta; Martinelli, Adriano | |
MMPs selectivity: Docking and 3D-QSAR evaluation | 1-gen-2007 | Tuccinardi, Tiziano; Ortore, GABRIELLA MARIA PIA; S. L., Baroncini; Martinelli, Adriano |
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