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Cell and Cell-Free Mechanistic Studies on Two Gold(III) Complexes with Proven Antitumor Properties 1-gen-2017 Nardon, Chiara; Boscutti, Giulia; Gabbiani, Chiara; Massai, Lara; Pettenuzzo, Nicolò; Fassina, Ambrogio; Messori, Luigi; Fregona, Dolores
ESI–MS studies of the reactions of novel platinum(II) complexes containing O,O′-chelated acetylacetonate and sulfur ligands with selected model proteins 1-gen-2017 Marzo, Tiziano; De Pascali, Sandra A.; Gabbiani, Chiara; Fanizzi, Francesco P.; Messori, Luigi; Pratesi, Alessandro
Gold compounds as cysteine protease inhibitors: perspectives for pharmaceutical application as antiparasitic agents 1-gen-2017 Massai, L; Messori, L; Micale, N; Schirmeister, T; Maes, L; Fregona, D; Cinellu, Ma; Gabbiani, Chiara
Ruthenium arene complexes with triphenylphosphane ligands: Cytotoxicity towards pancreatic cancer cells, interaction with model proteins, and effect of ethacrynic acid substitution 1-gen-2017 Biancalana, Lorenzo; Pratesi, Alessandro; Chiellini, Federica; Zacchini, Stefano; Funaioli, Tiziana; Gabbiani, Chiara; Marchetti, Fabio
Auranofin, Et3PAuCl, and Et3PAuI Are Highly Cytotoxic on Colorectal Cancer Cells: A Chemical and Biological Study 1-gen-2017 Marzo, Tiziano; Cirri, Damiano; Gabbiani, Chiara; Gamberi, Tania; Magherini, Francesca; Pratesi, Alessandro; Guerri, Annalisa; Biver, Tarita; Binacchi, Francesca; Stefanini, Matteo; Arcangeli, Annarosa; Messori, Luigi
Antiproliferative effects of two gold(I)-N-heterocyclic carbene complexes in A2780 human ovarian cancer cells: A comparative proteomic study 1-gen-2018 Magherini, Francesca; Fiaschi, Tania; Valocchia, Elisa; Becatti, Matteo; Pratesi, Alessandro; Marzo, Tiziano; Massai, Lara; Gabbiani, Chiara; Landini, Ida; Nobili, Stefania; Mini, Enrico; Messori, Luigi; Modesti, Alessandra; Gamberi, Tania
Chlorido and bromido oxaliplatin analogues as potential agents for CRC treatment: Solution behavior, protein binding and cytotoxicity evaluation 1-gen-2018 Marzo, Tiziano; Pratesi, Alessandro; Cirri, Damiano; Pillozzi, Serena; Petroni, Giulia; Guerri, Annalisa; Arcangeli, Annarosa; Messori, Luigi; Gabbiani, Chiara
Interaction of a Gold(I) Dicarbene Anticancer Drug with Human Telomeric DNA G-Quadruplex: Solution and Computationally Aided X-ray Diffraction Analysis 1-gen-2018 Guarra, Federica; Marzo, Tiziano; Ferraroni, Marta; Papi, Francesco; Bazzicalupi, Carla; Gratteri, Paola; Pescitelli, Gennaro; Messori, Luigi; Biver, Tarita; Gabbiani, Chiara
Synthesis, characterization and DNA interactions of [Pt3(TPymT)Cl3], the trinuclear platinum(II) complex of the TPymT ligand 1-gen-2018 Marzo, Tiziano; Cirri, Damiano; Ciofi, Lorenzo; Gabbiani, Chiara; Feis, Alessandro; Di Pasquale, Nancy; Stefanini, Matteo; Biver, Tarita; Messori, Luigi
Interaction of gold N-heterocyclic carbenes with nucleic acids 1-gen-2018 Biver, T.; Gabbiani, C.; Pescitelli, G.; Marzo, T.; Bazzicalupi, C.; Gratteri, P.; Messori, L.; Guarra, F.
Photocytotoxic Pt(iv) complexes as prospective anticancer agents 1-gen-2019 Canil, Giovanni; Braccini, Simona; Marzo, Tiziano; Marchetti, Lorella; Pratesi, Alessandro; Biver, Tarita; Funaioli, Tiziana; Chiellini, Federica; Hoeschele, James D; Gabbiani, Chiara
Interplay between Gold(I)-Ligand Bond Components and Hydrogen Bonding: A Combined Experimental/Computational Study 1-gen-2019 Marrazzini, G.; Gabbiani, C.; Ciancaleoni, G.
Cytotoxic Ag(I) and Au(I) NHC-carbenes bind DNA and show TrxR inhibition 1-gen-2020 Guarra, F.; Busto, N.; Guerri, A.; Marchetti, L.; Marzo, T.; Garcia, B.; Biver, T.; Gabbiani, C.
124I Radiolabeling of a AuIII-NHC Complex for In Vivo Biodistribution Studies 1-gen-2020 Guarra, F.; Terenzi, A.; Pirker, C.; Passannante, R.; Baier, D.; Zangrando, E.; Gomez-Vallejo, V.; Biver, T.; Gabbiani, C.; Berger, W.; Llop, J.; Salassa, L.
Mechanistic Insights Into the Anticancer Properties of the Auranofin Analog Au(PEt3)I: A Theoretical and Experimental Study 1-gen-2020 Tolbatov, I.; Cirri, D.; Marchetti, L.; Marrone, A.; Coletti, C.; Re, N.; La Mendola, D.; Messori, L.; Marzo, T.; Gabbiani, C.; Pratesi, A.
On the Different Mode of Action of Au(I)/Ag(I)-NHC Bis-Anthracenyl Complexes Towards Selected Target Biomolecules 1-gen-2020 Binacchi, F.; Guarra, F.; Cirri, D.; Marzo, T.; Pratesi, A.; Messori, L.; Gabbiani, C.; Biver, T.
Reactions of cisplatin and cis-[PtI2(NH3)2] with molecular models of relevant protein sidechains: A comparative analysis 1-gen-2020 Tolbatov, Iogann; Marzo, Tiziano; Cirri, Damiano; Gabbiani, Chiara; Coletti, Cecilia; Marrone, Alessandro; Paciotti, Roberto; Messori, Luigi; Re, Nazzareno
A focus on the biological targets for coinage metal-NHCs as potential anticancer complexes 1-gen-2021 Guarra, F.; Pratesi, A.; Gabbiani, C.; Biver, T.
Thermodynamic Evaluation of the Interactions between Anticancer Pt(II) Complexes and Model Proteins 1-gen-2021 Pelosi, Chiara; Saitta, Francesca; Zerino, Caterina; Canil, Giovanni; Biver, Tarita; Pratesi, Alessandro; Duce, Celia; Fessas, Dimitrios; Gabbiani, Chiara; Tiné, Maria Rosaria
Protein metalation by two structurally related gold(I) carbene complexes: An ESI MS study 1-gen-2021 Zoppi, C.; Massai, L.; Cirri, D.; Gabbiani, C.; Pratesi, A.; Messori, L.
Synthesis, chemical characterization, and biological evaluation of a novel auranofin derivative as an anticancer agent 1-gen-2022 Cirri, Damiano; Massai, Lara; Giacomelli, Chiara; Trincavelli, Maria Letizia; Guerri, Annalisa; Gabbiani, Chiara; Messori, Luigi; Pratesi, Alessandro
Synthesis, Characterization and Photoactivation Studies on the Novel Pt(IV)-Based [Pt(OCOCH3)3(phterpy)] Complex 1-gen-2023 Canil, Giovanni; Gurruchaga-Pereda, Juan; Braccini, Simona; Marchetti, Lorella; Funaioli, Tiziana; Marchetti, Fabio; Pratesi, Alessandro; Salassa, Luca; Gabbiani, Chiara
Highlights of New Strategies to Increase the Efficacy of Transition Metal Complexes for Cancer Treatments 1-gen-2023 Giorgi, Ester; Binacchi, Francesca; Marotta, Carlo; Cirri, Damiano; Gabbiani, Chiara; Pratesi, Alessandro
Cytotoxic auranofin analogues bearing phosphine, arsine and stibine ligands: A study on the possible role of the ligand on the biological activity 1-gen-2023 Giorgi, Ester; Mannelli, Michele; Gamberi, Tania; Durante, Maria; Gabbiani, Chiara; Cirri, Damiano; Pratesi, Alessandro
An overview of recent advancements in anticancer Pt(IV) prodrugs: New smart drug combinations, activation and delivery strategies 1-gen-2023 Marotta, Carlo; Giorgi, Ester; Binacchi, Francesca; Cirri, Damiano; Gabbiani, Chiara; Pratesi, Alessandro
Chemical Modification of Auranofin Yields a New Family of Anticancer Drug Candidates: The Gold(I) Phosphite Analogues 1-gen-2023 Cirri, Damiano; Geri, Andrea; Massai, Lara; Mannelli, Michele; Gamberi, Tania; Magherini, Francesca; Becatti, Matteo; Gabbiani, Chiara; Pratesi, Alessandro; Messori, Luigi
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