D'AGOSTINO, ILARIA Statistiche
D'AGOSTINO, ILARIA
DIPARTIMENTO DI FARMACIA
A Journey Around Boronic Acids: Sulfonyl Hydrazone-Containing Derivatives as Carbonic Anhydrase Inhibitors
2025-01-01 Anakök, Deniz A; Angeli, Andrea; D'Agostino, Ilaria; Renzi, Gioele; Massardi, Maria Luisa; Tavani, Camilla; Çete, Servet; Carradori, Simone; Ronca, Roberto; Capasso, Clemente; Carta, Fabrizio; Supuran, Claudiu T
A scaffold repositioning approach: dihydroBenzoImidazoTriazineDione (BITD) derivatives as selective ALDH1A1 inhibitors
2025-01-01 Bernardoni, Bianca Laura; D'Agostino, Ilaria; Siragusa, Sonia; Mori, Mattia; Garavaglia, Silvia; La Motta, Concettina
O-derivatization of natural tropolone and β-thujaplicin leading to effective inhibitors of human carbonic anhydrases IX and XII
2025-01-01 Melfi, Francesco; D'Agostino, Ilaria; Carradori, Simone; Carta, Fabrizio; Angeli, Andrea; Costa, Giosuè; Renzi, Gioele; Čikoš, Ana; Vullo, Daniela; Rešetar, Josip; Ferraroni, Marta; Baroni, Chiara; Mancuso, Francesca; Gitto, Rosaria; Ambrosio, Francesca Alessandra; Marchese, Emanuela; Torcasio, Roberta; Amodio, Nicola; Capasso, Clemente; Alcaro, Stefano; Supuran, Claudiu T.
Pegylation Approach Applied to Erlotinib-Carbonic Anhydrase Inhibitors Hybrids Towards Anticancer Agents
2025-01-01 Filiberti, Serena; Renzi, Gioele; Carta, Fabrizio; Fantacuzzi, Marialuigia; D'Agostino, Ilaria; Benito, German; Angeli, Andrea; Massardi, Marialuisa; Simsek, Rahime; Capasso, Clemente; Carradori, Simone; Ronca, Roberto; Supuran, Claudiu
Unprecedented carbonic anhydrase inhibition mechanism: Targeting histidine 64 side chain through a halogen bond
2025-01-01 Paciotti, Roberto; Carradori, Simone; Angeli, Andrea; D'Agostino, Ilaria; Ferraroni, Marta; Coletti, Cecilia; Supuran, Claudiu T.
β-Cyclodextrin nanosponges for the ocular delivery of therapeutic Micro-RNA in a Mouse model of retinitis Pigmentosa: A proof of concept study
2025-01-01 Piano, Ilaria; Polini, Beatrice; Corsi, Francesca; Carpi, Sara; Petrarolo, Giovanni; Quattrini, Luca; D'Agostino, Ilaria; Gamberini, Maria Cristina; Baraldi, Cecilia; Chiellini, Grazia; Nieri, Paola; Motta, Concettina La; Gargini, Claudia
A New Vista of Aldehyde Dehydrogenase 1A3 (ALDH1A3): New Specific Inhibitors and Activity-Based Probes Targeting ALDH1A3 Dependent Pathways in Glioblastoma, Mesothelioma and Other Cancers
2024-01-01 Magrassi, Lorenzo; Pinton, Giulia; Luzzi, Sabino; Comincini, Sergio; Scravaglieri, Andrea; Gigliotti, Valentina; Bernardoni, BIANCA LAURA; D'Agostino, Ilaria; Juretich, Francesca; LA MOTTA, Concettina; Garavaglia, Silvia
An insight into the last 5-year patents on Porphyromonas gingivalis and Streptococcus mutans, the pivotal pathogens in the oral cavity
2024-01-01 Bernardoni, B. L.; D'Agostino, I.; La Motta, C.; Angeli, A.
An update on antibacterial AlkylGuanidino Ureas: Design of new derivatives, synergism with colistin and data analysis of the whole library
2024-01-01 Ardino, Claudia; Sannio, Filomena; Poli, Giulio; Galati, Salvatore; Dreassi, Elena; Botta, Lorenzo; Docquier, Jean-Denis; D'Agostino, Ilaria
Azo derivatives of monoterpenes as anti-Helicobacter pylori agents: from synthesis to structure-based target investigation
2024-01-01 Melfi, F.; Fantacuzzi, M.; Carradori, S.; D'Agostino, I.; Ammazzalorso, A.; Mencarelli, N.; Gallorini, M.; Spano, M.; Guglielmi, P.; Agamennone, M.; Haji Ali, S.; Al-Samydai, A.; Sisto, F.
Azobenzenesulfonamide Carbonic Anhydrase Inhibitors as New Weapons to Fight Helicobacter pylori: Synthesis, Bioactivity Evaluation, In Vivo Toxicity, and Computational Studies
2024-01-01 Giampietro, Letizia; Marinacci, Beatrice; Della Valle, Alice; D'Agostino, Ilaria; Lauro, Aldo; Mori, Mattia; Carradori, Simone; Ammazzalorso, Alessandra; De Filippis, Barbara; Maccallini, Cristina; Angeli, Andrea; Capasso, Clemente; Francati, Santolo; Mollica, Adriano; Grande, Rossella; Supuran, Claudiu
Benzenesulfonamide decorated dihydropyrimidin(thi)ones: carbonic anhydrase profiling and antiproliferative activity
2024-01-01 Aslan, H.; Renzi, G.; Angeli, A.; D'Agostino, I.; Ronca, R.; Massardi, M. L.; Tavani, C.; Carradori, S.; Ferraroni, M.; Governa, P.; Manetti, F.; Carta, F.; Supuran, C. T.
Cyclization of acyl thiosemicarbazides led to new Helicobacter pylori α‐carbonic anhydrase inhibitors
2024-01-01 Gumus, Arzu; D'Agostino, Ilaria; Puca, Valentina; Crocetta, Valentina; Carradori, Simone; Cutarella, Luigi; Mori, Mattia; Carta, Fabrizio; Angeli, Andrea; Capasso, Clemente; Supuran, Claudiu T.
Early investigation of a novel SI306 theranostic prodrug for glioblastoma treatment
2024-01-01 Vagaggini, Chiara; Petroni, Debora; D'Agostino, Ilaria; Poggialini, Federica; Cavallini, Chiara; Cianciusi, Annarita; Salis, Annalisa; D'Antona, Lucia; Francesconi, Valeria; Manetti, Fabrizio; Damonte, Gianluca; Musumeci, Francesca; Menichetti, Luca; Dreassi, Elena; Carbone, Anna; Schenone, Silvia
Enzyme-mediated activation of prodrugs
2024-01-01 D'Agostino, Ilaria; Carradori, Simone; La Motta, Concettina
Exploring the Polypharmacological Potential of PCI-27483: A Selective Inhibitor of Carbonic Anhydrases IX and XII
2024-01-01 D'Agostino, Ilaria; Bonardi, Alessandro; Ferraroni, Marta; Gratteri, Paola; Angeli, Andrea; Supuran, Claudiu T.
Helicobacter pylori CAs inhibition
2024-01-01 Bernardoni, Bianca Laura; La Motta, Concettina; Carradori, Simone; D'Agostino, Ilaria
Inhibition of Pseudomonas aeruginosa Carbonic Anhydrases, Exploring Ciprofloxacin Functionalization Toward New Antibacterial Agents: An In-Depth Multidisciplinary Study
2024-01-01 Marinacci, Beatrice; D'Agostino, Ilaria; Angeli, Andrea; Carradori, Simone; Melfi, Francesco; Grande, Rossella; Corsiani, Micol; Ferraroni, Marta; Agamennone, Mariangela; Tondo, Anna Rita; Zara, Susi; Puca, Valentina; Pellegrini, Benedetta; Vagaggini, Chiara; Dreassi, Elena; Patrauchan, Marianna A.; Capasso, Clemente; Nicolotti, Orazio; Carta, Fabrizio; Supuran, Claudiu T.
Lasamide Containing Sulfonylpiperazines as Effective Agents for the Management of Glaucoma Associated Symptoms
2024-01-01 Kilbile, Jaydeo T.; Sapkal, Suryakant B.; Renzi, Gioele; D'Agostino, Ilaria; Boudjelal, Mohamed; Tamboli, Yasinalli; Cutarella, Luigi; Mori, Mattia; Sgambellone, Silvia; Villano, Serafina; Marri, Silvia; Lucarini, Laura; Carradori, Simone; Carta, Fabrizio; Supuran, Claudiu T.
Lasamide, a Potent Human Carbonic Anhydrase Inhibitor from the Market: Inhibition Profiling and Crystallographic Studies
2024-01-01 Baroni, Chiara; D'Agostino, Ilaria; Renzi, Gioele; Kilbile, Jaydeo T.; Tamboli, Yasinalli; Ferraroni, Marta; Carradori, Simone; Capasso, Clemente; Carta, Fabrizio; Supuran, Claudiu T.
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| A Journey Around Boronic Acids: Sulfonyl Hydrazone-Containing Derivatives as Carbonic Anhydrase Inhibitors | 1-gen-2025 | Anakök, Deniz A; Angeli, Andrea; D'Agostino, Ilaria; Renzi, Gioele; Massardi, Maria Luisa; Tavani, Camilla; Çete, Servet; Carradori, Simone; Ronca, Roberto; Capasso, Clemente; Carta, Fabrizio; Supuran, Claudiu T | |
| A scaffold repositioning approach: dihydroBenzoImidazoTriazineDione (BITD) derivatives as selective ALDH1A1 inhibitors | 1-gen-2025 | Bernardoni, Bianca Laura; D'Agostino, Ilaria; Siragusa, Sonia; Mori, Mattia; Garavaglia, Silvia; La Motta, Concettina | |
| O-derivatization of natural tropolone and β-thujaplicin leading to effective inhibitors of human carbonic anhydrases IX and XII | 1-gen-2025 | Melfi, Francesco; D'Agostino, Ilaria; Carradori, Simone; Carta, Fabrizio; Angeli, Andrea; Costa, Giosuè; Renzi, Gioele; Čikoš, Ana; Vullo, Daniela; Rešetar, Josip; Ferraroni, Marta; Baroni, Chiara; Mancuso, Francesca; Gitto, Rosaria; Ambrosio, Francesca Alessandra; Marchese, Emanuela; Torcasio, Roberta; Amodio, Nicola; Capasso, Clemente; Alcaro, Stefano; Supuran, Claudiu T. | |
| Pegylation Approach Applied to Erlotinib-Carbonic Anhydrase Inhibitors Hybrids Towards Anticancer Agents | 1-gen-2025 | Filiberti, Serena; Renzi, Gioele; Carta, Fabrizio; Fantacuzzi, Marialuigia; D'Agostino, Ilaria; Benito, German; Angeli, Andrea; Massardi, Marialuisa; Simsek, Rahime; Capasso, Clemente; Carradori, Simone; Ronca, Roberto; Supuran, Claudiu | |
| Unprecedented carbonic anhydrase inhibition mechanism: Targeting histidine 64 side chain through a halogen bond | 1-gen-2025 | Paciotti, Roberto; Carradori, Simone; Angeli, Andrea; D'Agostino, Ilaria; Ferraroni, Marta; Coletti, Cecilia; Supuran, Claudiu T. | |
| β-Cyclodextrin nanosponges for the ocular delivery of therapeutic Micro-RNA in a Mouse model of retinitis Pigmentosa: A proof of concept study | 1-gen-2025 | Piano, Ilaria; Polini, Beatrice; Corsi, Francesca; Carpi, Sara; Petrarolo, Giovanni; Quattrini, Luca; D'Agostino, Ilaria; Gamberini, Maria Cristina; Baraldi, Cecilia; Chiellini, Grazia; Nieri, Paola; Motta, Concettina La; Gargini, Claudia | |
| A New Vista of Aldehyde Dehydrogenase 1A3 (ALDH1A3): New Specific Inhibitors and Activity-Based Probes Targeting ALDH1A3 Dependent Pathways in Glioblastoma, Mesothelioma and Other Cancers | 1-gen-2024 | Magrassi, Lorenzo; Pinton, Giulia; Luzzi, Sabino; Comincini, Sergio; Scravaglieri, Andrea; Gigliotti, Valentina; Bernardoni, BIANCA LAURA; D'Agostino, Ilaria; Juretich, Francesca; LA MOTTA, Concettina; Garavaglia, Silvia | |
| An insight into the last 5-year patents on Porphyromonas gingivalis and Streptococcus mutans, the pivotal pathogens in the oral cavity | 1-gen-2024 | Bernardoni, B. L.; D'Agostino, I.; La Motta, C.; Angeli, A. | |
| An update on antibacterial AlkylGuanidino Ureas: Design of new derivatives, synergism with colistin and data analysis of the whole library | 1-gen-2024 | Ardino, Claudia; Sannio, Filomena; Poli, Giulio; Galati, Salvatore; Dreassi, Elena; Botta, Lorenzo; Docquier, Jean-Denis; D'Agostino, Ilaria | |
| Azo derivatives of monoterpenes as anti-Helicobacter pylori agents: from synthesis to structure-based target investigation | 1-gen-2024 | Melfi, F.; Fantacuzzi, M.; Carradori, S.; D'Agostino, I.; Ammazzalorso, A.; Mencarelli, N.; Gallorini, M.; Spano, M.; Guglielmi, P.; Agamennone, M.; Haji Ali, S.; Al-Samydai, A.; Sisto, F. | |
| Azobenzenesulfonamide Carbonic Anhydrase Inhibitors as New Weapons to Fight Helicobacter pylori: Synthesis, Bioactivity Evaluation, In Vivo Toxicity, and Computational Studies | 1-gen-2024 | Giampietro, Letizia; Marinacci, Beatrice; Della Valle, Alice; D'Agostino, Ilaria; Lauro, Aldo; Mori, Mattia; Carradori, Simone; Ammazzalorso, Alessandra; De Filippis, Barbara; Maccallini, Cristina; Angeli, Andrea; Capasso, Clemente; Francati, Santolo; Mollica, Adriano; Grande, Rossella; Supuran, Claudiu | |
| Benzenesulfonamide decorated dihydropyrimidin(thi)ones: carbonic anhydrase profiling and antiproliferative activity | 1-gen-2024 | Aslan, H.; Renzi, G.; Angeli, A.; D'Agostino, I.; Ronca, R.; Massardi, M. L.; Tavani, C.; Carradori, S.; Ferraroni, M.; Governa, P.; Manetti, F.; Carta, F.; Supuran, C. T. | |
| Cyclization of acyl thiosemicarbazides led to new Helicobacter pylori α‐carbonic anhydrase inhibitors | 1-gen-2024 | Gumus, Arzu; D'Agostino, Ilaria; Puca, Valentina; Crocetta, Valentina; Carradori, Simone; Cutarella, Luigi; Mori, Mattia; Carta, Fabrizio; Angeli, Andrea; Capasso, Clemente; Supuran, Claudiu T. | |
| Early investigation of a novel SI306 theranostic prodrug for glioblastoma treatment | 1-gen-2024 | Vagaggini, Chiara; Petroni, Debora; D'Agostino, Ilaria; Poggialini, Federica; Cavallini, Chiara; Cianciusi, Annarita; Salis, Annalisa; D'Antona, Lucia; Francesconi, Valeria; Manetti, Fabrizio; Damonte, Gianluca; Musumeci, Francesca; Menichetti, Luca; Dreassi, Elena; Carbone, Anna; Schenone, Silvia | |
| Enzyme-mediated activation of prodrugs | 1-gen-2024 | D'Agostino, Ilaria; Carradori, Simone; La Motta, Concettina | |
| Exploring the Polypharmacological Potential of PCI-27483: A Selective Inhibitor of Carbonic Anhydrases IX and XII | 1-gen-2024 | D'Agostino, Ilaria; Bonardi, Alessandro; Ferraroni, Marta; Gratteri, Paola; Angeli, Andrea; Supuran, Claudiu T. | |
| Helicobacter pylori CAs inhibition | 1-gen-2024 | Bernardoni, Bianca Laura; La Motta, Concettina; Carradori, Simone; D'Agostino, Ilaria | |
| Inhibition of Pseudomonas aeruginosa Carbonic Anhydrases, Exploring Ciprofloxacin Functionalization Toward New Antibacterial Agents: An In-Depth Multidisciplinary Study | 1-gen-2024 | Marinacci, Beatrice; D'Agostino, Ilaria; Angeli, Andrea; Carradori, Simone; Melfi, Francesco; Grande, Rossella; Corsiani, Micol; Ferraroni, Marta; Agamennone, Mariangela; Tondo, Anna Rita; Zara, Susi; Puca, Valentina; Pellegrini, Benedetta; Vagaggini, Chiara; Dreassi, Elena; Patrauchan, Marianna A.; Capasso, Clemente; Nicolotti, Orazio; Carta, Fabrizio; Supuran, Claudiu T. | |
| Lasamide Containing Sulfonylpiperazines as Effective Agents for the Management of Glaucoma Associated Symptoms | 1-gen-2024 | Kilbile, Jaydeo T.; Sapkal, Suryakant B.; Renzi, Gioele; D'Agostino, Ilaria; Boudjelal, Mohamed; Tamboli, Yasinalli; Cutarella, Luigi; Mori, Mattia; Sgambellone, Silvia; Villano, Serafina; Marri, Silvia; Lucarini, Laura; Carradori, Simone; Carta, Fabrizio; Supuran, Claudiu T. | |
| Lasamide, a Potent Human Carbonic Anhydrase Inhibitor from the Market: Inhibition Profiling and Crystallographic Studies | 1-gen-2024 | Baroni, Chiara; D'Agostino, Ilaria; Renzi, Gioele; Kilbile, Jaydeo T.; Tamboli, Yasinalli; Ferraroni, Marta; Carradori, Simone; Capasso, Clemente; Carta, Fabrizio; Supuran, Claudiu T. |