Some naphthol [1,2,-b]-s-triazolo[4,3-d]-1,4-thiazine and 1,5-thiazepine and s-triazolo[4',3'-4,5]-1, ,4-thiazino[3,2-c]quinoline derivatives have been synthesized and tested for their ability to displace [H-3]RO 15-1788 binding from bovine brain membranes. Several compounds showed moderate binding affinity for the benzodiazepine receptor.
Studies on annelated 1,4-benzothiazines and 1,5-benzothiazepines .10. Synthesis and inhibition of benzodiazepine receptor binding of new 1,4-thiazine and 1,5-thiazepine polycondensed heterocycles with steroidal structure
GIANNACCINI, GINO;LUCACCHINI, ANTONIO;MARTINI, CLAUDIA
1996-01-01
Abstract
Some naphthol [1,2,-b]-s-triazolo[4,3-d]-1,4-thiazine and 1,5-thiazepine and s-triazolo[4',3'-4,5]-1, ,4-thiazino[3,2-c]quinoline derivatives have been synthesized and tested for their ability to displace [H-3]RO 15-1788 binding from bovine brain membranes. Several compounds showed moderate binding affinity for the benzodiazepine receptor.File in questo prodotto:
Non ci sono file associati a questo prodotto.
I documenti in IRIS sono protetti da copyright e tutti i diritti sono riservati, salvo diversa indicazione.
