Several N-(indol-3-ylglyoxylyl)alanine and glycine ester derivatives were prepared to evaluate the influence of the ester group size both on affinity and on activity at the benzodiazepine receptor. Moreover, indol-3-ylglyoxylic acid esters, closely related to 3-alkoxy-β-carbolines, were synthesized and tested in vitro on the benzodiazepine receptor.
|Autori:||PRIMOFIORE G; DA SETTIMO F; MARINI AM; LA MOTTA C; MARTINI C; SENATORE G; LUCACCHINI A|
|Titolo:||N-(Indol-3-ylglyoxylyl)amino acid ester derivatives. Synthesis and interaction properties at the benzodiazepine receptor|
|Anno del prodotto:||1995|
|Appare nelle tipologie:||1.1 Articolo in rivista|