The one-pot synthesis and the benzodiazepine receptor binding activity of some imidazo[2,1-a]phthalazines bearing different substituents at position-2 and/or 3 and/or 6 is reported. The dissimilar binding results of the reported compounds are discussed in relation to the nature and/or position of the substituents on the tricyclic ring system.

REACTION OF 1-AMINOPHTHALAZINES WITH ALPHA-HALOCARBONYL COMPOUNDS - IMIDAZO[2,1-A]PHTHALAZINES AND THEIR BENZODIAZEPINE RECEPTOR ACTIVITIES

MARTINI, CLAUDIA;GIUSTI, LAURA;LUCACCHINI, ANTONIO
1993

Abstract

The one-pot synthesis and the benzodiazepine receptor binding activity of some imidazo[2,1-a]phthalazines bearing different substituents at position-2 and/or 3 and/or 6 is reported. The dissimilar binding results of the reported compounds are discussed in relation to the nature and/or position of the substituents on the tricyclic ring system.
Catarzi, D; Cecchi, L; Colotta, V; Conti, G; Melani, F; Filacchioni, G; Martini, Claudia; Giusti, Laura; Lucacchini, Antonio
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Utilizza questo identificativo per citare o creare un link a questo documento: http://hdl.handle.net/11568/205132
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