Sfoglia per Autore
Increased Lactate Secretion by Cancer Cells Sustains Non-cell-autonomous Adaptive Resistance to MET and EGFR Targeted Therapies
2018-01-01 Apicella, Maria; Giannoni, Elisa; Fiore, Stephany; Ferrari, Karin Johanna; Fernández-Pérez, Daniel; Isella, Claudio; Granchi, Carlotta; Minutolo, Filippo; Sottile, Antonino; Comoglio, Paolo Maria; Medico, Enzo; Pietrantonio, Filippo; Volante, Marco; Pasini, Diego; Chiarugi, Paola; Giordano, Silvia; Corso, Simona
ATP citrate lyase (ACLY) inhibitors: An anti-cancer strategy at the crossroads of glucose and lipid metabolism
2018-01-01 Granchi, Carlotta
Activators of Sirtuin-1 and their Involvement in Cardioprotection
2018-01-01 Granchi, Carlotta; Minutolo, Filippo
New phenylethanoid glycosides from Cistanche phelypaea and their activity as inhibitors of monoacylglycerol lipase (MAGL)
2018-01-01 Beladjila, K. A.; Berrehal, D.; De Tommasi, N.; Granchi, C.; Bononi, Giulia; Braca, A.; De Leo, M.
Discovery of 1,5-Diphenylpyrazole-3-Carboxamide Derivatives as Potent, Reversible, and Selective Monoacylglycerol Lipase (MAGL) Inhibitors
2018-01-01 Aghazadeh Tabrizi, Mojgan; Baraldi, Pier Giovanni; Baraldi, Stefania; Ruggiero, Emanuela; De Stefano, Lucia; Rizzolio, Flavio; Di Cesare Mannelli, Lorenzo; Ghelardini, Carla; Chicca, Andrea; Lapillo, Margherita; Gertsch, Jürg; Manera, Clementina; Macchia, Marco; Martinelli, Adriano; Granchi, Carlotta; Minutolo, Filippo; Tuccinardi, Tiziano
Liposomal delivery of a Pin1 inhibitor complexed with cyclodextrins as new therapy for high-grade serous ovarian cancer
2018-01-01 Russo Spena, Concetta; De Stefano, Lucia; Palazzolo, Stefano; Salis, Barbara; Granchi, Carlotta; Minutolo, Filippo; Tuccinardi, Tiziano; Fratamico, Roberto; Crotti, Sara; D'Aronco, Sara; Agostini, Marco; Corona, Giuseppe; Caligiuri, Isabella; Canzonieri, Vincenzo; Rizzolio, Flavio
Binding investigation and preliminary optimisation of the 3-amino-1,2,4-triazin-5(2H)-one core for the development of new Fyn inhibitors
2018-01-01 Poli, Giulio; Lapillo, Margherita; Granchi, Carlotta; Caciolla, Jessica; Mouawad, Nayla; Caligiuri, Isabella; Rizzolio, Flavio; Langer, Thierry; Minutolo, Filippo; Tuccinardi, Tiziano
Discovery of long-chain salicylketoxime derivatives as monoacylglycerol lipase (MAGL) inhibitors
2018-01-01 Bononi, Giulia; Granchi, Carlotta; Lapillo, Margherita; Giannotti, Massimiliano; Nieri, Daniela; Fortunato, Serena; Boustani, Maguie El; Caligiuri, Isabella; Poli, Giulio; Carlson, Kathryn E.; Kim, Sung Hoon; Macchia, Marco; Martinelli, Adriano; Rizzolio, Flavio; Chicca, Andrea; Katzenellenbogen, John A.; Minutolo, Filippo; Tuccinardi, Tiziano
Rational Development of MAGL Inhibitors
2018-01-01 Granchi, Carlotta; Rizzolio, Flavio; Caligiuri, Isabella; Macchia, Marco; Martinelli, Adriano; Minutolo, Filippo; Tuccinardi, Tiziano
Identification of Lactate Dehydrogenase 5 Inhibitors using Pharmacophore- Driven Consensus Docking
2018-01-01 Poli, Giulio; Scarpino, Andrea; Aissaoui, Mohamed; Granchi, Carlotta; Minutolo, Filippo; Martinelli, Adriano; Tuccinardi, Tiziano
Design, Synthesis, and Evaluation of GLUT Inhibitors
2018-01-01 Granchi, Carlotta; Tuccinardi, Tiziano; Minutolo, Filippo
An Update on Patents Covering Agents That Interfere with the Cancer Glycolytic Cascade
2018-01-01 Fortunato, Serena; Bononi, Giulia; Granchi, Carlotta; Minutolo, Filippo
New diterpenes from Salvia pseudorosmarinus and their activity as inhibitors of monoacylglycerol lipase (MAGL)
2018-01-01 De Leo, M.; Guillen Huallpa, C.; Alvarado, B.; Granchi, C.; Poli, G.; De Tommasi, N.; Braca, A.
Effect of Tumor Relevant Acidic Environment in the Interaction of a N-hydroxyindole-2-Carboxylic Derivative with the Phospholipid Bilayer
2018-01-01 Monti, Daniela; Tampucci, Silvia; Zucchetti, Erica; Granchi, Carlotta; Minutolo, Filippo; Piras, Anna Maria
New activators of SIRT1 enzyme for the treatment of cardiovascular and cardiometabolic pathologies
2019-01-01 Calderone, Vincenzo; Minutolo, Filippo; Tuccinardi, Tiziano; Testai, Lara; Granchi, Carlotta; Martelli, Alma; Citi, Valentina; DE LORENZO GARDINAL, Virginia; Lenzi, Giulia; Leo, Francesca; Malloggi, Giulia
The influence of Echinacea purpurea leaf microbiota on chicoric acid level
2019-01-01 Maggini, V.; De Leo, M.; Granchi, C.; Tuccinardi, T.; Mengoni, A.; Gallo, E. R.; Biffi, S.; Fani, R.; Pistelli, L.; Firenzuoli, F.; Bogani, P.
Abstract 3082: Targeting hypoxic pancreatic cancer cells with glucose conjugated lactate dehydrogenase inhibitor NHI-Glc-2
2019-01-01 Hassouni, Btissame El; Sciarrillo, Rocco; Gómez, Valentina Edith; Maftouh, Mina; Mantini, Giulia; Vonk, Christian M.; Granchi, Carlotta; Funel, Niccola; Minutolo, Filippo; Peters, Godefridus J.; Giovannetti, Elisa
First examples of H2S-releasing glycoconjugates: stereoselective synthesis and anticancer activities
2019-01-01 Fortunato, Serena; Lenzi, Chiara; Granchi, Carlotta; Citi, Valentina; Martelli, Alma; Calderone, Vincenzo; Di Pietro, Sebastiano; Signore, Giovanni; Di Bussolo, Valeria; Minutolo, Filippo
First-of-its-kind STARD 3 Inhibitor: In Silico Identification and Biological Evaluation as Anticancer Agent
2019-01-01 Lapillo, M.; Salis, B.; Palazzolo, S.; Poli, G.; Granchi, C.; Minutolo, F.; Rotondo, R.; Caligiuri, I.; Canzonieri, V.; Tuccinardi, T.; Rizzolio, F.
Synthesis and Biological Evaluation of New Glycoconjugated LDH Inhibitors as Anticancer Agents
2019-01-01 D'Andrea, Felicia; Giulia, Vagelli; Granchi, Carlotta; Guazzelli, Lorenzo; Tuccinardi, Tiziano; Poli, Giulio; Iacopini, Dalila; Minutolo, Filippo; DI BUSSOLO, Valeria
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Increased Lactate Secretion by Cancer Cells Sustains Non-cell-autonomous Adaptive Resistance to MET and EGFR Targeted Therapies | 1-gen-2018 | Apicella, Maria; Giannoni, Elisa; Fiore, Stephany; Ferrari, Karin Johanna; Fernández-Pérez, Daniel; Isella, Claudio; Granchi, Carlotta; Minutolo, Filippo; Sottile, Antonino; Comoglio, Paolo Maria; Medico, Enzo; Pietrantonio, Filippo; Volante, Marco; Pasini, Diego; Chiarugi, Paola; Giordano, Silvia; Corso, Simona | |
ATP citrate lyase (ACLY) inhibitors: An anti-cancer strategy at the crossroads of glucose and lipid metabolism | 1-gen-2018 | Granchi, Carlotta | |
Activators of Sirtuin-1 and their Involvement in Cardioprotection | 1-gen-2018 | Granchi, Carlotta; Minutolo, Filippo | |
New phenylethanoid glycosides from Cistanche phelypaea and their activity as inhibitors of monoacylglycerol lipase (MAGL) | 1-gen-2018 | Beladjila, K. A.; Berrehal, D.; De Tommasi, N.; Granchi, C.; Bononi, Giulia; Braca, A.; De Leo, M. | |
Discovery of 1,5-Diphenylpyrazole-3-Carboxamide Derivatives as Potent, Reversible, and Selective Monoacylglycerol Lipase (MAGL) Inhibitors | 1-gen-2018 | Aghazadeh Tabrizi, Mojgan; Baraldi, Pier Giovanni; Baraldi, Stefania; Ruggiero, Emanuela; De Stefano, Lucia; Rizzolio, Flavio; Di Cesare Mannelli, Lorenzo; Ghelardini, Carla; Chicca, Andrea; Lapillo, Margherita; Gertsch, Jürg; Manera, Clementina; Macchia, Marco; Martinelli, Adriano; Granchi, Carlotta; Minutolo, Filippo; Tuccinardi, Tiziano | |
Liposomal delivery of a Pin1 inhibitor complexed with cyclodextrins as new therapy for high-grade serous ovarian cancer | 1-gen-2018 | Russo Spena, Concetta; De Stefano, Lucia; Palazzolo, Stefano; Salis, Barbara; Granchi, Carlotta; Minutolo, Filippo; Tuccinardi, Tiziano; Fratamico, Roberto; Crotti, Sara; D'Aronco, Sara; Agostini, Marco; Corona, Giuseppe; Caligiuri, Isabella; Canzonieri, Vincenzo; Rizzolio, Flavio | |
Binding investigation and preliminary optimisation of the 3-amino-1,2,4-triazin-5(2H)-one core for the development of new Fyn inhibitors | 1-gen-2018 | Poli, Giulio; Lapillo, Margherita; Granchi, Carlotta; Caciolla, Jessica; Mouawad, Nayla; Caligiuri, Isabella; Rizzolio, Flavio; Langer, Thierry; Minutolo, Filippo; Tuccinardi, Tiziano | |
Discovery of long-chain salicylketoxime derivatives as monoacylglycerol lipase (MAGL) inhibitors | 1-gen-2018 | Bononi, Giulia; Granchi, Carlotta; Lapillo, Margherita; Giannotti, Massimiliano; Nieri, Daniela; Fortunato, Serena; Boustani, Maguie El; Caligiuri, Isabella; Poli, Giulio; Carlson, Kathryn E.; Kim, Sung Hoon; Macchia, Marco; Martinelli, Adriano; Rizzolio, Flavio; Chicca, Andrea; Katzenellenbogen, John A.; Minutolo, Filippo; Tuccinardi, Tiziano | |
Rational Development of MAGL Inhibitors | 1-gen-2018 | Granchi, Carlotta; Rizzolio, Flavio; Caligiuri, Isabella; Macchia, Marco; Martinelli, Adriano; Minutolo, Filippo; Tuccinardi, Tiziano | |
Identification of Lactate Dehydrogenase 5 Inhibitors using Pharmacophore- Driven Consensus Docking | 1-gen-2018 | Poli, Giulio; Scarpino, Andrea; Aissaoui, Mohamed; Granchi, Carlotta; Minutolo, Filippo; Martinelli, Adriano; Tuccinardi, Tiziano | |
Design, Synthesis, and Evaluation of GLUT Inhibitors | 1-gen-2018 | Granchi, Carlotta; Tuccinardi, Tiziano; Minutolo, Filippo | |
An Update on Patents Covering Agents That Interfere with the Cancer Glycolytic Cascade | 1-gen-2018 | Fortunato, Serena; Bononi, Giulia; Granchi, Carlotta; Minutolo, Filippo | |
New diterpenes from Salvia pseudorosmarinus and their activity as inhibitors of monoacylglycerol lipase (MAGL) | 1-gen-2018 | De Leo, M.; Guillen Huallpa, C.; Alvarado, B.; Granchi, C.; Poli, G.; De Tommasi, N.; Braca, A. | |
Effect of Tumor Relevant Acidic Environment in the Interaction of a N-hydroxyindole-2-Carboxylic Derivative with the Phospholipid Bilayer | 1-gen-2018 | Monti, Daniela; Tampucci, Silvia; Zucchetti, Erica; Granchi, Carlotta; Minutolo, Filippo; Piras, Anna Maria | |
New activators of SIRT1 enzyme for the treatment of cardiovascular and cardiometabolic pathologies | 1-gen-2019 | Calderone, Vincenzo; Minutolo, Filippo; Tuccinardi, Tiziano; Testai, Lara; Granchi, Carlotta; Martelli, Alma; Citi, Valentina; DE LORENZO GARDINAL, Virginia; Lenzi, Giulia; Leo, Francesca; Malloggi, Giulia | |
The influence of Echinacea purpurea leaf microbiota on chicoric acid level | 1-gen-2019 | Maggini, V.; De Leo, M.; Granchi, C.; Tuccinardi, T.; Mengoni, A.; Gallo, E. R.; Biffi, S.; Fani, R.; Pistelli, L.; Firenzuoli, F.; Bogani, P. | |
Abstract 3082: Targeting hypoxic pancreatic cancer cells with glucose conjugated lactate dehydrogenase inhibitor NHI-Glc-2 | 1-gen-2019 | Hassouni, Btissame El; Sciarrillo, Rocco; Gómez, Valentina Edith; Maftouh, Mina; Mantini, Giulia; Vonk, Christian M.; Granchi, Carlotta; Funel, Niccola; Minutolo, Filippo; Peters, Godefridus J.; Giovannetti, Elisa | |
First examples of H2S-releasing glycoconjugates: stereoselective synthesis and anticancer activities | 1-gen-2019 | Fortunato, Serena; Lenzi, Chiara; Granchi, Carlotta; Citi, Valentina; Martelli, Alma; Calderone, Vincenzo; Di Pietro, Sebastiano; Signore, Giovanni; Di Bussolo, Valeria; Minutolo, Filippo | |
First-of-its-kind STARD 3 Inhibitor: In Silico Identification and Biological Evaluation as Anticancer Agent | 1-gen-2019 | Lapillo, M.; Salis, B.; Palazzolo, S.; Poli, G.; Granchi, C.; Minutolo, F.; Rotondo, R.; Caligiuri, I.; Canzonieri, V.; Tuccinardi, T.; Rizzolio, F. | |
Synthesis and Biological Evaluation of New Glycoconjugated LDH Inhibitors as Anticancer Agents | 1-gen-2019 | D'Andrea, Felicia; Giulia, Vagelli; Granchi, Carlotta; Guazzelli, Lorenzo; Tuccinardi, Tiziano; Poli, Giulio; Iacopini, Dalila; Minutolo, Filippo; DI BUSSOLO, Valeria |
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