Sfoglia per Autore
2-(Methyleneaminoxy)methylmorpholine derivatives. Synthesis and antidepressant activity
1994-01-01 A., Balsamo; Lapucci, Annalina; Macchia, Marco; Martinelli, Adriano; Nencetti, Susanna; T., Cristina; Rossello, Armando
SYNTHESIS, ANTIINFLAMMATORY ACTIVITY AND MOLECULAR-ORBITAL STUDIES OF A SERIES OF BENZYLIDENEAMINOXYPROPIONIC ACIDS SUBSTITUTED ON THE PHENYL RING
1994-01-01 Lapucci, Annalina; Macchia, Marco; Martinelli, Adriano; Nencetti, Susanna; Orlandini, Elisabetta; Rossello, Armando; Baldacci, M; Soldani, G; Mengozzi, G.
(E)-(ARYLMETHYLENEAMINOXY)ACETAMIDES AS ANALOGS OF NEUROLEPTIC BENZAMIDES - SYNTHESIS AND D-2-DOPAMINERGIC BINDING-AFFINITY
1995-01-01 Macchia, Marco; Manera, Clementina; Martinelli, Adriano; Orlandini, Elisabetta; Romagnoli, F; Rossello, Armando; Chiellini, Grazia
SYNTHESIS AND BETA-ADRENERGIC ACTIVITY OF A SERIES OF 3-(SUBSTITUTED-BENZYLIDENEAMINOXY)PROPANOLAMINE DERIVATIVES
1995-01-01 Gentili, D; Lapucci, Annalina; Macchia, B; Macchia, Marco; Martinelli, Adriano; Nencetti, Susanna; Orlandini, Elisabetta; Ferni, G; Pinza, M.
SYNTHESIS, ANTIINFLAMMATORY ACTIVITY AND PLATELET ANTIAGGREGATING ACTIVITY OF A NEW SERIES OF BETA-AMINOXYPROPIONIC ACIDS
1995-01-01 Macchia, B; Macchia, Marco; Martinelli, Adriano; Orlandini, Elisabetta; Rossello, Armando; Bertini, S; Luchetti, E; Gervasi, G; Catalani, R.
Synthesis and ß-adrenergic properties of (E)-N-[3-(alkylamino)-2- hydroxypropilidene](methyloxy)amines substituted with an aromatic group on their [(methyloxy)imino]methyl moiety (MOIMM): an investigation into the biopharmacological effects of an aryl substitution in the class of MOIM ß-blocking drugs.
1995-01-01 Balsamo, A; Breschi, MARIA CRISTINA; Chiellini, Grazia; Favero, Lucilla; Macchia, Marco; Martinelli, Adriano; Martini, Claudia; Rossello, Armando; Scatizzi, R.
Conformationally restrained β -blocking oxime ethers. 4. Chiral 2-(3'-(5'-p-chlorophenyl)isoxazolidinyl)ethanolamines as conformationally restrained analogs of methyloxyiminomethyl (MOIM) β -adrenergic antagonists: synthesis, configuration and β -adrenergic properties
1996-01-01 Balsamo, Aldo; Breschi, M. C.; Chiellini, G; Cozzini, P; Domiano, P; Macchia, Marco; Manera, Clementina; Martinelli, A; Nencetti, S.
Chiral 2-(3'-(5'-p-chlorophenyl)isoxazolidinyl)ethanolamines as conformationally restrained analogs of methyloxyiminomethyl (MOIM) beta-adrenergic antagonists: Synthesis, configuration and beta-adrenergic properties
1996-01-01 Balsamo, A; Breschi, MARIA CRISTINA; Chiellini, Grazia; Cozzini, P; Domiano, P; Macchia, Marco; Manera, Clementina; Martinelli, Adriano; Nencetti, Susanna; Rossello, Armando; Sacca, P; Scatizzi, R.
1,2,3-triazolo[1.5-a]quinazolines: synthesis, benzodiazepine receptor binding and theoretical calculations
1996-01-01 Biagi, G; Giorgi, Irene; Livi, O; Scartoni, V; Velo, S; DE SANCTIS, B; Martinelli, Adriano; Martini, Claudia; Senatore, G.
Synthesis of pyrrolo[3,4-c]pyridine derivatives possessing an acid group and their in vitro and in vivo evaluation as aldose reductase inhibitors
1996-01-01 Dasettimo, A; Primofiore, G; DA SETTIMO PASSETTI, Federico; Simorini, Francesca; LA MOTTA, Concettina; Martinelli, Adriano; Boldrini, E.
1,2,3-Triazolo[1,5-a][1,3]benzodiazepine a new heterocyclic system: Synthesis, benzodiazepine receptor binding and theoretical calculations
1996-01-01 Biagi, G; Giorgi, Irene; Livi, O; Scartoni, V; Velo, S; Desantis, B; Martinelli, Adriano; Martini, Claudia; Senatore, G.
Conformational effects on the activity of drugs .19. Synthesis and alpha-adrenergic activity of 2- and 6-methyl-substituted (3,4-dihydroxyphenyl)-3-piperidinols
1997-01-01 Macchia, B; Macchia, Marco; Martinelli, Adriano; Martinotti, E; Orlandini, Elisabetta; Romagnoli, F; Scatizzi, R.
Unusual nitration of substituted 7-amino-1,8-naphthyridine in the synthesis of compounds with antiplatelet activity
1997-01-01 Ferrarini, Pl; Mori, C; Badawneh, M; Manera, Clementina; Clementina, M; Martinelli, Adriano; Miceli, M; Romagnoli, F; Saccomanni, Giuseppe
Stereoselective synthesis and beta-blocking activity of substituted (E)- and (Z)-4(1H)-[1-(3-alkylamino-2-hydroxypropyl)oximino]-2,3-dihydro-1,8-naphthyridine. Potential antihypertensive” agents. Part VI
1997-01-01 P. L., Ferrarini; C., Mori; M., Badawneh; Manera, Clementina; Martinelli, Adriano; M., Miceli; F., Romagnoli; Saccomanni, Giuseppe
N-n-propyl-substituted 3-(dimethylphenyl)piperidines display novel discriminative properties between dopamine receptor subtypes: synthesis and receptor binding studies
1998-01-01 Cervetto, L.; Demontis, GIAN CARLO ALFREDO GIUSEPPE; Giannaccini, Gino; Longoni, Biancamaria; Macchia, B.; Macchia, Marco; Martinelli, A.; Orlandini, Elisabetta
Derivati 1,8-naftiridinici con affinità verso i recettori A1 e A2A dell’adenosina.
1998-01-01 Ferrarini, P. L.; Manera, Clementina; Martinelli, Adriano; Mori, C.; Betti, Laura; Giannaccini, Gino; Lucacchini, Antonio
1,2-disubstituted cyclohexane derived tripeptide aldehydes as novel selective thrombin inhibitors
1998-01-01 Harmat, Njs; Di Bugno, C; Criscuoli, M; Giorgi, R; Lippi, A; Martinelli, Adriano; Monti, S; Subissi, A.
Synthesis and aldose reductase inhibitory activity of new N-(benzyloxy) glycine derivatives
1998-01-01 Macchia, Marco; Barontini, S; Martinelli, Adriano; Menchini, E; Nencetti, Susanna; Orlandini, Elisabetta; Romagnoli, F.
Synthesis and alpha-adrenergic and I-1-imidazoline activity of 3-phenylpiperidines dimethyl-substituted on the phenyl ring
1998-01-01 B., Macchia; D. B., Bylund; Calderone, Vincenzo; Giannaccini, Gino; Lucacchini, Antonio; Macchia, Marco; Martinelli, Adriano; E., Martinotti; Orlandini, Elisabetta; F., Romagnoli; Rossello, Armando
Toward the rational development of peptidomimetic analogs of the C-terminal endothelin hexapeptide: development of a theoretical model
1998-01-01 Macchia, Marco; Barontini, S; Ceccarelli, F; Galoppini, C; Giusti, Laura; Hamdan, M; Lucacchini, Antonio; Martinelli, Adriano; Menchini, E; Mazzoni, MARIA ROSA; Revoltella, Rp; Romagnoli, F; Rovero, P.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
2-(Methyleneaminoxy)methylmorpholine derivatives. Synthesis and antidepressant activity | 1-gen-1994 | A., Balsamo; Lapucci, Annalina; Macchia, Marco; Martinelli, Adriano; Nencetti, Susanna; T., Cristina; Rossello, Armando | |
SYNTHESIS, ANTIINFLAMMATORY ACTIVITY AND MOLECULAR-ORBITAL STUDIES OF A SERIES OF BENZYLIDENEAMINOXYPROPIONIC ACIDS SUBSTITUTED ON THE PHENYL RING | 1-gen-1994 | Lapucci, Annalina; Macchia, Marco; Martinelli, Adriano; Nencetti, Susanna; Orlandini, Elisabetta; Rossello, Armando; Baldacci, M; Soldani, G; Mengozzi, G. | |
(E)-(ARYLMETHYLENEAMINOXY)ACETAMIDES AS ANALOGS OF NEUROLEPTIC BENZAMIDES - SYNTHESIS AND D-2-DOPAMINERGIC BINDING-AFFINITY | 1-gen-1995 | Macchia, Marco; Manera, Clementina; Martinelli, Adriano; Orlandini, Elisabetta; Romagnoli, F; Rossello, Armando; Chiellini, Grazia | |
SYNTHESIS AND BETA-ADRENERGIC ACTIVITY OF A SERIES OF 3-(SUBSTITUTED-BENZYLIDENEAMINOXY)PROPANOLAMINE DERIVATIVES | 1-gen-1995 | Gentili, D; Lapucci, Annalina; Macchia, B; Macchia, Marco; Martinelli, Adriano; Nencetti, Susanna; Orlandini, Elisabetta; Ferni, G; Pinza, M. | |
SYNTHESIS, ANTIINFLAMMATORY ACTIVITY AND PLATELET ANTIAGGREGATING ACTIVITY OF A NEW SERIES OF BETA-AMINOXYPROPIONIC ACIDS | 1-gen-1995 | Macchia, B; Macchia, Marco; Martinelli, Adriano; Orlandini, Elisabetta; Rossello, Armando; Bertini, S; Luchetti, E; Gervasi, G; Catalani, R. | |
Synthesis and ß-adrenergic properties of (E)-N-[3-(alkylamino)-2- hydroxypropilidene](methyloxy)amines substituted with an aromatic group on their [(methyloxy)imino]methyl moiety (MOIMM): an investigation into the biopharmacological effects of an aryl substitution in the class of MOIM ß-blocking drugs. | 1-gen-1995 | Balsamo, A; Breschi, MARIA CRISTINA; Chiellini, Grazia; Favero, Lucilla; Macchia, Marco; Martinelli, Adriano; Martini, Claudia; Rossello, Armando; Scatizzi, R. | |
Conformationally restrained β -blocking oxime ethers. 4. Chiral 2-(3'-(5'-p-chlorophenyl)isoxazolidinyl)ethanolamines as conformationally restrained analogs of methyloxyiminomethyl (MOIM) β -adrenergic antagonists: synthesis, configuration and β -adrenergic properties | 1-gen-1996 | Balsamo, Aldo; Breschi, M. C.; Chiellini, G; Cozzini, P; Domiano, P; Macchia, Marco; Manera, Clementina; Martinelli, A; Nencetti, S. | |
Chiral 2-(3'-(5'-p-chlorophenyl)isoxazolidinyl)ethanolamines as conformationally restrained analogs of methyloxyiminomethyl (MOIM) beta-adrenergic antagonists: Synthesis, configuration and beta-adrenergic properties | 1-gen-1996 | Balsamo, A; Breschi, MARIA CRISTINA; Chiellini, Grazia; Cozzini, P; Domiano, P; Macchia, Marco; Manera, Clementina; Martinelli, Adriano; Nencetti, Susanna; Rossello, Armando; Sacca, P; Scatizzi, R. | |
1,2,3-triazolo[1.5-a]quinazolines: synthesis, benzodiazepine receptor binding and theoretical calculations | 1-gen-1996 | Biagi, G; Giorgi, Irene; Livi, O; Scartoni, V; Velo, S; DE SANCTIS, B; Martinelli, Adriano; Martini, Claudia; Senatore, G. | |
Synthesis of pyrrolo[3,4-c]pyridine derivatives possessing an acid group and their in vitro and in vivo evaluation as aldose reductase inhibitors | 1-gen-1996 | Dasettimo, A; Primofiore, G; DA SETTIMO PASSETTI, Federico; Simorini, Francesca; LA MOTTA, Concettina; Martinelli, Adriano; Boldrini, E. | |
1,2,3-Triazolo[1,5-a][1,3]benzodiazepine a new heterocyclic system: Synthesis, benzodiazepine receptor binding and theoretical calculations | 1-gen-1996 | Biagi, G; Giorgi, Irene; Livi, O; Scartoni, V; Velo, S; Desantis, B; Martinelli, Adriano; Martini, Claudia; Senatore, G. | |
Conformational effects on the activity of drugs .19. Synthesis and alpha-adrenergic activity of 2- and 6-methyl-substituted (3,4-dihydroxyphenyl)-3-piperidinols | 1-gen-1997 | Macchia, B; Macchia, Marco; Martinelli, Adriano; Martinotti, E; Orlandini, Elisabetta; Romagnoli, F; Scatizzi, R. | |
Unusual nitration of substituted 7-amino-1,8-naphthyridine in the synthesis of compounds with antiplatelet activity | 1-gen-1997 | Ferrarini, Pl; Mori, C; Badawneh, M; Manera, Clementina; Clementina, M; Martinelli, Adriano; Miceli, M; Romagnoli, F; Saccomanni, Giuseppe | |
Stereoselective synthesis and beta-blocking activity of substituted (E)- and (Z)-4(1H)-[1-(3-alkylamino-2-hydroxypropyl)oximino]-2,3-dihydro-1,8-naphthyridine. Potential antihypertensive” agents. Part VI | 1-gen-1997 | P. L., Ferrarini; C., Mori; M., Badawneh; Manera, Clementina; Martinelli, Adriano; M., Miceli; F., Romagnoli; Saccomanni, Giuseppe | |
N-n-propyl-substituted 3-(dimethylphenyl)piperidines display novel discriminative properties between dopamine receptor subtypes: synthesis and receptor binding studies | 1-gen-1998 | Cervetto, L.; Demontis, GIAN CARLO ALFREDO GIUSEPPE; Giannaccini, Gino; Longoni, Biancamaria; Macchia, B.; Macchia, Marco; Martinelli, A.; Orlandini, Elisabetta | |
Derivati 1,8-naftiridinici con affinità verso i recettori A1 e A2A dell’adenosina. | 1-gen-1998 | Ferrarini, P. L.; Manera, Clementina; Martinelli, Adriano; Mori, C.; Betti, Laura; Giannaccini, Gino; Lucacchini, Antonio | |
1,2-disubstituted cyclohexane derived tripeptide aldehydes as novel selective thrombin inhibitors | 1-gen-1998 | Harmat, Njs; Di Bugno, C; Criscuoli, M; Giorgi, R; Lippi, A; Martinelli, Adriano; Monti, S; Subissi, A. | |
Synthesis and aldose reductase inhibitory activity of new N-(benzyloxy) glycine derivatives | 1-gen-1998 | Macchia, Marco; Barontini, S; Martinelli, Adriano; Menchini, E; Nencetti, Susanna; Orlandini, Elisabetta; Romagnoli, F. | |
Synthesis and alpha-adrenergic and I-1-imidazoline activity of 3-phenylpiperidines dimethyl-substituted on the phenyl ring | 1-gen-1998 | B., Macchia; D. B., Bylund; Calderone, Vincenzo; Giannaccini, Gino; Lucacchini, Antonio; Macchia, Marco; Martinelli, Adriano; E., Martinotti; Orlandini, Elisabetta; F., Romagnoli; Rossello, Armando | |
Toward the rational development of peptidomimetic analogs of the C-terminal endothelin hexapeptide: development of a theoretical model | 1-gen-1998 | Macchia, Marco; Barontini, S; Ceccarelli, F; Galoppini, C; Giusti, Laura; Hamdan, M; Lucacchini, Antonio; Martinelli, Adriano; Menchini, E; Mazzoni, MARIA ROSA; Revoltella, Rp; Romagnoli, F; Rovero, P. |
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