Sfoglia per Autore
Synthesis and antimicrobial properties of substituted 3-aminoxy-(E)-2-methoxyiminopropionyl penicillins and cephalosporins
1990-01-01 A., Balsamo; B., Macchia; Martinelli, Adriano; Orlandini, Elisabetta; F., Macchia; G., Broccali; P., Domiano; Rossello, Armando
Acidi benzilideneamminossipropionici sostituiti sul fenile. Sintesi e proprietà antiinfiammatorie.
1991-01-01 A., Balsamo; Lapucci, Annalina; B., Macchia; Martinelli, Adriano; Nencetti, Susanna; Orlandini, Elisabetta; Rossello, Armando; Soldani, G. M. e. n. g. o. z. z. i. G.; M., Baldacci
1-benzilossiimmino-3- ammino-2-propanoli: sintesi e proprietà ß-adrenergiche
1991-01-01 Balsamo, A; Macchia, B; Macchia, Marco; Martinelli, Adriano; Rossello, Armando; Breschi, MARIA CRISTINA; Nieri, Paola; Scatizzi, R.
Conformational effects on the activity of drugs. 13. A revision of previously proposed models for the activation of a- and ß-adrenergic receptors
1992-01-01 Macchia, B; Balsamo, A; Breschi, MARIA CRISTINA; Lapucci, Annalina; Lucacchini, Antonio; Macchia, F; Manera, Clementina; Martinelli, Adriano; Martini, Claudia; Martinotti, E; Nencetti, Susanna
CONFORMATIONAL EFFECTS ON THE ACTIVITY OF DRUGS .13. A REVISION OF PREVIOUSLY PROPOSED MODELS FOR THE ACTIVATION OF ALPHA-ADRENERGIC AND BETA-ADRENERGIC RECEPTORS
1992-01-01 Macchia, Bruno; Balsamo, A; Breschi, MARIA CRISTINA; Lapucci, Annalina; Lucacchini, Antonio; Macchia, F; Manera, Clementina; Martinelli, Adriano; Martini, Claudia; Martinotti, E; Nencetti, Susanna
X-Ray analysis, theoretical studies and alfa-adrenergic biopharmacological properties of 1-(2,5-dimethoxyphenyl)-2-aminoethanol and its morpholine analogue.
1992-01-01 Manera, Clementina; Martinelli, Adriano; Nencetti, Susanna; Rossello, Armando; Giannaccini, Gino; R., Scatizzi; P., Domiano
CONFORMATIONALLY RESTRAINED BETA-BLOCKING OXIME ETHERS - SYNTHESIS AND BETA-ADRENERGIC PROPERTIES OF DIASTEREOISOMERIC ANTI AND SYN 2-(5'-ISOXAZOLIDINYL)-ETHANOLAMINES
1992-01-01 Balsamo, A; Breschi, Mc; Chini, M; Domiano, P; Giannaccini, Gino; Lucacchini, Antonio; Macchia, B; Macchia, Marco; Manera, Clementina; Martinelli, A; Martini, Claudia; Martinotti, E; Nieri, Paola; Rossello, Armando
Conformational effects on the activity of drugs. 13. A revision of previously proposed models for the activation of alfa- and beta-adrenergic receptors
1992-01-01 Macchia, B; Balsamo, Aldo; Breschi, M. C.; Lapucci, A; Lucacchini, Antonio; Macchia, F; Manera, Clementina; Martinelli, A; Martinotti, E; Nencetti, S.
N-ALKYL-NOR-TROPINE ESTERS OF 2-PHENYL-CYCLOHEXENIC ACIDS AS NEW BRONCHODILATOR AGENTS - EFFECT OF STRUCTURAL AND CONFORMATIONAL MODIFICATIONS ON AFFINITY FOR MUSCARINIC RECEPTORS
1992-01-01 Turbanti, L; Cerbai, G; Garzelli, G; Renzetti, Ar; Criscuoli, M; Subissi, A; Bramanti, G; Martinelli, Adriano
Conformationally restrained β -blocking oxime ethers: synthesis and β -adrenergic properties of diastereoisomeric anti and syn 2-(5-isoxazolidinyl)ethanolamines
1992-01-01 A., Balsamo; Breschi, MARIA CRISTINA; M., Chini; P., Domiano; Giannaccini, Gino; Lucacchini, Antonio; B., Macchia; Macchia, Marco; Manera, Clementina; Martinelli, Adriano; Martini, Claudia; E., Martinotti; Nieri, Paola; Rossello, Armando
Conformationally Restrained Analogs of Sympathomimetic Catecholamines. Synthesis, Conformational Analysis, and Adrenergic Activity of Isochroman Derivatives
1993-01-01 Macchia, B; Balsamo, A; Breschi, MARIA CRISTINA; Chiellini, Grazia; Lapucci, Annalina; Macchia, Marco; Manera, Clementina; Martinelli, Adriano; Martini, Claudia; Scatizzi, R; UCCELLO BARRETTA, Gloria
Sintesi e proprietà alfa-adrenergiche di derivati cromanici, quali analoghi conformazionalmente ristretti dell’1-(2,5-dimetossifenil)-2-amminoetanolo
1994-01-01 B., Macchia; Chiellini, Grazia; Lapucci, Annalina; Manera, Clementina; Martinelli, Adriano; Nencetti, Susanna; R., Scatizzi
The [(Methyloxy)imino]methyl Moiety as a Bioisoster of Aryl. A Novel Class of Completely Aliphatic Beta-Adrenergic Receptor Antagonists
1994-01-01 Macchia, Bruno; Balsamo, Aldo; Breschi, MARIA CRISTINA; Chiellini, Grazia; Macchia, Marco; Martinelli, Adriano; Martini, Claudia; Nardini, C; Nencetti, Susanna; Rossello, Armando; Scatizzi, R.
Conformationally restrained analogs of sympathomimetic catecholamine. Synthesis and adrenergic activity of tetrahydrobenzocycloheptene derivatives
1994-01-01 Macchia, B; Breschi, MARIA CRISTINA; Gentili, D; Lapucci, Annalina; Macchia, Marco; Manera, Clementina; Martinelli, Adriano; Martinotti, E; Nencetti, Susanna; Nieri, Paola
AROMATIC SUBSTITUENT EFFECT ON THE STEREOSELECTIVITY OF THE ACID-INDUCED RING-OPENING OF 1,2-EPOXIDES DERIVED FROM 3,4-DIHYDRONAPHTHALENE - IMPORTANCE OF THE REACTIVE CONFORMATIONS FOR THE STEREOSELECTIVITY
1994-01-01 Chini, M; Crotti, Paolo; Minutolo, Filippo; Martinelli, Adriano; Micali, E.
SYNTHESIS, ANTIINFLAMMATORY ACTIVITY AND MOLECULAR-ORBITAL STUDIES OF A SERIES OF BENZYLIDENEAMINOXYPROPIONIC ACIDS SUBSTITUTED ON THE PHENYL RING
1994-01-01 Lapucci, Annalina; Macchia, Marco; Martinelli, Adriano; Nencetti, Susanna; Orlandini, Elisabetta; Rossello, Armando; Baldacci, M; Soldani, G; Mengozzi, G.
Conformationally restrained ß-blocking oxime ethers. 2. Synthesis and ß-adrenergic properties of diastereoisomeric anti and syn 2-(5’-(3’-aryl-substituted)isoxazolidinyl)-N-alkylethanolamines
1994-01-01 A., Balsamo; Breschi, MARIA CRISTINA; Chiellini, Grazia; Lucacchini, Antonio; Macchia, Marco; Martinelli, Adriano; Martini, Claudia; C., Nardini; Orlandini, Elisabetta; F., Romagnoli; Rossello, Armando
BIOISOSTERS OF THE DIPHOSPHATE GROUP IN ACTIVATED FORMS OF ANTIHERPES VIRUS AGENTS - A THEORETICAL-STUDY
1994-01-01 Macchia, Marco; Martinelli, Adriano; Parkin, A; Rossello, Armando
SYNTHESIS AND BETA-ADRENERGIC ACTIVITY OF NEW COMPLETELY ALIPHATIC 3-(METHYLENEAMINOXY)PROPANOLAMINE DERIVATIVES
1994-01-01 Balsamo, A; Gentili, D; Lapucci, Annalina; Macchia, Marco; Martinelli, Adriano; Orlandini, Elisabetta
CONFORMATIONALLY RESTRAINED ANALOGS OF SYMPATHOMIMETIC CATECHOLAMINES - SYNTHESIS AND ADRENERGIC ACTIVITY OF TETRAHYDROBENZOCYCLOHEPTENE DERIVATIVES
1994-01-01 Macchia, B; Breschi, MARIA CRISTINA; Gentili, D; Lapucci, Annalina; Macchia, Marco; Manera, Clementina; Martinelli, Adriano; Martinotti, E; Nencetti, Susanna; Nieri, Paola
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Synthesis and antimicrobial properties of substituted 3-aminoxy-(E)-2-methoxyiminopropionyl penicillins and cephalosporins | 1-gen-1990 | A., Balsamo; B., Macchia; Martinelli, Adriano; Orlandini, Elisabetta; F., Macchia; G., Broccali; P., Domiano; Rossello, Armando | |
Acidi benzilideneamminossipropionici sostituiti sul fenile. Sintesi e proprietà antiinfiammatorie. | 1-gen-1991 | A., Balsamo; Lapucci, Annalina; B., Macchia; Martinelli, Adriano; Nencetti, Susanna; Orlandini, Elisabetta; Rossello, Armando; Soldani, G. M. e. n. g. o. z. z. i. G.; M., Baldacci | |
1-benzilossiimmino-3- ammino-2-propanoli: sintesi e proprietà ß-adrenergiche | 1-gen-1991 | Balsamo, A; Macchia, B; Macchia, Marco; Martinelli, Adriano; Rossello, Armando; Breschi, MARIA CRISTINA; Nieri, Paola; Scatizzi, R. | |
Conformational effects on the activity of drugs. 13. A revision of previously proposed models for the activation of a- and ß-adrenergic receptors | 1-gen-1992 | Macchia, B; Balsamo, A; Breschi, MARIA CRISTINA; Lapucci, Annalina; Lucacchini, Antonio; Macchia, F; Manera, Clementina; Martinelli, Adriano; Martini, Claudia; Martinotti, E; Nencetti, Susanna | |
CONFORMATIONAL EFFECTS ON THE ACTIVITY OF DRUGS .13. A REVISION OF PREVIOUSLY PROPOSED MODELS FOR THE ACTIVATION OF ALPHA-ADRENERGIC AND BETA-ADRENERGIC RECEPTORS | 1-gen-1992 | Macchia, Bruno; Balsamo, A; Breschi, MARIA CRISTINA; Lapucci, Annalina; Lucacchini, Antonio; Macchia, F; Manera, Clementina; Martinelli, Adriano; Martini, Claudia; Martinotti, E; Nencetti, Susanna | |
X-Ray analysis, theoretical studies and alfa-adrenergic biopharmacological properties of 1-(2,5-dimethoxyphenyl)-2-aminoethanol and its morpholine analogue. | 1-gen-1992 | Manera, Clementina; Martinelli, Adriano; Nencetti, Susanna; Rossello, Armando; Giannaccini, Gino; R., Scatizzi; P., Domiano | |
CONFORMATIONALLY RESTRAINED BETA-BLOCKING OXIME ETHERS - SYNTHESIS AND BETA-ADRENERGIC PROPERTIES OF DIASTEREOISOMERIC ANTI AND SYN 2-(5'-ISOXAZOLIDINYL)-ETHANOLAMINES | 1-gen-1992 | Balsamo, A; Breschi, Mc; Chini, M; Domiano, P; Giannaccini, Gino; Lucacchini, Antonio; Macchia, B; Macchia, Marco; Manera, Clementina; Martinelli, A; Martini, Claudia; Martinotti, E; Nieri, Paola; Rossello, Armando | |
Conformational effects on the activity of drugs. 13. A revision of previously proposed models for the activation of alfa- and beta-adrenergic receptors | 1-gen-1992 | Macchia, B; Balsamo, Aldo; Breschi, M. C.; Lapucci, A; Lucacchini, Antonio; Macchia, F; Manera, Clementina; Martinelli, A; Martinotti, E; Nencetti, S. | |
N-ALKYL-NOR-TROPINE ESTERS OF 2-PHENYL-CYCLOHEXENIC ACIDS AS NEW BRONCHODILATOR AGENTS - EFFECT OF STRUCTURAL AND CONFORMATIONAL MODIFICATIONS ON AFFINITY FOR MUSCARINIC RECEPTORS | 1-gen-1992 | Turbanti, L; Cerbai, G; Garzelli, G; Renzetti, Ar; Criscuoli, M; Subissi, A; Bramanti, G; Martinelli, Adriano | |
Conformationally restrained β -blocking oxime ethers: synthesis and β -adrenergic properties of diastereoisomeric anti and syn 2-(5-isoxazolidinyl)ethanolamines | 1-gen-1992 | A., Balsamo; Breschi, MARIA CRISTINA; M., Chini; P., Domiano; Giannaccini, Gino; Lucacchini, Antonio; B., Macchia; Macchia, Marco; Manera, Clementina; Martinelli, Adriano; Martini, Claudia; E., Martinotti; Nieri, Paola; Rossello, Armando | |
Conformationally Restrained Analogs of Sympathomimetic Catecholamines. Synthesis, Conformational Analysis, and Adrenergic Activity of Isochroman Derivatives | 1-gen-1993 | Macchia, B; Balsamo, A; Breschi, MARIA CRISTINA; Chiellini, Grazia; Lapucci, Annalina; Macchia, Marco; Manera, Clementina; Martinelli, Adriano; Martini, Claudia; Scatizzi, R; UCCELLO BARRETTA, Gloria | |
Sintesi e proprietà alfa-adrenergiche di derivati cromanici, quali analoghi conformazionalmente ristretti dell’1-(2,5-dimetossifenil)-2-amminoetanolo | 1-gen-1994 | B., Macchia; Chiellini, Grazia; Lapucci, Annalina; Manera, Clementina; Martinelli, Adriano; Nencetti, Susanna; R., Scatizzi | |
The [(Methyloxy)imino]methyl Moiety as a Bioisoster of Aryl. A Novel Class of Completely Aliphatic Beta-Adrenergic Receptor Antagonists | 1-gen-1994 | Macchia, Bruno; Balsamo, Aldo; Breschi, MARIA CRISTINA; Chiellini, Grazia; Macchia, Marco; Martinelli, Adriano; Martini, Claudia; Nardini, C; Nencetti, Susanna; Rossello, Armando; Scatizzi, R. | |
Conformationally restrained analogs of sympathomimetic catecholamine. Synthesis and adrenergic activity of tetrahydrobenzocycloheptene derivatives | 1-gen-1994 | Macchia, B; Breschi, MARIA CRISTINA; Gentili, D; Lapucci, Annalina; Macchia, Marco; Manera, Clementina; Martinelli, Adriano; Martinotti, E; Nencetti, Susanna; Nieri, Paola | |
AROMATIC SUBSTITUENT EFFECT ON THE STEREOSELECTIVITY OF THE ACID-INDUCED RING-OPENING OF 1,2-EPOXIDES DERIVED FROM 3,4-DIHYDRONAPHTHALENE - IMPORTANCE OF THE REACTIVE CONFORMATIONS FOR THE STEREOSELECTIVITY | 1-gen-1994 | Chini, M; Crotti, Paolo; Minutolo, Filippo; Martinelli, Adriano; Micali, E. | |
SYNTHESIS, ANTIINFLAMMATORY ACTIVITY AND MOLECULAR-ORBITAL STUDIES OF A SERIES OF BENZYLIDENEAMINOXYPROPIONIC ACIDS SUBSTITUTED ON THE PHENYL RING | 1-gen-1994 | Lapucci, Annalina; Macchia, Marco; Martinelli, Adriano; Nencetti, Susanna; Orlandini, Elisabetta; Rossello, Armando; Baldacci, M; Soldani, G; Mengozzi, G. | |
Conformationally restrained ß-blocking oxime ethers. 2. Synthesis and ß-adrenergic properties of diastereoisomeric anti and syn 2-(5’-(3’-aryl-substituted)isoxazolidinyl)-N-alkylethanolamines | 1-gen-1994 | A., Balsamo; Breschi, MARIA CRISTINA; Chiellini, Grazia; Lucacchini, Antonio; Macchia, Marco; Martinelli, Adriano; Martini, Claudia; C., Nardini; Orlandini, Elisabetta; F., Romagnoli; Rossello, Armando | |
BIOISOSTERS OF THE DIPHOSPHATE GROUP IN ACTIVATED FORMS OF ANTIHERPES VIRUS AGENTS - A THEORETICAL-STUDY | 1-gen-1994 | Macchia, Marco; Martinelli, Adriano; Parkin, A; Rossello, Armando | |
SYNTHESIS AND BETA-ADRENERGIC ACTIVITY OF NEW COMPLETELY ALIPHATIC 3-(METHYLENEAMINOXY)PROPANOLAMINE DERIVATIVES | 1-gen-1994 | Balsamo, A; Gentili, D; Lapucci, Annalina; Macchia, Marco; Martinelli, Adriano; Orlandini, Elisabetta | |
CONFORMATIONALLY RESTRAINED ANALOGS OF SYMPATHOMIMETIC CATECHOLAMINES - SYNTHESIS AND ADRENERGIC ACTIVITY OF TETRAHYDROBENZOCYCLOHEPTENE DERIVATIVES | 1-gen-1994 | Macchia, B; Breschi, MARIA CRISTINA; Gentili, D; Lapucci, Annalina; Macchia, Marco; Manera, Clementina; Martinelli, Adriano; Martinotti, E; Nencetti, Susanna; Nieri, Paola |
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