Sfoglia per Autore
SYNTHESIS AND ANTIMICROBIAL ACTIVITY OF 7-BETA-[N-(ARYLMETHYLOXYIMINO) ACETAMIDO]CEPHALOSPORANIC ACID-DERIVATIVES
1995-01-01 Macchia, Marco; Menchini, E; Orlandini, Elisabetta; Rossello, Armando; Broccali, G; Visconti, M.
Synthesis and adrenergic beta-blocking activity of ortho-, meta- and para-oxypropanolamino-substituted [(benzylideneamino)oxy]propanolamines.
1995-01-01 A., Balsamo; Lapucci, Annalina; B., Macchia; Macchia, Marco; Orlandini, Elisabetta; G., Ferni; M., Pinza; Rossello, Armando
(E)-(ARYLMETHYLENEAMINOXY)ACETAMIDES AS ANALOGS OF NEUROLEPTIC BENZAMIDES - SYNTHESIS AND D-2-DOPAMINERGIC BINDING-AFFINITY
1995-01-01 Macchia, Marco; Manera, Clementina; Martinelli, Adriano; Orlandini, Elisabetta; Romagnoli, F; Rossello, Armando; Chiellini, Grazia
Role of the benzylic hydroxyl group of adrenergic catecholamines in eliciting a-adrenergic activity. Synthesis and a1- and a2-adrenergic activity of 3-phenyl-3-piperidinols and of their desoxy analogs
1995-01-01 B., Macchia; Macchia, Marco; Manera, Clementina; E., Martinotti; Nencetti, Susanna; Orlandini, Elisabetta; R., Scatizzi; Rossello, Armando
SYNTHESIS AND BETA-ADRENERGIC ACTIVITY OF A SERIES OF 3-(SUBSTITUTED-BENZYLIDENEAMINOXY)PROPANOLAMINE DERIVATIVES
1995-01-01 Gentili, D; Lapucci, Annalina; Macchia, B; Macchia, Marco; Martinelli, Adriano; Nencetti, Susanna; Orlandini, Elisabetta; Ferni, G; Pinza, M.
Sintesi e proprietà beta-adrenergiche di [(benzilideneammino)ossi] propanolammine orto-ossipropanolammine sostituite chirali,
1996-01-01 Lapucci, Annalina; Macchia, Marco; Orlandini, Elisabetta; Nencetti, Susanna; Chiellini, Grazia; Nieri, Paola
Synthesis and aldose reductase inhibitory activity of some N-(aroyl)-N-(arylalkyloxy)-glycines and -beta-alanines
1996-01-01 Macchia, Marco; Menchini, E; Nencetti, Susanna; Orlandini, Elisabetta; Rossello, Armando
Synthesis and antimicrobial activity of 7ß-(S) and 7ß-(R)-3-(methyleneaminoxy)-2-methylpropionamido substituted cephalosporanic acid derivatives
1996-01-01 Macchia, Marco; E., Menchini; Orlandini, Elisabetta; G., Broccali; M., Visconti; Rossello, Armando
(E)-(methyloxyimino)acetamides as analogues of neuroleptic benzamides: Synthesis and D-2-dopaminergic binding affinity
1996-01-01 Lapucci, Annalina; Macchia, Marco; Orlandini, Elisabetta; Romagnoli, F; Rossello, Armando; Chiellini, Grazia; Cozzini, P; Domiano, P.
Conformational effects on the activity of drugs .19. Synthesis and alpha-adrenergic activity of 2- and 6-methyl-substituted (3,4-dihydroxyphenyl)-3-piperidinols
1997-01-01 Macchia, B; Macchia, Marco; Martinelli, Adriano; Martinotti, E; Orlandini, Elisabetta; Romagnoli, F; Scatizzi, R.
Effects on the antimicrobial properties of structural modifications on the C(7)-amidic side chain of cephalosporins
1997-01-01 Macchia, Marco; E., Menchini; Nencetti, Susanna; Orlandini, Elisabetta; Rossello, Armando; G:, Broccali; D:, Limonta
New beta-lactam monocyclic inhibitors of human elastases: synthesis and anti-elastase properties of 1-carbamoyl-4-methyleneaminoxyazetidinone derivatives
1997-01-01 Balsamo, A; Asti, C; BELFIORE M., S; Brandolini, L; Cercignani, G; Gentili, D.; Macchia, Marco; Mantovanini, M; Orlandini, Elisabetta; Rossello, Armando
Synthesis and aldose reductase inhibitory activity of new N-(benzyloxy) glycine derivatives
1998-01-01 Macchia, Marco; Barontini, S; Martinelli, Adriano; Menchini, E; Nencetti, Susanna; Orlandini, Elisabetta; Romagnoli, F.
Synthesis and alpha-adrenergic and I-1-imidazoline activity of 3-phenylpiperidines dimethyl-substituted on the phenyl ring
1998-01-01 B., Macchia; D. B., Bylund; Calderone, Vincenzo; Giannaccini, Gino; Lucacchini, Antonio; Macchia, Marco; Martinelli, Adriano; E., Martinotti; Orlandini, Elisabetta; F., Romagnoli; Rossello, Armando
N-n-propyl-substituted 3-(dimethylphenyl)piperidines display novel discriminative properties between dopamine receptor subtypes: synthesis and receptor binding studies
1998-01-01 Cervetto, L.; Demontis, GIAN CARLO ALFREDO GIUSEPPE; Giannaccini, Gino; Longoni, Biancamaria; Macchia, B.; Macchia, Marco; Martinelli, A.; Orlandini, Elisabetta
Synthesis And Antimicrobial Property Of Cephalosporin Derivatives Substituted On The C(7) Nitrogen With Arylmethyloxyimino Or Arylmethyloxyamino Alkanoyl Groups
1999-01-01 Gentili, D.; Macchia, Marco; E., Menchini; Nencetti, Susanna; Orlandini, Elisabetta; Rossello, Armando; G., Broccali; D., Limonta
Synthesis and prostaglandin synthase inhibitory activity of new aromatic O-alkyloxime ethers substituted with methylsulfonamidic and methylsulfonyl groups on their aliphatic portion
2000-01-01 A., Balsamo; Orlandini, Elisabetta; Rapposelli, Simona; M., Pinza; C., Milanese; F., Mancini
Synthesis and antiviral properties of 9-[(2-methyleneaminoxyethoxy)methyl]guanine derivatives as novel acyclovir analogues
2000-01-01 Macchia, Marco; G., Antonelli; F., Calvani; DI BUSSOLO, Valeria; Minutolo, Filippo; Orlandini, Elisabetta; R., Tesoro; O., Turriziani
Synthesis, Inhibitory Activity Towards Human Leukocyte Elastase and Molecular Modelling Studies of Carbamoyl-4-methyleneaminoxyazetidinones
2000-01-01 B., Macchia; D., Gentili; Macchia, Marco; F., Mamone; Martinelli, Adriano; Orlandini, Elisabetta; Rossello, Armando; G., Cercignani; R., Pierotti; M., Allegretti; C., Asti; G., Caselli
Enantiopure 3-(arylmethylidene)aminoxy-2-methylpropionic acids: synthesis and antiinflammatory properties
2001-01-01 Aldo, Balsamo; Simone, Bertini; Giambattista, Gervasi; Lapucci, Annalina; Nencetti, Susanna; Orlandini, Elisabetta; Rapposelli, Simona; Rossello, Armando; Giulio, Soldani
Titolo | Data di pubblicazione | Autore(i) | File |
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SYNTHESIS AND ANTIMICROBIAL ACTIVITY OF 7-BETA-[N-(ARYLMETHYLOXYIMINO) ACETAMIDO]CEPHALOSPORANIC ACID-DERIVATIVES | 1-gen-1995 | Macchia, Marco; Menchini, E; Orlandini, Elisabetta; Rossello, Armando; Broccali, G; Visconti, M. | |
Synthesis and adrenergic beta-blocking activity of ortho-, meta- and para-oxypropanolamino-substituted [(benzylideneamino)oxy]propanolamines. | 1-gen-1995 | A., Balsamo; Lapucci, Annalina; B., Macchia; Macchia, Marco; Orlandini, Elisabetta; G., Ferni; M., Pinza; Rossello, Armando | |
(E)-(ARYLMETHYLENEAMINOXY)ACETAMIDES AS ANALOGS OF NEUROLEPTIC BENZAMIDES - SYNTHESIS AND D-2-DOPAMINERGIC BINDING-AFFINITY | 1-gen-1995 | Macchia, Marco; Manera, Clementina; Martinelli, Adriano; Orlandini, Elisabetta; Romagnoli, F; Rossello, Armando; Chiellini, Grazia | |
Role of the benzylic hydroxyl group of adrenergic catecholamines in eliciting a-adrenergic activity. Synthesis and a1- and a2-adrenergic activity of 3-phenyl-3-piperidinols and of their desoxy analogs | 1-gen-1995 | B., Macchia; Macchia, Marco; Manera, Clementina; E., Martinotti; Nencetti, Susanna; Orlandini, Elisabetta; R., Scatizzi; Rossello, Armando | |
SYNTHESIS AND BETA-ADRENERGIC ACTIVITY OF A SERIES OF 3-(SUBSTITUTED-BENZYLIDENEAMINOXY)PROPANOLAMINE DERIVATIVES | 1-gen-1995 | Gentili, D; Lapucci, Annalina; Macchia, B; Macchia, Marco; Martinelli, Adriano; Nencetti, Susanna; Orlandini, Elisabetta; Ferni, G; Pinza, M. | |
Sintesi e proprietà beta-adrenergiche di [(benzilideneammino)ossi] propanolammine orto-ossipropanolammine sostituite chirali, | 1-gen-1996 | Lapucci, Annalina; Macchia, Marco; Orlandini, Elisabetta; Nencetti, Susanna; Chiellini, Grazia; Nieri, Paola | |
Synthesis and aldose reductase inhibitory activity of some N-(aroyl)-N-(arylalkyloxy)-glycines and -beta-alanines | 1-gen-1996 | Macchia, Marco; Menchini, E; Nencetti, Susanna; Orlandini, Elisabetta; Rossello, Armando | |
Synthesis and antimicrobial activity of 7ß-(S) and 7ß-(R)-3-(methyleneaminoxy)-2-methylpropionamido substituted cephalosporanic acid derivatives | 1-gen-1996 | Macchia, Marco; E., Menchini; Orlandini, Elisabetta; G., Broccali; M., Visconti; Rossello, Armando | |
(E)-(methyloxyimino)acetamides as analogues of neuroleptic benzamides: Synthesis and D-2-dopaminergic binding affinity | 1-gen-1996 | Lapucci, Annalina; Macchia, Marco; Orlandini, Elisabetta; Romagnoli, F; Rossello, Armando; Chiellini, Grazia; Cozzini, P; Domiano, P. | |
Conformational effects on the activity of drugs .19. Synthesis and alpha-adrenergic activity of 2- and 6-methyl-substituted (3,4-dihydroxyphenyl)-3-piperidinols | 1-gen-1997 | Macchia, B; Macchia, Marco; Martinelli, Adriano; Martinotti, E; Orlandini, Elisabetta; Romagnoli, F; Scatizzi, R. | |
Effects on the antimicrobial properties of structural modifications on the C(7)-amidic side chain of cephalosporins | 1-gen-1997 | Macchia, Marco; E., Menchini; Nencetti, Susanna; Orlandini, Elisabetta; Rossello, Armando; G:, Broccali; D:, Limonta | |
New beta-lactam monocyclic inhibitors of human elastases: synthesis and anti-elastase properties of 1-carbamoyl-4-methyleneaminoxyazetidinone derivatives | 1-gen-1997 | Balsamo, A; Asti, C; BELFIORE M., S; Brandolini, L; Cercignani, G; Gentili, D.; Macchia, Marco; Mantovanini, M; Orlandini, Elisabetta; Rossello, Armando | |
Synthesis and aldose reductase inhibitory activity of new N-(benzyloxy) glycine derivatives | 1-gen-1998 | Macchia, Marco; Barontini, S; Martinelli, Adriano; Menchini, E; Nencetti, Susanna; Orlandini, Elisabetta; Romagnoli, F. | |
Synthesis and alpha-adrenergic and I-1-imidazoline activity of 3-phenylpiperidines dimethyl-substituted on the phenyl ring | 1-gen-1998 | B., Macchia; D. B., Bylund; Calderone, Vincenzo; Giannaccini, Gino; Lucacchini, Antonio; Macchia, Marco; Martinelli, Adriano; E., Martinotti; Orlandini, Elisabetta; F., Romagnoli; Rossello, Armando | |
N-n-propyl-substituted 3-(dimethylphenyl)piperidines display novel discriminative properties between dopamine receptor subtypes: synthesis and receptor binding studies | 1-gen-1998 | Cervetto, L.; Demontis, GIAN CARLO ALFREDO GIUSEPPE; Giannaccini, Gino; Longoni, Biancamaria; Macchia, B.; Macchia, Marco; Martinelli, A.; Orlandini, Elisabetta | |
Synthesis And Antimicrobial Property Of Cephalosporin Derivatives Substituted On The C(7) Nitrogen With Arylmethyloxyimino Or Arylmethyloxyamino Alkanoyl Groups | 1-gen-1999 | Gentili, D.; Macchia, Marco; E., Menchini; Nencetti, Susanna; Orlandini, Elisabetta; Rossello, Armando; G., Broccali; D., Limonta | |
Synthesis and prostaglandin synthase inhibitory activity of new aromatic O-alkyloxime ethers substituted with methylsulfonamidic and methylsulfonyl groups on their aliphatic portion | 1-gen-2000 | A., Balsamo; Orlandini, Elisabetta; Rapposelli, Simona; M., Pinza; C., Milanese; F., Mancini | |
Synthesis and antiviral properties of 9-[(2-methyleneaminoxyethoxy)methyl]guanine derivatives as novel acyclovir analogues | 1-gen-2000 | Macchia, Marco; G., Antonelli; F., Calvani; DI BUSSOLO, Valeria; Minutolo, Filippo; Orlandini, Elisabetta; R., Tesoro; O., Turriziani | |
Synthesis, Inhibitory Activity Towards Human Leukocyte Elastase and Molecular Modelling Studies of Carbamoyl-4-methyleneaminoxyazetidinones | 1-gen-2000 | B., Macchia; D., Gentili; Macchia, Marco; F., Mamone; Martinelli, Adriano; Orlandini, Elisabetta; Rossello, Armando; G., Cercignani; R., Pierotti; M., Allegretti; C., Asti; G., Caselli | |
Enantiopure 3-(arylmethylidene)aminoxy-2-methylpropionic acids: synthesis and antiinflammatory properties | 1-gen-2001 | Aldo, Balsamo; Simone, Bertini; Giambattista, Gervasi; Lapucci, Annalina; Nencetti, Susanna; Orlandini, Elisabetta; Rapposelli, Simona; Rossello, Armando; Giulio, Soldani |
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