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CONFORMATIONALLY RESTRAINED ANALOGS OF SYMPATHOMIMETIC CATECHOLAMINES - SYNTHESIS AND ADRENERGIC ACTIVITY OF TETRAHYDROBENZOCYCLOHEPTENE DERIVATIVES 1-gen-1994 Macchia, B; Breschi, MARIA CRISTINA; Gentili, D; Lapucci, Annalina; Macchia, Marco; Manera, Clementina; Martinelli, Adriano; Martinotti, E; Nencetti, Susanna; Nieri, Paola
X-ray analisis, theoretical studies and a-adrenergic biopharmacological properties of 1-(2,5-dimethoxyphenyl)-2-aminoethanol and its morpholine analogue 1-gen-1994 Manera, Clementina; Martinelli, Adriano; Nencetti, Susanna; F., Romagnoli; Rossello, Armando; Giannaccini, Gino; R., Scatizzi; P., Cozzini; P., Domiano
(E)-(ARYLMETHYLENEAMINOXY)ACETAMIDES AS ANALOGS OF NEUROLEPTIC BENZAMIDES - SYNTHESIS AND D-2-DOPAMINERGIC BINDING-AFFINITY 1-gen-1995 Macchia, Marco; Manera, Clementina; Martinelli, Adriano; Orlandini, Elisabetta; Romagnoli, F; Rossello, Armando; Chiellini, Grazia
Role of the benzylic hydroxyl group of adrenergic catecholamines in eliciting a-adrenergic activity. Synthesis and a1- and a2-adrenergic activity of 3-phenyl-3-piperidinols and of their desoxy analogs 1-gen-1995 B., Macchia; Macchia, Marco; Manera, Clementina; E., Martinotti; Nencetti, Susanna; Orlandini, Elisabetta; R., Scatizzi; Rossello, Armando
Role of the benzylic hydroxyl group of adrenergic cattecholamines in eliciting alpha-adrenergic activity. Synthesis and alpha1- and alpha2-adrenergic activity of 3-phenyl-3-piperidinols and of their desoxy analogs 1-gen-1995 Macchia, Bruno; Macchia, Marco; Manera, Clementina; Martinotti, E.
Conformationally restrained beta-blocking oxime ethers. 3. Synthesis and beta-adrenergic antagonistic activity of diastereomeric anti and syn 2-(5’-(3’-methyl)isoxazolidinyl)-N-alkylethanolamines”. 1-gen-1996 Breschi, MARIA CRISTINA; Macchia, Marco; Manera, Clementina; E., Micali; C., Nardini; Nencetti, Susanna; Rossello, Armando; R., Scatizzi
Chiral 2-(3'-(5'-p-chlorophenyl)isoxazolidinyl)ethanolamines as conformationally restrained analogs of methyloxyiminomethyl (MOIM) beta-adrenergic antagonists: Synthesis, configuration and beta-adrenergic properties 1-gen-1996 Balsamo, A; Breschi, MARIA CRISTINA; Chiellini, Grazia; Cozzini, P; Domiano, P; Macchia, Marco; Manera, Clementina; Martinelli, Adriano; Nencetti, Susanna; Rossello, Armando; Sacca, P; Scatizzi, R.
Synthesis and antimicrobial activity of benzo[a]dihydrocarbazole and benzotetrahydrocyclohept[1,2-b]indole derivatives 1-gen-1996 Macchia, Marco; Manera, Clementina; Nencetti, Susanna; Rossello, Armando; Broccali, G; Limonta, D.
Stereochemistry and dynamics of the hydrobromide of 1-(aminomethyl)-5,6-dihydroxyisochroman, semirigid analogue of catecholamines 1-gen-1996 DI BARI, Lorenzo; UCCELLO BARRETTA, Gloria; Manera, Clementina
1,2,3-triazolo [4,5-d] pyridazines-V. Preparation and adenosine receptor binding of new 4-amino derivatives. 1-gen-1996 Biagi, G; Giorgi, Irene; Livi, O; Scartoni, V; Manera, Clementina; Lucacchini, Antonio; Senatore, G.
Conformationally restrained β -blocking oxime ethers. 4. Chiral 2-(3'-(5'-p-chlorophenyl)isoxazolidinyl)ethanolamines as conformationally restrained analogs of methyloxyiminomethyl (MOIM) β -adrenergic antagonists: synthesis, configuration and β -adrenergic properties 1-gen-1996 Balsamo, Aldo; Breschi, M. C.; Chiellini, G; Cozzini, P; Domiano, P; Macchia, Marco; Manera, Clementina; Martinelli, A; Nencetti, S.
New chiral methyloxyiminomethyl(MOIM) beta-adrenergic antagonists. (S)- and (R)-N-[3-(alkylamino)-2-hydroxypropylidene](p-chlorophenylmethyloxy)amines as probes for determining enantiomeric specificity in the class of MOIM-type beta-adrenergic blocking agents 1-gen-1996 Balsamo, A; Breschi, MARIA CRISTINA; Chiellini, Grazia; Macchia, B; Macchia, Marco; Manera, Clementina; Sacca, P; Scatizzi, R.
Stereoselective synthesis and beta-blocking activity of substituted (E)- and (Z)-4(1H)-[1-(3-alkylamino-2-hydroxypropyl)oximino]-2,3-dihydro-1,8-naphthyridine. Potential antihypertensive” agents. Part VI 1-gen-1997 P. L., Ferrarini; C., Mori; M., Badawneh; Manera, Clementina; Martinelli, Adriano; M., Miceli; F., Romagnoli; Saccomanni, Giuseppe
Unusual nitration of substituted 7-amino-1,8-naphthyridine in the synthesis of compounds with antiplatelet activity 1-gen-1997 Ferrarini, Pl; Mori, C; Badawneh, M; Manera, Clementina; Clementina, M; Martinelli, Adriano; Miceli, M; Romagnoli, F; Saccomanni, Giuseppe
Synthesis of New 1,2,3-triazolo[1,2-a]benzotriazole derivatives or substituted 2,3-benzo-1,3a,6,6a-tetraazapentalenes. II” 1-gen-1997 G., Biagi; Giorgi, Irene; O., Livi; Manera, Clementina; V., Scartoni; P. L., Barili
1,2,3-Triazolo[4,5-d]-1,2,4-triazolo[4,3-b]pyridazines 1-gen-1997 Biagi, G; Giorgi, Irene; Livi, O; Manera, Clementina; Scartoni, V.
Stereoselective synthesis and beta-blocking activity of substituted (E)- and (Z)- 4(1H) - [1- (3 - alkylamino - 2 - hydroxypropyl) oximino - 2,3 - dihydro - 1,8 - naphthyridine. Potential antihypertensive agents. Part VI 1-gen-1997 Ferrarini, Pl; Mori, C; Badawneh, M; Manera, Clementina; Saccomanni, Giuseppe; Calderone, Vincenzo; Scatizzi, R; Barili, Pl
Derivati 1,8-naftiridinici con affinità verso i recettori A1 e A2A dell’adenosina. 1-gen-1998 Ferrarini, P. L.; Manera, Clementina; Martinelli, Adriano; Mori, C.; Betti, Laura; Giannaccini, Gino; Lucacchini, Antonio
Novel 3-aralkyl-7-(amino-substituted)-1,2,3-triazolo[4,5-d]pyramidines with high affinity toward A(1) adenosine receptors 1-gen-1998 Betti, Laura; Biagi, G.; Giannaccini, Gino; Giorgi, Irene; Livi, O.; Lucacchini, Antonio; Manera, Clementina; Scartoni, V.
1,2,3-Triazolo[1,5-a]quinoxalines: synthesis and binding to benzodiazepine and adenosine receptors 1-gen-1998 Bertelli, L; Biagi, G; Giorgi, Irene; Manera, Clementina; Livi, O; Scartoni, V; Betti, Laura; Giannaccini, Gino; Trincavelli, MARIA LETIZIA; Barili, Pl
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