MACCHIA, MARCO Statistiche
MACCHIA, MARCO
DIPARTIMENTO DI FARMACIA
"Soft Drugs" Based on Cannabinoid Receptor Ligands as Potential Local Analgesic and Antiglaucoma Agents
2007-01-01 Minutolo, Filippo; CASCIO M., G; Carboni, I; Bisogno, T; Prota, G; Bertini, Simone; Digiacomo, Maria; Bifulco, M; DI MARZO, V; Macchia, Marco
(E)-(ARYLMETHYLENEAMINOXY)ACETAMIDES AS ANALOGS OF NEUROLEPTIC BENZAMIDES - SYNTHESIS AND D-2-DOPAMINERGIC BINDING-AFFINITY
1995-01-01 Macchia, Marco; Manera, Clementina; Martinelli, Adriano; Orlandini, Elisabetta; Romagnoli, F; Rossello, Armando; Chiellini, Grazia
(E)-(methyloxyimino)acetamides as analogues of neuroleptic benzamides: Synthesis and D-2-dopaminergic binding affinity
1996-01-01 Lapucci, Annalina; Macchia, Marco; Orlandini, Elisabetta; Romagnoli, F; Rossello, Armando; Chiellini, Grazia; Cozzini, P; Domiano, P.
(Z)-(Methyloxyiminomethyl)ethanolamines. Effects of the configuration around the iminic double bond on the beta-adrenergic affinity of moim-type beta-adrenergic blocking agents
1995-01-01 Chiellini, Grazia; Lapucci, Annalina; Macchia, Marco; F., Romagnoli; Rossello, Armando; Nencetti, Susanna
1,2-Dihydro-2-oxopyridine-3-carboxamides: the C-5 substituent is responsible for functionality switch at CB2 cannabinoid receptor
2014-01-01 Valentina, Lucchesi; Teija, Parkkari; Juha R., Savinainen; Anna Maria, Malfitano; Marco, Allarà; Bertini, Simone; Francesca, Castelli; Sara Del, Carlo; Chiara, Laezza; Alessia, Ligresti; Saccomanni, Giuseppe; Maurizio, Bifulco; Vincenzo Di, Marzo; Macchia, Marco; Manera, Clementina
1-benzilossiimmino-3- ammino-2-propanoli: sintesi e proprietà ß-adrenergiche
1991-01-01 Balsamo, A; Macchia, B; Macchia, Marco; Martinelli, Adriano; Rossello, Armando; Breschi, MARIA CRISTINA; Nieri, Paola; Scatizzi, R.
18FLUORINE-LABELED NITROGEN HETEROCYCLIC DERIVATIVES AS NEW CANDIDATE FOR CANNABINOID CB2 RECEPTOR PET IMAGING
2011-01-01 Castelli, Francesca; Bertini, Simone; DEL CARLO, Sara; Lucchesi, Valentina; Manera, Clementina; Pascali, Giancarlo; Saccomanni, Giuseppe; DI MARZO, Vincenzo; Salvadori, Piero; Macchia, Marco
2-(Methyleneaminoxy)methylmorpholine derivatives. Synthesis and antidepressant activity
1994-01-01 A., Balsamo; Lapucci, Annalina; Macchia, Marco; Martinelli, Adriano; Nencetti, Susanna; T., Cristina; Rossello, Armando
3-(Methyleneaminoxy)methylpiperidine derivatives as uptake inhibitors of biogenic amines in the brain synaptosomal fraction
1994-01-01 Balsamo, A; Lapucci, Annalina; Lucacchini, Antonio; Macchia, Marco; Martini, Claudia; Nardini, C; Nencetti, Susanna
3-(METHYLENEAMINOXY)METHYLPIPERIDINE DERIVATIVES AS UPTAKE INHIBITORS OF BIOGENIC-AMINES IN THE BRAIN SYNAPTOSOMAL FRACTION
1994-01-01 Balsamo, A; Lapucci, Annalina; Lucacchini, Antonio; Macchia, Marco; Martini, Claudia; Nardini, C; Nencetti, Susanna
4-[6-(dansylamino)hexylamino]-7-methyl-2-phenyl-1,8-naphthyridine as a new potential fluorescent probe for studying A1-adenosine receptor
2002-01-01 Macchia, Marco; Bertini, Simone; DI BUSSOLO, Valeria; Manera, Clementina; Martini, Claudia; Minutolo, Filippo; C., Mori; Saccomanni, Giuseppe; D., Tuscano; Ferrarini, P.
4-Aryliden-2-methyloxazol-5(4H)-one as a new scaffold for selective reversible MAGL inhibitors
2016-01-01 Granchi, Carlotta; Rizzolio, F; Bordoni, Vittorio; Caligiuri, I; Manera, Clementina; Macchia, Marco; Minutolo, Filippo; Martinelli, Adriano; Giordano, A; Tuccinardi, Tiziano
7-Nitrobenzofurazan (NBD)-Derivatives Of 5'-N-Ethylcarboxamidoadenosine (NECA) As New Fluorescent Probes For Human A3 Adenosine Receptors
2001-01-01 Macchia, Marco; Salvetti, F; Bertini, Simone; DI BUSSOLO, Valeria; Gattuso, L; Gesi, Marco; Hamdan, M; KLOTZ K., N; Laragione, T; Lucacchini, Antonio; Minutolo, Filippo; Nencetti, Susanna; Papi, C; Tuscano, D; Martini, Claudia
A new D2 dopamine receptor agonist allosterically modulates A2A adenosine receptor signalling by interacting with the A2A/D2 receptor heteromer
2012-01-01 Trincavelli, MARIA LETIZIA; Daniele, Simona; Orlandini, Elisabetta; Navarro, G.; Casado, V.; Giacomelli, Chiara; Nencetti, Susanna; Nuti, Elisa; Macchia, Marco; Huebner, H.; Gmeiner, P.; Rossello, Armando; Lluis, C.; Martini, Claudia
A new small molecule, D2 dopamine receptor agonist, as an allosteric modulator of A2A adenosine receptor signalling
2010-01-01 Trincavelli, MARIA LETIZIA; Orlandini, Elisabetta; Daniele, Simona; Nencetti, Susanna; Nuti, Elisa; Macchia, Marco; Huebner, H; Gmeiner, P; Rossello, Armando; Martini, Claudia
A new small molecule, D2 dopamine receptor agonist, as an allosteric modulator of A2A adenosine receptor signalling
2010-01-01 Trincavelli, MARIA LETIZIA; Orlandini, Elisabetta; Daniele, Simona; Nencetti, Susanna; Nuti, Elisa; Macchia, Marco; Huebner, H; Gmeiner, P; Rossello, Armando; Martini, Claudia
A Proteomic Approach to Uncover Neuroprotective Mechanisms of Oleocanthal against Oxidative Stress
2018-01-01 Giusti, Laura; Angeloni, Cristina; Barbalace, Maria Cristina; Lacerenza, Serena; Ciregia, Federica; Ronci, Maurizio; Urbani, Andrea; Manera, Clementina; Digiacomo, Maria; Macchia, Marco; Mazzoni, Maria Rosa; Lucacchini, Antonio; Hrelia, Silvana
A structure-activity study of a C-terminal endothelin analogue
1998-01-01 Cassano, E; Galoppini, C; Giusti, Laura; Hamdan, M; Macchia, Marco; Mazzoni, MARIA ROSA; Menchini, E; Pegoraro, S; Rovero, P.
A Virtual Screening Study for Lactate Dehydrogenase 5 Inhibitors by using a Pharmacophore-Based Approach
2016-01-01 Tuccinardi, Tiziano; Poli, Giulio; Corchia, Isacco; Granchi, Carlotta; Lapillo, Margherita; Macchia, Marco; Minutolo, Filippo; Ortore, GABRIELLA MARIA PIA; Martinelli, Adriano
A(1) adenosine receptors in human neutrophils: Direct binding and electron microscope visualization
1999-01-01 Falleni, Alessandra; Trincavelli, MARIA LETIZIA; Macchia, Marco; Salvetti, F.; Hamdan, M.; Calvani, F.; Gremigni, Vittorio; Lucacchini, Antonio; Martini, Claudia
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
"Soft Drugs" Based on Cannabinoid Receptor Ligands as Potential Local Analgesic and Antiglaucoma Agents | 1-gen-2007 | Minutolo, Filippo; CASCIO M., G; Carboni, I; Bisogno, T; Prota, G; Bertini, Simone; Digiacomo, Maria; Bifulco, M; DI MARZO, V; Macchia, Marco | |
(E)-(ARYLMETHYLENEAMINOXY)ACETAMIDES AS ANALOGS OF NEUROLEPTIC BENZAMIDES - SYNTHESIS AND D-2-DOPAMINERGIC BINDING-AFFINITY | 1-gen-1995 | Macchia, Marco; Manera, Clementina; Martinelli, Adriano; Orlandini, Elisabetta; Romagnoli, F; Rossello, Armando; Chiellini, Grazia | |
(E)-(methyloxyimino)acetamides as analogues of neuroleptic benzamides: Synthesis and D-2-dopaminergic binding affinity | 1-gen-1996 | Lapucci, Annalina; Macchia, Marco; Orlandini, Elisabetta; Romagnoli, F; Rossello, Armando; Chiellini, Grazia; Cozzini, P; Domiano, P. | |
(Z)-(Methyloxyiminomethyl)ethanolamines. Effects of the configuration around the iminic double bond on the beta-adrenergic affinity of moim-type beta-adrenergic blocking agents | 1-gen-1995 | Chiellini, Grazia; Lapucci, Annalina; Macchia, Marco; F., Romagnoli; Rossello, Armando; Nencetti, Susanna | |
1,2-Dihydro-2-oxopyridine-3-carboxamides: the C-5 substituent is responsible for functionality switch at CB2 cannabinoid receptor | 1-gen-2014 | Valentina, Lucchesi; Teija, Parkkari; Juha R., Savinainen; Anna Maria, Malfitano; Marco, Allarà; Bertini, Simone; Francesca, Castelli; Sara Del, Carlo; Chiara, Laezza; Alessia, Ligresti; Saccomanni, Giuseppe; Maurizio, Bifulco; Vincenzo Di, Marzo; Macchia, Marco; Manera, Clementina | |
1-benzilossiimmino-3- ammino-2-propanoli: sintesi e proprietà ß-adrenergiche | 1-gen-1991 | Balsamo, A; Macchia, B; Macchia, Marco; Martinelli, Adriano; Rossello, Armando; Breschi, MARIA CRISTINA; Nieri, Paola; Scatizzi, R. | |
18FLUORINE-LABELED NITROGEN HETEROCYCLIC DERIVATIVES AS NEW CANDIDATE FOR CANNABINOID CB2 RECEPTOR PET IMAGING | 1-gen-2011 | Castelli, Francesca; Bertini, Simone; DEL CARLO, Sara; Lucchesi, Valentina; Manera, Clementina; Pascali, Giancarlo; Saccomanni, Giuseppe; DI MARZO, Vincenzo; Salvadori, Piero; Macchia, Marco | |
2-(Methyleneaminoxy)methylmorpholine derivatives. Synthesis and antidepressant activity | 1-gen-1994 | A., Balsamo; Lapucci, Annalina; Macchia, Marco; Martinelli, Adriano; Nencetti, Susanna; T., Cristina; Rossello, Armando | |
3-(Methyleneaminoxy)methylpiperidine derivatives as uptake inhibitors of biogenic amines in the brain synaptosomal fraction | 1-gen-1994 | Balsamo, A; Lapucci, Annalina; Lucacchini, Antonio; Macchia, Marco; Martini, Claudia; Nardini, C; Nencetti, Susanna | |
3-(METHYLENEAMINOXY)METHYLPIPERIDINE DERIVATIVES AS UPTAKE INHIBITORS OF BIOGENIC-AMINES IN THE BRAIN SYNAPTOSOMAL FRACTION | 1-gen-1994 | Balsamo, A; Lapucci, Annalina; Lucacchini, Antonio; Macchia, Marco; Martini, Claudia; Nardini, C; Nencetti, Susanna | |
4-[6-(dansylamino)hexylamino]-7-methyl-2-phenyl-1,8-naphthyridine as a new potential fluorescent probe for studying A1-adenosine receptor | 1-gen-2002 | Macchia, Marco; Bertini, Simone; DI BUSSOLO, Valeria; Manera, Clementina; Martini, Claudia; Minutolo, Filippo; C., Mori; Saccomanni, Giuseppe; D., Tuscano; Ferrarini, P. | |
4-Aryliden-2-methyloxazol-5(4H)-one as a new scaffold for selective reversible MAGL inhibitors | 1-gen-2016 | Granchi, Carlotta; Rizzolio, F; Bordoni, Vittorio; Caligiuri, I; Manera, Clementina; Macchia, Marco; Minutolo, Filippo; Martinelli, Adriano; Giordano, A; Tuccinardi, Tiziano | |
7-Nitrobenzofurazan (NBD)-Derivatives Of 5'-N-Ethylcarboxamidoadenosine (NECA) As New Fluorescent Probes For Human A3 Adenosine Receptors | 1-gen-2001 | Macchia, Marco; Salvetti, F; Bertini, Simone; DI BUSSOLO, Valeria; Gattuso, L; Gesi, Marco; Hamdan, M; KLOTZ K., N; Laragione, T; Lucacchini, Antonio; Minutolo, Filippo; Nencetti, Susanna; Papi, C; Tuscano, D; Martini, Claudia | |
A new D2 dopamine receptor agonist allosterically modulates A2A adenosine receptor signalling by interacting with the A2A/D2 receptor heteromer | 1-gen-2012 | Trincavelli, MARIA LETIZIA; Daniele, Simona; Orlandini, Elisabetta; Navarro, G.; Casado, V.; Giacomelli, Chiara; Nencetti, Susanna; Nuti, Elisa; Macchia, Marco; Huebner, H.; Gmeiner, P.; Rossello, Armando; Lluis, C.; Martini, Claudia | |
A new small molecule, D2 dopamine receptor agonist, as an allosteric modulator of A2A adenosine receptor signalling | 1-gen-2010 | Trincavelli, MARIA LETIZIA; Orlandini, Elisabetta; Daniele, Simona; Nencetti, Susanna; Nuti, Elisa; Macchia, Marco; Huebner, H; Gmeiner, P; Rossello, Armando; Martini, Claudia | |
A new small molecule, D2 dopamine receptor agonist, as an allosteric modulator of A2A adenosine receptor signalling | 1-gen-2010 | Trincavelli, MARIA LETIZIA; Orlandini, Elisabetta; Daniele, Simona; Nencetti, Susanna; Nuti, Elisa; Macchia, Marco; Huebner, H; Gmeiner, P; Rossello, Armando; Martini, Claudia | |
A Proteomic Approach to Uncover Neuroprotective Mechanisms of Oleocanthal against Oxidative Stress | 1-gen-2018 | Giusti, Laura; Angeloni, Cristina; Barbalace, Maria Cristina; Lacerenza, Serena; Ciregia, Federica; Ronci, Maurizio; Urbani, Andrea; Manera, Clementina; Digiacomo, Maria; Macchia, Marco; Mazzoni, Maria Rosa; Lucacchini, Antonio; Hrelia, Silvana | |
A structure-activity study of a C-terminal endothelin analogue | 1-gen-1998 | Cassano, E; Galoppini, C; Giusti, Laura; Hamdan, M; Macchia, Marco; Mazzoni, MARIA ROSA; Menchini, E; Pegoraro, S; Rovero, P. | |
A Virtual Screening Study for Lactate Dehydrogenase 5 Inhibitors by using a Pharmacophore-Based Approach | 1-gen-2016 | Tuccinardi, Tiziano; Poli, Giulio; Corchia, Isacco; Granchi, Carlotta; Lapillo, Margherita; Macchia, Marco; Minutolo, Filippo; Ortore, GABRIELLA MARIA PIA; Martinelli, Adriano | |
A(1) adenosine receptors in human neutrophils: Direct binding and electron microscope visualization | 1-gen-1999 | Falleni, Alessandra; Trincavelli, MARIA LETIZIA; Macchia, Marco; Salvetti, F.; Hamdan, M.; Calvani, F.; Gremigni, Vittorio; Lucacchini, Antonio; Martini, Claudia |