MACCHIA, MARCO Statistiche
MACCHIA, MARCO
DIPARTIMENTO DI FARMACIA
Enhanced Nutraceutical Properties of Extra Virgin Olive Oil Extract by Olive Leaf Enrichment
2023-01-01 Cuffaro, Doretta; Bertini, Simone; Macchia, Marco; Digiacomo, Maria
The phenolic compounds tyrosol and hydroxytyrosol counteract liver fibrogenesis via the transcriptional modulation of NADPH oxidases and oxidative stress-related miRNAs
2023-01-01 Gabbia, Daniela; Carpi, Sara; Sarcognato, Samantha; Zanotto, Ilaria; Sayaf, Katia; Colognesi, Martina; Polini, Beatrice; Digiacomo, Maria; Macchia, Marco; Nieri, Paola; Carrara, Maria; Cazzagon, Nora; Russo, Francesco Paolo; Guido, Maria; De Martin, Sara
CB1 receptor binding sites for NAM and PAM: A first approach for studying, new n‑butyl‑diphenylcarboxamides as allosteric modulators
2022-01-01 Gado, F.; Ceni, C.; Ferrisi, R.; Sbrana, G.; Stevenson, L. A.; Macchia, M.; Pertwee, R. G.; Bertini, S.; Manera, C.; Ortore, G.
Content Variations in Oleocanthalic Acid and Other Phenolic Compounds in Extra-Virgin Olive Oil during Storage
2022-01-01 Esposito Salsano, Jasmine; Digiacomo, Maria; Cuffaro, Doretta; Bertini, Simone; Macchia, Marco
Electrospun Poly(3-Hydroxybutyrate-Co-3-Hydroxyvalerate)/Olive Leaf Extract Fiber Mesh as Prospective Bio-Based Scaffold for Wound Healing
2022-01-01 De la Ossa, J. G.; Danti, S.; Esposito Salsano, J.; Azimi, B.; Tempesti, V.; Barbani, N.; Digiacomo, M.; Macchia, M.; Uddin, M. J.; Cristallini, C.; Di Stefano, R.; Lazzeri, A.
Machine Learning-Based Virtual Screening for the Identification of Cdk5 Inhibitors
2022-01-01 Di Stefano, Miriana; Galati, Salvatore; Ortore, Gabriella; Caligiuri, Isabella; Rizzolio, Flavio; Ceni, Costanza; Bertini, Simone; Bononi, Giulia; Granchi, Carlotta; Macchia, Marco; Poli, Giulio; Tuccinardi, Tiziano
New PIN1 inhibitors identified through a pharmacophore-driven, hierarchical consensus docking strategy
2022-01-01 Poli, Giulio; Di Stefano, Miriana; Estevez, Joan Arias; Minutolo, Filippo; Granchi, Carlotta; Giordano, Antonio; Parisi, Salvatore; Mauceri, Matteo; Canzonieri, Vincenzo; Macchia, Marco; Caligiuri, Isabella; Tuccinardi, Tiziano; Rizzolio, Flavio
Novel Potent and Selective Agonists of the GPR55 Receptor Based on the 3-Benzylquinolin-2(1H)-One Scaffold
2022-01-01 Ceni, Costanza; Benko, Michael J; Mohamed, Kawthar A; Poli, Giulio; Di Stefano, Miriana; Tuccinardi, Tiziano; Digiacomo, Maria; Valoti, Massimo; Laprairie, Robert B; Macchia, Marco; Bertini, Simone
Oleocanthalic acid from extra-virgin olive oil: Analysis, preparative isolation and radical scavenging activity
2022-01-01 Esposito Salsano, J.; Pinto, D.; Rodrigues, F.; Saba, A.; Manera, C.; Digiacomo, M.; Macchia, M.
Predicting potentially pathogenic effects of hRPE65 missense mutations: a computational strategy based on molecular dynamics simulations
2022-01-01 Poli, Giulio; Barravecchia, Ivana; Demontis, Gian Carlo; Sodi, Andrea; Saba, Alessandro; Rizzo, Stanislao; Macchia, Marco; Tuccinardi, Tiziano
Reversible Monoacylglycerol Lipase Inhibitors: Discovery of a New Class of Benzylpiperidine Derivatives
2022-01-01 Bononi, Giulia; Di Stefano, Miriana; Poli, Giulio; Ortore, Gabriella; Meier, Philip; Masetto, Francesca; Caligiuri, Isabella; Rizzolio, Flavio; Macchia, Marco; Chicca, Andrea; Avan, Amir; Giovannetti, Elisa; Vagaggini, Chiara; Brai, Annalaura; Dreassi, Elena; Valoti, Massimo; Minutolo, Filippo; Granchi, Carlotta; Gertsch, Jürg; Tuccinardi, Tiziano
VenomPred: A Machine Learning Based Platform for Molecular Toxicity Predictions
2022-01-01 Galati, Salvatore; Di Stefano, Miriana; Martinelli, Elisa; Macchia, Marco; Martinelli, Adriano; Poli, Giulio; Tuccinardi, Tiziano
An updated patent review of monoacylglycerol lipase (MAGL) inhibitors (2018-present)
2021-01-01 Bononi, G.; Poli, G.; Rizzolio, F.; Tuccinardi, T.; Macchia, M.; Minutolo, F.; Granchi, C.
Antioxidant and neuroprotective activity of extra virgin olive oil extracts obtained from quercetano cultivar trees grown in different areas of the tuscany region (Italy)
2021-01-01 Barbalace, M. C.; Zallocco, L.; Beghelli, D.; Ronci, M.; Scortichini, S.; Digiacomo, M.; Macchia, M.; Mazzoni, M. R.; Fiorini, D.; Lucacchini, A.; Hrelia, S.; Giusti, L.; Angeloni, C.
Design, synthesis and biological evaluation of second-generation benzoylpiperidine derivatives as reversible monoacylglycerol lipase (MAGL) inhibitors
2021-01-01 Granchi, C.; Bononi, G.; Ferrisi, R.; Gori, E.; Mantini, G.; Glasmacher, S.; Poli, G.; Palazzolo, S.; Caligiuri, I.; Rizzolio, F.; Canzonieri, V.; Perin, T.; Gertsch, J.; Sodi, A.; Giovannetti, E.; Macchia, M.; Minutolo, F.; Tuccinardi, T.; Chicca, A.
Discovery of monoacylglycerol lipase (MAGL) inhibitors based on a pharmacophore-guided virtual screening study
2021-01-01 Jha, V.; Biagi, M.; Spinelli, V.; Di Stefano, M. D.; Macchia, M.; Minutolo, F.; Granchi, C.; Poli, G.; Tuccinardi, T.
Immunomodulatory activity of electrospun polyhydroxyalkanoate fiber scaffolds incorporating olive leaf extract
2021-01-01 De la Ossa, J. G.; Fusco, A.; Azimi, B.; Salsano, J. E.; Digiacomo, M.; Coltelli, M. B.; De Clerck, K.; Roy, I.; Macchia, M.; Lazzeri, A.; Donnarumma, G.; Danti, S.; Di Stefano, R.
Medicinal Chemistry approach, pharmacology and neuroprotective benefits of CB2R modulators in neurodegenerative diseases
2021-01-01 Ferrisi, R.; Ceni, C.; Bertini, S.; Macchia, M.; Manera, C.; Gado, F.
Monoacylglycerol lipase (MAGL) Inhibitors
2021-01-01 Granchi, C; Bononi, G; Macchia, M; Minutolo, F; Poli, G; Scalabrini, D; Tuccinardi, T; Rizzolio, F; Giordano, A
Monoacylglycerol lipase (MAGL) inhibitors based on a diphenylsulfide-benzoylpiperidine scaffold
2021-01-01 Bononi, G.; Tonarini, G.; Poli, G.; Barravecchia, I.; Caligiuri, I.; Macchia, M.; Rizzolio, F.; Demontis, G. C. A. G.; Minutolo, F.; Granchi, C.; Tuccinardi, T.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Enhanced Nutraceutical Properties of Extra Virgin Olive Oil Extract by Olive Leaf Enrichment | 1-gen-2023 | Cuffaro, Doretta; Bertini, Simone; Macchia, Marco; Digiacomo, Maria | |
The phenolic compounds tyrosol and hydroxytyrosol counteract liver fibrogenesis via the transcriptional modulation of NADPH oxidases and oxidative stress-related miRNAs | 1-gen-2023 | Gabbia, Daniela; Carpi, Sara; Sarcognato, Samantha; Zanotto, Ilaria; Sayaf, Katia; Colognesi, Martina; Polini, Beatrice; Digiacomo, Maria; Macchia, Marco; Nieri, Paola; Carrara, Maria; Cazzagon, Nora; Russo, Francesco Paolo; Guido, Maria; De Martin, Sara | |
CB1 receptor binding sites for NAM and PAM: A first approach for studying, new n‑butyl‑diphenylcarboxamides as allosteric modulators | 1-gen-2022 | Gado, F.; Ceni, C.; Ferrisi, R.; Sbrana, G.; Stevenson, L. A.; Macchia, M.; Pertwee, R. G.; Bertini, S.; Manera, C.; Ortore, G. | |
Content Variations in Oleocanthalic Acid and Other Phenolic Compounds in Extra-Virgin Olive Oil during Storage | 1-gen-2022 | Esposito Salsano, Jasmine; Digiacomo, Maria; Cuffaro, Doretta; Bertini, Simone; Macchia, Marco | |
Electrospun Poly(3-Hydroxybutyrate-Co-3-Hydroxyvalerate)/Olive Leaf Extract Fiber Mesh as Prospective Bio-Based Scaffold for Wound Healing | 1-gen-2022 | De la Ossa, J. G.; Danti, S.; Esposito Salsano, J.; Azimi, B.; Tempesti, V.; Barbani, N.; Digiacomo, M.; Macchia, M.; Uddin, M. J.; Cristallini, C.; Di Stefano, R.; Lazzeri, A. | |
Machine Learning-Based Virtual Screening for the Identification of Cdk5 Inhibitors | 1-gen-2022 | Di Stefano, Miriana; Galati, Salvatore; Ortore, Gabriella; Caligiuri, Isabella; Rizzolio, Flavio; Ceni, Costanza; Bertini, Simone; Bononi, Giulia; Granchi, Carlotta; Macchia, Marco; Poli, Giulio; Tuccinardi, Tiziano | |
New PIN1 inhibitors identified through a pharmacophore-driven, hierarchical consensus docking strategy | 1-gen-2022 | Poli, Giulio; Di Stefano, Miriana; Estevez, Joan Arias; Minutolo, Filippo; Granchi, Carlotta; Giordano, Antonio; Parisi, Salvatore; Mauceri, Matteo; Canzonieri, Vincenzo; Macchia, Marco; Caligiuri, Isabella; Tuccinardi, Tiziano; Rizzolio, Flavio | |
Novel Potent and Selective Agonists of the GPR55 Receptor Based on the 3-Benzylquinolin-2(1H)-One Scaffold | 1-gen-2022 | Ceni, Costanza; Benko, Michael J; Mohamed, Kawthar A; Poli, Giulio; Di Stefano, Miriana; Tuccinardi, Tiziano; Digiacomo, Maria; Valoti, Massimo; Laprairie, Robert B; Macchia, Marco; Bertini, Simone | |
Oleocanthalic acid from extra-virgin olive oil: Analysis, preparative isolation and radical scavenging activity | 1-gen-2022 | Esposito Salsano, J.; Pinto, D.; Rodrigues, F.; Saba, A.; Manera, C.; Digiacomo, M.; Macchia, M. | |
Predicting potentially pathogenic effects of hRPE65 missense mutations: a computational strategy based on molecular dynamics simulations | 1-gen-2022 | Poli, Giulio; Barravecchia, Ivana; Demontis, Gian Carlo; Sodi, Andrea; Saba, Alessandro; Rizzo, Stanislao; Macchia, Marco; Tuccinardi, Tiziano | |
Reversible Monoacylglycerol Lipase Inhibitors: Discovery of a New Class of Benzylpiperidine Derivatives | 1-gen-2022 | Bononi, Giulia; Di Stefano, Miriana; Poli, Giulio; Ortore, Gabriella; Meier, Philip; Masetto, Francesca; Caligiuri, Isabella; Rizzolio, Flavio; Macchia, Marco; Chicca, Andrea; Avan, Amir; Giovannetti, Elisa; Vagaggini, Chiara; Brai, Annalaura; Dreassi, Elena; Valoti, Massimo; Minutolo, Filippo; Granchi, Carlotta; Gertsch, Jürg; Tuccinardi, Tiziano | |
VenomPred: A Machine Learning Based Platform for Molecular Toxicity Predictions | 1-gen-2022 | Galati, Salvatore; Di Stefano, Miriana; Martinelli, Elisa; Macchia, Marco; Martinelli, Adriano; Poli, Giulio; Tuccinardi, Tiziano | |
An updated patent review of monoacylglycerol lipase (MAGL) inhibitors (2018-present) | 1-gen-2021 | Bononi, G.; Poli, G.; Rizzolio, F.; Tuccinardi, T.; Macchia, M.; Minutolo, F.; Granchi, C. | |
Antioxidant and neuroprotective activity of extra virgin olive oil extracts obtained from quercetano cultivar trees grown in different areas of the tuscany region (Italy) | 1-gen-2021 | Barbalace, M. C.; Zallocco, L.; Beghelli, D.; Ronci, M.; Scortichini, S.; Digiacomo, M.; Macchia, M.; Mazzoni, M. R.; Fiorini, D.; Lucacchini, A.; Hrelia, S.; Giusti, L.; Angeloni, C. | |
Design, synthesis and biological evaluation of second-generation benzoylpiperidine derivatives as reversible monoacylglycerol lipase (MAGL) inhibitors | 1-gen-2021 | Granchi, C.; Bononi, G.; Ferrisi, R.; Gori, E.; Mantini, G.; Glasmacher, S.; Poli, G.; Palazzolo, S.; Caligiuri, I.; Rizzolio, F.; Canzonieri, V.; Perin, T.; Gertsch, J.; Sodi, A.; Giovannetti, E.; Macchia, M.; Minutolo, F.; Tuccinardi, T.; Chicca, A. | |
Discovery of monoacylglycerol lipase (MAGL) inhibitors based on a pharmacophore-guided virtual screening study | 1-gen-2021 | Jha, V.; Biagi, M.; Spinelli, V.; Di Stefano, M. D.; Macchia, M.; Minutolo, F.; Granchi, C.; Poli, G.; Tuccinardi, T. | |
Immunomodulatory activity of electrospun polyhydroxyalkanoate fiber scaffolds incorporating olive leaf extract | 1-gen-2021 | De la Ossa, J. G.; Fusco, A.; Azimi, B.; Salsano, J. E.; Digiacomo, M.; Coltelli, M. B.; De Clerck, K.; Roy, I.; Macchia, M.; Lazzeri, A.; Donnarumma, G.; Danti, S.; Di Stefano, R. | |
Medicinal Chemistry approach, pharmacology and neuroprotective benefits of CB2R modulators in neurodegenerative diseases | 1-gen-2021 | Ferrisi, R.; Ceni, C.; Bertini, S.; Macchia, M.; Manera, C.; Gado, F. | |
Monoacylglycerol lipase (MAGL) Inhibitors | 1-gen-2021 | Granchi, C; Bononi, G; Macchia, M; Minutolo, F; Poli, G; Scalabrini, D; Tuccinardi, T; Rizzolio, F; Giordano, A | |
Monoacylglycerol lipase (MAGL) inhibitors based on a diphenylsulfide-benzoylpiperidine scaffold | 1-gen-2021 | Bononi, G.; Tonarini, G.; Poli, G.; Barravecchia, I.; Caligiuri, I.; Macchia, M.; Rizzolio, F.; Demontis, G. C. A. G.; Minutolo, F.; Granchi, C.; Tuccinardi, T. |