MACCHIA, MARCO Statistiche
MACCHIA, MARCO
DIPARTIMENTO DI FARMACIA
A series of benzensulfonamide derivatives as new potent carbonic anhydrase IX and XII inhibitors
2025-01-01 Nencetti, Susanna; Cuffaro, Doretta; Ciccone, Lidia; Nocentini, Alessio; Di Stefano, Miriana; Poli, Giulio; Macchia, Marco; Tuccinardi, Tiziano; Nuti, Elisa; Supuran, Claudiu T.; Rossello, Armando; Orlandini, Elisabetta
Discovery of reversible monoacylglycerol lipase (MAGL) inhibitors based on ortho-hydroxyanilide scaffold
2025-01-01 Bononi, Giulia; Gado, Francesca; Masoni, Samuele; Scalabrini, Diana; Vedova, Larissa Della; Di Stefano, Miriana; Piazza, Lisa; Poles, Clarissa; Lonzi, Chiara; Landucci, Eva; Vagaggini, Chiara; Poggialini, Federica; Brai, Annalaura; Caligiuri, Isabella; Rizzolio, Flavio; Mohamed, Kawthar A; Bertini, Simone; De Lorenzi, Ersilia; Dreassi, Elena; Macchia, Marco; Minutolo, Filippo; Laprairie, Robert B; Granchi, Carlotta; Tuccinardi, Tiziano
Fast, sensitive, and sustainable colorimetric detection of chlorogenic acid in artichoke waste material
2025-01-01 Cuffaro, Doretta; Palladino, Pasquale; Digiacomo, Maria; Bertini, Simone; Minunni, Maria; Macchia, Marco
JG26 attenuates ADAM17 metalloproteinase-mediated ACE2 receptor processing and SARS-CoV-2 infection in vitro
2025-01-01 Gentili, Valentina; Beltrami, Silvia; Cuffaro, Doretta; Cianci, Giorgia; Maini, Gloria; Rizzo, Roberta; Macchia, Marco; Rossello, Armando; Bortolotti, Daria; Nuti, Elisa
KinasePred: A Computational Tool for Small-Molecule Kinase Target Prediction
2025-01-01 Di Stefano, Miriana; Piazza, Lisa; Poles, Clarissa; Galati, Salvatore; Granchi, Carlotta; Giordano, Antonio; Campisi, Luca; Macchia, Marco; Poli, Giulio; Tuccinardi, Tiziano
Methods for Assessing MAGL Enzymatic Activity: An Extensive Review of Past and Emerging Approaches
2025-01-01 Bononi, Giulia; Landucci, Eva; Di Stefano, Miriana; Piazza, Lisa; Bertini, Simone; Macchia, Marco; Granchi, Carlotta
Multivalent MMP-12 inhibitors as a valuable approach to counteract the intestinal epithelial barrier impairment and inflammation in an in vitro model mimicking intestinal high-fat exposure
2025-01-01 Cuffaro, D.; D'Antongiovanni, V.; Mangini, C.; Di Salvo, C.; Benvenuti, L.; Vandooren, J.; Macchia, M.; Antonioli, L.; Rossello, A.; Fornai, M.; Nuti, E.
Neuroprotective Potential of Polyphenol-Rich Artichoke Waste Extract: Exploring Antioxidant and Immunomodulatory Activities in Cell Models
2025-01-01 Cuffaro, D.; Ceni, C.; Capitini, C.; Gabbia, D.; Zanotto, I.; Bertolini, A.; Mirabeni, M.; Bertini, S.; Saba, A.; De Martin, S.; Calamai, M.; Digiacomo, M.; Macchia, M.
Oleocanthalic acid improves MASH features via a NOX1-dependent mechanism
2025-01-01 Frion-Herrera, Yahima; Zanotto, Ilaria; Colognesi, Martina; Signor, Anna; Cuffaro, Doretta; Chilin, Adriana; Macchia, Marco; Marzaro, Giovanni; Digiacomo, Maria; Gabbia, Daniela; De Martin, Sara
Solid-State Fermented Cereals: Increased Phenolics and Their Role in Attenuating Liver Diseases
2025-01-01 Wijaya, Ganesha Yanuar Arief; Vornoli, Andrea; Giambastiani, Lucia; Digiacomo, Maria; Macchia, Marco; Szymczak, Bartłomiej; Wójcik, Marta; Pozzo, Luisa; Longo, Vincenzo
Valorization of olive mill wastewater: improving the polyphenolic content, antioxidant potential, and cytotoxicity profile of extra virgin olive oil extract
2025-01-01 Rodrigues, Francisca; Cuffaro, Doretta; Silva, Ana Margarida; Mirabeni, Massimiliano; Bertini, Simone; Macchia, Marco; Digiacomo, Maria
1-Acetoxypinoresinol, a Lignan from Olives: Insight into Its Characterization, Identification, and Nutraceutical Properties
2024-01-01 Yanuar Arief Wijaya, Ganesha; Cuffaro, Doretta; Bertini, Simone; Digiacomo, Maria; Macchia, Marco
Comparative Analysis on Polyphenolic Composition of Different Olive Mill Wastewater and Related Extra Virgin Olive Oil Extracts and Evaluation of Nutraceutical Properties by Cell-Based Studies
2024-01-01 Cuffaro, D.; Bertolini, A.; Silva, A. M.; Rodrigues, F.; Gabbia, D.; De Martin, S.; Saba, A.; Bertini, S.; Digiacomo, M.; Macchia, M.
Design, synthesis and biological evaluation of arylsulfonamides as ADAMTS7 inhibitors
2024-01-01 Cuffaro, Doretta; Burkhard, Tina; Bernardoni, Bianca Laura; Di Leo, Riccardo; Zhang, Xiaohan; Galati, Salvatore; Tuccinardi, Tiziano; Macchia, Marco; Rossello, Armando; Santamaria, Salvatore; de Groot, Rens; Nuti, Elisa
Design, synthesis, ADME and biological evaluation of benzylpiperidine and benzylpiperazine derivatives as novel reversible monoacylglycerol lipase (MAGL) inhibitors
2024-01-01 Di Stefano, Miriana; Masoni, Samuele; Bononi, Giulia; Poli, Giulio; Galati, Salvatore; Gado, Francesca; Manzi, Simone; Vagaggini, Chiara; Brai, Annalaura; Caligiuri, Isabella; Asif, Kanwal; Rizzolio, Flavio; Macchia, Marco; Chicca, Andrea; Sodi, Andrea; Di Bussolo, Valeria; Minutolo, Filippo; Meier, Philip; Gertsch, Jürg; Granchi, Carlotta; Dreassi, Elena; Tuccinardi, Tiziano
Unraveling the Protective Role of Oleocanthal and Its Oxidation Product, Oleocanthalic Acid, against Neuroinflammation
2024-01-01 Barbalace, Maria Cristina; Freschi, Michela; Rinaldi, Irene; Zallocco, Lorenzo; Malaguti, Marco; Manera, Clementina; Ortore, Gabriella; Zuccarini, Mariachiara; Ronci, Maurizio; Cuffaro, Doretta; Macchia, Marco; Hrelia, Silvana; Giusti, Laura; Digiacomo, Maria; Angeloni, Cristina
VenomPred 2.0: A Novel In Silico Platform for an Extended and Human Interpretable Toxicological Profiling of Small Molecules
2024-01-01 Di Stefano, Miriana; Galati, Salvatore; Piazza, Lisa; Granchi, Carlotta; Mancini, Simone; Fratini, Filippo; Macchia, Marco; Poli, Giulio; Tuccinardi, Tiziano
WaSPred: A reliable AI-based water solubility predictor for small molecules
2024-01-01 Di Stefano, Miriana; Galati, Salvatore; Lonzi, Chiara; Granchi, Carlotta; Poli, Giulio; Tuccinardi, Tiziano; Macchia, Marco
Watermelon: setup and validation of an in silico fragment-based approach
2024-01-01 Di Stefano, Miriana; Galati, Salvatore; Piazza, Lisa; Gado, Francesca; Granchi, Carlotta; Macchia, Marco; Giordano, Antonio; Tuccinardi, Tiziano; Poli, Giulio
An in silico toolbox for the prediction of the potential pathogenic effects of missense mutations in the dimeric region of hRPE65
2023-01-01 Poli, Giulio; Demontis, Gian Carlo; Sodi, Andrea; Saba, Alessandro; Rizzo, Stanislao; Macchia, Marco; Tuccinardi, Tiziano
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| A series of benzensulfonamide derivatives as new potent carbonic anhydrase IX and XII inhibitors | 1-gen-2025 | Nencetti, Susanna; Cuffaro, Doretta; Ciccone, Lidia; Nocentini, Alessio; Di Stefano, Miriana; Poli, Giulio; Macchia, Marco; Tuccinardi, Tiziano; Nuti, Elisa; Supuran, Claudiu T.; Rossello, Armando; Orlandini, Elisabetta | |
| Discovery of reversible monoacylglycerol lipase (MAGL) inhibitors based on ortho-hydroxyanilide scaffold | 1-gen-2025 | Bononi, Giulia; Gado, Francesca; Masoni, Samuele; Scalabrini, Diana; Vedova, Larissa Della; Di Stefano, Miriana; Piazza, Lisa; Poles, Clarissa; Lonzi, Chiara; Landucci, Eva; Vagaggini, Chiara; Poggialini, Federica; Brai, Annalaura; Caligiuri, Isabella; Rizzolio, Flavio; Mohamed, Kawthar A; Bertini, Simone; De Lorenzi, Ersilia; Dreassi, Elena; Macchia, Marco; Minutolo, Filippo; Laprairie, Robert B; Granchi, Carlotta; Tuccinardi, Tiziano | |
| Fast, sensitive, and sustainable colorimetric detection of chlorogenic acid in artichoke waste material | 1-gen-2025 | Cuffaro, Doretta; Palladino, Pasquale; Digiacomo, Maria; Bertini, Simone; Minunni, Maria; Macchia, Marco | |
| JG26 attenuates ADAM17 metalloproteinase-mediated ACE2 receptor processing and SARS-CoV-2 infection in vitro | 1-gen-2025 | Gentili, Valentina; Beltrami, Silvia; Cuffaro, Doretta; Cianci, Giorgia; Maini, Gloria; Rizzo, Roberta; Macchia, Marco; Rossello, Armando; Bortolotti, Daria; Nuti, Elisa | |
| KinasePred: A Computational Tool for Small-Molecule Kinase Target Prediction | 1-gen-2025 | Di Stefano, Miriana; Piazza, Lisa; Poles, Clarissa; Galati, Salvatore; Granchi, Carlotta; Giordano, Antonio; Campisi, Luca; Macchia, Marco; Poli, Giulio; Tuccinardi, Tiziano | |
| Methods for Assessing MAGL Enzymatic Activity: An Extensive Review of Past and Emerging Approaches | 1-gen-2025 | Bononi, Giulia; Landucci, Eva; Di Stefano, Miriana; Piazza, Lisa; Bertini, Simone; Macchia, Marco; Granchi, Carlotta | |
| Multivalent MMP-12 inhibitors as a valuable approach to counteract the intestinal epithelial barrier impairment and inflammation in an in vitro model mimicking intestinal high-fat exposure | 1-gen-2025 | Cuffaro, D.; D'Antongiovanni, V.; Mangini, C.; Di Salvo, C.; Benvenuti, L.; Vandooren, J.; Macchia, M.; Antonioli, L.; Rossello, A.; Fornai, M.; Nuti, E. | |
| Neuroprotective Potential of Polyphenol-Rich Artichoke Waste Extract: Exploring Antioxidant and Immunomodulatory Activities in Cell Models | 1-gen-2025 | Cuffaro, D.; Ceni, C.; Capitini, C.; Gabbia, D.; Zanotto, I.; Bertolini, A.; Mirabeni, M.; Bertini, S.; Saba, A.; De Martin, S.; Calamai, M.; Digiacomo, M.; Macchia, M. | |
| Oleocanthalic acid improves MASH features via a NOX1-dependent mechanism | 1-gen-2025 | Frion-Herrera, Yahima; Zanotto, Ilaria; Colognesi, Martina; Signor, Anna; Cuffaro, Doretta; Chilin, Adriana; Macchia, Marco; Marzaro, Giovanni; Digiacomo, Maria; Gabbia, Daniela; De Martin, Sara | |
| Solid-State Fermented Cereals: Increased Phenolics and Their Role in Attenuating Liver Diseases | 1-gen-2025 | Wijaya, Ganesha Yanuar Arief; Vornoli, Andrea; Giambastiani, Lucia; Digiacomo, Maria; Macchia, Marco; Szymczak, Bartłomiej; Wójcik, Marta; Pozzo, Luisa; Longo, Vincenzo | |
| Valorization of olive mill wastewater: improving the polyphenolic content, antioxidant potential, and cytotoxicity profile of extra virgin olive oil extract | 1-gen-2025 | Rodrigues, Francisca; Cuffaro, Doretta; Silva, Ana Margarida; Mirabeni, Massimiliano; Bertini, Simone; Macchia, Marco; Digiacomo, Maria | |
| 1-Acetoxypinoresinol, a Lignan from Olives: Insight into Its Characterization, Identification, and Nutraceutical Properties | 1-gen-2024 | Yanuar Arief Wijaya, Ganesha; Cuffaro, Doretta; Bertini, Simone; Digiacomo, Maria; Macchia, Marco | |
| Comparative Analysis on Polyphenolic Composition of Different Olive Mill Wastewater and Related Extra Virgin Olive Oil Extracts and Evaluation of Nutraceutical Properties by Cell-Based Studies | 1-gen-2024 | Cuffaro, D.; Bertolini, A.; Silva, A. M.; Rodrigues, F.; Gabbia, D.; De Martin, S.; Saba, A.; Bertini, S.; Digiacomo, M.; Macchia, M. | |
| Design, synthesis and biological evaluation of arylsulfonamides as ADAMTS7 inhibitors | 1-gen-2024 | Cuffaro, Doretta; Burkhard, Tina; Bernardoni, Bianca Laura; Di Leo, Riccardo; Zhang, Xiaohan; Galati, Salvatore; Tuccinardi, Tiziano; Macchia, Marco; Rossello, Armando; Santamaria, Salvatore; de Groot, Rens; Nuti, Elisa | |
| Design, synthesis, ADME and biological evaluation of benzylpiperidine and benzylpiperazine derivatives as novel reversible monoacylglycerol lipase (MAGL) inhibitors | 1-gen-2024 | Di Stefano, Miriana; Masoni, Samuele; Bononi, Giulia; Poli, Giulio; Galati, Salvatore; Gado, Francesca; Manzi, Simone; Vagaggini, Chiara; Brai, Annalaura; Caligiuri, Isabella; Asif, Kanwal; Rizzolio, Flavio; Macchia, Marco; Chicca, Andrea; Sodi, Andrea; Di Bussolo, Valeria; Minutolo, Filippo; Meier, Philip; Gertsch, Jürg; Granchi, Carlotta; Dreassi, Elena; Tuccinardi, Tiziano | |
| Unraveling the Protective Role of Oleocanthal and Its Oxidation Product, Oleocanthalic Acid, against Neuroinflammation | 1-gen-2024 | Barbalace, Maria Cristina; Freschi, Michela; Rinaldi, Irene; Zallocco, Lorenzo; Malaguti, Marco; Manera, Clementina; Ortore, Gabriella; Zuccarini, Mariachiara; Ronci, Maurizio; Cuffaro, Doretta; Macchia, Marco; Hrelia, Silvana; Giusti, Laura; Digiacomo, Maria; Angeloni, Cristina | |
| VenomPred 2.0: A Novel In Silico Platform for an Extended and Human Interpretable Toxicological Profiling of Small Molecules | 1-gen-2024 | Di Stefano, Miriana; Galati, Salvatore; Piazza, Lisa; Granchi, Carlotta; Mancini, Simone; Fratini, Filippo; Macchia, Marco; Poli, Giulio; Tuccinardi, Tiziano | |
| WaSPred: A reliable AI-based water solubility predictor for small molecules | 1-gen-2024 | Di Stefano, Miriana; Galati, Salvatore; Lonzi, Chiara; Granchi, Carlotta; Poli, Giulio; Tuccinardi, Tiziano; Macchia, Marco | |
| Watermelon: setup and validation of an in silico fragment-based approach | 1-gen-2024 | Di Stefano, Miriana; Galati, Salvatore; Piazza, Lisa; Gado, Francesca; Granchi, Carlotta; Macchia, Marco; Giordano, Antonio; Tuccinardi, Tiziano; Poli, Giulio | |
| An in silico toolbox for the prediction of the potential pathogenic effects of missense mutations in the dimeric region of hRPE65 | 1-gen-2023 | Poli, Giulio; Demontis, Gian Carlo; Sodi, Andrea; Saba, Alessandro; Rizzo, Stanislao; Macchia, Marco; Tuccinardi, Tiziano |