NUTI, ELISA Statistiche
NUTI, ELISA
DIPARTIMENTO DI FARMACIA
Bacterial Zinc Metalloenzyme Inhibitors: Recent Advances and Future Perspectives
2023-01-01 Di Leo, Riccardo; Cuffaro, Doretta; Rossello, Armando; Nuti, Elisa
New isoxazolidinyl-based N-alkylethanolamines as new activators of human brain carbonic anhydrases
2023-01-01 Cuffaro, Doretta; Di Leo, Riccardo; Ciccone, Lidia; Nocentini, Alessio; Supuran, Claudiu T; Nuti, Elisa; Rossello, Armando
Compounds with a benzo [a]carbazole structure for use in the prevention and/or treatment of infectious diseases
2022-01-01 Rossello, Armando; Nencetti, Susanna; Nuti, Elisa; Orlandini, Elisabetta; Martini, Claudia; Costa, Barbara; Daniele, Simona; Giacomelli, Chiara; Ciccone, Lidia; Cuffaro, Doretta; Comar, Manola
Identification of a Novel p53 Modulator Endowed with Antitumoural and Antibacterial Activity through a Scaffold Repurposing Approach
2022-01-01 Nuti, Elisa; La Pietra, Valeria; Daniele, Simona; Cuffaro, Doretta; Ciccone, Lidia; Giacomelli, Chiara; Cason, Carolina; Carotenuto, Alfonso; D'Amore, Vincenzo Maria; Pozzo, Eleonora Da; Costa, Barbara; Di Leo, Riccardo; Comar, Manola; Marinelli, Luciana; Martini, Claudia; Rossello, Armando
Inhibitors of A Disintegrin And Metalloproteinases-10 reduce Hodgkin lymphoma cell growth in 3D microenvironments and enhance brentuximab-vedotin effect
2022-01-01 Pece, Roberta; Tavella, Sara; Costa, Delfina; Varesano, Serena; Camodeca, Caterina; Cuffaro, Doretta; Nuti, Elisa; Rossello, Armando; Alfano, Massimo; D'Arrigo, Cristina; Galante, Denise; Ravetti, Jean-Louis; Gobbi, Marco; Tosetti, Francesca; Poggi, Alessandro; Zocchi, Maria Raffaella
Targeting Aggrecanases for Osteoarthritis Therapy: From Zinc Chelation to Exosite Inhibition
2022-01-01 Cuffaro, Doretta; Ciccone, Lidia; Rossello, Armando; Nuti, Elisa; Santamaria, Salvatore
Activation of carbonic anhydrases from human brain by amino alcohol oxime ethers: towards human carbonic anhydrase VII selective activators
2021-01-01 Nocentini, A.; Cuffaro, D.; Ciccone, L.; Orlandini, E.; Nencetti, S.; Nuti, E.; Rossello, A.; Supuran, C. T.
Crystal structure of a dimeric based inhibitor JG34 in complex with the MMP-12 catalytic domain
2021-01-01 Ciccone, L.; Rossello, A.; Vera, L.; Nuti, E.; Stura, E. A.
Development of a fluorogenic ADAMTS-7 substrate
2021-01-01 Santamaria, S.; Buemi, F.; Nuti, E.; Cuffaro, D.; De Vita, E.; Tuccinardi, T.; Rossello, A.; Howell, S.; Mehmood, S.; Snijders, A. P.; de Groot, R.
Discovery of Dimeric Arylsulfonamides as Potent ADAM8 Inhibitors
2021-01-01 Cuffaro, Doretta; Camodeca, Caterina; Tuccinardi, Tiziano; Ciccone, Lidia; Bartsch, Jörg W.; Kellermann, Tanja; Cook, Lena; Nuti, Elisa; Rossello, Armando
Exosite inhibition of ADAMTS-5 by a glycoconjugated arylsulfonamide
2021-01-01 Santamaria, S.; Cuffaro, D.; Nuti, E.; Ciccone, L.; Tuccinardi, T.; Liva, F.; D'Andrea, F.; de Groot, R.; Rossello, A.; Ahnstrom, J.
Identification of broad-spectrum mmp inhibitors by virtual screening
2021-01-01 Gimeno, A.; Cuffaro, D.; Nuti, E.; Ojeda-Montes, M. J.; Beltran-Debon, R.; Mulero, M.; Rossello, A.; Pujadas, G.; Garcia-Vallve, S.
Strategies to target ADAM17 in disease: From its discovery to the iRhom revolution
2021-01-01 Calligaris, M.; Cuffaro, D.; Bonelli, S.; Spano, D. P.; Rossello, A.; Nuti, E.; Scilabra, S. D.
The metalloproteinase ADAM10 requires its activity to sustain surface expression
2021-01-01 Seifert, A.; Dusterhoft, S.; Wozniak, J.; Koo, C. Z.; Tomlinson, M. G.; Nuti, E.; Rossello, A.; Cuffaro, D.; Yildiz, D.; Ludwig, A.
An overview of carbohydrate-based carbonic anhydrase inhibitors
2020-01-01 Cuffaro, D.; Nuti, E.; Rossello, A.
Bivalent Inhibitor with Selectivity for Trimeric MMP-9 Amplifies Neutrophil Chemotaxis and Enables Functional Studies on MMP-9 Proteoforms
2020-01-01 Nuti, E.; Rossello, A.; Cuffaro, D.; Camodeca, C.; Van Bael, J.; van der Maat, D.; Martens, E.; Fiten, P.; Pereira, R. V. S.; Ugarte-Berzal, E.; Gouwy, M.; Opdenakker, G.; Vandooren, J.
Developments in carbohydrate-based metzincin inhibitors
2020-01-01 Cuffaro, D.; Nuti, E.; D'Andrea, F.; Rossello, A.
Identification of histone deacetylase inhibitors with (arylidene)aminoxy scaffold active in uveal melanoma cell lines
2020-01-01 Nencetti, S.; Cuffaro, D.; Nuti, E.; Ciccone, L.; Rossello, A.; Fabbi, M.; Ballante, F.; Ortore, G.; Carbotti, G.; Campelli, F.; Banti, I.; Gangemi, R.; Marshall, G. R.; Orlandini, E.
Ionic liquid-promoted green synthesis of biologically relevant diaryl thioethers
2020-01-01 Cuffaro, Doretta; D'Andrea, Felicia; Mezzetta, Andrea; Guazzelli, Lorenzo; Chiappe, Cinzia; Nuti, Elisa; Rossello, Armando
Monoaryl derivatives as transthyretin fibril formation inhibitors: Design, synthesis, biological evaluation and structural analysis
2020-01-01 Ciccone, L.; Nencetti, S.; Tonali, Nicolo; Fruchart-Gaillard, C.; Shepard, W.; Nuti, E.; Camodeca, C.; Rossello, A.; Orlandini, E.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Bacterial Zinc Metalloenzyme Inhibitors: Recent Advances and Future Perspectives | 1-gen-2023 | Di Leo, Riccardo; Cuffaro, Doretta; Rossello, Armando; Nuti, Elisa | |
New isoxazolidinyl-based N-alkylethanolamines as new activators of human brain carbonic anhydrases | 1-gen-2023 | Cuffaro, Doretta; Di Leo, Riccardo; Ciccone, Lidia; Nocentini, Alessio; Supuran, Claudiu T; Nuti, Elisa; Rossello, Armando | |
Compounds with a benzo [a]carbazole structure for use in the prevention and/or treatment of infectious diseases | 1-gen-2022 | Rossello, Armando; Nencetti, Susanna; Nuti, Elisa; Orlandini, Elisabetta; Martini, Claudia; Costa, Barbara; Daniele, Simona; Giacomelli, Chiara; Ciccone, Lidia; Cuffaro, Doretta; Comar, Manola | |
Identification of a Novel p53 Modulator Endowed with Antitumoural and Antibacterial Activity through a Scaffold Repurposing Approach | 1-gen-2022 | Nuti, Elisa; La Pietra, Valeria; Daniele, Simona; Cuffaro, Doretta; Ciccone, Lidia; Giacomelli, Chiara; Cason, Carolina; Carotenuto, Alfonso; D'Amore, Vincenzo Maria; Pozzo, Eleonora Da; Costa, Barbara; Di Leo, Riccardo; Comar, Manola; Marinelli, Luciana; Martini, Claudia; Rossello, Armando | |
Inhibitors of A Disintegrin And Metalloproteinases-10 reduce Hodgkin lymphoma cell growth in 3D microenvironments and enhance brentuximab-vedotin effect | 1-gen-2022 | Pece, Roberta; Tavella, Sara; Costa, Delfina; Varesano, Serena; Camodeca, Caterina; Cuffaro, Doretta; Nuti, Elisa; Rossello, Armando; Alfano, Massimo; D'Arrigo, Cristina; Galante, Denise; Ravetti, Jean-Louis; Gobbi, Marco; Tosetti, Francesca; Poggi, Alessandro; Zocchi, Maria Raffaella | |
Targeting Aggrecanases for Osteoarthritis Therapy: From Zinc Chelation to Exosite Inhibition | 1-gen-2022 | Cuffaro, Doretta; Ciccone, Lidia; Rossello, Armando; Nuti, Elisa; Santamaria, Salvatore | |
Activation of carbonic anhydrases from human brain by amino alcohol oxime ethers: towards human carbonic anhydrase VII selective activators | 1-gen-2021 | Nocentini, A.; Cuffaro, D.; Ciccone, L.; Orlandini, E.; Nencetti, S.; Nuti, E.; Rossello, A.; Supuran, C. T. | |
Crystal structure of a dimeric based inhibitor JG34 in complex with the MMP-12 catalytic domain | 1-gen-2021 | Ciccone, L.; Rossello, A.; Vera, L.; Nuti, E.; Stura, E. A. | |
Development of a fluorogenic ADAMTS-7 substrate | 1-gen-2021 | Santamaria, S.; Buemi, F.; Nuti, E.; Cuffaro, D.; De Vita, E.; Tuccinardi, T.; Rossello, A.; Howell, S.; Mehmood, S.; Snijders, A. P.; de Groot, R. | |
Discovery of Dimeric Arylsulfonamides as Potent ADAM8 Inhibitors | 1-gen-2021 | Cuffaro, Doretta; Camodeca, Caterina; Tuccinardi, Tiziano; Ciccone, Lidia; Bartsch, Jörg W.; Kellermann, Tanja; Cook, Lena; Nuti, Elisa; Rossello, Armando | |
Exosite inhibition of ADAMTS-5 by a glycoconjugated arylsulfonamide | 1-gen-2021 | Santamaria, S.; Cuffaro, D.; Nuti, E.; Ciccone, L.; Tuccinardi, T.; Liva, F.; D'Andrea, F.; de Groot, R.; Rossello, A.; Ahnstrom, J. | |
Identification of broad-spectrum mmp inhibitors by virtual screening | 1-gen-2021 | Gimeno, A.; Cuffaro, D.; Nuti, E.; Ojeda-Montes, M. J.; Beltran-Debon, R.; Mulero, M.; Rossello, A.; Pujadas, G.; Garcia-Vallve, S. | |
Strategies to target ADAM17 in disease: From its discovery to the iRhom revolution | 1-gen-2021 | Calligaris, M.; Cuffaro, D.; Bonelli, S.; Spano, D. P.; Rossello, A.; Nuti, E.; Scilabra, S. D. | |
The metalloproteinase ADAM10 requires its activity to sustain surface expression | 1-gen-2021 | Seifert, A.; Dusterhoft, S.; Wozniak, J.; Koo, C. Z.; Tomlinson, M. G.; Nuti, E.; Rossello, A.; Cuffaro, D.; Yildiz, D.; Ludwig, A. | |
An overview of carbohydrate-based carbonic anhydrase inhibitors | 1-gen-2020 | Cuffaro, D.; Nuti, E.; Rossello, A. | |
Bivalent Inhibitor with Selectivity for Trimeric MMP-9 Amplifies Neutrophil Chemotaxis and Enables Functional Studies on MMP-9 Proteoforms | 1-gen-2020 | Nuti, E.; Rossello, A.; Cuffaro, D.; Camodeca, C.; Van Bael, J.; van der Maat, D.; Martens, E.; Fiten, P.; Pereira, R. V. S.; Ugarte-Berzal, E.; Gouwy, M.; Opdenakker, G.; Vandooren, J. | |
Developments in carbohydrate-based metzincin inhibitors | 1-gen-2020 | Cuffaro, D.; Nuti, E.; D'Andrea, F.; Rossello, A. | |
Identification of histone deacetylase inhibitors with (arylidene)aminoxy scaffold active in uveal melanoma cell lines | 1-gen-2020 | Nencetti, S.; Cuffaro, D.; Nuti, E.; Ciccone, L.; Rossello, A.; Fabbi, M.; Ballante, F.; Ortore, G.; Carbotti, G.; Campelli, F.; Banti, I.; Gangemi, R.; Marshall, G. R.; Orlandini, E. | |
Ionic liquid-promoted green synthesis of biologically relevant diaryl thioethers | 1-gen-2020 | Cuffaro, Doretta; D'Andrea, Felicia; Mezzetta, Andrea; Guazzelli, Lorenzo; Chiappe, Cinzia; Nuti, Elisa; Rossello, Armando | |
Monoaryl derivatives as transthyretin fibril formation inhibitors: Design, synthesis, biological evaluation and structural analysis | 1-gen-2020 | Ciccone, L.; Nencetti, S.; Tonali, Nicolo; Fruchart-Gaillard, C.; Shepard, W.; Nuti, E.; Camodeca, C.; Rossello, A.; Orlandini, E. |