NUTI, ELISA Statistiche
NUTI, ELISA
DIPARTIMENTO DI FARMACIA
Design, synthesis and biological activity of glycoconjugated ADAMTS5 exosite inhibitors: applications in osteoarthritis and ovarian cancer models
2026-01-01 Cuffaro, Doretta; Blagg, Sophie; Yamamoto, Kazuhiro; Pinzi, Luca; Bacchetti, Rachele; Yuan, Shengnan; Tew, Simon; Campagnolo, Paola; D'Andrea, Felicia; Crispino, Enrico; Rastelli, Giulio; Rossello, Armando; Rainero, Elena; Nuti, Elisa; Santamaria, Salvatore
Synthesis and Properties of Chemically Modified Cyclodextrins as Drug Delivery Systems: An Update
2026-01-01 Castagnoli, Jacopo; Nuti, Elisa; Piras, Anna Maria; Taliani, Sabrina
Towards circular analytical chemistry: Optimization of colorimetric assay for sustainable and selective dopamine detection in pharmaceutical formulations using green solvents
2026-01-01 Cuffaro, Doretta; Spiaggia, Fabio; Crispino, Enrico; Mezzetta, Andrea; Nuti, Elisa; Calderone, Vincenzo; Guazzelli, Lorenzo; Palladino, Pasquale; Minunni, Maria
A series of benzensulfonamide derivatives as new potent carbonic anhydrase IX and XII inhibitors
2025-01-01 Nencetti, Susanna; Cuffaro, Doretta; Ciccone, Lidia; Nocentini, Alessio; Di Stefano, Miriana; Poli, Giulio; Macchia, Marco; Tuccinardi, Tiziano; Nuti, Elisa; Supuran, Claudiu T.; Rossello, Armando; Orlandini, Elisabetta
Anti-tumor efficacy and Vδ2 T-cell activation via EGFR antibody-drug conjugates featuring novel aminobisphosphonates
2025-01-01 Cuffaro, Doretta; Di Gregorio, Linda; Mangini, Camilla; Taglieri, Martina; Matis, Serena; Benelli, Roberto; Ardy, Massimo; Salvini, Laura; Rossello, Armando; Poggi, Alessandro; Raffaghello, Lizzia; Nuti, Elisa
Identification of novel N-benzyloxy-amino acid hydroxamates as inhibitors of the virulence factor LasB from Pseudomonas aeruginosa
2025-01-01 Di Leo, Riccardo; Crispino, Enrico; Cuffaro, Doretta; Maisetta, Giuseppantonio; Bertacca, Andrea; Bianchi, Marta; Batoni, Giovanna; Wushur, Imin; Rahman, Fatema Amatur; Winberg, Jan-Olof; Sylte, Ingebrigt; Rossello, Armando; Nuti, Elisa
JG26 attenuates ADAM17 metalloproteinase-mediated ACE2 receptor processing and SARS-CoV-2 infection in vitro
2025-01-01 Gentili, Valentina; Beltrami, Silvia; Cuffaro, Doretta; Cianci, Giorgia; Maini, Gloria; Rizzo, Roberta; Macchia, Marco; Rossello, Armando; Bortolotti, Daria; Nuti, Elisa
Multivalent MMP-12 inhibitors as a valuable approach to counteract the intestinal epithelial barrier impairment and inflammation in an in vitro model mimicking intestinal high-fat exposure
2025-01-01 Cuffaro, D.; D'Antongiovanni, V.; Mangini, C.; Di Salvo, C.; Benvenuti, L.; Vandooren, J.; Macchia, M.; Antonioli, L.; Rossello, A.; Fornai, M.; Nuti, E.
The protease ADAMTS5 controls ovarian cancer cell invasion, downstream of Rab25
2025-01-01 Yuan, Shengnan; Bacchetti, Rachele; Adams, Jamie; Cuffaro, Doretta; Rossello, Armando; Nuti, Elisa; Santamaria, Salvatore; Rainero, Elena
TSPO Modulation Prevents Photoreceptor Degeneration and Produces Neuroprotective Effects in an Animal Model of Retinitis Pigmentosa
2025-01-01 Corsi, Francesca; Castagnoli, Jacopo; Galante, Alessia; Fabiano, Angela; Nuti, Elisa; Piras, Anna Maria; Taliani, Sabrina; Piano, Ilaria; Gargini, Claudia
Design, synthesis and biological evaluation of arylsulfonamides as ADAMTS7 inhibitors
2024-01-01 Cuffaro, Doretta; Burkhard, Tina; Bernardoni, Bianca Laura; Di Leo, Riccardo; Zhang, Xiaohan; Galati, Salvatore; Tuccinardi, Tiziano; Macchia, Marco; Rossello, Armando; Santamaria, Salvatore; de Groot, Rens; Nuti, Elisa
iRhom2 regulates ectodomain shedding and surface expression of the major histocompatibility complex (MHC) class I
2024-01-01 Calligaris, Matteo; Spanò, Donatella P; Bonelli, Simone; Müller, Stephan A; Carcione, Claudia; D'Apolito, Danilo; Amico, Giandomenico; Miele, Monica; Di Bella, Mariangela; Zito, Giovanni; Nuti, Elisa; Rossello, Armando; Blobel, Carl P; Lichtenthaler, Stefan F; Scilabra, Simone D
A disintegrin and metalloproteinases (ADAMs) and tumor necrosis factor-alpha-converting enzyme (TACE)
2023-01-01 Cuffaro, Doretta; Scilabra, Simone D.; Spanò, Donatella P.; Calligaris, Matteo; Nuti, Elisa; Rossello, Armando
Bacterial Zinc Metalloenzyme Inhibitors: Recent Advances and Future Perspectives
2023-01-01 Di Leo, Riccardo; Cuffaro, Doretta; Rossello, Armando; Nuti, Elisa
Identification of N-Acyl Hydrazones as New Non-Zinc-Binding MMP-13 Inhibitors by Structure-Based Virtual Screening Studies and Chemical Optimization
2023-01-01 Cuffaro, Doretta; Gimeno, Aleix; Bernardoni, Bianca Laura; Di Leo, Riccardo; Pujadas, Gerard; Garcia-Vallvé, Santiago; Nencetti, Susanna; Rossello, Armando; Nuti, Elisa
New isoxazolidinyl-based N-alkylethanolamines as new activators of human brain carbonic anhydrases
2023-01-01 Cuffaro, Doretta; Di Leo, Riccardo; Ciccone, Lidia; Nocentini, Alessio; Supuran, Claudiu T; Nuti, Elisa; Rossello, Armando
Compounds with a benzo [a]carbazole structure for use in the prevention and/or treatment of infectious diseases
2022-01-01 Rossello, Armando; Nencetti, Susanna; Nuti, Elisa; Orlandini, Elisabetta; Martini, Claudia; Costa, Barbara; Daniele, Simona; Giacomelli, Chiara; Ciccone, Lidia; Cuffaro, Doretta; Comar, Manola
Identification of a Novel p53 Modulator Endowed with Antitumoural and Antibacterial Activity through a Scaffold Repurposing Approach
2022-01-01 Nuti, Elisa; La Pietra, Valeria; Daniele, Simona; Cuffaro, Doretta; Ciccone, Lidia; Giacomelli, Chiara; Cason, Carolina; Carotenuto, Alfonso; D'Amore, Vincenzo Maria; Pozzo, Eleonora Da; Costa, Barbara; Di Leo, Riccardo; Comar, Manola; Marinelli, Luciana; Martini, Claudia; Rossello, Armando
Inhibitors of A Disintegrin And Metalloproteinases-10 reduce Hodgkin lymphoma cell growth in 3D microenvironments and enhance brentuximab-vedotin effect
2022-01-01 Pece, Roberta; Tavella, Sara; Costa, Delfina; Varesano, Serena; Camodeca, Caterina; Cuffaro, Doretta; Nuti, Elisa; Rossello, Armando; Alfano, Massimo; D'Arrigo, Cristina; Galante, Denise; Ravetti, Jean-Louis; Gobbi, Marco; Tosetti, Francesca; Poggi, Alessandro; Zocchi, Maria Raffaella
Targeting Aggrecanases for Osteoarthritis Therapy: From Zinc Chelation to Exosite Inhibition
2022-01-01 Cuffaro, Doretta; Ciccone, Lidia; Rossello, Armando; Nuti, Elisa; Santamaria, Salvatore
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Design, synthesis and biological activity of glycoconjugated ADAMTS5 exosite inhibitors: applications in osteoarthritis and ovarian cancer models | 1-gen-2026 | Cuffaro, Doretta; Blagg, Sophie; Yamamoto, Kazuhiro; Pinzi, Luca; Bacchetti, Rachele; Yuan, Shengnan; Tew, Simon; Campagnolo, Paola; D'Andrea, Felicia; Crispino, Enrico; Rastelli, Giulio; Rossello, Armando; Rainero, Elena; Nuti, Elisa; Santamaria, Salvatore | |
| Synthesis and Properties of Chemically Modified Cyclodextrins as Drug Delivery Systems: An Update | 1-gen-2026 | Castagnoli, Jacopo; Nuti, Elisa; Piras, Anna Maria; Taliani, Sabrina | |
| Towards circular analytical chemistry: Optimization of colorimetric assay for sustainable and selective dopamine detection in pharmaceutical formulations using green solvents | 1-gen-2026 | Cuffaro, Doretta; Spiaggia, Fabio; Crispino, Enrico; Mezzetta, Andrea; Nuti, Elisa; Calderone, Vincenzo; Guazzelli, Lorenzo; Palladino, Pasquale; Minunni, Maria | |
| A series of benzensulfonamide derivatives as new potent carbonic anhydrase IX and XII inhibitors | 1-gen-2025 | Nencetti, Susanna; Cuffaro, Doretta; Ciccone, Lidia; Nocentini, Alessio; Di Stefano, Miriana; Poli, Giulio; Macchia, Marco; Tuccinardi, Tiziano; Nuti, Elisa; Supuran, Claudiu T.; Rossello, Armando; Orlandini, Elisabetta | |
| Anti-tumor efficacy and Vδ2 T-cell activation via EGFR antibody-drug conjugates featuring novel aminobisphosphonates | 1-gen-2025 | Cuffaro, Doretta; Di Gregorio, Linda; Mangini, Camilla; Taglieri, Martina; Matis, Serena; Benelli, Roberto; Ardy, Massimo; Salvini, Laura; Rossello, Armando; Poggi, Alessandro; Raffaghello, Lizzia; Nuti, Elisa | |
| Identification of novel N-benzyloxy-amino acid hydroxamates as inhibitors of the virulence factor LasB from Pseudomonas aeruginosa | 1-gen-2025 | Di Leo, Riccardo; Crispino, Enrico; Cuffaro, Doretta; Maisetta, Giuseppantonio; Bertacca, Andrea; Bianchi, Marta; Batoni, Giovanna; Wushur, Imin; Rahman, Fatema Amatur; Winberg, Jan-Olof; Sylte, Ingebrigt; Rossello, Armando; Nuti, Elisa | |
| JG26 attenuates ADAM17 metalloproteinase-mediated ACE2 receptor processing and SARS-CoV-2 infection in vitro | 1-gen-2025 | Gentili, Valentina; Beltrami, Silvia; Cuffaro, Doretta; Cianci, Giorgia; Maini, Gloria; Rizzo, Roberta; Macchia, Marco; Rossello, Armando; Bortolotti, Daria; Nuti, Elisa | |
| Multivalent MMP-12 inhibitors as a valuable approach to counteract the intestinal epithelial barrier impairment and inflammation in an in vitro model mimicking intestinal high-fat exposure | 1-gen-2025 | Cuffaro, D.; D'Antongiovanni, V.; Mangini, C.; Di Salvo, C.; Benvenuti, L.; Vandooren, J.; Macchia, M.; Antonioli, L.; Rossello, A.; Fornai, M.; Nuti, E. | |
| The protease ADAMTS5 controls ovarian cancer cell invasion, downstream of Rab25 | 1-gen-2025 | Yuan, Shengnan; Bacchetti, Rachele; Adams, Jamie; Cuffaro, Doretta; Rossello, Armando; Nuti, Elisa; Santamaria, Salvatore; Rainero, Elena | |
| TSPO Modulation Prevents Photoreceptor Degeneration and Produces Neuroprotective Effects in an Animal Model of Retinitis Pigmentosa | 1-gen-2025 | Corsi, Francesca; Castagnoli, Jacopo; Galante, Alessia; Fabiano, Angela; Nuti, Elisa; Piras, Anna Maria; Taliani, Sabrina; Piano, Ilaria; Gargini, Claudia | |
| Design, synthesis and biological evaluation of arylsulfonamides as ADAMTS7 inhibitors | 1-gen-2024 | Cuffaro, Doretta; Burkhard, Tina; Bernardoni, Bianca Laura; Di Leo, Riccardo; Zhang, Xiaohan; Galati, Salvatore; Tuccinardi, Tiziano; Macchia, Marco; Rossello, Armando; Santamaria, Salvatore; de Groot, Rens; Nuti, Elisa | |
| iRhom2 regulates ectodomain shedding and surface expression of the major histocompatibility complex (MHC) class I | 1-gen-2024 | Calligaris, Matteo; Spanò, Donatella P; Bonelli, Simone; Müller, Stephan A; Carcione, Claudia; D'Apolito, Danilo; Amico, Giandomenico; Miele, Monica; Di Bella, Mariangela; Zito, Giovanni; Nuti, Elisa; Rossello, Armando; Blobel, Carl P; Lichtenthaler, Stefan F; Scilabra, Simone D | |
| A disintegrin and metalloproteinases (ADAMs) and tumor necrosis factor-alpha-converting enzyme (TACE) | 1-gen-2023 | Cuffaro, Doretta; Scilabra, Simone D.; Spanò, Donatella P.; Calligaris, Matteo; Nuti, Elisa; Rossello, Armando | |
| Bacterial Zinc Metalloenzyme Inhibitors: Recent Advances and Future Perspectives | 1-gen-2023 | Di Leo, Riccardo; Cuffaro, Doretta; Rossello, Armando; Nuti, Elisa | |
| Identification of N-Acyl Hydrazones as New Non-Zinc-Binding MMP-13 Inhibitors by Structure-Based Virtual Screening Studies and Chemical Optimization | 1-gen-2023 | Cuffaro, Doretta; Gimeno, Aleix; Bernardoni, Bianca Laura; Di Leo, Riccardo; Pujadas, Gerard; Garcia-Vallvé, Santiago; Nencetti, Susanna; Rossello, Armando; Nuti, Elisa | |
| New isoxazolidinyl-based N-alkylethanolamines as new activators of human brain carbonic anhydrases | 1-gen-2023 | Cuffaro, Doretta; Di Leo, Riccardo; Ciccone, Lidia; Nocentini, Alessio; Supuran, Claudiu T; Nuti, Elisa; Rossello, Armando | |
| Compounds with a benzo [a]carbazole structure for use in the prevention and/or treatment of infectious diseases | 1-gen-2022 | Rossello, Armando; Nencetti, Susanna; Nuti, Elisa; Orlandini, Elisabetta; Martini, Claudia; Costa, Barbara; Daniele, Simona; Giacomelli, Chiara; Ciccone, Lidia; Cuffaro, Doretta; Comar, Manola | |
| Identification of a Novel p53 Modulator Endowed with Antitumoural and Antibacterial Activity through a Scaffold Repurposing Approach | 1-gen-2022 | Nuti, Elisa; La Pietra, Valeria; Daniele, Simona; Cuffaro, Doretta; Ciccone, Lidia; Giacomelli, Chiara; Cason, Carolina; Carotenuto, Alfonso; D'Amore, Vincenzo Maria; Pozzo, Eleonora Da; Costa, Barbara; Di Leo, Riccardo; Comar, Manola; Marinelli, Luciana; Martini, Claudia; Rossello, Armando | |
| Inhibitors of A Disintegrin And Metalloproteinases-10 reduce Hodgkin lymphoma cell growth in 3D microenvironments and enhance brentuximab-vedotin effect | 1-gen-2022 | Pece, Roberta; Tavella, Sara; Costa, Delfina; Varesano, Serena; Camodeca, Caterina; Cuffaro, Doretta; Nuti, Elisa; Rossello, Armando; Alfano, Massimo; D'Arrigo, Cristina; Galante, Denise; Ravetti, Jean-Louis; Gobbi, Marco; Tosetti, Francesca; Poggi, Alessandro; Zocchi, Maria Raffaella | |
| Targeting Aggrecanases for Osteoarthritis Therapy: From Zinc Chelation to Exosite Inhibition | 1-gen-2022 | Cuffaro, Doretta; Ciccone, Lidia; Rossello, Armando; Nuti, Elisa; Santamaria, Salvatore |