BERTINI, SIMONE Statistiche
BERTINI, SIMONE
DIPARTIMENTO DI FARMACIA
"Soft Drugs" Based on Cannabinoid Receptor Ligands as Potential Local Analgesic and Antiglaucoma Agents
2007-01-01 Minutolo, Filippo; CASCIO M., G; Carboni, I; Bisogno, T; Prota, G; Bertini, Simone; Digiacomo, Maria; Bifulco, M; DI MARZO, V; Macchia, Marco
1,2-Dihydro-2-oxopyridine-3-carboxamides: the C-5 substituent is responsible for functionality switch at CB2 cannabinoid receptor
2014-01-01 Valentina, Lucchesi; Teija, Parkkari; Juha R., Savinainen; Anna Maria, Malfitano; Marco, Allarà; Bertini, Simone; Francesca, Castelli; Sara Del, Carlo; Chiara, Laezza; Alessia, Ligresti; Saccomanni, Giuseppe; Maurizio, Bifulco; Vincenzo Di, Marzo; Macchia, Marco; Manera, Clementina
18FLUORINE-LABELED NITROGEN HETEROCYCLIC DERIVATIVES AS NEW CANDIDATE FOR CANNABINOID CB2 RECEPTOR PET IMAGING
2011-01-01 Castelli, Francesca; Bertini, Simone; DEL CARLO, Sara; Lucchesi, Valentina; Manera, Clementina; Pascali, Giancarlo; Saccomanni, Giuseppe; DI MARZO, Vincenzo; Salvadori, Piero; Macchia, Marco
200 Esercizi Risolti di Chimica Generale ed Inorganica
2006-01-01 Bertini, Simone
4-[6-(dansylamino)hexylamino]-7-methyl-2-phenyl-1,8-naphthyridine as a new potential fluorescent probe for studying A1-adenosine receptor
2002-01-01 Macchia, Marco; Bertini, Simone; DI BUSSOLO, Valeria; Manera, Clementina; Martini, Claudia; Minutolo, Filippo; C., Mori; Saccomanni, Giuseppe; D., Tuscano; Ferrarini, P.
7-Nitrobenzofurazan (NBD)-Derivatives Of 5'-N-Ethylcarboxamidoadenosine (NECA) As New Fluorescent Probes For Human A3 Adenosine Receptors
2001-01-01 Macchia, Marco; Salvetti, F; Bertini, Simone; DI BUSSOLO, Valeria; Gattuso, L; Gesi, Marco; Hamdan, M; KLOTZ K., N; Laragione, T; Lucacchini, Antonio; Minutolo, Filippo; Nencetti, Susanna; Papi, C; Tuscano, D; Martini, Claudia
A theoretical study to investigate D2DAR/D4DAR selectivity: Receptor modeling and molecular docking of dopaminergic ligands
2006-01-01 Ortore, GABRIELLA MARIA PIA; Tuccinardi, Tiziano; Bertini, Simone; Martinelli, Adriano
Allosteric modulators targeting cannabinoid cb1 and cb2 receptors: Implications for drug discovery
2019-01-01 Gado, F.; Meini, S.; Bertini, S.; Digiacomo, M.; Macchia, M.; Manera, C.
alpha-Naphthylaminopropan-2-ol Derivatives as BACE1 Inhibitors
2008-01-01 V., Asso; E., Ghilardi; Bertini, Simone; Digiacomo, Maria; Granchi, Carlotta; Minutolo, Filippo; Rapposelli, Simona; A., Bortolato; S., Moro; Macchia, Marco
alpha-Naphtylaminopropan-2-ol derivatives as BACE1 inhibitors
2008-01-01 V., Asso; E., Ghilardi; Bertini, Simone; Digiacomo, Maria; Granchi, Carlotta; Minutolo, Filippo; Rapposelli, Simona; A., Bortolato; S., Moro; Macchia, Marco
Alternatives to phenol-based estrogen receptor ligands
2003-01-01 Minutolo, Filippo; Antonello, M; Bertini, Simone; Ortore, GABRIELLA MARIA PIA; Rapposelli, Simona; Sheng, S; CARLSON K., E; KATZENELLENBOGEN B., S; KATZENELLENBOGEN J., A; Macchia, Marco
Alzheimer Diseases: Design and synthesis of new BACE inhibitors
2006-01-01 Ghilardi, E; Pericot, G; Asso, V; Bertini, Simone; Minutolo, Filippo; LA ROSA, S; Power, E; Porcari, V; Macchia, Marco; Thomas, R.
Aminobenzothiazoles as beta-Selective Estrogen Receptor Ligands
2006-01-01 Minutolo, Filippo; Bertini, Simone; Rapposelli, Simona; K. E., Carlson; J. A., Katzenellenbogen; F., Stossi; B. S., Katzenellenbogen; Macchia, Marco
Aminobenzothiazoles as inhibitors of tau-fibril formation in Alzheimer's and other neurodegenerative diseases
2008-01-01 Minutolo, Filippo; G., Bellini; Bertini, Simone; Granchi, Carlotta; Macchia, Marco; C., Ballatore; A., Crowe; E., Hyde; K., Brunden; J. Q., Trojanowski; V. M. Y., Lee
Anti-proliferative activity of oleocanthal in human malignant cutaneous melanoma cells
2015-01-01 Arena, C.; Carpi, Sara; Fogli, Stefano; Bertini, S.; Gado, Francesca; Saba, Alessandro; Saccomanni, Giuseppe; Nieri, Paola; Manera, Clementina; Macchia, Marco
Antiproliferative activity and cell cycle analysis of 2-(3,5-dihydroxyphenyl)-6-hydroxybenzothiazole on MCF-7 breast and HCT-15 colon cancer cell lines.
2011-01-01 M., Rajabi; Minutolo, Filippo; Bertini, Simone; Macchia, Marco; R., Ghidoni
Antiproliferative oxime derivatives that inhibit glucose transporter 1 (GLUT1) in cancer cells
2013-01-01 Tuccinardi, Tiziano; Granchi, Carlotta; Jessica, Iegre; Paterni, Ilaria; Bertini, Simone; Macchia, Marco; Martinelli, Adriano; Yanrong, Qian; Xiaozhuo, Chen; Minutolo, Filippo
Application of An Improved HPLC-FL Method to Screen Serine Palmitoyl Transferase Inhibitors
2017-01-01 Bertini, Simone; Saccomanni, Giuseppe; Carlo, Sara Del; Digiacomo, Maria; Gargini, MARIA CLAUDIA; Piano, Ilaria; Campisi, Giuseppe Matteo; Ghidoni, Riccardo; Macchia, Marco; Manera, Clementina
Aromatic aldoximes as Estrogen Receptor Beta–Selective Ligands
2007-01-01 Minutolo, Filippo; Bellini, R; Bertini, Simone; Carboni, I; Gambini, M; Pistolesi, L; Prota, G; Solati, F; Ortore, GABRIELLA MARIA PIA; Tuccinardi, Tiziano; Martinelli, Adriano; CARLSON K., E; KATZENELLENBOGEN J., A; Macchia, Marco
Assessment of a HPLC assay for monoacylglycerol lipase activity
2013-01-01 DEL CARLO, Sara; Arena, Chiara; Chicca, A; Bertini, Simone; Chidini, S; Manera, Clementina; Saccomanni, Giuseppe; Gertsch, J; Macchia, Marco
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
"Soft Drugs" Based on Cannabinoid Receptor Ligands as Potential Local Analgesic and Antiglaucoma Agents | 1-gen-2007 | Minutolo, Filippo; CASCIO M., G; Carboni, I; Bisogno, T; Prota, G; Bertini, Simone; Digiacomo, Maria; Bifulco, M; DI MARZO, V; Macchia, Marco | |
1,2-Dihydro-2-oxopyridine-3-carboxamides: the C-5 substituent is responsible for functionality switch at CB2 cannabinoid receptor | 1-gen-2014 | Valentina, Lucchesi; Teija, Parkkari; Juha R., Savinainen; Anna Maria, Malfitano; Marco, Allarà; Bertini, Simone; Francesca, Castelli; Sara Del, Carlo; Chiara, Laezza; Alessia, Ligresti; Saccomanni, Giuseppe; Maurizio, Bifulco; Vincenzo Di, Marzo; Macchia, Marco; Manera, Clementina | |
18FLUORINE-LABELED NITROGEN HETEROCYCLIC DERIVATIVES AS NEW CANDIDATE FOR CANNABINOID CB2 RECEPTOR PET IMAGING | 1-gen-2011 | Castelli, Francesca; Bertini, Simone; DEL CARLO, Sara; Lucchesi, Valentina; Manera, Clementina; Pascali, Giancarlo; Saccomanni, Giuseppe; DI MARZO, Vincenzo; Salvadori, Piero; Macchia, Marco | |
200 Esercizi Risolti di Chimica Generale ed Inorganica | 1-gen-2006 | Bertini, Simone | |
4-[6-(dansylamino)hexylamino]-7-methyl-2-phenyl-1,8-naphthyridine as a new potential fluorescent probe for studying A1-adenosine receptor | 1-gen-2002 | Macchia, Marco; Bertini, Simone; DI BUSSOLO, Valeria; Manera, Clementina; Martini, Claudia; Minutolo, Filippo; C., Mori; Saccomanni, Giuseppe; D., Tuscano; Ferrarini, P. | |
7-Nitrobenzofurazan (NBD)-Derivatives Of 5'-N-Ethylcarboxamidoadenosine (NECA) As New Fluorescent Probes For Human A3 Adenosine Receptors | 1-gen-2001 | Macchia, Marco; Salvetti, F; Bertini, Simone; DI BUSSOLO, Valeria; Gattuso, L; Gesi, Marco; Hamdan, M; KLOTZ K., N; Laragione, T; Lucacchini, Antonio; Minutolo, Filippo; Nencetti, Susanna; Papi, C; Tuscano, D; Martini, Claudia | |
A theoretical study to investigate D2DAR/D4DAR selectivity: Receptor modeling and molecular docking of dopaminergic ligands | 1-gen-2006 | Ortore, GABRIELLA MARIA PIA; Tuccinardi, Tiziano; Bertini, Simone; Martinelli, Adriano | |
Allosteric modulators targeting cannabinoid cb1 and cb2 receptors: Implications for drug discovery | 1-gen-2019 | Gado, F.; Meini, S.; Bertini, S.; Digiacomo, M.; Macchia, M.; Manera, C. | |
alpha-Naphthylaminopropan-2-ol Derivatives as BACE1 Inhibitors | 1-gen-2008 | V., Asso; E., Ghilardi; Bertini, Simone; Digiacomo, Maria; Granchi, Carlotta; Minutolo, Filippo; Rapposelli, Simona; A., Bortolato; S., Moro; Macchia, Marco | |
alpha-Naphtylaminopropan-2-ol derivatives as BACE1 inhibitors | 1-gen-2008 | V., Asso; E., Ghilardi; Bertini, Simone; Digiacomo, Maria; Granchi, Carlotta; Minutolo, Filippo; Rapposelli, Simona; A., Bortolato; S., Moro; Macchia, Marco | |
Alternatives to phenol-based estrogen receptor ligands | 1-gen-2003 | Minutolo, Filippo; Antonello, M; Bertini, Simone; Ortore, GABRIELLA MARIA PIA; Rapposelli, Simona; Sheng, S; CARLSON K., E; KATZENELLENBOGEN B., S; KATZENELLENBOGEN J., A; Macchia, Marco | |
Alzheimer Diseases: Design and synthesis of new BACE inhibitors | 1-gen-2006 | Ghilardi, E; Pericot, G; Asso, V; Bertini, Simone; Minutolo, Filippo; LA ROSA, S; Power, E; Porcari, V; Macchia, Marco; Thomas, R. | |
Aminobenzothiazoles as beta-Selective Estrogen Receptor Ligands | 1-gen-2006 | Minutolo, Filippo; Bertini, Simone; Rapposelli, Simona; K. E., Carlson; J. A., Katzenellenbogen; F., Stossi; B. S., Katzenellenbogen; Macchia, Marco | |
Aminobenzothiazoles as inhibitors of tau-fibril formation in Alzheimer's and other neurodegenerative diseases | 1-gen-2008 | Minutolo, Filippo; G., Bellini; Bertini, Simone; Granchi, Carlotta; Macchia, Marco; C., Ballatore; A., Crowe; E., Hyde; K., Brunden; J. Q., Trojanowski; V. M. Y., Lee | |
Anti-proliferative activity of oleocanthal in human malignant cutaneous melanoma cells | 1-gen-2015 | Arena, C.; Carpi, Sara; Fogli, Stefano; Bertini, S.; Gado, Francesca; Saba, Alessandro; Saccomanni, Giuseppe; Nieri, Paola; Manera, Clementina; Macchia, Marco | |
Antiproliferative activity and cell cycle analysis of 2-(3,5-dihydroxyphenyl)-6-hydroxybenzothiazole on MCF-7 breast and HCT-15 colon cancer cell lines. | 1-gen-2011 | M., Rajabi; Minutolo, Filippo; Bertini, Simone; Macchia, Marco; R., Ghidoni | |
Antiproliferative oxime derivatives that inhibit glucose transporter 1 (GLUT1) in cancer cells | 1-gen-2013 | Tuccinardi, Tiziano; Granchi, Carlotta; Jessica, Iegre; Paterni, Ilaria; Bertini, Simone; Macchia, Marco; Martinelli, Adriano; Yanrong, Qian; Xiaozhuo, Chen; Minutolo, Filippo | |
Application of An Improved HPLC-FL Method to Screen Serine Palmitoyl Transferase Inhibitors | 1-gen-2017 | Bertini, Simone; Saccomanni, Giuseppe; Carlo, Sara Del; Digiacomo, Maria; Gargini, MARIA CLAUDIA; Piano, Ilaria; Campisi, Giuseppe Matteo; Ghidoni, Riccardo; Macchia, Marco; Manera, Clementina | |
Aromatic aldoximes as Estrogen Receptor Beta–Selective Ligands | 1-gen-2007 | Minutolo, Filippo; Bellini, R; Bertini, Simone; Carboni, I; Gambini, M; Pistolesi, L; Prota, G; Solati, F; Ortore, GABRIELLA MARIA PIA; Tuccinardi, Tiziano; Martinelli, Adriano; CARLSON K., E; KATZENELLENBOGEN J., A; Macchia, Marco | |
Assessment of a HPLC assay for monoacylglycerol lipase activity | 1-gen-2013 | DEL CARLO, Sara; Arena, Chiara; Chicca, A; Bertini, Simone; Chidini, S; Manera, Clementina; Saccomanni, Giuseppe; Gertsch, J; Macchia, Marco |