MARTINELLI, ADRIANO Statistiche

MARTINELLI, ADRIANO  

DIPARTIMENTO DI FARMACIA  

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Titolo Data di pubblicazione Autore(i) File
From Anti-infective Agents to Cancer Therapy: a Drug Repositioning Study Revealed a New Use for Nitrofuran Derivatives 1-gen-2022 Ortore, Gabriella; Poli, Giulio; Martinelli, Adriano; Tuccinardi, Tiziano; Rizzolio, Flavio; Caligiuri, Isabella
VenomPred: A Machine Learning Based Platform for Molecular Toxicity Predictions 1-gen-2022 Galati, Salvatore; Di Stefano, Miriana; Martinelli, Elisa; Macchia, Marco; Martinelli, Adriano; Poli, Giulio; Tuccinardi, Tiziano
Development of a cheminformatics platform for selectivity analyses of carbonic anhydrase inhibitors 1-gen-2020 Poli, G.; Galati, S.; Martinelli, A.; Supuran, C. T.; Tuccinardi, T.
Extensive reliability evaluation of docking-based target-fishing strategies 1-gen-2019 Lapillo, M.; Tuccinardi, T.; Martinelli, A.; Macchia, M.; Giordano, A.; Poli, G.
Development of a Fingerprint-Based Scoring Function for the Prediction of the Binding Mode of Carbonic Anhydrase II Inhibitors 1-gen-2018 Poli, Giulio; Jha, Vibhu; Martinelli, Adriano; Supuran, Claudiu T; Tuccinardi, Tiziano
Discovery of 1,5-Diphenylpyrazole-3-Carboxamide Derivatives as Potent, Reversible, and Selective Monoacylglycerol Lipase (MAGL) Inhibitors 1-gen-2018 Aghazadeh Tabrizi, Mojgan; Baraldi, Pier Giovanni; Baraldi, Stefania; Ruggiero, Emanuela; De Stefano, Lucia; Rizzolio, Flavio; Di Cesare Mannelli, Lorenzo; Ghelardini, Carla; Chicca, Andrea; Lapillo, Margherita; Gertsch, Jürg; Manera, Clementina; Macchia, Marco; Martinelli, Adriano; Granchi, Carlotta; Minutolo, Filippo; Tuccinardi, Tiziano
Discovery of long-chain salicylketoxime derivatives as monoacylglycerol lipase (MAGL) inhibitors 1-gen-2018 Bononi, Giulia; Granchi, Carlotta; Lapillo, Margherita; Giannotti, Massimiliano; Nieri, Daniela; Fortunato, Serena; Boustani, Maguie El; Caligiuri, Isabella; Poli, Giulio; Carlson, Kathryn E.; Kim, Sung Hoon; Macchia, Marco; Martinelli, Adriano; Rizzolio, Flavio; Chicca, Andrea; Katzenellenbogen, John A.; Minutolo, Filippo; Tuccinardi, Tiziano
Identification of Lactate Dehydrogenase 5 Inhibitors using Pharmacophore- Driven Consensus Docking 1-gen-2018 Poli, Giulio; Scarpino, Andrea; Aissaoui, Mohamed; Granchi, Carlotta; Minutolo, Filippo; Martinelli, Adriano; Tuccinardi, Tiziano
Rational Development of MAGL Inhibitors 1-gen-2018 Granchi, Carlotta; Rizzolio, Flavio; Caligiuri, Isabella; Macchia, Marco; Martinelli, Adriano; Minutolo, Filippo; Tuccinardi, Tiziano
Chimica - VI Edizione Copyright © 2017, EdiSES srl - Napoli 1-gen-2017 Battistuzzi, Gianantonio; Bergamini, Paola; Botta, Mauro; Carbonaro, Laura; Carcelli, Mauro; De Guidi, Guido; Pia Donzello, Maria; Drava, Giuliana; Ennas, Guido; Favero, Lucilla; Fiore, Tiziana; Assunta Girasolo, Maria; Iannelli, Pio; Lamastra, Lucrezia; Leone, Gemma; Magnani, Agnese; Martinelli, Adriano; Monzani, Enrico; Operti, Lorenza; Panzavolta, Silvia; Ruffo, Francesco; Tarallo, Oresto; Terreno, Enzo
Development of terphenyl-2-methyloxazol-5(4H)-one derivatives as selective reversible MAGL inhibitors 1-gen-2017 Granchi, Carlotta; Caligiuri, Isabella; Bertelli, Eleonora; Poli, Giulio; Rizzolio, Flavio; Macchia, Marco; Martinelli, Adriano; Minutolo, Filippo; Tuccinardi, Tiziano
Identification of Transthyretin Fibril Formation Inhibitors Using Structure-Based Virtual Screening 1-gen-2017 Ortore, GABRIELLA MARIA PIA; Martinelli, Adriano
4-Aryliden-2-methyloxazol-5(4H)-one as a new scaffold for selective reversible MAGL inhibitors 1-gen-2016 Granchi, Carlotta; Rizzolio, F; Bordoni, Vittorio; Caligiuri, I; Manera, Clementina; Macchia, Marco; Minutolo, Filippo; Martinelli, Adriano; Giordano, A; Tuccinardi, Tiziano
A STRUCTURE-BASED VIRTUAL SCREENING TO IDENTIFY NEW SCAFFOLDS FOR TRANSTHYRETIN FIBRIL FORMATION INHIBITORS 1-gen-2016 Ortore, G.; Martinelli, A.
A Virtual Screening Study for Lactate Dehydrogenase 5 Inhibitors by using a Pharmacophore-Based Approach 1-gen-2016 Tuccinardi, Tiziano; Poli, Giulio; Corchia, Isacco; Granchi, Carlotta; Lapillo, Margherita; Macchia, Marco; Minutolo, Filippo; Ortore, GABRIELLA MARIA PIA; Martinelli, Adriano
Identification of a new STAT3 dimerization inhibitor through a pharmacophore-based virtual screening approach 1-gen-2016 Poli, Giulio; Gelain, Arianna; Porta, Federica; Asai, Akira; Martinelli, Adriano; Tuccinardi, Tiziano
Reliability analysis and optimization of the consensus docking approach for the development of virtual screening studies 1-gen-2016 Poli, Giulio; Martinelli, Adriano; Tuccinardi, Tiziano
Structural optimization of 4-chlorobenzoylpiperidine derivatives for the development of potent, reversible and selective monoacylglycerol lipase (MAGL) inhibitors 1-gen-2016 Granchi, Carlotta; Rizzolio, Flavio; Palazzolo, Stefano; Carmignani, Sara; Macchia, Marco; Saccomanni, Giuseppe; Manera, Clementina; Martinelli, Adriano; Minutolo, Filippo; Tuccinardi, Tiziano
Targeting Different Transthyretin Binding Sites with Unusual Natural Compounds 1-gen-2016 Ortore, GABRIELLA MARIA PIA; Orlandini, Elisabetta; Braca, Alessandra; Ciccone, Lidia; Rossello, Armando; Martinelli, Adriano; Nencetti, Susanna
Application of a FLAP-Consensus Docking Mixed Strategy for the Identification of New FAAH Inhibitors 1-gen-2015 Poli, Giulio; Giuntini, N; Martinelli, Adriano; Tuccinardi, Tiziano