CHIELLINI, GRAZIA Statistiche
CHIELLINI, GRAZIA
DIPARTIMENTO DI PATOLOGIA CHIRURGICA, MEDICA, MOLECOLARE E DELL'AREA CRITICA
New Insights into Bitopic Orthosteric/Allosteric Ligands of Cannabinoid Receptor Type 2
2023-01-01 Ferrisi, Rebecca; Polini, Beatrice; Ricardi, Caterina; Gado, Francesca; Mohamed, Kawthar A; Baron, Giovanna; Faiella, Salvatore; Poli, Giulio; Rapposelli, Simona; Saccomanni, Giuseppe; Aldini, Giancarlo; Chiellini, Grazia; Laprairie, Robert B; Manera, Clementina; Ortore, Gabriella
New Insights into Bitopic Orthosteric/Allosteric Ligands of Cannabinoid Receptor Type 2
2023-01-01 Ferrisi, Rebecca; Polini, Beatrice; Ricardi, Caterina; Gado, Francesca; Mohamed, Kawthar A; Baron, Giovanna; Faiella, Salvatore; Poli, Giulio; Rapposelli, Simona; Saccomanni, Giuseppe; Aldini, Giancarlo; Chiellini, Grazia; Laprairie, Robert B; Manera, Clementina; Ortore, Gabriella
An Efficient Aequorea victoria Green Fluorescent Protein for Stimulated Emission Depletion Super-Resolution Microscopy
2022-01-01 Storti, B.; Carlotti, B.; Chiellini, G.; Ruglioni, M.; Salvadori, T.; Scotto, M.; Elisei, F.; Diaspro, A.; Bianchini, P.; Bizzarri, R.
Design, synthesis and biological evaluation of novel orthosteric-allosteric ligands of the cannabinoid receptor type 2 (CB2R)
2022-01-01 Ferrisi, Rebecca; Gado, Francesca; Polini, Beatrice; Ricardi, Caterina; Mohamed, Kawthar A.; Stevenson, Lesley A.; Ortore, GABRIELLA MARIA PIA; Rapposelli, Simona; Saccomanni, Giuseppe; Pertwee, Roger G.; Laprairie, Robert B.; Manera, Clementina; Chiellini, Grazia
Design, Synthesis, and Biological Activity of New CB2 Receptor Ligands: from Orthosteric and Allosteric Modulators to Dualsteric/Bitopic Ligands
2022-01-01 Gado, Francesca; Ferrisi, Rebecca; Polini, Beatrice; Mohamed, Kawthar A.; Ricardi, Caterina; Lucarini, Elena; Carpi, Sara; Domenichini, Federica; Stevenson, Lesley A.; Rapposelli, Simona; Saccomanni, Giuseppe; Nieri, Paola; Ortore, GABRIELLA MARIA PIA; Pertwee, Roger G.; Ghelardini, Carla; Di Cesare Mannelli, Lorenzo; Chiellini, Grazia; Laprairie, Robert B.; Manera, Clementina
Editorial: Calcium Metabolism: Hormonal Crosstalk, Pathophysiology and Disease
2022-01-01 Battafarano, Giulia; Chiellini, Grazia; Saponaro, Federica
Delivery of thyronamines (Tams) to the brain: A preliminary study
2021-01-01 Di Leo, N.; Moscato, S.; Borso', M.; Sestito, S.; Polini, B.; Bandini, L.; Grillone, A.; Battaglini, M.; Saba, A.; Mattii, L.; Ciofani, G.; Chiellini, G.
Diphenyl-methane based thyromimetic inhibitors for transthyretin amyloidosis
2021-01-01 Kim, B.; Ko, Y. H.; Runfola, M.; Rapposelli, S.; Ortore, G.; Chiellini, G.; Kim, J. H.
Identification of a Thyroid Hormone Derivative as a Pleiotropic Agent for the Treatment of Alzheimer's Disease
2021-01-01 Runfola, Massimiliano; Perni, Michele; Yang, Xiaoting; Marchese, Maria; Bacci, Andrea; Mero, Serena; Santorelli, Filippo M; Polini, Beatrice; Chiellini, Grazia; Giuliani, Daniela; Vilella, Antonietta; Bodria, Martina; Daini, Eleonora; Vandini, Eleonora; Rudge, Simon; Gul, Sheraz; Wakelam, Michale O J; Vendruscolo, Michele; Rapposelli, Simona
SG‐2: A SYNTHETIC ANALOG OF THYROID HORMONE METABOLITE 3‐IODOTHYRONAMINE (T1AM), PREVENTS β‐AMYLOID NEUROTOXICITY IN VITRO
2021-01-01 Polini, Beatrice; Carnicelli, Vittoria; Runfola, Massimiliano; Rapposelli, Simona; Zucchi, Riccardo; Chiellini, Grazia
The role of cannabinoids in bone metabolism: A new perspective for bone disorders
2021-01-01 Saponaro, F.; Ferrisi, R.; Gado, F.; Polini, B.; Saba, A.; Manera, C.; Chiellini, G.
Understanding amyloid structures and disease: A continuing challenge in health research
2021-01-01 Chiellini, G.
3-iodothyronamine affects thermogenic substrates’ mobilization in brown adipocytes
2020-01-01 Gencarelli, M.; Laurino, A.; Landucci, E.; Buonvicino, D.; Mazzantini, C.; Chiellini, G.; Raimondi, L.
3-Iodothyronamine and Derivatives: New Allies Against Metabolic Syndrome?
2020-01-01 Rutigliano, Grazia; Bandini, Lavinia; Sestito, Simona; Chiellini, Grazia
Collecting data through high throughput in vitro early toxicity and off-target liability assays to rapidly identify limitations of novel thyromimetics
2020-01-01 Runfola, M.; Sestito, S.; Gul, S.; Chiellini, G.; Rapposelli, S.
Design, synthesis and biological evaluation of novel TRβ selective agonists sustained by ADME-toxicity analysis
2020-01-01 Runfola, Massimiliano; Sestito, Simona; Bellusci, Lorenza; La Pietra, Valeria; D'Amore, Vincenzo Maria; Kowalik, Marta Anna; Chiellini, Grazia; Gul, Sheraz; Perra, Andrea; Columbano, Amedeo; Marinelli, Luciana; Novellino, Ettore; Rapposelli, Simona
Endogenous 3-iodothyronamine (T1Am) and synthetic thyronamine-like analog SG-2 act as novel pleiotropic neuroprotective agents through the modulation of SIRT6
2020-01-01 Bellusci, L.; Runfola, M.; Carnicelli, V.; Sestito, S.; Fulceri, F.; Santucci, F.; Lenzi, P.; Fornai, F.; Rapposelli, S.; Origlia, N.; Zucchi, R.; Chiellini, G.
Late Breaker: Posters
2020-01-01 Perra, Andrea; Anna Kowalik, Marta; Cabras, Lavinia; Onali, Simona; Migliore, Cristina; Giordano, Silvia; Chiellini, Grazia; Rapposelli, Simona; Columbano., Amedeo
Metabolic Reprogramming in Health and Disease
2020-01-01 Chiellini, Grazia
NOVEL THYROMIMETICS WITH A BIPHENYLMETHANE SCAFFOLD AND THEIR USE
2020-01-01 Puricelli, Guido; Rapposelli, Simona; Chiellini, Grazia; Columbano, Amedeo; Perra, Andrea; Runfola, Massimiliano; Gul, Sheraz
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
New Insights into Bitopic Orthosteric/Allosteric Ligands of Cannabinoid Receptor Type 2 | 1-gen-2023 | Ferrisi, Rebecca; Polini, Beatrice; Ricardi, Caterina; Gado, Francesca; Mohamed, Kawthar A; Baron, Giovanna; Faiella, Salvatore; Poli, Giulio; Rapposelli, Simona; Saccomanni, Giuseppe; Aldini, Giancarlo; Chiellini, Grazia; Laprairie, Robert B; Manera, Clementina; Ortore, Gabriella | |
New Insights into Bitopic Orthosteric/Allosteric Ligands of Cannabinoid Receptor Type 2 | 1-gen-2023 | Ferrisi, Rebecca; Polini, Beatrice; Ricardi, Caterina; Gado, Francesca; Mohamed, Kawthar A; Baron, Giovanna; Faiella, Salvatore; Poli, Giulio; Rapposelli, Simona; Saccomanni, Giuseppe; Aldini, Giancarlo; Chiellini, Grazia; Laprairie, Robert B; Manera, Clementina; Ortore, Gabriella | |
An Efficient Aequorea victoria Green Fluorescent Protein for Stimulated Emission Depletion Super-Resolution Microscopy | 1-gen-2022 | Storti, B.; Carlotti, B.; Chiellini, G.; Ruglioni, M.; Salvadori, T.; Scotto, M.; Elisei, F.; Diaspro, A.; Bianchini, P.; Bizzarri, R. | |
Design, synthesis and biological evaluation of novel orthosteric-allosteric ligands of the cannabinoid receptor type 2 (CB2R) | 1-gen-2022 | Ferrisi, Rebecca; Gado, Francesca; Polini, Beatrice; Ricardi, Caterina; Mohamed, Kawthar A.; Stevenson, Lesley A.; Ortore, GABRIELLA MARIA PIA; Rapposelli, Simona; Saccomanni, Giuseppe; Pertwee, Roger G.; Laprairie, Robert B.; Manera, Clementina; Chiellini, Grazia | |
Design, Synthesis, and Biological Activity of New CB2 Receptor Ligands: from Orthosteric and Allosteric Modulators to Dualsteric/Bitopic Ligands | 1-gen-2022 | Gado, Francesca; Ferrisi, Rebecca; Polini, Beatrice; Mohamed, Kawthar A.; Ricardi, Caterina; Lucarini, Elena; Carpi, Sara; Domenichini, Federica; Stevenson, Lesley A.; Rapposelli, Simona; Saccomanni, Giuseppe; Nieri, Paola; Ortore, GABRIELLA MARIA PIA; Pertwee, Roger G.; Ghelardini, Carla; Di Cesare Mannelli, Lorenzo; Chiellini, Grazia; Laprairie, Robert B.; Manera, Clementina | |
Editorial: Calcium Metabolism: Hormonal Crosstalk, Pathophysiology and Disease | 1-gen-2022 | Battafarano, Giulia; Chiellini, Grazia; Saponaro, Federica | |
Delivery of thyronamines (Tams) to the brain: A preliminary study | 1-gen-2021 | Di Leo, N.; Moscato, S.; Borso', M.; Sestito, S.; Polini, B.; Bandini, L.; Grillone, A.; Battaglini, M.; Saba, A.; Mattii, L.; Ciofani, G.; Chiellini, G. | |
Diphenyl-methane based thyromimetic inhibitors for transthyretin amyloidosis | 1-gen-2021 | Kim, B.; Ko, Y. H.; Runfola, M.; Rapposelli, S.; Ortore, G.; Chiellini, G.; Kim, J. H. | |
Identification of a Thyroid Hormone Derivative as a Pleiotropic Agent for the Treatment of Alzheimer's Disease | 1-gen-2021 | Runfola, Massimiliano; Perni, Michele; Yang, Xiaoting; Marchese, Maria; Bacci, Andrea; Mero, Serena; Santorelli, Filippo M; Polini, Beatrice; Chiellini, Grazia; Giuliani, Daniela; Vilella, Antonietta; Bodria, Martina; Daini, Eleonora; Vandini, Eleonora; Rudge, Simon; Gul, Sheraz; Wakelam, Michale O J; Vendruscolo, Michele; Rapposelli, Simona | |
SG‐2: A SYNTHETIC ANALOG OF THYROID HORMONE METABOLITE 3‐IODOTHYRONAMINE (T1AM), PREVENTS β‐AMYLOID NEUROTOXICITY IN VITRO | 1-gen-2021 | Polini, Beatrice; Carnicelli, Vittoria; Runfola, Massimiliano; Rapposelli, Simona; Zucchi, Riccardo; Chiellini, Grazia | |
The role of cannabinoids in bone metabolism: A new perspective for bone disorders | 1-gen-2021 | Saponaro, F.; Ferrisi, R.; Gado, F.; Polini, B.; Saba, A.; Manera, C.; Chiellini, G. | |
Understanding amyloid structures and disease: A continuing challenge in health research | 1-gen-2021 | Chiellini, G. | |
3-iodothyronamine affects thermogenic substrates’ mobilization in brown adipocytes | 1-gen-2020 | Gencarelli, M.; Laurino, A.; Landucci, E.; Buonvicino, D.; Mazzantini, C.; Chiellini, G.; Raimondi, L. | |
3-Iodothyronamine and Derivatives: New Allies Against Metabolic Syndrome? | 1-gen-2020 | Rutigliano, Grazia; Bandini, Lavinia; Sestito, Simona; Chiellini, Grazia | |
Collecting data through high throughput in vitro early toxicity and off-target liability assays to rapidly identify limitations of novel thyromimetics | 1-gen-2020 | Runfola, M.; Sestito, S.; Gul, S.; Chiellini, G.; Rapposelli, S. | |
Design, synthesis and biological evaluation of novel TRβ selective agonists sustained by ADME-toxicity analysis | 1-gen-2020 | Runfola, Massimiliano; Sestito, Simona; Bellusci, Lorenza; La Pietra, Valeria; D'Amore, Vincenzo Maria; Kowalik, Marta Anna; Chiellini, Grazia; Gul, Sheraz; Perra, Andrea; Columbano, Amedeo; Marinelli, Luciana; Novellino, Ettore; Rapposelli, Simona | |
Endogenous 3-iodothyronamine (T1Am) and synthetic thyronamine-like analog SG-2 act as novel pleiotropic neuroprotective agents through the modulation of SIRT6 | 1-gen-2020 | Bellusci, L.; Runfola, M.; Carnicelli, V.; Sestito, S.; Fulceri, F.; Santucci, F.; Lenzi, P.; Fornai, F.; Rapposelli, S.; Origlia, N.; Zucchi, R.; Chiellini, G. | |
Late Breaker: Posters | 1-gen-2020 | Perra, Andrea; Anna Kowalik, Marta; Cabras, Lavinia; Onali, Simona; Migliore, Cristina; Giordano, Silvia; Chiellini, Grazia; Rapposelli, Simona; Columbano., Amedeo | |
Metabolic Reprogramming in Health and Disease | 1-gen-2020 | Chiellini, Grazia | |
NOVEL THYROMIMETICS WITH A BIPHENYLMETHANE SCAFFOLD AND THEIR USE | 1-gen-2020 | Puricelli, Guido; Rapposelli, Simona; Chiellini, Grazia; Columbano, Amedeo; Perra, Andrea; Runfola, Massimiliano; Gul, Sheraz |