GALATI, SALVATORE Statistiche
GALATI, SALVATORE
DIPARTIMENTO DI CHIMICA E CHIMICA INDUSTRIALE
An update on antibacterial AlkylGuanidino Ureas: Design of new derivatives, synergism with colistin and data analysis of the whole library
2024-01-01 Ardino, Claudia; Sannio, Filomena; Poli, Giulio; Galati, Salvatore; Dreassi, Elena; Botta, Lorenzo; Docquier, Jean-Denis; D'Agostino, Ilaria
Design, synthesis and biological evaluation of arylsulfonamides as ADAMTS7 inhibitors
2024-01-01 Cuffaro, Doretta; Burkhard, Tina; Bernardoni, Bianca Laura; Di Leo, Riccardo; Zhang, Xiaohan; Galati, Salvatore; Tuccinardi, Tiziano; Macchia, Marco; Rossello, Armando; Santamaria, Salvatore; de Groot, Rens; Nuti, Elisa
Design, synthesis, ADME and biological evaluation of benzylpiperidine and benzylpiperazine derivatives as novel reversible monoacylglycerol lipase (MAGL) inhibitors
2024-01-01 Di Stefano, Miriana; Masoni, Samuele; Bononi, Giulia; Poli, Giulio; Galati, Salvatore; Gado, Francesca; Manzi, Simone; Vagaggini, Chiara; Brai, Annalaura; Caligiuri, Isabella; Asif, Kanwal; Rizzolio, Flavio; Macchia, Marco; Chicca, Andrea; Sodi, Andrea; Di Bussolo, Valeria; Minutolo, Filippo; Meier, Philip; Gertsch, Jürg; Granchi, Carlotta; Dreassi, Elena; Tuccinardi, Tiziano
VenomPred 2.0: A Novel In Silico Platform for an Extended and Human Interpretable Toxicological Profiling of Small Molecules
2024-01-01 Di Stefano, Miriana; Galati, Salvatore; Piazza, Lisa; Granchi, Carlotta; Mancini, Simone; Fratini, Filippo; Macchia, Marco; Poli, Giulio; Tuccinardi, Tiziano
WaSPred: A reliable AI-based water solubility predictor for small molecules
2024-01-01 Di Stefano, Miriana; Galati, Salvatore; Lonzi, Chiara; Granchi, Carlotta; Poli, Giulio; Tuccinardi, Tiziano; Macchia, Marco
Watermelon: setup and validation of an in silico fragment-based approach
2024-01-01 Di Stefano, Miriana; Galati, Salvatore; Piazza, Lisa; Gado, Francesca; Granchi, Carlotta; Macchia, Marco; Giordano, Antonio; Tuccinardi, Tiziano; Poli, Giulio
Identification of New GSK3β Inhibitors through a Consensus Machine Learning-Based Virtual Screening
2023-01-01 Galati, Salvatore; Di Stefano, Miriana; Bertini, Simone; Granchi, Carlotta; Giordano, Antonio; Gado, Francesca; Macchia, Marco; Tuccinardi, Tiziano; Poli, Giulio
MolBook UNIPI─Create, Manage, Analyze, and Share Your Chemical Data for Free
2023-01-01 Galati, Salvatore; Di Stefano, Miriana; Macchia, Marco; Poli, Giulio; Tuccinardi, Tiziano
Identification of Human Dihydroorotate Dehydrogenase Inhibitor by a Pharmacophore-Based Virtual Screening Study
2022-01-01 Galati, Salvatore; Sainas, Stefano; Giorgis, Marta; Boschi, Donatella; Lolli, Marco L; Ortore, Gabriella; Poli, Giulio; Tuccinardi, Tiziano
Machine Learning-Based Virtual Screening for the Identification of Cdk5 Inhibitors
2022-01-01 Di Stefano, Miriana; Galati, Salvatore; Ortore, Gabriella; Caligiuri, Isabella; Rizzolio, Flavio; Ceni, Costanza; Bertini, Simone; Bononi, Giulia; Granchi, Carlotta; Macchia, Marco; Poli, Giulio; Tuccinardi, Tiziano
Resveratrol Analogues as Dual Inhibitors of Monoamine Oxidase B and Carbonic Anhydrase VII: A New Multi-Target Combination for Neurodegenerative Diseases?
2022-01-01 Carradori, Simone; Fantacuzzi, Marialuigia; Ammazzalorso, Alessandra; Angeli, Andrea; De Filippis, Barbara; Galati, Salvatore; Petzer, Anél; Petzer, Jacobus P; Poli, Giulio; Tuccinardi, Tiziano; Agamennone, Mariangela; Supuran, Claudiu T
VenomPred: A Machine Learning Based Platform for Molecular Toxicity Predictions
2022-01-01 Galati, Salvatore; Di Stefano, Miriana; Martinelli, Elisa; Macchia, Marco; Martinelli, Adriano; Poli, Giulio; Tuccinardi, Tiziano
Discovery of a new ATP-citrate lyase (ACLY) inhibitor identified by a pharmacophore-based virtual screening study
2021-01-01 Jha, V.; Galati, S.; Volpi, V.; Ciccone, L.; Minutolo, F.; Rizzolio, F.; Granchi, C.; Poli, G.; Tuccinardi, T.
Predicting Isoform-Selective Carbonic Anhydrase Inhibitors via Machine Learning and Rationalizing Structural Features Important for Selectivity
2021-01-01 Galati, S.; Yonchev, D.; Rodriguez-Perez, R.; Vogt, M.; Tuccinardi, T.; Bajorath, J.
Recent advances in in silico target fishing
2021-01-01 Galati, S.; Di Stefano, M.; Martinelli, E.; Poli, G.; Tuccinardi, T.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
An update on antibacterial AlkylGuanidino Ureas: Design of new derivatives, synergism with colistin and data analysis of the whole library | 1-gen-2024 | Ardino, Claudia; Sannio, Filomena; Poli, Giulio; Galati, Salvatore; Dreassi, Elena; Botta, Lorenzo; Docquier, Jean-Denis; D'Agostino, Ilaria | |
Design, synthesis and biological evaluation of arylsulfonamides as ADAMTS7 inhibitors | 1-gen-2024 | Cuffaro, Doretta; Burkhard, Tina; Bernardoni, Bianca Laura; Di Leo, Riccardo; Zhang, Xiaohan; Galati, Salvatore; Tuccinardi, Tiziano; Macchia, Marco; Rossello, Armando; Santamaria, Salvatore; de Groot, Rens; Nuti, Elisa | |
Design, synthesis, ADME and biological evaluation of benzylpiperidine and benzylpiperazine derivatives as novel reversible monoacylglycerol lipase (MAGL) inhibitors | 1-gen-2024 | Di Stefano, Miriana; Masoni, Samuele; Bononi, Giulia; Poli, Giulio; Galati, Salvatore; Gado, Francesca; Manzi, Simone; Vagaggini, Chiara; Brai, Annalaura; Caligiuri, Isabella; Asif, Kanwal; Rizzolio, Flavio; Macchia, Marco; Chicca, Andrea; Sodi, Andrea; Di Bussolo, Valeria; Minutolo, Filippo; Meier, Philip; Gertsch, Jürg; Granchi, Carlotta; Dreassi, Elena; Tuccinardi, Tiziano | |
VenomPred 2.0: A Novel In Silico Platform for an Extended and Human Interpretable Toxicological Profiling of Small Molecules | 1-gen-2024 | Di Stefano, Miriana; Galati, Salvatore; Piazza, Lisa; Granchi, Carlotta; Mancini, Simone; Fratini, Filippo; Macchia, Marco; Poli, Giulio; Tuccinardi, Tiziano | |
WaSPred: A reliable AI-based water solubility predictor for small molecules | 1-gen-2024 | Di Stefano, Miriana; Galati, Salvatore; Lonzi, Chiara; Granchi, Carlotta; Poli, Giulio; Tuccinardi, Tiziano; Macchia, Marco | |
Watermelon: setup and validation of an in silico fragment-based approach | 1-gen-2024 | Di Stefano, Miriana; Galati, Salvatore; Piazza, Lisa; Gado, Francesca; Granchi, Carlotta; Macchia, Marco; Giordano, Antonio; Tuccinardi, Tiziano; Poli, Giulio | |
Identification of New GSK3β Inhibitors through a Consensus Machine Learning-Based Virtual Screening | 1-gen-2023 | Galati, Salvatore; Di Stefano, Miriana; Bertini, Simone; Granchi, Carlotta; Giordano, Antonio; Gado, Francesca; Macchia, Marco; Tuccinardi, Tiziano; Poli, Giulio | |
MolBook UNIPI─Create, Manage, Analyze, and Share Your Chemical Data for Free | 1-gen-2023 | Galati, Salvatore; Di Stefano, Miriana; Macchia, Marco; Poli, Giulio; Tuccinardi, Tiziano | |
Identification of Human Dihydroorotate Dehydrogenase Inhibitor by a Pharmacophore-Based Virtual Screening Study | 1-gen-2022 | Galati, Salvatore; Sainas, Stefano; Giorgis, Marta; Boschi, Donatella; Lolli, Marco L; Ortore, Gabriella; Poli, Giulio; Tuccinardi, Tiziano | |
Machine Learning-Based Virtual Screening for the Identification of Cdk5 Inhibitors | 1-gen-2022 | Di Stefano, Miriana; Galati, Salvatore; Ortore, Gabriella; Caligiuri, Isabella; Rizzolio, Flavio; Ceni, Costanza; Bertini, Simone; Bononi, Giulia; Granchi, Carlotta; Macchia, Marco; Poli, Giulio; Tuccinardi, Tiziano | |
Resveratrol Analogues as Dual Inhibitors of Monoamine Oxidase B and Carbonic Anhydrase VII: A New Multi-Target Combination for Neurodegenerative Diseases? | 1-gen-2022 | Carradori, Simone; Fantacuzzi, Marialuigia; Ammazzalorso, Alessandra; Angeli, Andrea; De Filippis, Barbara; Galati, Salvatore; Petzer, Anél; Petzer, Jacobus P; Poli, Giulio; Tuccinardi, Tiziano; Agamennone, Mariangela; Supuran, Claudiu T | |
VenomPred: A Machine Learning Based Platform for Molecular Toxicity Predictions | 1-gen-2022 | Galati, Salvatore; Di Stefano, Miriana; Martinelli, Elisa; Macchia, Marco; Martinelli, Adriano; Poli, Giulio; Tuccinardi, Tiziano | |
Discovery of a new ATP-citrate lyase (ACLY) inhibitor identified by a pharmacophore-based virtual screening study | 1-gen-2021 | Jha, V.; Galati, S.; Volpi, V.; Ciccone, L.; Minutolo, F.; Rizzolio, F.; Granchi, C.; Poli, G.; Tuccinardi, T. | |
Predicting Isoform-Selective Carbonic Anhydrase Inhibitors via Machine Learning and Rationalizing Structural Features Important for Selectivity | 1-gen-2021 | Galati, S.; Yonchev, D.; Rodriguez-Perez, R.; Vogt, M.; Tuccinardi, T.; Bajorath, J. | |
Recent advances in in silico target fishing | 1-gen-2021 | Galati, S.; Di Stefano, M.; Martinelli, E.; Poli, G.; Tuccinardi, T. |