Sfoglia per Autore
Synthesis and β-adrenergic properties of tetrahydronaphthalene analogs of dichloroisoproterenol
1993-01-01 Balsamo, A; Breschi, MARIA CRISTINA; Giannaccini, Gino; Lapucci, Annalina; Lucacchini, Antonio; Macchia, B; Manera, Clementina; Martini, Claudia; Martinotti, E; Nencetti, Susanna; Rossello, Armando; Scatizzi, R.
The [(Methyloxy)imino]methyl Moiety as a Bioisoster of Aryl. A Novel Class of Completely Aliphatic Beta-Adrenergic Receptor Antagonists
1994-01-01 Macchia, Bruno; Balsamo, Aldo; Breschi, MARIA CRISTINA; Chiellini, Grazia; Macchia, Marco; Martinelli, Adriano; Martini, Claudia; Nardini, C; Nencetti, Susanna; Rossello, Armando; Scatizzi, R.
SYNTHESIS, ANTIINFLAMMATORY ACTIVITY AND MOLECULAR-ORBITAL STUDIES OF A SERIES OF BENZYLIDENEAMINOXYPROPIONIC ACIDS SUBSTITUTED ON THE PHENYL RING
1994-01-01 Lapucci, Annalina; Macchia, Marco; Martinelli, Adriano; Nencetti, Susanna; Orlandini, Elisabetta; Rossello, Armando; Baldacci, M; Soldani, G; Mengozzi, G.
Conformationally restrained ß-blocking oxime ethers. 2. Synthesis and ß-adrenergic properties of diastereoisomeric anti and syn 2-(5’-(3’-aryl-substituted)isoxazolidinyl)-N-alkylethanolamines
1994-01-01 A., Balsamo; Breschi, MARIA CRISTINA; Chiellini, Grazia; Lucacchini, Antonio; Macchia, Marco; Martinelli, Adriano; Martini, Claudia; C., Nardini; Orlandini, Elisabetta; F., Romagnoli; Rossello, Armando
BIOISOSTERS OF THE DIPHOSPHATE GROUP IN ACTIVATED FORMS OF ANTIHERPES VIRUS AGENTS - A THEORETICAL-STUDY
1994-01-01 Macchia, Marco; Martinelli, Adriano; Parkin, A; Rossello, Armando
SYNTHESIS, PLATELET ANTI-AGGREGATING ACTIVITY AND ANTIINFLAMMATORY ACTIVITY OF A SERIES OF BETA-AMINOXYPROPIONIC ACIDS
1994-01-01 Macchia, Marco; Orlandini, Elisabetta; Rossello, Armando; Bertini, S; Soldani, G; Baldacci, M; Gervasi, G.
Synthesis and aldose reductase inhibitory activity of N-(arylsulfonyl)- and N-(aroyl)-N-(arylmethyloxy)glycines
1994-01-01 Balsamo, A; Belfiore, M. S.; Macchia, Marco; Martini, Claudia; Nencetti, Susanna; Orlandini, Elisabetta; Rossello, Armando
X-ray analisis, theoretical studies and a-adrenergic biopharmacological properties of 1-(2,5-dimethoxyphenyl)-2-aminoethanol and its morpholine analogue
1994-01-01 Manera, Clementina; Martinelli, Adriano; Nencetti, Susanna; F., Romagnoli; Rossello, Armando; Giannaccini, Gino; R., Scatizzi; P., Cozzini; P., Domiano
2-(Methyleneaminoxy)methylmorpholine derivatives. Synthesis and antidepressant activity
1994-01-01 A., Balsamo; Lapucci, Annalina; Macchia, Marco; Martinelli, Adriano; Nencetti, Susanna; T., Cristina; Rossello, Armando
Synthesis and adrenergic ß-blocking activity of (oxypropanolamino)-substituted [(benzylideneamino)oxy]propanolamines
1995-01-01 Balsamo, A; Lapucci, Annalina; Macchia, Bruno; Macchia, Marco; Orlandini, Elisabetta; Rossello, Armando; Ferni, Giovanni; Pinza, Mario
(Z)-(Methyloxyiminomethyl)ethanolamines. Effects of the configuration around the iminic double bond on the beta-adrenergic affinity of moim-type beta-adrenergic blocking agents
1995-01-01 Chiellini, Grazia; Lapucci, Annalina; Macchia, Marco; F., Romagnoli; Rossello, Armando; Nencetti, Susanna
composti dotati di attivita' antivirale e antitumorale, loro preparazione e loro uso farmaceutico
1995-01-01 Balsamo, Aldo; Drago, Lorenzo; GISMONDO MARIA, Rita; Macchia, Franco; Macchia, Bruno; Macchia, Marco; Rossello, Armando
SYNTHESIS AND ANTIMICROBIAL ACTIVITY OF 7-BETA-[N-(ARYLMETHYLOXYIMINO) ACETAMIDO]CEPHALOSPORANIC ACID-DERIVATIVES
1995-01-01 Macchia, Marco; Menchini, E; Orlandini, Elisabetta; Rossello, Armando; Broccali, G; Visconti, M.
SYNTHESIS, ANTIINFLAMMATORY ACTIVITY AND PLATELET ANTIAGGREGATING ACTIVITY OF A NEW SERIES OF BETA-AMINOXYPROPIONIC ACIDS
1995-01-01 Macchia, B; Macchia, Marco; Martinelli, Adriano; Orlandini, Elisabetta; Rossello, Armando; Bertini, S; Luchetti, E; Gervasi, G; Catalani, R.
Synthesis And Antiviral Activity Of Dihydroxycyclohexyl Pirimidine And Purine Carbocyclic Nucleosides
1995-01-01 Rossello, Armando; Calvani, F; Macchia, Marco; Gismondo, Mr; Drago, L; Fassina, Mc; Cisternino, M; Domiano, P.
Synthesis and adrenergic beta-blocking activity of ortho-, meta- and para-oxypropanolamino-substituted [(benzylideneamino)oxy]propanolamines.
1995-01-01 A., Balsamo; Lapucci, Annalina; B., Macchia; Macchia, Marco; Orlandini, Elisabetta; G., Ferni; M., Pinza; Rossello, Armando
Synthesis and ß-adrenergic properties of (E)-N-[3-(alkylamino)-2- hydroxypropilidene](methyloxy)amines substituted with an aromatic group on their [(methyloxy)imino]methyl moiety (MOIMM): an investigation into the biopharmacological effects of an aryl substitution in the class of MOIM ß-blocking drugs.
1995-01-01 Balsamo, A; Breschi, MARIA CRISTINA; Chiellini, Grazia; Favero, Lucilla; Macchia, Marco; Martinelli, Adriano; Martini, Claudia; Rossello, Armando; Scatizzi, R.
(E)-(ARYLMETHYLENEAMINOXY)ACETAMIDES AS ANALOGS OF NEUROLEPTIC BENZAMIDES - SYNTHESIS AND D-2-DOPAMINERGIC BINDING-AFFINITY
1995-01-01 Macchia, Marco; Manera, Clementina; Martinelli, Adriano; Orlandini, Elisabetta; Romagnoli, F; Rossello, Armando; Chiellini, Grazia
Role of the benzylic hydroxyl group of adrenergic catecholamines in eliciting a-adrenergic activity. Synthesis and a1- and a2-adrenergic activity of 3-phenyl-3-piperidinols and of their desoxy analogs
1995-01-01 B., Macchia; Macchia, Marco; Manera, Clementina; E., Martinotti; Nencetti, Susanna; Orlandini, Elisabetta; R., Scatizzi; Rossello, Armando
Conformationally restrained beta-blocking oxime ethers. 3. Synthesis and beta-adrenergic antagonistic activity of diastereomeric anti and syn 2-(5’-(3’-methyl)isoxazolidinyl)-N-alkylethanolamines”.
1996-01-01 Breschi, MARIA CRISTINA; Macchia, Marco; Manera, Clementina; E., Micali; C., Nardini; Nencetti, Susanna; Rossello, Armando; R., Scatizzi
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Synthesis and β-adrenergic properties of tetrahydronaphthalene analogs of dichloroisoproterenol | 1-gen-1993 | Balsamo, A; Breschi, MARIA CRISTINA; Giannaccini, Gino; Lapucci, Annalina; Lucacchini, Antonio; Macchia, B; Manera, Clementina; Martini, Claudia; Martinotti, E; Nencetti, Susanna; Rossello, Armando; Scatizzi, R. | |
The [(Methyloxy)imino]methyl Moiety as a Bioisoster of Aryl. A Novel Class of Completely Aliphatic Beta-Adrenergic Receptor Antagonists | 1-gen-1994 | Macchia, Bruno; Balsamo, Aldo; Breschi, MARIA CRISTINA; Chiellini, Grazia; Macchia, Marco; Martinelli, Adriano; Martini, Claudia; Nardini, C; Nencetti, Susanna; Rossello, Armando; Scatizzi, R. | |
SYNTHESIS, ANTIINFLAMMATORY ACTIVITY AND MOLECULAR-ORBITAL STUDIES OF A SERIES OF BENZYLIDENEAMINOXYPROPIONIC ACIDS SUBSTITUTED ON THE PHENYL RING | 1-gen-1994 | Lapucci, Annalina; Macchia, Marco; Martinelli, Adriano; Nencetti, Susanna; Orlandini, Elisabetta; Rossello, Armando; Baldacci, M; Soldani, G; Mengozzi, G. | |
Conformationally restrained ß-blocking oxime ethers. 2. Synthesis and ß-adrenergic properties of diastereoisomeric anti and syn 2-(5’-(3’-aryl-substituted)isoxazolidinyl)-N-alkylethanolamines | 1-gen-1994 | A., Balsamo; Breschi, MARIA CRISTINA; Chiellini, Grazia; Lucacchini, Antonio; Macchia, Marco; Martinelli, Adriano; Martini, Claudia; C., Nardini; Orlandini, Elisabetta; F., Romagnoli; Rossello, Armando | |
BIOISOSTERS OF THE DIPHOSPHATE GROUP IN ACTIVATED FORMS OF ANTIHERPES VIRUS AGENTS - A THEORETICAL-STUDY | 1-gen-1994 | Macchia, Marco; Martinelli, Adriano; Parkin, A; Rossello, Armando | |
SYNTHESIS, PLATELET ANTI-AGGREGATING ACTIVITY AND ANTIINFLAMMATORY ACTIVITY OF A SERIES OF BETA-AMINOXYPROPIONIC ACIDS | 1-gen-1994 | Macchia, Marco; Orlandini, Elisabetta; Rossello, Armando; Bertini, S; Soldani, G; Baldacci, M; Gervasi, G. | |
Synthesis and aldose reductase inhibitory activity of N-(arylsulfonyl)- and N-(aroyl)-N-(arylmethyloxy)glycines | 1-gen-1994 | Balsamo, A; Belfiore, M. S.; Macchia, Marco; Martini, Claudia; Nencetti, Susanna; Orlandini, Elisabetta; Rossello, Armando | |
X-ray analisis, theoretical studies and a-adrenergic biopharmacological properties of 1-(2,5-dimethoxyphenyl)-2-aminoethanol and its morpholine analogue | 1-gen-1994 | Manera, Clementina; Martinelli, Adriano; Nencetti, Susanna; F., Romagnoli; Rossello, Armando; Giannaccini, Gino; R., Scatizzi; P., Cozzini; P., Domiano | |
2-(Methyleneaminoxy)methylmorpholine derivatives. Synthesis and antidepressant activity | 1-gen-1994 | A., Balsamo; Lapucci, Annalina; Macchia, Marco; Martinelli, Adriano; Nencetti, Susanna; T., Cristina; Rossello, Armando | |
Synthesis and adrenergic ß-blocking activity of (oxypropanolamino)-substituted [(benzylideneamino)oxy]propanolamines | 1-gen-1995 | Balsamo, A; Lapucci, Annalina; Macchia, Bruno; Macchia, Marco; Orlandini, Elisabetta; Rossello, Armando; Ferni, Giovanni; Pinza, Mario | |
(Z)-(Methyloxyiminomethyl)ethanolamines. Effects of the configuration around the iminic double bond on the beta-adrenergic affinity of moim-type beta-adrenergic blocking agents | 1-gen-1995 | Chiellini, Grazia; Lapucci, Annalina; Macchia, Marco; F., Romagnoli; Rossello, Armando; Nencetti, Susanna | |
composti dotati di attivita' antivirale e antitumorale, loro preparazione e loro uso farmaceutico | 1-gen-1995 | Balsamo, Aldo; Drago, Lorenzo; GISMONDO MARIA, Rita; Macchia, Franco; Macchia, Bruno; Macchia, Marco; Rossello, Armando | |
SYNTHESIS AND ANTIMICROBIAL ACTIVITY OF 7-BETA-[N-(ARYLMETHYLOXYIMINO) ACETAMIDO]CEPHALOSPORANIC ACID-DERIVATIVES | 1-gen-1995 | Macchia, Marco; Menchini, E; Orlandini, Elisabetta; Rossello, Armando; Broccali, G; Visconti, M. | |
SYNTHESIS, ANTIINFLAMMATORY ACTIVITY AND PLATELET ANTIAGGREGATING ACTIVITY OF A NEW SERIES OF BETA-AMINOXYPROPIONIC ACIDS | 1-gen-1995 | Macchia, B; Macchia, Marco; Martinelli, Adriano; Orlandini, Elisabetta; Rossello, Armando; Bertini, S; Luchetti, E; Gervasi, G; Catalani, R. | |
Synthesis And Antiviral Activity Of Dihydroxycyclohexyl Pirimidine And Purine Carbocyclic Nucleosides | 1-gen-1995 | Rossello, Armando; Calvani, F; Macchia, Marco; Gismondo, Mr; Drago, L; Fassina, Mc; Cisternino, M; Domiano, P. | |
Synthesis and adrenergic beta-blocking activity of ortho-, meta- and para-oxypropanolamino-substituted [(benzylideneamino)oxy]propanolamines. | 1-gen-1995 | A., Balsamo; Lapucci, Annalina; B., Macchia; Macchia, Marco; Orlandini, Elisabetta; G., Ferni; M., Pinza; Rossello, Armando | |
Synthesis and ß-adrenergic properties of (E)-N-[3-(alkylamino)-2- hydroxypropilidene](methyloxy)amines substituted with an aromatic group on their [(methyloxy)imino]methyl moiety (MOIMM): an investigation into the biopharmacological effects of an aryl substitution in the class of MOIM ß-blocking drugs. | 1-gen-1995 | Balsamo, A; Breschi, MARIA CRISTINA; Chiellini, Grazia; Favero, Lucilla; Macchia, Marco; Martinelli, Adriano; Martini, Claudia; Rossello, Armando; Scatizzi, R. | |
(E)-(ARYLMETHYLENEAMINOXY)ACETAMIDES AS ANALOGS OF NEUROLEPTIC BENZAMIDES - SYNTHESIS AND D-2-DOPAMINERGIC BINDING-AFFINITY | 1-gen-1995 | Macchia, Marco; Manera, Clementina; Martinelli, Adriano; Orlandini, Elisabetta; Romagnoli, F; Rossello, Armando; Chiellini, Grazia | |
Role of the benzylic hydroxyl group of adrenergic catecholamines in eliciting a-adrenergic activity. Synthesis and a1- and a2-adrenergic activity of 3-phenyl-3-piperidinols and of their desoxy analogs | 1-gen-1995 | B., Macchia; Macchia, Marco; Manera, Clementina; E., Martinotti; Nencetti, Susanna; Orlandini, Elisabetta; R., Scatizzi; Rossello, Armando | |
Conformationally restrained beta-blocking oxime ethers. 3. Synthesis and beta-adrenergic antagonistic activity of diastereomeric anti and syn 2-(5’-(3’-methyl)isoxazolidinyl)-N-alkylethanolamines”. | 1-gen-1996 | Breschi, MARIA CRISTINA; Macchia, Marco; Manera, Clementina; E., Micali; C., Nardini; Nencetti, Susanna; Rossello, Armando; R., Scatizzi |
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