MARTINI, CLAUDIA Statistiche
MARTINI, CLAUDIA
DIPARTIMENTO DI FARMACIA
"Indol-3-ylglyoxylylamide derivatives probing the existence of a hydrogen acceptor/donor group in the S1 region of the benzodiazepine receptor binding site"
2000-01-01 G., Primofiore; DA SETTIMO PASSETTI, Federico; Taliani, Sabrina; Marini, ANNA MARIA; G., Greco; E., Novellino; Trincavelli, MARIA LETIZIA; Martini, Claudia
"Interaction at BzR of closed-chain anlogues of N-benzyl-indol-3-ylglyoxylylamide derivatives"
1999-01-01 G., Primofiore; DA SETTIMO PASSETTI, Federico; Marini, ANNA MARIA; Taliani, Sabrina; G., Greco; E., Novellino; Martini, Claudia; Trincavelli, MARIA LETIZIA
1,2,3-Triazole[4,5-d]pyridazines II. New Derivatives Tested on the Adenosine Receptors
1994-01-01 Biagi, Giuliana; Giorgi, Irene; Livi, Oreste; Scartoni, Valerio; Martini, Claudia; Tacchi, P; Merlino, Stefano; Pasero, Marco
1,2,3-Triazole[4,5-d]pyridazines IV. Preparation and Adenosine Receptor Binding of New 4-and /or 7-Aminoderivatives
1995-01-01 Biagi, G; Giorgi, Irene; Livi, O; Scartoni, V; Velo, S; Martini, Claudia; Senatore, G; Barili, P. L.; Lucacchini, Antonio
1,2,3-Triazolo[1,5-a][1,3]benzodiazepine a new heterocyclic system: Synthesis, benzodiazepine receptor binding and theoretical calculations
1996-01-01 Biagi, G; Giorgi, Irene; Livi, O; Scartoni, V; Velo, S; Desantis, B; Martinelli, Adriano; Martini, Claudia; Senatore, G.
1,2,3-Triazolo[1,5-a][1,4]- and 1,2,3-Triazolo[1,5-a][1,5]benzodiazepine derivatives: synthesis and benzodiazepine receptor binding.
1998-01-01 Bertelli, L; Biagi, G; Giorgi, Irene; Livi, O; Manera, Clementina; Scartoni, V; Martini, Claudia; Giannaccini, Gino; Trincavelli, MARIA LETIZIA; Barili, Pl
1,2,3-triazolo[1.5-a]quinazolines: synthesis, benzodiazepine receptor binding and theoretical calculations
1996-01-01 Biagi, G; Giorgi, Irene; Livi, O; Scartoni, V; Velo, S; DE SANCTIS, B; Martinelli, Adriano; Martini, Claudia; Senatore, G.
1,2,4-Triazolo[1,5-a]quinoxaline as a versatile tool for the design of selective human A3 adenosine receptor antagonists: synthesis, biological evaluation, and molecular modeling studies of 2-(hetero)aryl- and 2-carboxy-substituted derivatives
2005-01-01 Catarzi, D; Colotta, V; Varano, F; Lenzi, O; Filacchioni, G; Trincavelli, MARIA LETIZIA; Martini, Claudia; Montopoli, C; Moro, S.
1,2,4-Triazolo[1,5-a]quinoxaline derivatives and their simplified analogues as adenosine A3 receptor antagonists. Synthesis, structure-affinity relationships and molecular modeling studies.
2015-01-01 Catarzi, D; Varano, F; Poli, D; Squarcialupi, L; Betti, M; Trincavelli, MARIA LETIZIA; Martini, Claudia; Dal Ben, D; Thomas, A; Volpini, R; Colotta, V.
1,2,4-Triazolo[1,5-a]quinoxaline derivatives: synthesis and biological evaluation as adenosine receptor antagonists
2004-01-01 Catarzi, D.; Colotta, V.; Varano, F.; Filiacchioni, G.; Martini, Claudia; Trincavelli, MARIA LETIZIA; Lucacchini, Antonio
1,2,4-triazolo[4,3-a]quinoxalin-1-one moiety as an attractive scaffold to develop new potent and selective human A3 adenosine receptor antagonists: synthesis, pharmacological, and ligand-receptor modeling studies.
2004-01-01 Colotta, V.; Catarzi, D.; Varano, F.; Calabri, F. R.; Lenzi, O.; Filacchioni, G.; Martini, Claudia; Trincavelli, MARIA LETIZIA; Deflorian, F.; Moro, S.
1,2,4-Triazolo[4,3-a]quinoxalin-1-one: a versatile tool for the synthesis of potent and selective adenosine receptor antagonists
2000-01-01 Colotta, V; Catarzi, D; Varano, F; Cecchi, L; Filacchioni, G; Martini, Claudia; Trincavelli, MARIA LETIZIA; Lucacchini, Antonio
1,3-DIARYLPYRAZOLO[4,5-C]QUINOLIN-4-ONES AND 1,3-DIARYLPYRAZOLO[5,4-C]QUINOLIN-4-ONES .4. SYNTHESIS AND SPECIFIC-INHIBITION OF BENZODIAZEPINE RECEPTOR-BINDING
1987-01-01 Palazzino, G; Cecchi, L; Melani, F; Colotta, V; Filacchioni, G; Martini, Claudia; Lucacchini, Antonio
1-(3-AMINOPHENYL)-3-METHYL [1]BENZOPYRANO[2,3-C]PYRAZOL-4-ONE: A NEW SELECTIVE a2 ADENOSINE RECEPTOR ANTAGONIST.
1992-01-01 Colotta, V; Cecchi, L; Catarzi, D; Melani, F; Filacchioni, G; Martini, Claudia; Tacchi, P; Lucacchini, Antonio
18-kDa translocator protein association complexes in the brain: From structure to function
2020-01-01 Costa, B.; Da Pozzo, E.; Martini, C.
2 '-C-methyl analogues of selective adenosine receptor agonists: Synthesis and binding studies
1998-01-01 Franchetti, P; Cappellacci, L; Marchetti, S; Trincavelli, MARIA LETIZIA; Martini, Claudia; Mazzoni, MARIA ROSA; Lucacchini, Antonio; Grifantini, M.
2,3-butanedione inactivates the [H-3]nitrendipine binding sites, whereas diethylpyrocarbonate does not
1996-01-01 Costa, Barbara; Giusti, L.; Martini, Claudia; Lucacchini, Antonio
2- and 8-alkynyl-9-ethyladenines: synthesis and biological activity at human and rat adenosine receptors
2005-01-01 Volpini, R.; Costanzi, S.; Lambertucci, K.; Vittori, S.; Martini, Claudia; Trincavelli, MARIA LETIZIA; Klotz, K. N.; Cristalli, G.
2-(Benzimidazol-2-yl)quinoxalines: A Novel Class of selective Antagonists at Human A1 and A3 Adenosine Receptors Designed by 3D Database Searching
2005-01-01 Novellino, E.; Cosimelli, B.; Ehlardo, M.; Greco, G.; Iadanza, M.; Lavecchia, A.; Rimoli, M. G.; Sala, A.; DA SETTIMO, A.; Primofiore, G.; DA SETTIMO PASSETTI, Federico; Taliani, Sabrina; LA MOTTA, Concettina; Klotz, K. N.; Tuscano, D.; Trincavelli, MARIA LETIZIA; Martini, Claudia
2-Aryl-8-Azaadenosines: Structure-Activity Relationships in the Binding with A1 and A2 Receptors. A Comparison with the Corresponding 9-Benzyl-8-Azaadenines
1994-01-01 Biagi, G; Giorgi, Irene; Livi, O; Scartoni, V; Lucacchini, Antonio; Martini, Claudia; Tacchi, P.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
"Indol-3-ylglyoxylylamide derivatives probing the existence of a hydrogen acceptor/donor group in the S1 region of the benzodiazepine receptor binding site" | 1-gen-2000 | G., Primofiore; DA SETTIMO PASSETTI, Federico; Taliani, Sabrina; Marini, ANNA MARIA; G., Greco; E., Novellino; Trincavelli, MARIA LETIZIA; Martini, Claudia | |
"Interaction at BzR of closed-chain anlogues of N-benzyl-indol-3-ylglyoxylylamide derivatives" | 1-gen-1999 | G., Primofiore; DA SETTIMO PASSETTI, Federico; Marini, ANNA MARIA; Taliani, Sabrina; G., Greco; E., Novellino; Martini, Claudia; Trincavelli, MARIA LETIZIA | |
1,2,3-Triazole[4,5-d]pyridazines II. New Derivatives Tested on the Adenosine Receptors | 1-gen-1994 | Biagi, Giuliana; Giorgi, Irene; Livi, Oreste; Scartoni, Valerio; Martini, Claudia; Tacchi, P; Merlino, Stefano; Pasero, Marco | |
1,2,3-Triazole[4,5-d]pyridazines IV. Preparation and Adenosine Receptor Binding of New 4-and /or 7-Aminoderivatives | 1-gen-1995 | Biagi, G; Giorgi, Irene; Livi, O; Scartoni, V; Velo, S; Martini, Claudia; Senatore, G; Barili, P. L.; Lucacchini, Antonio | |
1,2,3-Triazolo[1,5-a][1,3]benzodiazepine a new heterocyclic system: Synthesis, benzodiazepine receptor binding and theoretical calculations | 1-gen-1996 | Biagi, G; Giorgi, Irene; Livi, O; Scartoni, V; Velo, S; Desantis, B; Martinelli, Adriano; Martini, Claudia; Senatore, G. | |
1,2,3-Triazolo[1,5-a][1,4]- and 1,2,3-Triazolo[1,5-a][1,5]benzodiazepine derivatives: synthesis and benzodiazepine receptor binding. | 1-gen-1998 | Bertelli, L; Biagi, G; Giorgi, Irene; Livi, O; Manera, Clementina; Scartoni, V; Martini, Claudia; Giannaccini, Gino; Trincavelli, MARIA LETIZIA; Barili, Pl | |
1,2,3-triazolo[1.5-a]quinazolines: synthesis, benzodiazepine receptor binding and theoretical calculations | 1-gen-1996 | Biagi, G; Giorgi, Irene; Livi, O; Scartoni, V; Velo, S; DE SANCTIS, B; Martinelli, Adriano; Martini, Claudia; Senatore, G. | |
1,2,4-Triazolo[1,5-a]quinoxaline as a versatile tool for the design of selective human A3 adenosine receptor antagonists: synthesis, biological evaluation, and molecular modeling studies of 2-(hetero)aryl- and 2-carboxy-substituted derivatives | 1-gen-2005 | Catarzi, D; Colotta, V; Varano, F; Lenzi, O; Filacchioni, G; Trincavelli, MARIA LETIZIA; Martini, Claudia; Montopoli, C; Moro, S. | |
1,2,4-Triazolo[1,5-a]quinoxaline derivatives and their simplified analogues as adenosine A3 receptor antagonists. Synthesis, structure-affinity relationships and molecular modeling studies. | 1-gen-2015 | Catarzi, D; Varano, F; Poli, D; Squarcialupi, L; Betti, M; Trincavelli, MARIA LETIZIA; Martini, Claudia; Dal Ben, D; Thomas, A; Volpini, R; Colotta, V. | |
1,2,4-Triazolo[1,5-a]quinoxaline derivatives: synthesis and biological evaluation as adenosine receptor antagonists | 1-gen-2004 | Catarzi, D.; Colotta, V.; Varano, F.; Filiacchioni, G.; Martini, Claudia; Trincavelli, MARIA LETIZIA; Lucacchini, Antonio | |
1,2,4-triazolo[4,3-a]quinoxalin-1-one moiety as an attractive scaffold to develop new potent and selective human A3 adenosine receptor antagonists: synthesis, pharmacological, and ligand-receptor modeling studies. | 1-gen-2004 | Colotta, V.; Catarzi, D.; Varano, F.; Calabri, F. R.; Lenzi, O.; Filacchioni, G.; Martini, Claudia; Trincavelli, MARIA LETIZIA; Deflorian, F.; Moro, S. | |
1,2,4-Triazolo[4,3-a]quinoxalin-1-one: a versatile tool for the synthesis of potent and selective adenosine receptor antagonists | 1-gen-2000 | Colotta, V; Catarzi, D; Varano, F; Cecchi, L; Filacchioni, G; Martini, Claudia; Trincavelli, MARIA LETIZIA; Lucacchini, Antonio | |
1,3-DIARYLPYRAZOLO[4,5-C]QUINOLIN-4-ONES AND 1,3-DIARYLPYRAZOLO[5,4-C]QUINOLIN-4-ONES .4. SYNTHESIS AND SPECIFIC-INHIBITION OF BENZODIAZEPINE RECEPTOR-BINDING | 1-gen-1987 | Palazzino, G; Cecchi, L; Melani, F; Colotta, V; Filacchioni, G; Martini, Claudia; Lucacchini, Antonio | |
1-(3-AMINOPHENYL)-3-METHYL [1]BENZOPYRANO[2,3-C]PYRAZOL-4-ONE: A NEW SELECTIVE a2 ADENOSINE RECEPTOR ANTAGONIST. | 1-gen-1992 | Colotta, V; Cecchi, L; Catarzi, D; Melani, F; Filacchioni, G; Martini, Claudia; Tacchi, P; Lucacchini, Antonio | |
18-kDa translocator protein association complexes in the brain: From structure to function | 1-gen-2020 | Costa, B.; Da Pozzo, E.; Martini, C. | |
2 '-C-methyl analogues of selective adenosine receptor agonists: Synthesis and binding studies | 1-gen-1998 | Franchetti, P; Cappellacci, L; Marchetti, S; Trincavelli, MARIA LETIZIA; Martini, Claudia; Mazzoni, MARIA ROSA; Lucacchini, Antonio; Grifantini, M. | |
2,3-butanedione inactivates the [H-3]nitrendipine binding sites, whereas diethylpyrocarbonate does not | 1-gen-1996 | Costa, Barbara; Giusti, L.; Martini, Claudia; Lucacchini, Antonio | |
2- and 8-alkynyl-9-ethyladenines: synthesis and biological activity at human and rat adenosine receptors | 1-gen-2005 | Volpini, R.; Costanzi, S.; Lambertucci, K.; Vittori, S.; Martini, Claudia; Trincavelli, MARIA LETIZIA; Klotz, K. N.; Cristalli, G. | |
2-(Benzimidazol-2-yl)quinoxalines: A Novel Class of selective Antagonists at Human A1 and A3 Adenosine Receptors Designed by 3D Database Searching | 1-gen-2005 | Novellino, E.; Cosimelli, B.; Ehlardo, M.; Greco, G.; Iadanza, M.; Lavecchia, A.; Rimoli, M. G.; Sala, A.; DA SETTIMO, A.; Primofiore, G.; DA SETTIMO PASSETTI, Federico; Taliani, Sabrina; LA MOTTA, Concettina; Klotz, K. N.; Tuscano, D.; Trincavelli, MARIA LETIZIA; Martini, Claudia | |
2-Aryl-8-Azaadenosines: Structure-Activity Relationships in the Binding with A1 and A2 Receptors. A Comparison with the Corresponding 9-Benzyl-8-Azaadenines | 1-gen-1994 | Biagi, G; Giorgi, Irene; Livi, O; Scartoni, V; Lucacchini, Antonio; Martini, Claudia; Tacchi, P. |