LAPUCCI, ANNALINA Statistiche

LAPUCCI, ANNALINA  

DIPARTIMENTO DI FARMACIA  

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Risultati 1 - 20 di 97 (tempo di esecuzione: 0.034 secondi).
Titolo Data di pubblicazione Autore(i) File
Locking PDK1 in DFG-out conformation through 2-oxo-indole containing molecules: Another tools to fight glioblastoma 1-gen-2016 Sestito, Simona; Daniele, Simona; Nesi, Giulia; Zappelli, Elisa; Di Maio, D; Marinelli, L; Digiacomo, Maria; Lapucci, Annalina; Martini, Claudia; Novellino, E; Rapposelli, Simona
Synthesis and In Vivo Imaging of N-(3-[11C]Methoxybenzyl)-2-(3-Methoxyphenyl)ethylaniline as a Potential Targeting Agent for P-glycoprotein 1-gen-2016 Petroni, Debora; Bartoli, Antonietta; Rapposelli, Simona; Digiacomo, Maria; Burchielli, Silvia; Nesi, Giulia; Lapucci, Annalina; Pardini, Silvia; Fucci, Sabrina; Macchia, Marco; Salvadori, Piero A.; Menichetti, Luca
Design and synthesis of 2-oxindole based multi-targeted inhibitors of PDK1/Akt signaling pathway for the treatment of glioblastoma multiforme 1-gen-2015 Sestito, Simona; Nesi, Giulia; Daniele, Simona; Martelli, Alma; Digiacomo, Maria; Borghini, Alice; Pietra, Daniele; Calderone, Vincenzo; Lapucci, Annalina; Falasca, Marco; Parrella, Paola; Notarangelo, Angelantonio; Breschi, MARIA CRISTINA; Macchia, Marco; Martini, Claudia; Rapposelli, Simona
Synthesis and evaluation of multi-functional NO-donor/insulin-secretagogue derivatives for the treatment of type II diabetes and its cardiovascular complications 1-gen-2015 Digiacomo, Maria; Martelli, Alma; Testai, Lara; Lapucci, Annalina; Breschi, MARIA CRISTINA; Calderone, Vincenzo; Rapposelli, Simona
Synthesis and pharmacological evaluation of multifunctional tacrine derivatives against several disease pathways of AD 1-gen-2015 Digiacomo, Maria; Chen, Ziwei; Wang, Shengnan; Lapucci, Annalina; Macchia, Marco; Yang, Xiaohong; Chu, Jiaqi; Han, Yifan; Pi, Rongbiao; Rapposelli, Simona
SAR study on arylmethyloxyphenyl scaffold: Looking for a P-gp nanomolar affinity 1-gen-2014 Nesi, Giulia; Colabufo, N. A.; Contino, M.; Perrone, M. G.; Digiacomo, Maria; Perrone, R.; Lapucci, Annalina; Macchia, Marco; Rapposelli, Simona
Synthesis and biological evaluation of (Hetero)aryl-methyloxyphenyl derivatives as potent P-glycoprotein modulating agents. 1-gen-2013 Nesi, Giulia; Colabufo, N. A.; Contino, M.; Perrone, M. G.; Digiacomo, Maria; Perrone, R.; Lapucci, Annalina; Macchia, Marco; Rapposelli, Simona
Synthesis of Novel 3,5-Disubstituted-2-oxindole Derivatives As Antitumor Agents against Human Nonsmall Cell Lung Cancer 1-gen-2013 Nesi, Giulia; Sestito, Simona; Mey, V.; Ricciardi, S.; Falasca, M.; Danesi, Romano; Lapucci, Annalina; Breschi, MARIA CRISTINA; Fogli, Stefano; Rapposelli, Simona
Targeting the upregulated PI3K-PDK1-Akt pathway: a drug discovery approach of treating cancer. 1-gen-2012 Nesi, Giulia; Danesi, Romano; Lapucci, Annalina; Ricciardi, S; Sestito, Simona; Rapposelli, Simona
Synthesis and Biological Evaluation of 2'-Oxo-2,3-dihydro-3'H-spiro[chromene-4,5'-[1,3]oxazolidin]3'il]acetic Acid Derivatives as Aldose reductase Inhibitors 1-gen-2011 Rapposelli, Simona; DA SETTIMO PASSETTI, Federico; Digiacomo, Maria; LA MOTTA, Concettina; Lapucci, Annalina; Sartini, Stefania; Vanni, M.
Synthesis, molecular docking and binding studies of selective serotonin transporter inhibitors 1-gen-2011 Nencetti, Susanna; Mazzoni, MARIA ROSA; Ortore, GABRIELLA MARIA PIA; Lapucci, Annalina; Giuntini, Janette; Orlandini, Elisabetta; Banti, Irene; Nuti, Elisa; Lucacchini, Antonio; Giannaccini, Gino; Rossello, Armando
Therapeutic potential of sulindac hydroxamic acid against human pancreatic and colonic cancer cells 1-gen-2010 Fogli, Stefano; Banti, I; Stefanelli, Fabio; Picchianti, L; Digiacomo, Maria; Macchia, Marco; Breschi, MARIA CRISTINA; Lapucci, Annalina
In vitro investigation of sulindac derivatives as potential anticancer agents 1-gen-2009 Fogli, Stefano; Banti, I; Digiacomo, Maria; Macchia, Marco; Lapucci, Annalina; Breschi, MARIA CRISTINA
Novel Transthyretin Amyloid Fibril Formation Inhibitors: Synthesis, Biological Evaluation, and X-Ray Structural Analysis 1-gen-2009 Palaninathan, S. K.; Mohamedmohaideen, N. N.; Orlandini, Elisabetta; Ortore, GABRIELLA MARIA PIA; Nencetti, Susanna; Lapucci, Annalina; Rossello, Armando; FREUNDLINCH JL, S; Sacchettini, J. C.
Synthesis and in-vitro antitumour activity of new naphthyridine derivatives on human pancreatic cancer cells 1-gen-2009 Banti, I; Nencetti, Susanna; Orlandini, Elisabetta; Lapucci, Annalina; Breschi, MARIA CRISTINA; Fogli, Stefano
Allosteric inhibition of (125I) ET-1 binding to ET(A) receptors by aldoxime and hydroxamic acid derivatives 1-gen-2008 Ahmed, M; Nencetti, Susanna; Mazzoni, MARIA ROSA; Porchia, F; Antonelli, F; Lapucci, Annalina
Allosteric inhibition of ET-1 binding to ETA receptors by aldoxime derivatives 1-gen-2008 Ahmed, Musa; Nencetti, Susanna; Mazzoni, MARIA ROSA; Porchia, Francesca; Antonelli, Federica; Lapucci, Annalina
Inhibition of [125] ET-1 binding to ETA receptors by salicilic acid dimers 1-gen-2008 Musa, Ahmed; Nencetti, Susanna; Mazzoni, MARIA ROSA; Francesca, Porchia; Federica, Antonelli; Lapucci, Annalina
Monoaryl-substituted Salicylaldoximes as Ligands for Estrogen Receptor Beta 1-gen-2008 Minutolo, Filippo; Bellini, R; Bertini, Simone; Carboni, I; Lapucci, Annalina; Pistolesi, L; Prota, G; Rapposelli, Simona; Solati, F; Tuccinardi, Tiziano; Martinelli, Adriano; Stossi, F; Carlson, K. E.; Katzenellenbogen, B. S.; Katzenellenbogen, J. A.; Macchia, Marco
Synthesis and AT1 affinity evaluation of benzamidophenyl analogs of known AT1 receptor ligands with similar aromatic skeleton 1-gen-2008 Rapposelli, Simona; Cuboni, S; Digiacomo, Maria; Lapucci, Annalina; Trincavelli, MARIA LETIZIA; Tuccinardi, Tiziano; Balsamo, A.