LAPUCCI, ANNALINA Statistiche
LAPUCCI, ANNALINA
DIPARTIMENTO DI FARMACIA
(E)-(methyloxyimino)acetamides as analogues of neuroleptic benzamides: Synthesis and D-2-dopaminergic binding affinity
1996-01-01 Lapucci, Annalina; Macchia, Marco; Orlandini, Elisabetta; Romagnoli, F; Rossello, Armando; Chiellini, Grazia; Cozzini, P; Domiano, P.
(Z)-(Methyloxyiminomethyl)ethanolamines. Effects of the configuration around the iminic double bond on the beta-adrenergic affinity of moim-type beta-adrenergic blocking agents
1995-01-01 Chiellini, Grazia; Lapucci, Annalina; Macchia, Marco; F., Romagnoli; Rossello, Armando; Nencetti, Susanna
1-(1-pirril)-3- ammino-2-propanoli N-sostituiti: sintesi e proprietà ß-adrenergiche
1989-01-01 Lapucci, Annalina; Nencetti, Susanna; Orlandini, Elisabetta; Rossello, Armando; Macchia, F; Breschi, MARIA CRISTINA; Ciucci, Ma; Martinotti, E.
2-(Methyleneaminoxy)methylmorpholine derivatives. Synthesis and antidepressant activity
1994-01-01 A., Balsamo; Lapucci, Annalina; Macchia, Marco; Martinelli, Adriano; Nencetti, Susanna; T., Cristina; Rossello, Armando
2-Imminossimetil morfoline attive sul sistema nervoso centrale. Sintesi e proprietà antidepressive.
1986-01-01 A., Balsamo; T., Cristina; Lapucci, Annalina; B., Macchia; F., Macchia; Martinelli, Adriano; Nencetti, Susanna; M., Riva
3-(Methyleneaminoxy)methylpiperidine derivatives as uptake inhibitors of biogenic amines in the brain synaptosomal fraction
1994-01-01 Balsamo, A; Lapucci, Annalina; Lucacchini, Antonio; Macchia, Marco; Martini, Claudia; Nardini, C; Nencetti, Susanna
3-(METHYLENEAMINOXY)METHYLPIPERIDINE DERIVATIVES AS UPTAKE INHIBITORS OF BIOGENIC-AMINES IN THE BRAIN SYNAPTOSOMAL FRACTION
1994-01-01 Balsamo, A; Lapucci, Annalina; Lucacchini, Antonio; Macchia, Marco; Martini, Claudia; Nardini, C; Nencetti, Susanna
3-[(2-Ethoxyphenoxy)methyl]piperidine derivatives. Synthesis and antidepressant activity
1987-01-01 Balsamo, A; Giorgi, Irene; Lapucci, Annalina; Lucacchini, Antonio; Macchia, B; Macchia, F; Martini, Claudia; Rossi, A.
3-[(aryl)(4-fluorobenzyloxy)methyl]piperidine derivatives: high-affinity ligands for the serotonin transporter
2007-01-01 Nencetti, Susanna; Demontis, GIAN CARLO ALFREDO GIUSEPPE; Mazzoni, MARIA ROSA; Betti, Laura; Banti, I; Rossello, Armando; Lapucci, Annalina
4-ARYLPIPERIDINE DERIVATIVES AND USE THEREOF FOR PREPARING A MEDICAMENT FOR THE TREATMENT OF CNS DISEASE
2006-01-01 Nencetti, Susanna; Lapucci, Annalina; Orlandini, Elisabetta; Balsamo, Aldo; Mazzoni, MARIA ROSA
Acidi benzilideneamminossipropionici sostituiti sul fenile. Sintesi e proprietà antiinfiammatorie.
1991-01-01 A., Balsamo; Lapucci, Annalina; B., Macchia; Martinelli, Adriano; Nencetti, Susanna; Orlandini, Elisabetta; Rossello, Armando; Soldani, G. M. e. n. g. o. z. z. i. G.; M., Baldacci
Allosteric inhibition of (125I) ET-1 binding to ET(A) receptors by aldoxime and hydroxamic acid derivatives
2008-01-01 Ahmed, M; Nencetti, Susanna; Mazzoni, MARIA ROSA; Porchia, F; Antonelli, F; Lapucci, Annalina
Allosteric inhibition of ET-1 binding to ETA receptors by aldoxime derivatives
2008-01-01 Ahmed, Musa; Nencetti, Susanna; Mazzoni, MARIA ROSA; Porchia, Francesca; Antonelli, Federica; Lapucci, Annalina
An anomalous effect of N-isopropyl substitution in determining beta-adrenergic activity
1988-01-01 B., Macchia; A., Balsamo; Lapucci, Annalina; F., Macchia; Manera, Clementina; Nencetti, Susanna; Breschi, MARIA CRISTINA; Lucacchini, Antonio; Martini, Claudia; E., Martinotti
An approach to the knowledge of the steric requirements for alpha-adrenoreceptor direct activation. alpha-Adrenergic properties of new 3-piperidinols
1981-01-01 Balsamo, A; Lapucci, Annalina; Macchia, Bruno; Macchia, Franco; Ceserani, Roberto; Longiave, Daniela
An interdisciplinary approach to the design of new structures active at the beta-adrenergic receptor. Aliphatic oxime ether derivatives
1985-01-01 Macchia, B; Balsamo, A; Lapucci, Annalina; Martinelli, Adriano; Macchia, F; Breschi, MARIA CRISTINA; Fantoni, B; Martinotti, E.
Antiherpes virus agents: A review
1993-01-01 Lapucci, Annalina; Macchia, Marco; Parkin, A.
Aryl-substituted methyleneaminoxymethyl (MAOM) analogues of diarylcyclopentenyl cyclooxygenase-2 inhibitors: effects of some structural modifications on their biological properties
2002-01-01 Balsamo, A; Coletta, I; Guglielmotti, A; Landolfi, C; Lapucci, Annalina; Mancini, F; Milanese, C; Minutolo, Filippo; Orlandini, Elisabetta; Ortore, GABRIELLA MARIA PIA; Pinza, M; Rapposelli, Simona
Chemistry of the Dihydrothiazine Ring Moiety of Cephalosporins. A Route to 3-Formoxymethyl-3-Cephem Derivatives
1981-01-01 Balsamo, A; Epifani, E; Giorgi, Irene; Lapucci, Annalina; Macchia, B; Macchia, F.
CONFORMATIONAL EFFECTS ON DRUG ACTIVITY .6. SYNTHESIS AND PHARMACOLOGICAL PROPERTIES OF 2-(PARANITROPHENYL) SUBSTITUTED MORPHOLINES
1975-01-01 Balsamo, A; Crotti, Paolo; Lapucci, Annalina; Macchia, B; Macchia, F; Deltacca, M; Mazzanti, L.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
(E)-(methyloxyimino)acetamides as analogues of neuroleptic benzamides: Synthesis and D-2-dopaminergic binding affinity | 1-gen-1996 | Lapucci, Annalina; Macchia, Marco; Orlandini, Elisabetta; Romagnoli, F; Rossello, Armando; Chiellini, Grazia; Cozzini, P; Domiano, P. | |
(Z)-(Methyloxyiminomethyl)ethanolamines. Effects of the configuration around the iminic double bond on the beta-adrenergic affinity of moim-type beta-adrenergic blocking agents | 1-gen-1995 | Chiellini, Grazia; Lapucci, Annalina; Macchia, Marco; F., Romagnoli; Rossello, Armando; Nencetti, Susanna | |
1-(1-pirril)-3- ammino-2-propanoli N-sostituiti: sintesi e proprietà ß-adrenergiche | 1-gen-1989 | Lapucci, Annalina; Nencetti, Susanna; Orlandini, Elisabetta; Rossello, Armando; Macchia, F; Breschi, MARIA CRISTINA; Ciucci, Ma; Martinotti, E. | |
2-(Methyleneaminoxy)methylmorpholine derivatives. Synthesis and antidepressant activity | 1-gen-1994 | A., Balsamo; Lapucci, Annalina; Macchia, Marco; Martinelli, Adriano; Nencetti, Susanna; T., Cristina; Rossello, Armando | |
2-Imminossimetil morfoline attive sul sistema nervoso centrale. Sintesi e proprietà antidepressive. | 1-gen-1986 | A., Balsamo; T., Cristina; Lapucci, Annalina; B., Macchia; F., Macchia; Martinelli, Adriano; Nencetti, Susanna; M., Riva | |
3-(Methyleneaminoxy)methylpiperidine derivatives as uptake inhibitors of biogenic amines in the brain synaptosomal fraction | 1-gen-1994 | Balsamo, A; Lapucci, Annalina; Lucacchini, Antonio; Macchia, Marco; Martini, Claudia; Nardini, C; Nencetti, Susanna | |
3-(METHYLENEAMINOXY)METHYLPIPERIDINE DERIVATIVES AS UPTAKE INHIBITORS OF BIOGENIC-AMINES IN THE BRAIN SYNAPTOSOMAL FRACTION | 1-gen-1994 | Balsamo, A; Lapucci, Annalina; Lucacchini, Antonio; Macchia, Marco; Martini, Claudia; Nardini, C; Nencetti, Susanna | |
3-[(2-Ethoxyphenoxy)methyl]piperidine derivatives. Synthesis and antidepressant activity | 1-gen-1987 | Balsamo, A; Giorgi, Irene; Lapucci, Annalina; Lucacchini, Antonio; Macchia, B; Macchia, F; Martini, Claudia; Rossi, A. | |
3-[(aryl)(4-fluorobenzyloxy)methyl]piperidine derivatives: high-affinity ligands for the serotonin transporter | 1-gen-2007 | Nencetti, Susanna; Demontis, GIAN CARLO ALFREDO GIUSEPPE; Mazzoni, MARIA ROSA; Betti, Laura; Banti, I; Rossello, Armando; Lapucci, Annalina | |
4-ARYLPIPERIDINE DERIVATIVES AND USE THEREOF FOR PREPARING A MEDICAMENT FOR THE TREATMENT OF CNS DISEASE | 1-gen-2006 | Nencetti, Susanna; Lapucci, Annalina; Orlandini, Elisabetta; Balsamo, Aldo; Mazzoni, MARIA ROSA | |
Acidi benzilideneamminossipropionici sostituiti sul fenile. Sintesi e proprietà antiinfiammatorie. | 1-gen-1991 | A., Balsamo; Lapucci, Annalina; B., Macchia; Martinelli, Adriano; Nencetti, Susanna; Orlandini, Elisabetta; Rossello, Armando; Soldani, G. M. e. n. g. o. z. z. i. G.; M., Baldacci | |
Allosteric inhibition of (125I) ET-1 binding to ET(A) receptors by aldoxime and hydroxamic acid derivatives | 1-gen-2008 | Ahmed, M; Nencetti, Susanna; Mazzoni, MARIA ROSA; Porchia, F; Antonelli, F; Lapucci, Annalina | |
Allosteric inhibition of ET-1 binding to ETA receptors by aldoxime derivatives | 1-gen-2008 | Ahmed, Musa; Nencetti, Susanna; Mazzoni, MARIA ROSA; Porchia, Francesca; Antonelli, Federica; Lapucci, Annalina | |
An anomalous effect of N-isopropyl substitution in determining beta-adrenergic activity | 1-gen-1988 | B., Macchia; A., Balsamo; Lapucci, Annalina; F., Macchia; Manera, Clementina; Nencetti, Susanna; Breschi, MARIA CRISTINA; Lucacchini, Antonio; Martini, Claudia; E., Martinotti | |
An approach to the knowledge of the steric requirements for alpha-adrenoreceptor direct activation. alpha-Adrenergic properties of new 3-piperidinols | 1-gen-1981 | Balsamo, A; Lapucci, Annalina; Macchia, Bruno; Macchia, Franco; Ceserani, Roberto; Longiave, Daniela | |
An interdisciplinary approach to the design of new structures active at the beta-adrenergic receptor. Aliphatic oxime ether derivatives | 1-gen-1985 | Macchia, B; Balsamo, A; Lapucci, Annalina; Martinelli, Adriano; Macchia, F; Breschi, MARIA CRISTINA; Fantoni, B; Martinotti, E. | |
Antiherpes virus agents: A review | 1-gen-1993 | Lapucci, Annalina; Macchia, Marco; Parkin, A. | |
Aryl-substituted methyleneaminoxymethyl (MAOM) analogues of diarylcyclopentenyl cyclooxygenase-2 inhibitors: effects of some structural modifications on their biological properties | 1-gen-2002 | Balsamo, A; Coletta, I; Guglielmotti, A; Landolfi, C; Lapucci, Annalina; Mancini, F; Milanese, C; Minutolo, Filippo; Orlandini, Elisabetta; Ortore, GABRIELLA MARIA PIA; Pinza, M; Rapposelli, Simona | |
Chemistry of the Dihydrothiazine Ring Moiety of Cephalosporins. A Route to 3-Formoxymethyl-3-Cephem Derivatives | 1-gen-1981 | Balsamo, A; Epifani, E; Giorgi, Irene; Lapucci, Annalina; Macchia, B; Macchia, F. | |
CONFORMATIONAL EFFECTS ON DRUG ACTIVITY .6. SYNTHESIS AND PHARMACOLOGICAL PROPERTIES OF 2-(PARANITROPHENYL) SUBSTITUTED MORPHOLINES | 1-gen-1975 | Balsamo, A; Crotti, Paolo; Lapucci, Annalina; Macchia, B; Macchia, F; Deltacca, M; Mazzanti, L. |