CINECA IRIS Institutional Research Information System

LAPUCCI, ANNALINA
 Distribuzione geografica
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Continente #
NA - Nord America 5.803
EU - Europa 2.557
AS - Asia 1.202
AF - Africa 67
SA - Sud America 34
OC - Oceania 5
Continente sconosciuto - Info sul continente non disponibili 1
Totale 9.669
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Nazione #
US - Stati Uniti d'America 5.628
IT - Italia 763
SE - Svezia 585
CN - Cina 495
DE - Germania 365
SG - Singapore 272
BG - Bulgaria 259
TR - Turchia 249
CA - Canada 173
UA - Ucraina 138
GB - Regno Unito 119
FI - Finlandia 116
VN - Vietnam 65
IN - India 58
FR - Francia 54
CH - Svizzera 53
CI - Costa d'Avorio 37
HK - Hong Kong 35
BR - Brasile 31
RU - Federazione Russa 30
BE - Belgio 21
SN - Senegal 16
PL - Polonia 13
CZ - Repubblica Ceca 9
GR - Grecia 8
JP - Giappone 6
TW - Taiwan 6
AT - Austria 5
BJ - Benin 5
KR - Corea 4
ZA - Sudafrica 4
AU - Australia 3
NL - Olanda 3
BY - Bielorussia 2
EC - Ecuador 2
ES - Italia 2
HU - Ungheria 2
IE - Irlanda 2
IQ - Iraq 2
IR - Iran 2
MX - Messico 2
NG - Nigeria 2
NZ - Nuova Zelanda 2
RO - Romania 2
RS - Serbia 2
SC - Seychelles 2
BD - Bangladesh 1
BN - Brunei Darussalam 1
CO - Colombia 1
DK - Danimarca 1
EU - Europa 1
HR - Croazia 1
ID - Indonesia 1
IL - Israele 1
LB - Libano 1
NO - Norvegia 1
PK - Pakistan 1
PS - Palestinian Territory 1
PT - Portogallo 1
SA - Arabia Saudita 1
TN - Tunisia 1
Totale 9.669
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Città #
Woodbridge 931
Ann Arbor 730
Houston 536
Chandler 464
Fairfield 426
Santa Clara 291
Sofia 258
Serra 249
Ashburn 248
Izmir 196
Milan 179
Jacksonville 175
Beijing 174
Ottawa 160
Wilmington 157
Seattle 149
Singapore 135
Cambridge 127
New York 121
Princeton 112
Boardman 102
Lawrence 95
Medford 94
Nanjing 91
Des Moines 69
Dearborn 67
Bern 51
Istanbul 48
Boulder 45
Dong Ket 43
Abidjan 37
Nanchang 33
Marseille 30
Hong Kong 28
Jüchen 27
Redwood City 26
London 24
Brussels 21
Frankfurt am Main 21
San Diego 21
Florence 20
Ogden 18
Tianjin 18
Kunming 17
Norwalk 17
Auburn Hills 16
Bremen 16
Dakar 16
Changsha 15
Grafing 15
Nürnberg 15
Rome 15
Hefei 13
Shenyang 13
Dallas 12
Fuzhou 12
Los Angeles 12
Warsaw 12
Hebei 11
Jiaxing 10
Shanghai 10
Lancaster 9
Orange 9
Pune 9
Hyderabad 8
Padova 8
Hangzhou 7
Fremont 6
Indiana 6
Nottingham 6
Phoenix 6
Taipei 6
Washington 6
Brno 5
Cerveteri 5
Chicago 5
Cotonou 5
Düsseldorf 5
Manchester 5
Pisa 5
Quanzhou 5
San Francisco 5
Tokyo 5
Vienna 5
Augusta 4
Chengdu 4
Falls Church 4
Guangzhou 4
Haikou 4
Johannesburg 4
San Jose 4
Verona 4
Wuhan 4
Zhengzhou 4
Belo Horizonte 3
Changchun 3
Chongqing 3
Jinan 3
Kocaeli 3
Lanzhou 3
Totale 7.293
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Nome #
Design and synthesis of 2-oxindole based multi-targeted inhibitors of PDK1/Akt signaling pathway for the treatment of glioblastoma multiforme 220
Synthesis of Novel 3,5-Disubstituted-2-oxindole Derivatives As Antitumor Agents against Human Nonsmall Cell Lung Cancer 217
An approach to the knowledge of the steric requirements for alpha-adrenoreceptor direct activation. alpha-Adrenergic properties of new 3-piperidinols 173
Locking PDK1 in DFG-out conformation through 2-oxo-indole containing molecules: Another tools to fight glioblastoma 162
Synthesis and evaluation of multi-functional NO-donor/insulin-secretagogue derivatives for the treatment of type II diabetes and its cardiovascular complications 160
3-[(aryl)(4-fluorobenzyloxy)methyl]piperidine derivatives: high-affinity ligands for the serotonin transporter 155
SYNTHESIS AND EVALUATION OF THE PHARMACOLOGICAL ACTIVITY OF RIGID ANALOGUES OF SYMPATHOMIMETIC DERIVED FROM BICYCLO[2.2.1]HEPTANE 151
3-(METHYLENEAMINOXY)METHYLPIPERIDINE DERIVATIVES AS UPTAKE INHIBITORS OF BIOGENIC-AMINES IN THE BRAIN SYNAPTOSOMAL FRACTION 149
Enantiopure 3-(arylmethylidene)aminoxy-2-methylpropionic acids: synthesis and antiinflammatory properties 148
Synthesis and AT1 affinity evaluation of benzamidophenyl analogs of known AT1 receptor ligands with similar aromatic skeleton 146
CONFORMATIONALLY RESTRAINED ANALOGS OF SYMPATHOMIMETIC CATECHOLAMINES - SYNTHESIS AND ADRENERGIC ACTIVITY OF TETRAHYDROBENZOCYCLOHEPTENE DERIVATIVES 144
Inhibition of [125] ET-1 binding to ETA receptors by salicilic acid dimers 142
3-(Methyleneaminoxy)methylpiperidine derivatives as uptake inhibitors of biogenic amines in the brain synaptosomal fraction 139
Structure of 2-hydroxy-3-isopropylaminopropyl 3,4-methylenedioxybenzoate hydrochloride 138
Role of the acyloxymethyl moiety in eliciting the adrenergic ß-blocking activity of 3-acyloxypropanolamines 134
4-ARYLPIPERIDINE DERIVATIVES AND USE THEREOF FOR PREPARING A MEDICAMENT FOR THE TREATMENT OF CNS DISEASE 130
Synthesis and in-vitro antitumour activity of new naphthyridine derivatives on human pancreatic cancer cells 129
SYNTHESIS, ANTIINFLAMMATORY ACTIVITY AND MOLECULAR-ORBITAL STUDIES OF A SERIES OF BENZYLIDENEAMINOXYPROPIONIC ACIDS SUBSTITUTED ON THE PHENYL RING 128
Synthesis and In Vivo Imaging of N-(3-[11C]Methoxybenzyl)-2-(3-Methoxyphenyl)ethylaniline as a Potential Targeting Agent for P-glycoprotein 127
SYNTHESIS AND EVALUATION OF THE PHARMACOLOGICAL ACTIVITY OF RIGID ANALOGS OF SYMPATHOMIMETIC CATECHOLAMINES DERIVED FROM BICYCLO[2.2.1]HEPTANE 126
Conformationally restrained analogues of sympathomimetic catecholamines: Synthesis and adrenergic activity of 5,6- and 6,7-dihydroxy-3,4-dihydrospiro[naphthalen-1(2H)-2′,5′- morpholines] 125
Conformationally Restrained Analogs of Sympathomimetic Catecholamines. Synthesis, Conformational Analysis, and Adrenergic Activity of Isochroman Derivatives 125
Sintesi e proprietà farmacologiche di analoghi semirigidi morfolinici e piperidinici di catecolamine simpatomimetiche. Modelli sterici per l'attivazione diretta dei recettori a- e ß-adrenergici. 124
Synthesis and β-adrenergic properties of tetrahydronaphthalene analogs of dichloroisoproterenol 124
Conformational effects on the activity of drugs. 7. Synthesis and pharmacological properties of 2-(p-nitrophenyl)-substituted morpholines 123
SAR study on arylmethyloxyphenyl scaffold: Looking for a P-gp nanomolar affinity 123
3-[(2-Ethoxyphenoxy)methyl]piperidine derivatives. Synthesis and antidepressant activity 122
An interdisciplinary approach to the design of new structures active at the beta-adrenergic receptor. Aliphatic oxime ether derivatives 120
2-(Methyleneaminoxy)methylmorpholine derivatives. Synthesis and antidepressant activity 119
Synthesis and adrenergic beta-blocking activity of diastereoisomeric 3-(p-nitrophenyl)-6-methyl-3-piperidinols 119
Synthesis and adrenergic ß-blocking activity of (oxypropanolamino)-substituted [(benzylideneamino)oxy]propanolamines 116
MOLECULAR DESIGN, SYNTHESIS, AND ANTIINFLAMMATORY ACTIVITY OF A SERIES OF BETA-AMINOXYPROPIONIC ACIDS 114
Synthesis and affinity for serotonin and dopamine transporters of some benzophenone oxime ether derivatives 114
Novel Transthyretin Amyloid Fibril Formation Inhibitors: Synthesis, Biological Evaluation, and X-Ray Structural Analysis 114
(Z)-(Methyloxyiminomethyl)ethanolamines. Effects of the configuration around the iminic double bond on the beta-adrenergic affinity of moim-type beta-adrenergic blocking agents 113
Targeting the upregulated PI3K-PDK1-Akt pathway: a drug discovery approach of treating cancer. 109
Synthesis, Antifungal Activity, and Molecular Modeling Studies of New Inverted Oxime Ethers of Oxiconazole 109
ROLE OF THE (ACYLOXY)METHYL MOIETY IN ELICITING THE ADRENERGIC BETA-BLOCKING ACTIVITY OF 3-(ACYLOXY)PROPANOLAMINES 109
Therapeutic potential of sulindac hydroxamic acid against human pancreatic and colonic cancer cells 109
1-(1-pirril)-3- ammino-2-propanoli N-sostituiti: sintesi e proprietà ß-adrenergiche 108
Synthesis and COX2 inhibitory properties of N-Phenyl-and N-benzyl-substituted amides of 2-(4-methylsulfonylphenyl)cyclopent-1-ene-1-carboxylic acid and of their pyrazole, thiophene, and isoxazole analogs 106
Aryl-substituted methyleneaminoxymethyl (MAOM) analogues of diarylcyclopentenyl cyclooxygenase-2 inhibitors: effects of some structural modifications on their biological properties 105
Nuovi agenti ß-bloccanti: Derivati propanolamminici di eteri di ossime completamente alifatiche 103
Sintesi e proprietà beta-adrenergiche di [(benzilideneammino)ossi] propanolammine orto-ossipropanolammine sostituite chirali, 103
null 103
Synthesis and ß-Adrenergic Properties Of (Z)-N-[3-(Alkylamino)-2-hydroxypropilidene](aryl-methyloxy)amines: Effects Of The Configuration Around The Methyloxyiminomethyl(MOIM) Double Bond On The Biopharmacological Properties Of MOIM-type ß-Blocking Agents 102
Conformationally restrained analogs of sympathomimetic catecholamine. Synthesis and adrenergic activity of tetrahydrobenzocycloheptene derivatives 102
CONFORMATIONAL EFFECTS ON THE ACTIVITY OF DRUGS .13. A REVISION OF PREVIOUSLY PROPOSED MODELS FOR THE ACTIVATION OF ALPHA-ADRENERGIC AND BETA-ADRENERGIC RECEPTORS 101
Structure-activity relationship in cinnamamides. 3. Synthesis and anticonvulsant activity evaluation of some derivatives of (E)- and (Z)-m-(trifluoromethyl)cinnamamide 98
Conformational effects on the activity of drugs. Synthesis and adrenergic properties of 2-methyl-substituted 3-(3,4- dihydroxyphenyl)-3-piperidinols 97
Sintesi e attività recettoriale adrenergica di analoghi tetraidronaftalenici di catecolamine simpatomimetiche 94
Synthesis and pharmacological evaluation of multifunctional tacrine derivatives against several disease pathways of AD 94
Allosteric inhibition of ET-1 binding to ETA receptors by aldoxime derivatives 92
In vitro investigation of sulindac derivatives as potential anticancer agents 91
Uncommon formation of spiro orthoesters in the bromomethoxylation reaction of a 4-[(aroyloxy)methyl]-3-cephem derivative 91
Effetti conformazionali sull'attività dei farmaci. Sintesi e proprietà farmacologiche di cis-2-aril-3-metilmorfoline 88
Conformational effects on the activity of drugs. Synthesis and a and ß-adrenergic receptor activity of new terahydronaphthalene analogs of sympathomimetic catecholamines 88
Synthesis and biological evaluation of (Hetero)aryl-methyloxyphenyl derivatives as potent P-glycoprotein modulating agents. 88
Synthesis and evaluation of beta3-adrenergic affinity of new oximethereal derivative 86
Synthesis and inhibitory activity towards human leukocyte elastase of new 7 alpha-methoxy and 7 alpha-chloro (2-acyloxymethyl) cephem derivatives 86
(E)-(methyloxyimino)acetamides as analogues of neuroleptic benzamides: Synthesis and D-2-dopaminergic binding affinity 86
Conformational effects on the activity of drugs. 11. Stereostructural models for the direct activation of the a- and ß-adrenergic receptor 84
Conformational effects on the activity of drugs. 13. A revision of previously proposed models for the activation of a- and ß-adrenergic receptors 82
Chemistry of the Dihydrothiazine Ring Moiety of Cephalosporins. A Route to 3-Formoxymethyl-3-Cephem Derivatives 82
Effetti conformazionali sull'attività dei farmaci. Sintesi e valutazione dell'attività farmacologica di analoghi rigidi di catecolamine simpatomimetiche derivati dal norbornano 81
Synthesis and adrenergic beta-blocking activity of ortho-, meta- and para-oxypropanolamino-substituted [(benzylideneamino)oxy]propanolamines. 81
SYNTHESIS AND BETA-ADRENERGIC ACTIVITY OF NEW COMPLETELY ALIPHATIC 3-(METHYLENEAMINOXY)PROPANOLAMINE DERIVATIVES 81
Conformational effects on the activity of drugs. 10. Synthesis, conformation, and pharmacological properties of 1-(2,5-dimethoxyphenyl)-2-aminoethanols and their morpholine analogues 81
Synthesis and pharmacological activity of 1-phenyl-2-oxa-5-azabicyclo[4.4.0]decane derivatives 80
Sintesi ed attività adrenergica di analoghi ciclici dell’1-(2,5-dimetossifenil)-2-amminoetanolo 78
Oximethereal piperidinic derivatives: synthesis and affinity for serotonin and dopamine transporters 77
Synthesis and antimicrobial properties of substituted ß-aminoxypropionyl penicillins and cephalosporins 76
An anomalous effect of N-isopropyl substitution in determining beta-adrenergic activity 75
SYNTHESIS AND BETA-ADRENERGIC ACTIVITY OF A SERIES OF 3-(SUBSTITUTED-BENZYLIDENEAMINOXY)PROPANOLAMINE DERIVATIVES 74
Monoaryl-substituted Salicylaldoximes as Ligands for Estrogen Receptor Beta 73
Sintesi ed attività α- e ß-adrenergica di analoghi benzocicloeptanici di catecolamine simpatomimetiche 72
Antiherpes virus agents: A review 71
SYNTHESIS AND AFFINITY FOR SEROTONIN TRANSPORTER OF NEW PIPERIDINE BASED BIVALENT LIGANDS 70
Synthesis and ß-adrenergic properties of tetrahydronaphthalene analogs of dichloroisoproterenol 70
Synthesis and binding affinity at beta-adrenergic receptors of semirigid dichloroisoproterenol analogues, 70
Acidi benzilideneamminossipropionici sostituiti sul fenile. Sintesi e proprietà antiinfiammatorie. 69
Synthesis and Biological Evaluation of 2'-Oxo-2,3-dihydro-3'H-spiro[chromene-4,5'-[1,3]oxazolidin]3'il]acetic Acid Derivatives as Aldose reductase Inhibitors 67
Conformationally restrained analogues of sympathomimetic catecholamines. Synthesis and adrenergic activity of 5,6- and 6,7-dihydroxy-3,4-dihydrospiro[naphthalen-1(2H)-2',5'-morpholines] 65
Sintesi e proprietà inibitrici nei confronti delle cicloossigenasi di ammidi dell'acido 2-(4-metilsulfonilfenil)-1-ciclopentenico e di suoi analoghi eteroaromatici 64
Allosteric inhibition of (125I) ET-1 binding to ET(A) receptors by aldoxime and hydroxamic acid derivatives 64
Derivati della 3-imminossimetilpiperidina inibitori dell’uptake delle monoammine nelle frazioni sinaptosomiali cerebrali. 63
Sintesi e affinità per il trasportatore della serotonina di nuovi derivati piperidinici ossimeterei 60
Sintesi e proprietà alfa-adrenergiche di derivati cromanici, quali analoghi conformazionalmente ristretti dell’1-(2,5-dimetossifenil)-2-amminoetanolo 59
Synthesis and biological evaluation of sulindac derivatives as potential anticancer agents 58
Synthesis and pharmacological properties of cis-2-(2,5-dimethoxyphenyl)-3-methylmorpholine and its N-isopropyl derivative 57
2-Imminossimetil morfoline attive sul sistema nervoso centrale. Sintesi e proprietà antidepressive. 55
Sintesi, conformazione e proprietà farmacologiche di 1-(2,5-dimetossi fenil)-2-amminoetanoli e dei loro analoghi morfolinici. Un contributo alla conoscenza delle richieste steriche del recettore a-adrenergico 55
Derivati 4-arilpiperidinici e loro uso per la preparazione di un medicamento per il trattamento di disordini del SNC 50
Synthesis and stereochemistry of (Z)- and (E)-(3,4,5-trimethoxy)-a,ß-dimethylcinnamic acids and diastereoisomeric intermediate ß-hydroxy esters 48
CONFORMATIONAL EFFECTS ON DRUG ACTIVITY .6. SYNTHESIS AND PHARMACOLOGICAL PROPERTIES OF 2-(PARANITROPHENYL) SUBSTITUTED MORPHOLINES 48
Sintesi e stereochimica degli acidi (Z)- e (E)-(3,4,5-trimetossi)-alfa,beta-dimetilcinnamico e dei beta-idrossiesteri diastereoisomeri intermedi. 46
Nuovi derivati piperidinici: sintesi e proprietà biologiche 41
Synthesis, molecular docking and binding studies of selective serotonin transporter inhibitors 23
Totale 9.811
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Categoria #
all - tutte 24.797
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 24.797
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2019/2020891 0 0 0 0 116 170 162 81 117 94 116 35
2020/2021665 53 22 66 42 98 32 52 80 54 51 24 91
2021/20221.160 22 80 17 91 227 135 26 52 49 42 77 342
2022/20231.328 195 154 105 142 136 194 16 83 210 11 70 12
2023/2024848 128 91 113 47 95 155 38 30 13 21 24 93
2024/2025758 14 119 45 196 384 0 0 0 0 0 0 0
Totale 9.811